Meibom, Daniel

Solution Conformations Shed Light on PROTAC Cell Permeability

Atilaw, Y., Poongavanam, V., Svensson Nilsson, C., Nguyen, D., Giese, A., Meibom, D., Erdelyi, M., & Kihlberg, J. (2021) · ACS Medicinal Chemistry Letters

Protein Degradation and InhibitorsChemical Synthesis and Analysis

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Freezing the Bioactive Conformation to Boost Potency: The Identification of BAY 85‐8501, a Selective and Potent Inhibitor of Human Neutrophil Elastase for Pulmonary Diseases

von Nussbaum, F., Li, V. M. ‐., Allerheiligen, S., Anlauf, S., Bärfacker, L., Bechem, M., Delbeck, M., Fitzgerald, M. F., Gerisch, M., Gielen‐Haertwig, H., et al. (2015) · ChemMedChem

Protease and Inhibitor MechanismsEnzyme function and inhibition

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