Petros, Andrew M.

Structural biology of the Bcl-2 family of proteins

Petros, A. M., Olejniczak, E. T., & Fesik, S. W. (2004) · Biochimica et Biophysica Acta (BBA) - Molecular Cell Research

Cell death mechanisms and regulationEnzyme Structure and Function

Cited by 745

The EED protein–protein interaction inhibitor A-395 inactivates the PRC2 complex

He, Y., Selvaraju, S., Curtin, M. L., Jakob, C. G., Zhu, H., Comess, K. M., Shaw, B., The, J., Lima-Fernandes, E., Szewczyk, M. M., et al. (2017) · Nature Chemical Biology

Epigenetics and DNA MethylationCancer-related gene regulation

Cited by 224

Discovery and Development of Potent and Selective Inhibitors of Histone Methyltransferase G9a

Sweis, R. F., Pliushchev, M., Brown, P. J., Guo, J., Li, F., Maag, D., Petros, A. M., Soni, N. B., Tse, C., Vedadi, M., et al. (2014) · ACS Medicinal Chemistry Letters

Epigenetics and DNA MethylationCancer-related gene regulation

Cited by 193

Structure-Guided Design of a Series of MCL-1 Inhibitors with High Affinity and Selectivity

Bruncko, M., Wang, L., Sheppard, G. S., Phillips, D. C., Tahir, S. K., Xue, J., Erickson, S., Fidanze, S., Fry, E., Hasvold, L., et al. (2015) · Journal of Medicinal Chemistry

Cell death mechanisms and regulationComputational Drug Discovery Methods

Cited by 164

Fragment-Based Discovery of an Apolipoprotein E4 (apoE4) Stabilizer

Petros, A. M., Korepanova, A., Jakob, C. G., Qiu, W., Panchal, S. C., Wang, J., Dietrich, J. D., Brewer, J. T., Pohlki, F., Kling, A., et al. (2019) · Journal of Medicinal Chemistry

Alzheimer's disease research and treatmentsProtein Interaction Studies and Fluorescence Analysis

Cited by 32