Whitty, Adrian

The resurgence of covalent drugs

Singh, J., Petter, R. C., Baillie, T. A., & Whitty, A. (2011) · Nature Reviews Drug Discovery

Click Chemistry and ApplicationsProtein Degradation and Inhibitors

Cited by 1,873

Structural and Functional Differences Between Glycosylated and Non-glycosylated Forms of Human Interferon-β (IFN-β)

Runkel, L., Meier, W., Pepinsky, R. B., Karpusas, M., Whitty, A., Kimball, K., Brickelmaier, M., Muldowney, C., Jones, W., & Goelz, S. E. (1998) · Pharmaceutical Research

interferon and immune responsesMultiple Sclerosis Research Studies

Cited by 304

The road less traveled: modulating signal transduction enzymes by inhibiting their protein–protein interactions

Arkin, M. R., & Whitty, A. (2009) · Current Opinion in Chemical Biology

Protein Kinase Regulation and GTPase SignalingChemical Synthesis and Analysis

Cited by 190

Comprehensive Experimental and Computational Analysis of Binding Energy Hot Spots at the NF-κB Essential Modulator/IKKβ Protein–Protein Interface

Golden, M. S., Cote, S. M., Sayeg, M., Zerbe, B. S., Villar, E. A., Beglov, D., Sazinsky, S. L., Georgiadis, R. M., Vajda, S., Kozakov, D., et al. (2013) · Journal of the American Chemical Society

NF-κB Signaling PathwaysComputational Drug Discovery Methods

Cited by 47