Dicaffeoyltartaric Acid and Dicaffeoylquinic Acid HIV Integrase Inhibitors
Abstract
This chapter contains sections titled: Introduction Discovery Characterization of L-CA as a Selective IN Inhibitor Controversy Surrounding In Vivo Site of Action For L-CA Mechanisms of Viral Resistance Stucture-Activity Relationship Studies L-CA in Combination with Reverse Transcriptase and Protease Inhibitors Summary Acknowledgments References
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- Authors
- Crosby, D. C., & Robinson, W. E.
- Affiliations
- University of California, Irvine (US)
- Venue
- HIV‐1 Integrase
- Publisher
- Wiley
- Published
- 2011-09-09
- Pages
- 341-362
- OpenAlex
- W1569339539
- Cited by
- 2
- References
- 2
- Citations by year
- 2015: 1 · 2012: 1
- Type
- other
- Language
- en
- Open access
- closed
- Topics
- Health Sciences › Medicine › Infectious Diseases › HIV/AIDS drug development and treatment
- Life Sciences › Immunology and Microbiology › Virology › HIV Research and Treatment
- Health Sciences › Medicine › Oncology › Drug Transport and Resistance Mechanisms
- Keywords
- dicaffeoylquinic acids, HIV integrase inhibitors, integrase inhibitors, virus resistance, structure-activity relationship, reverse transcriptase inhibitors, protease inhibitors, highly active antiretroviral therapy
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