Structure–Activity Studies in a Family of β‐Hairpin Protein Epitope Mimetic Inhibitors of the p53–HDM2 Protein–Protein Interaction

Fasan, Rudi, Dias, Ricardo L. A., Moehle, Kerstin, Zerbe, Oliver, Obrecht, Daniel, Mittl, Peer R. E., Grütter, Markus G., Robinson, John A.·2006·ChemBioChem

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  10. Protein–Protein Interaction Inhibitors in Cancer
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  11. Targeting the MDM2–p53 Protein–Protein Interaction
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  14. Peptidomimetics of α‐Helical and β‐Strand Protein Binding Epitopes
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  16. β-Hairpin Peptidomimetics for Protein-Protein Interaction Inhibition
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  17. Lp...π Interactions involving π-systems with different degrees of electron density delocalization: uracil and isocyanurate
    Julia К. Voronina, Igor A. Litvinov · 2015 · Russian Chemical Bulletin
  18. Disrupting Protein–Protein Interfaces Using GRID Molecular Interaction Fields
    Simon Cross, Massimo Baroni, Francesco Ortuso, Stefano Alcaro, Gabriele Cruciani · 2013 · Springer eBooks
  19. Macrocyclic Organo‐Peptide Hybrids by Intein‐Mediated Ligation: Synthesis and Applications
    John R. Frost, Rudi Fasan · 2017 · Wiley eBooks
  20. Inhibition of the MDM2/p53 Interaction Design, Synthesis and Evaluation of MDM2 Inhibitors
    Mariell Pettersson · 2015 · Gothenburg University Publications Electronic Archive (Gothenburg University)
  21. Discovery of Inhibitors of Protein–Protein Interactions by Screening Chemical Libraries
    Carlos Garcı́a-Echeverrı́a · 2010 · Wiley eBooks
  22. Accurate Docking is Achieved by Decoupling Systematic Sampling from Scoring
    Jianwen A. Feng · 2009 · Open Scholarship Institutional Repository (Washington University in St. Louis)
  23. Parallel Interactions of Aromatic Molecules at Large Horizontal Displacements
    Dušan P. Malenov, Snežana D. Zarić · 2016
  24. 17 The protein epitope mimetic approach to protein-protein interaction inhibitors
    John A. Robinson, Kerstin Moehle · 2011 · De Gruyter eBooks
  25. Mit organischen Substanzen hemmen
    Thorsten Berg · 2016 · Nachrichten aus der Chemie
  26. Interface Peptides
    Mark W. Peczuh, Richard T. Desmond · 2010
  27. Diameter Is a Key 3D Characteristic for Assessments of Efficient Inhibitors of Protein–Protein Interactions
    Masakazu Nakadai, Shuta Tomida · 2020 · Journal of Chemical Information and Modeling
  28. Solvent effects on the NMR shieldings of stacked DNA base pairs
    Fernando A. Martínez, Natalia S. Adler, Claudio N. Cavasotto, Gustavo A. Aucar · 2022 · Physical Chemistry Chemical Physics
  29. Protein-protein interaction inhibitors in cancer
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  30. BindingDB Entry 50012111: hDM2 protein-binding peptides screened from stapled α-helical peptide phage display libraries with different types of staple linkers.
    BindingDB · 2022 · UC San Diego
  31. BindingDB Entry 3460: N-acylpolyamine inhibitors of HDM2 and HDMX binding to p53.
    BindingDB · 2009 · UC San Diego
  32. BindingDB Entry 50046974: Peptide-based inhibitors of protein-protein interactions.
    BindingDB · 2017 · UC San Diego
  33. BindingDB Entry 50009576: Selective Targeting of Integrin αvβ8 by a Highly Active Cyclic Peptide.
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  34. BindingDB Entry 50040300: An ultrahigh affinity d-peptide antagonist Of MDM2.
    BindingDB · 2013 · UC San Diego