50 years of oral lipid-based formulations: provenance, progress and future perspectives

Feeney, Orlagh M., Crum, Matthew F., McEvoy, Claire L., Trevaskis, Natalie L., Williams, Hywel D., Pouton, Colin W., Charman, William N., Bergström, Christel A.S. +1 more·2016·Advanced Drug Delivery Reviews

DOI 10.1016/j.addr.2016.04.007

Cited by (432)

Items 101–200 of 432

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The artificial membrane insert system as predictive tool for formulation performance evaluation
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Development of ternary solid dispersions with hydrophilic polymer and surface adsorbent for improving dissolution rate of carbamazepine
Tanja Vojinović, Djordje P. Medarević, Edina Vranić, Zorica Potpara, Marko Krstić, Jelena Djuriš, Svetlana R. Ibric · 2018 · Saudi Pharmaceutical Journal
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Espérance Moine, Philippe Brabet, Laurent Guillou, Thierry Durand, Joseph Vercauteren, Céline Crauste · 2018 · Antioxidants
In Vitro Evaluation of Self-Nano-Emulsifying Drug Delivery Systems (SNEDDS) Containing Room Temperature Ionic Liquids (RTILs) for the Oral Delivery of Amphotericin B
Eleni Kontogiannidou, Thomas Meikopoulos, Helen Gika, Emmanuel Panteris, Ioannis S. Vizirianakis, Anette Müllertz, Dimitrios G. Fatouros · 2020 · Pharmaceutics
From Quantum Chemistry to Prediction of Drug Solubility in Glycerides
Jochem Alsenz, Martin Kuentz · 2019 · Molecular Pharmaceutics
A Retrospective Biopharmaceutical Analysis of >800 Approved Oral Drug Products: Are Drug Properties of Solid Dispersions and Lipid-Based Formulations Distinctive?
Harriet Bennett-Lenane, Joseph P. O’Shea, Caitríona M. O’Driscoll, Brendan T. Griffin · 2020 · Journal of Pharmaceutical Sciences
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Alskär, Linda C., Parrow, Albin, Keemink, Janneke, Johansson, Pernilla, Abrahamsson, Bertil, Bergström, Christel A.S. · 2019 · Journal of Controlled Release
Lipid-Based Formulations Can Enable the Model Poorly Water-Soluble Weakly Basic Drug Cinnarizine To Precipitate in an Amorphous-Salt Form During In Vitro Digestion
Jamal Khan, Thomas Rades, Ben J. Boyd · 2016 · Molecular Pharmaceutics
Oleochemistry potential from Brazil northeastern exotic plants
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Endang Wahyu Fitriani, Christina Avanti, Yeva Rosana, Silvia Surini · 2024 · Pharmacia
AI-directed formulation strategy design initiates rational drug development
Nannan Wang, Jie Dong, Defang Ouyang · 2024 · Journal of Controlled Release
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Niklas J. Koehl, René Holm, Martin Kuentz, Brendan T. Griffin · 2019 · Pharmaceutical Research
Enhancing the oral bioavailability of simvastatin with silica-lipid hybrid particles: The effect of supersaturation and silica geometry
Tahlia R. Meola, Hayley B. Schultz, Karl F. Peressin, Clive A. Prestidge · 2020 · European Journal of Pharmaceutical Sciences
Novel amorphous solid dispersion based on natural deep eutectic solvent for enhancing delivery of anti-tumor RA-XII by oral administration in rats
Mingyu Liu, Zhixing Lai, Lijun Zhu, Xin Ding, Xiyang Tong, Zhen Wang, Qirui Bi, Ning‐Hua Tan · 2021 · European Journal of Pharmaceutical Sciences
Exploring impact of supersaturated lipid-based drug delivery systems of celecoxib on in vitro permeation across PermeapadⓇ membrane and in vivo absorption
Ilie, Alexandra-Roxana, Griffin, Brendan T., Brandl, Martin, Bauer-Brandl, Annette, Jacobsen, Ann-Christin, Vertzoni, Maria, Kuentz, Martin, Kolakovic, Ruzica, Holm, René · 2020 · European Journal of Pharmaceutical Sciences
Potent and Selective Human Prostaglandin F (FP) Receptor Antagonist (BAY-6672) for the Treatment of Idiopathic Pulmonary Fibrosis (IPF)
Hartmut Beck, Tobias Thaler, Daniel Meibom, Mark Meininghaus, Hannah Jörißen, Lisa Dietz, Carsten Terjung, Michaela Bairlein, Clemens-Jeremias von Bühler, Sonja Anlauf et al. · 2020 · Journal of Medicinal Chemistry
Rational Selection of Bio-Enabling Oral Drug Formulations – A PEARRL Commentary
Martin Kuentz, René Holm, Christian Kronseder, Christoph Saal, Brendan T. Griffin · 2021 · Journal of Pharmaceutical Sciences
Estimating the Oral Absorption from Self-Nanoemulsifying Drug Delivery Systems Using an In Vitro Lipolysis-Permeation Method
Mette Klitgaard, Anette Müllertz, Ragna Berthelsen · 2021 · Pharmaceutics
Rapid determination of drug solubilization versus supersaturation in natural and digested lipids
Nicolas Gautschi, Christel A. S. Bergström, Martin Kuentz · 2016 · International Journal of Pharmaceutics
Formulating a single thioether-bridged oleate prodrug into a self-nanoemulsifying drug delivery system to facilitate oral absorption of docetaxel
Weiping Cui, Shenwu Zhang, Hanqing Zhao, Cong Luo, Bingjun Sun, Zhenbao Li, Mengchi Sun, Qing Ye, Jin Sun, Zhonggui He · 2018 · Biomaterials Science
Thermal stability of indomethacin increases with the amount of polyvinylpyrrolidone in solid dispersion
Dijana Jelić, Tatsiana Liavitskaya, Sergey Vyazovkin · 2019 · Thermochimica Acta
A bubble bursting-mediated oral drug delivery system that enables concurrent delivery of lipophilic and hydrophilic chemotherapeutics for treating pancreatic tumors in rats
Kuan‐Hung Chen, Yang‐Bao Miao, Chun-Yu Shang, Tring-Yo Huang, Yu‐Tzu Yu, Chun‐Nan Yeh, Hsiang‐Lin Song, Chiung-Tong Chen, Fwu‐Long Mi, Kun‐Ju Lin et al. · 2020 · Biomaterials
Opportunities for milk and milk-related systems as ‘new’ low-cost excipient drug delivery materials
Malinda Salim, Thomas Eason, Ben J. Boyd · 2022 · Advanced Drug Delivery Reviews
Mechanistic aspects of drug loading in liquisolid systems with hydrophilic lipid-based mixtures
Barbora Vraníková, Andreas Niederquell, Felix Ditzinger, Zdeňka Šklubalová, Martin Kuentz · 2020 · International Journal of Pharmaceutics
A Nonionic Polyethylene Oxide (PEO) Surfactant Model: Experimental and Molecular Dynamics Studies of Kolliphor EL
Estelle J. A. Suys, Dallas B. Warren, Anna C. Pham, Cameron J. Nowell, Andrew J. Clulow, Hassan Benameur, Christopher J. H. Porter, Colin William Pouton, David K. Chalmers · 2018 · Journal of Pharmaceutical Sciences
Enhancement of abiraterone acetate oral bioavailability by supersaturated-silica lipid hybrids
Hayley B. Schultz, Anthony D. Wignall, Nicky Thomas, Clive A. Prestidge · 2020 · International Journal of Pharmaceutics
Aqueous Dissolution and Dispersion Behavior of Polyvinylpyrrolidone Vinyl Acetate-based Amorphous Solid Dispersion of Ritonavir Prepared by Hot-Melt Extrusion with and without Added Surfactants
Nitprapa Siriwannakij, Tycho Heimbach, Abu T.M. Serajuddin · 2020 · Journal of Pharmaceutical Sciences
Interactions of Artefenomel (OZ439) with Milk during Digestion: Insights into Digestion-Driven Solubilization and Polymorphic Transformations
Malinda Salim, Jamal Khan, Gisela Ramirez, Andrew J. Clulow, Adrian M. Hawley, Hanu Ramachandruni, Ben J. Boyd · 2018 · Molecular Pharmaceutics
Comparison of different chemometric methods to extract chemical and physical information from Raman images of homogeneous and heterogeneous semi-solid pharmaceutical formulations
Hery Mitsutake, Simone R. Castro, Eneida de Paula, Ronei J. Poppi, Douglas Neil Rutledge, Márcia Cristina Breitkreitz · 2018 · International Journal of Pharmaceutics
Supersaturated lipid-based drug delivery systems – exploring impact of lipid composition type and drug properties on supersaturability and physical stability
Alexandra-Roxana Ilie, Brendan T. Griffin, Ruzica Kolakovic, Maria Vertzoni, Martin Kuentz, René Holm · 2020 · Drug Development and Industrial Pharmacy
Recent Options and Techniques to Assess Improved Bioavailability: In Vitro and Ex Vivo Methods
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Orlagh M. Feeney, Gracia Gracia, Daniel H.S. Brundel, Natalie L. Trevaskis, Enyuan Cao, Lisa M. Kaminskas, Christopher J. H. Porter · 2020 · Advanced Drug Delivery Reviews
Montmorillonite-lipid hybrid carriers for ionizable and neutral poorly water-soluble drugs: Formulation, characterization and in vitro lipolysis studies
Tahnee J. Dening, Shasha Rao, Nicky Thomas, Clive A. Prestidge · 2017 · International Journal of Pharmaceutics
Labrasol® and Salts of Medium-Chain Fatty Acids Can Be Combined in Low Concentrations to Increase the Permeability of a Macromolecule Marker Across Isolated Rat Intestinal Mucosae
Joanne Heade, Sam Maher, Sinéad B. Bleiel, David J. Brayden · 2018 · Journal of Pharmaceutical Sciences
Alginate-coating of artemisinin-loaded cochleates results in better control over gastro-intestinal release for effective oral delivery
Shuddhodana Shuddhodana, Zaher M. A. Judeh · 2019 · Journal of Drug Delivery Science and Technology
API ionic liquids: probing the effect of counterion structure on physical form and lipid solubility
Leigh Ford, Erin Tay, Tri‐Hung Nguyen, Hywel D. Williams, Hassan Benameur, Peter J. Scammells, Christopher J. H. Porter · 2020 · RSC Advances
Solidification of SMEDDS by fluid bed granulation and manufacturing of fast drug release tablets
Jelena Mandić, Vesna Pirnat, Matevž Luštrik, Ilija German Ilić, Franc Vrečer, Mirjana Gašperlin, Alenka Zvonar Pobirk · 2020 · International Journal of Pharmaceutics
Development of solid SEDDS, VII: Effect of pore size of silica on drug release from adsorbed self-emulsifying lipid-based formulations
Suhas G. Gumaste, Abu T.M. Serajuddin · 2017 · European Journal of Pharmaceutical Sciences
An in vitro dissolution–digestion–permeation assay for the study of advanced drug delivery systems
Caroline Alvebratt, Janneke Keemink, Khadijah Edueng, Ocean Y. H. Cheung, Maria Strømme, Christel A. S. Bergström · 2020 · European Journal of Pharmaceutics and Biopharmaceutics
Novel Strategies for the Formulation of Poorly Water-Soluble Drug Substances by Different Physical Modification Strategies with a Focus on Peroral Applications
Julian Quodbach, Eduard Preis, Frank Karkossa, Judith Winck, Jan Henrik Finke, Denise Steiner · 2025 · Pharmaceuticals
Novel Biphasic Lipolysis Method To Predict <i>in Vivo</i> Performance of Lipid-Based Formulations
O’Dwyer, Patrick J., Box, Karl J., Koehl, Niklas J., Bennett-Lenane, Harriet, Reppas, Christos, Holm, Rene, Kuentz, Martin, Griffin, Brendan T. · 2020 · Molecular Pharmaceutics
Novel Phenobarbital-Loaded Nanostructured Lipid Carriers for Epilepsy Treatment: From QbD to In Vivo Evaluation
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Revisiting dispersible milk-drug tablets as a solid lipid formulation in the context of digestion
Syaza Y. Binte Abu Bakar, Malinda Salim, Andrew J. Clulow, Adrian M. Hawley, Ben J. Boyd · 2018 · International Journal of Pharmaceutics
Suitability of Artificial Membranes in Lipolysis-Permeation Assays of Oral Lipid-Based Formulations
Oliver J. Hedge, Christel A. S. Bergström · 2020 · Pharmaceutical Research
Incorporation of lipolysis in monolayer permeability studies of lipid-based oral drug delivery systems
Tanmoy Sadhukha, Buddhadev Layek, Swayam Prabha · 2017 · Drug Delivery and Translational Research
Size characterization of lipid-based self-emulsifying pharmaceutical excipients during lipolysis using Taylor dispersion analysis with fluorescence detection
Joseph Chamieh, Habib Merdassi, Jean‐Christophe Rossi, Vincent Jannin, Frédéric Demarne, Hervé Cottet · 2017 · International Journal of Pharmaceutics
Transient Supersaturation Supports Drug Absorption from Lipid-Based Formulations for Short Periods of Time, but Ongoing Solubilization Is Required for Longer Absorption Periods
Matthew Crum, Natalie L. Trevaskis, Colin William Pouton, Christopher J. H. Porter · 2016 · Molecular Pharmaceutics
Spray Encapsulation as a Formulation Strategy for Drug-Based Room Temperature Ionic Liquids: Exploiting Drug–Polymer Immiscibility to Enable Processing for Solid Dosage Forms
Michael W. Stocker, Anne Marie Healy, Steven Ferguson · 2020 · Molecular Pharmaceutics
Is oral lipid-based delivery for drug targeting to the brain feasible?
Alice Brookes, Liuhang Ji, Tracey Dawn Bradshaw, Michael J. Stocks, David A. Gray, James Butler, Pavel Gershkovich · 2022 · European Journal of Pharmaceutics and Biopharmaceutics
Combined effects of the drug distribution and mucus diffusion properties of self-microemulsifying drug delivery systems on the oral absorption of fenofibrate
Yushi Sunazuka, Keisuke Ueda, Kenjirou Higashi, Yusuke Tanaka, Kunikazu Moribe · 2018 · International Journal of Pharmaceutics
Montmorillonite and Laponite Clay Materials for the Solidification of Lipid-Based Formulations for the Basic Drug Blonanserin: In Vitro and in Vivo Investigations
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Synergistic Computational Modeling Approaches as Team Players in the Game of Solubility Predictions
Martin Kuentz, Christel A. S. Bergström · 2020 · Journal of Pharmaceutical Sciences
Enhanced Stability and Improved Oral Absorption of Enzalutamide with Self-Nanoemulsifying Drug Delivery System
Su-Min Lee, Jeong-Gyun Lee, Tae-Han Yun, Jung Hyun Cho, Kyeong Soo Kim · 2024 · International Journal of Molecular Sciences
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Yaping Huang, Sisi Zhang, Huifen Shen, Jinqing Li, Chongkai Gao · 2018 · AAPS PharmSciTech
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Ljiljana Đekić, Jovana Janković, Aleksandar Rašković, Marija Primorac · 2018 · European Journal of Pharmaceutical Sciences
Improvement of the bioavailability of curcumin by a supersaturatable self nanoemulsifying drug delivery system with incorporation of a hydrophilic polymer: in vitro and in vivo characterisation
Xulong Chen, Xin‐Li Liang, Guowei Zhao, Qing-yun Zeng, Wei Dong, Liquan Ou, Haonan Zhang, Qie-Ying Jiang, Zheng‐Gen Liao · 2021 · Journal of Pharmacy and Pharmacology
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Supersaturated-Silica Lipid Hybrids Improve in Vitro Solubilization of Abiraterone Acetate
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Eleonora Maretti, Barbara Pavan, Cecilia Rustichelli, Monica Montanari, Alessandro Dalpiaz, Valentina Iannuccelli, Eliana Leo · 2020 · Colloids and Surfaces A Physicochemical and Engineering Aspects
Improving Correlations Between Drug Solubilization and In Vitro Lipolysis by Monitoring the Phase Partitioning of Lipolytic Species for Lipid-Based Formulations
Tahnee J. Dening, Paul Joyce, Clive A. Prestidge · 2018 · Journal of Pharmaceutical Sciences
High-Shear Wet Granulation of SMEDDS Based on Mesoporous Carriers for Improved Carvedilol Solubility
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