50 years of oral lipid-based formulations: provenance, progress and future perspectives
Feeney, Orlagh M., Crum, Matthew F., McEvoy, Claire L., Trevaskis, Natalie L., Williams, Hywel D., Pouton, Colin W., Charman, William N., Bergström, Christel A.S. +1 more·2016·Advanced Drug Delivery Reviews
Cites (289)
Items 201–285 of 285
- Visualization by freeze fracture, in vitro and in vivo, of the products of fat digestion.Mark W. Rigler, Richard E. Honkanen, J. Scott Patton · 1988 · Journal of Lipid Research
- Lipophilic Prodrugs of SN38: Synthesis and in Vitro Characterization toward Oral ChemotherapyVaskor Bala, Shasha Rao, Peng Li, Shudong Wang, Clive A. Prestidge · 2015 · Molecular Pharmaceutics
- Lipid Absorption Triggers Drug Supersaturation at the Intestinal Unstirred Water Layer and Promotes Drug Absorption from Mixed MicellesYan Yan Yeap, Natalie L. Trevaskis, Christopher J. H. Porter · 2013 · Pharmaceutical Research
- Analysis of the enhanced oral bioavailability of fenofibrate lipid formulations in fasted humans using an in vitro–in silico–in vivo approachYang Fei, Edmund S. Kostewicz, Ming‐Thau Sheu, Jennifer Dressman · 2013 · European Journal of Pharmaceutics and Biopharmaceutics
- Toward an Improved Understanding of the Precipitation Behavior of Weakly Basic Drugs from Oral Lipid-Based FormulationsCordula Stillhart, Désirée Dürr, Martin Kuentz · 2014 · Journal of Pharmaceutical Sciences
- Insights into Intermediate Phases of Human Intestinal Fluids Visualized by Atomic Force Microscopy and Cryo-Transmission Electron Microscopy ex VivoAnette Müllertz, Dimitrios G. Fatouros, James R. Smith, Maria Vertzoni, Christos I. Reppas · 2011 · Molecular Pharmaceutics
- Development of Clinical Dosage Forms for a Poorly Water-Soluble Drug II: Formulation and Characterization of a Novel Solid Microemulsion Preconcentrate System for Oral Delivery of a Poorly Water-Soluble DrugPing Li, Sara Royce Hynes, Thomas Haefele, Madhu Pudipeddi, Alan E. Royce, Abu T.M. Serajuddin · 2008 · Journal of Pharmaceutical Sciences
- Comparative bioavailability of neoral and sandimmune in cardiac transplant recipients over 1 yearGerard F. Cooney, Valluvan Jeevanandam, S Choudhury, Gilles Feutren, E. Mueller, Howard J. Eisen · 1998 · Transplantation Proceedings
- Characterization of mucin – lipid droplet interactions: Influence on potential fate of fish oil-in-water emulsions under simulated gastrointestinal conditionsYaoguang Chang, David Julian McClements · 2016 · Food Hydrocolloids
- Prediction of dissolution-absorption relationships from a continuous dissolution/Caco-2 systemMark J. Ginski, Rajneesh Taneja, James E. Polli · 1999 · AAPS PharmSci
- Development of Solid Self-Emulsifying Drug Delivery System (SEDDS) I: Use of Poloxamer 188 as Both Solidifying and Emulsifying Agent for LipidsAnkita V. Shah, Abu T.M. Serajuddin · 2012 · Pharmaceutical Research
- Cyclosporin absorption from microemulsion formulation in liver transplant recipientAndrew K. Trull, Keith Tan, Julie A. Uttridge, T. Bauer, Graeme Alexander, Neville V. Jamieson · 1993 · The Lancet
- Association of Halofantrine with Postprandially Derived Plasma Lipoproteins Decreases Its Clearance Relative To Administration in the Fasted StateAndrew Humberstone, Christopher J. H. Porter, Glenn Anthony Edwards, William N. Charman · 1998 · Journal of Pharmaceutical Sciences
- The conflict between in vitro release studies in human biorelevant media and the in vivo exposure in rats of the lipophilic compound fenofibrateThao Do Thi, Michiel Van Speybroeck, Raf Mols, Pieter Annaert, Johan A. Martens, Jan Van Humbeeck, Jan Vermant, Patrick Augustijns, Guy Van den Mooter · 2011 · International Journal of Pharmaceutics
- In-vitro permeability of poorly water soluble drugs in the phospholipid vesicle-based permeation assay: the influence of nonionic surfactantsSarah Maud Fischer, Gøril Eide Flaten, Ellen Hagesæther, Gert Fricker, Martin Brandl · 2011 · Journal of Pharmacy and Pharmacology
- Insights into Drug Precipitation Kinetics during In Vitro Digestion of a Lipid-Based Drug Delivery System Using In-Line Raman Spectroscopy and Mathematical ModelingCordula Stillhart, Georgios Imanidis, Martin Kuentz · 2013 · Pharmaceutical Research
- The effect of drug lipophilicity and lipid vehicles on the lymphatic absorption of various testosterone estersT. Noguchi, William N. Charman, Valentino J. Stella · 1985 · International Journal of Pharmaceutics
- Evaluation of the Structural Determinants of Polymeric Precipitation Inhibitors Using Solvent Shift Methods and Principle Component AnalysisDallas B. Warren, Christel A. S. Bergström, Hassan Benameur, Christopher J. H. Porter, Colin William Pouton · 2013 · Molecular Pharmaceutics
- Enhancement of Bioavailability of a Hydrophobic Amine Antimalarial by Formulation with Oleic Acid in a Soft Gelatin CapsuleValentine J. Stella, John L. Haslam, Noboru Yata, Hiroaki Okada, Siegfried Lindenbaum, Tsunehiko Higuchi · 1978 · Journal of Pharmaceutical Sciences
- The effect of digestion and drug load on halofantrine absorption from self-nanoemulsifying drug delivery system (SNEDDS)Michaelsen, Maria Høtoft, Wasan, Kishor M., Sivak, Olena, Müllertz, Anette, Rades, Thomas · 2016 · The AAPS Journal
- Mechanisms of intestinal fat absorptionY. F. Shiau · 1981 · American Journal of Physiology-Gastrointestinal and Liver Physiology
- A New Method for Dissolution Studies of Lipid-Filled Capsules Employing Nifedipine as a Model DrugViness Pillay, Reza Fassihi · 1999 · Pharmaceutical Research
- Hybrid Nanomaterials that Mimic the Food Effect: Controlling Enzymatic Digestion for Enhanced Oral Drug AbsorptionAngel Tan, Amanda L. Martin, Tri‐Hung Nguyen, Ben J. Boyd, Clive A. Prestidge · 2012 · Angewandte Chemie International Edition
- Bioavailability of phenytoin in lipid containing dosage forms in ratsSasanka Chakrabarti, F. M. Belpaire · 1978 · Journal of Pharmacy and Pharmacology
- Drug release from lipid-based dosage forms. IN. Anthony Armstrong, Kenneth James · 1980 · International Journal of Pharmaceutics
- Hot-melt extruded ethylcellulose cylinders containing a HPMC–Gelucire® core for sustained drug deliveryEls Mehuys, Chris Vervaet, Jean Paul Remon · 2004 · Journal of Controlled Release
- In Situ Lipolysis and Synchrotron Small-Angle X-ray Scattering for the Direct Determination of the Precipitation and Solid-State Form of a Poorly Water-Soluble Drug During Digestion of a Lipid-Based FormulationJamal Khan, Adrian M. Hawley, Thomas Rades, Ben J. Boyd · 2015 · Journal of Pharmaceutical Sciences
- The self-emulsifying action of mixed surfactants in oil.Groves Mj, D A de Galindez · 1976 · PubMed
- Rapid (1 hour) high performance gel filtration chromatography resolves coexisting simple micelles, mixed micelles, and vesicles in bile.DE Cohen, M C Carey · 1990 · Journal of Lipid Research
- Impact of Cremophor-EL and Polysorbate-80 on Digoxin Permeability across Rat Jejunum: Delineation of Thermodynamic and Transporter Related Events Using the Reciprocal Permeability ApproachKasiram Katneni, Susan A. Charman, Christopher J. H. Porter · 2006 · Journal of Pharmaceutical Sciences
- Effects of lipids on bioavailability of sulfisoxazole acetyl, dicumarol, and griseofulvin in ratsDuane C. Bloedow, William L. Hayton · 1976 · Journal of Pharmaceutical Sciences
- Toward the Establishment of Standardized In Vitro Tests for Lipid-Based Formulations, Part 4: Proposing a New Lipid Formulation Performance Classification SystemHywel D. Williams, Philip Jonas Sassene, Karen Kleberg, Marilyn Calderone, Annabel Igonin, Eduardo Jule, Jan Vertommen, Ross Blundell, Hassan Benameur, Anette Müllertz et al. · 2014 · Journal of Pharmaceutical Sciences
- Bioavailability and pharmacokinetics of cyclosporine formulations: Neoral® vs Sandimmune®Miles G. Choc · 1997 · International Journal of Dermatology
- Development of a high-throughput in vitro intestinal lipolysis model for rapid screening of lipid-based drug delivery systemsMette Dalskov Mosgaard, Philip Jonas Sassene, Huiling Mu, Thomas Rades, Anette Müllertz · 2015 · European Journal of Pharmaceutics and Biopharmaceutics
- Measurement of the ‘spontaneity’ of self-emulsifiable oilsMichael J. Groves, R M A Mustafa · 1974 · Journal of Pharmacy and Pharmacology
- Characteristics of lipid substances activating the ileal brake in the rat.Nicola Jane Brown, N. W. Read, Alan Richardson, R.D.E. Rumsey, Conny B. Bogentoft · 1990 · Gut
- Ionic Liquid Versus Prodrug Strategy to Address Formulation ChallengesAnja Balk, Toni Widmer, Johannes M. Wiest, H. D. Bruhn, J.-C. Rybak, Philipp R. Matthes, Klaus Müller‐Buschbaum, Anastasios Sakalis, Tessa C. Lühmann, Jörg Berghausen et al. · 2014 · Pharmaceutical Research
- Drug release from lipid-based dosage forms. IIN.A. Armstrong, Kenneth James · 1980 · International Journal of Pharmaceutics
- Analytical technologies for real-time drug dissolution and precipitation testing on a small scaleMartin Kuentz · 2014 · Journal of Pharmacy and Pharmacology
- In vivo evaluation of tablets and capsules containing spray-dried o/w-emulsions for oral delivery of poorly soluble drugsTue Hansen, Per Holm, Morten Rohde, Kirsten Schultz · 2005 · International Journal of Pharmaceutics
- Lipophilic prodrugs of apomorphine I: Preparation, characterisation, and in vitro enzymatic hydrolysis in biorelevant mediaNrupa Borkar, Boyang Li, René Holm, Anders E. Håkansson, Anette Müllertz, Mingshi Yang, Huiling Mu · 2014 · European Journal of Pharmaceutics and Biopharmaceutics
- GASTROINTESTINAL ABSORPTION OF GRISEOFULVIN: I. EFFECT OF PARTICLE SIZE, ADDITION OF SURFACTANTS, AND CORN OIL ON THE LEVEL OF GRISEOFULVIN IN THE SERUM OF RATSM. Kraml, Jean Dubuc, Desmond Beall, Nicole L'Heureux · 1962 · Canadian Journal of Biochemistry and Physiology
- The Mechanism of Lymphatic Access of Two Cholesteryl Ester Transfer Protein Inhibitors (CP524,515 and CP532,623) and Evaluation of Their Impact on Lymph Lipoprotein ProfilesNatalie L. Trevaskis, Ravi M. Shanker, William N. Charman, Christopher J. H. Porter · 2010 · Pharmaceutical Research
- Pluronic and Tetronic Copolymers with Polyglycolyzed Oils as Self-Emulsifying Drug Delivery SystemsMarta Fernandez-Tarrio, Fernando Yáñez, Kristof Immesoete, Carmen Alvarez‐Lorenzo, Ángel Concheiro · 2008 · AAPS PharmSciTech
- The Potential for Drug Supersaturation during Intestinal Processing of Lipid-Based Formulations May Be Enhanced for Basic DrugsYan Yan Yeap, Natalie L. Trevaskis, Christopher J. H. Porter · 2013 · Molecular Pharmaceutics
- Profiling the Role of Deacylation-Reacylation in the Lymphatic Transport of a Triglyceride-Mimetic ProdrugSifei Han, Luojuan Hu, Tim Quach, Jamie S. Simpson, Natalie L. Trevaskis, Christopher J. H. Porter · 2014 · Pharmaceutical Research
- Glyceride Lipid Formulations: Molecular Dynamics Modeling of Phase Behavior During Dispersion and Molecular Interactions Between Drugs and ExcipientsDallas B. Warren, Dylan T. King, Hassan Benameur, Colin William Pouton, David K. Chalmers · 2013 · Pharmaceutical Research
- Biorelevant media resistant co-culture model mimicking permeability of human intestineDelphine Antoine, Yann Pellequer, Camille Tempesta, Stefan Lorscheidt, Bernadette Kettel, Lana Tamaddon, Vincent Jannin, Frédéric Demarne, Alf Lamprecht, Arnaud Béduneau · 2015 · International Journal of Pharmaceutics
- AN EXAMINATION OF THE INTERPLAY BETWEEN ENTEROCYTE-BASED METABOLISM AND LYMPHATIC DRUG TRANSPORT IN THE RATNatalie L. Trevaskis, Christopher J. H. Porter, William N. Charman · 2006 · Drug Metabolism and Disposition
- Proposal of stability categories for nano-dispersions obtained from pharmaceutical self-emulsifying formulationsAndreas Niederquell, Martin Kuentz · 2013 · International Journal of Pharmaceutics
- Drug migration into soft gelatin capsule shells and its effect on in-vitro availabilityN A Armstrong, Kenneth James, W K L Pugh · 1984 · Journal of Pharmacy and Pharmacology
- Elucidating the Molecular Interactions Occurring during Drug Precipitation of Weak Bases from Lipid-Based Formulations: A Case Study with Cinnarizine and a Long Chain Self-Nanoemulsifying Drug Delivery SystemPhilip Jonas Sassene, Mette Dalskov Mosgaard, Korbinian Löbmann, Huiling Mu, Flemming Hofmann Larsen, Thomas Rades, Anette Müllertz · 2015 · Molecular Pharmaceutics
- Biopharmaceutical Modeling of Drug Supersaturation During Lipid-Based Formulation Digestion Considering an Absorption SinkCordula Stillhart, Georgios Imanidis, Brendan T. Griffin, Martin Kuentz · 2014 · Pharmaceutical Research
- The effect of oral lipids and circulating lipoproteins on the metabolism of drugsJigar P. Patel, Dion R. Brocks · 2009 · Expert Opinion on Drug Metabolism & Toxicology
- Lipidic dispersion to reduce food dependent oral bioavailability of fenofibrate: In vitro, in vivo and in silico assessmentsJoseph P. O’Shea, Waleed Faisal, Therese Ruane-O’Hora, Ken J. Devine, Edmund S. Kostewicz, Caitríona M. O’Driscoll, Brendan T. Griffin · 2015 · European Journal of Pharmaceutics and Biopharmaceutics
- The disintegration behaviour of capsules in fed subjects: A comparison of hypromellose (carrageenan) capsules and standard gelatin capsulesBrian E. Jones, Abdul W. Basit, Catherine Tuleu · 2011 · International Journal of Pharmaceutics
- Comparison of high-resolution ultrasonic resonator technology and Raman spectroscopy as novel process analytical tools for drug quantification in self-emulsifying drug delivery systemsCordula Stillhart, Martin Kuentz · 2011 · Journal of Pharmaceutical and Biomedical Analysis
- Effect of food intake and co-administration of placebo self-nanoemulsifying drug delivery systems on the absorption of cinnarizine in healthy human volunteersMartin Lau Christiansen, René Holm, Bertil Abrahamsson, Jette Bredahl Jacobsen, Jakob Kristensen, Jens Rikardt Andersen, Anette Müllertz · 2016 · European Journal of Pharmaceutical Sciences
- An in Vitro Digestion Test That Reflects Rat Intestinal Conditions To Probe the Importance of Formulation Digestion vs First Pass Metabolism in Danazol Bioavailability from Lipid Based FormulationsMette U. Anby, Tri‐Hung Nguyen, Yan Yan Yeap, Orlagh M. Feeney, Hywel D. Williams, Hassan Benameur, Colin William Pouton, Christopher J. H. Porter · 2014 · Molecular Pharmaceutics
- In vitro and in vivo evaluation of a matrix-in-cylinder system for sustained drug deliveryEls Mehuys, Chris Vervaet, Ingrid Gielen, Henri van Bree, Jean Paul Remon · 2004 · Journal of Controlled Release
- Tableting Lipid-Based Formulations for Oral Drug Delivery: A Case Study with Silica Nanoparticle–Lipid–Mannitol Hybrid MicroparticlesKristen E. Bremmell, Angel Tan, Amanda L. Martin, Clive A. Prestidge · 2012 · Journal of Pharmaceutical Sciences
- Biopharmaceutical studies of lipid-containing oral dosage forms: Relationship between drug absorption rate and digestibility of vehiclesYoshiya Yamahira, Noguchi Takeshi, Hiroshi Takenaka, Maeda Tadao · 1979 · International Journal of Pharmaceutics
- Trends in the Assessment of Drug Supersaturation and Precipitation In Vitro Using Lipid-Based Delivery SystemsCordula Stillhart, Martin Kuentz · 2016 · Journal of Pharmaceutical Sciences
- Acidic mucin layer facilitates micelle dissociation and fatty acid diffusionY. F. Shiau, R. J. Kelemen, M. A. Reed · 1990 · American Journal of Physiology-Gastrointestinal and Liver Physiology
- In vitro and in vivo preclinical evaluation of a minisphere emulsion-based formulation (SmPill®) of salmon calcitoninTanira Alessandra Silveira Aguirre, Mónica Rosa, Ivan S. Coulter, David J. Brayden · 2015 · European Journal of Pharmaceutical Sciences
- Chemical Drug Stability in Lipids, Modified Lipids, and Polyethylene Oxide-Containing FormulationsValentino J. Stella · 2013 · Pharmaceutical Research
- In Vivo Formation of Cubic Phase in Situ after Oral Administration of Cubic Phase Precursor Formulation Provides Long Duration Gastric Retention and Absorption for Poorly Water-Soluble DrugsAnna C. Pham, Linda Hong, Oliver D. Montagnat, Cameron J. Nowell, Tri‐Hung Nguyen, Ben J. Boyd · 2015 · Molecular Pharmaceutics
- Human bioavailability of propranolol from a matrix-in-cylinder system with a HPMC-Gelucire® coreEls Mehuys, Jean Paul Remon, Annelies E. C. Korst, Luc MAB. Van Bortel, Raf Mols, Patrick Augustijns, Christopher J. H. Porter, Chris Vervaet · 2005 · Journal of Controlled Release
- The use of supports in the lyophilization of oil-in-water emulsionsM Lladser, Claudia Alejandra Medrano, A Arancibia · 1968 · Journal of Pharmacy and Pharmacology
- In vitro–in vivo evaluation of lipid based formulations of the CETP inhibitors CP-529,414 (torcetrapib) and CP-532,623Claire L. McEvoy, Natalie L. Trevaskis, Glenn Anthony Edwards, Michael E. Perlman, Catherine M. Ambler, Mary Catherine Mack, Barbara Brockhurst, Christopher J. H. Porter · 2014 · European Journal of Pharmaceutics and Biopharmaceutics
- In vitro and in vivo evaluations of the performance of an indirubin derivative, formulated in four different self-emulsifying drug delivery systemsNasim Heshmati, Xinlai Cheng, Else Dapat, Philip Jonas Sassene, Gerhard Eisenbrand, Gert Fricker, Anette Müllertz · 2014 · Journal of Pharmacy and Pharmacology
- A simplified method to screen for in-vivo performance of oral lipid formulationsMurat Kilic, Jennifer Dressman · 2013 · Journal of Pharmacy and Pharmacology
- Study of drug supersaturation for rational early formulation screening of surfactant/co-solvent drug delivery systemsCordula Stillhart, Martin Cavegn, Martin Kuentz · 2012 · Journal of Pharmacy and Pharmacology
- In Vitro Lipolysis and Intestinal Transport of β-Arteether-Loaded Lipid-Based Drug Delivery SystemsPatrick B. Memvanga, Pierre Eloy, Éric M. Gaigneaux, Véronique Préat A · 2013 · Pharmaceutical Research
- Pancreatic Lipase-Catalyzed Hydrolysis of Esters of Hydroxymethyl Phenytoin Dissolved in Various Metabolizable Vehicles, Dispersed in Micellar Systems, and in Aqueous SuspensionsFrancisco J. Álvarez, Valentine J. Stella · 1989 · Pharmaceutical Research
- Physicochemical Characterization of Simulated Intestinal Fed-State Fluids Containing Lyso-Phosphatidylcholine and CholesterolDimitris G. Fatouros, Isabelle Walrand, Björn Bergenståhl, Anette Müllertz · 2009 · Dissolution Technologies
- Biopharmaceutical studies of lipid-containing oral dosage forms: Relationship between drug absorption and gastric emptying of lipid formulations.Yoshiya Yamahira, TAKESHI NOGUCHI, Hiroshi Takenaka, TADAO MAEDA · 1978 · Journal of Pharmacobio-Dynamics
- A prodrug strategy for the oral delivery of a poorly soluble HCV NS5B thumb pocket 1 polymerase inhibitor using self-emulsifying drug delivery systems (SEDDS)Pierre L. Beaulieu, Josie De Marte, Michel Garneau, Laibin Luo, Timothy A. Stammers, Chitra Telang, Dominik Wernic, George Kukolj, Jianmin Duan · 2014 · Bioorganic & Medicinal Chemistry Letters
- Preliminary development and evaluation of a parenteral emulsion formulation of penclomedine (NSC-338720; 3,5-dichloro-2,4-dimethoxy-6-trichloromethylpyridine): a novel, practically water insoluble cytotoxic agent.R.J. Prankerd, Sylvan G. Frank, Valentine J. Stella · 1989 · PubMed
- Novel semisolid SNEDDS based on PEG-30-di-(polyhydroxystearate): Progesterone incorporation and in vitro digestionTamer H. Hassan, Karsten Mäder · 2015 · International Journal of Pharmaceutics
- [Research on the spray drying of emulsified medical preparations. 1].A RICHTER, K Steiger-Trippi · 1961 · PubMed
- Plasma concentrations after oral administration of different pharmaceutical preparations of clomethiazole.M Fischler, Frisch Ep, B. Örtengren · 1973 · PubMed
- Oral Sulfonamides in Lipid EmulsionC. W. Daeschner · 1957 · A M A Journal of Diseases of Children
- Steroidal ethers: urinary excretion of pregnanediols in man after ingestion of quingestrone in fasting or non-fasting conditions.G Bruni, F Galletti · 1970 · PubMed
- Absorption and chemotherapeutic activity of acetyl sulfisoxazole suspended in an oil in water emulsion.Svenson Se, W. F. DeLorenzo, Recha Engelberg, MILDRED E. SPOONER, L O RANDALL · 1956 · PubMed