50 years of oral lipid-based formulations: provenance, progress and future perspectives

Feeney, Orlagh M., Crum, Matthew F., McEvoy, Claire L., Trevaskis, Natalie L., Williams, Hywel D., Pouton, Colin W., Charman, William N., Bergström, Christel A.S. +1 more·2016·Advanced Drug Delivery Reviews

Cites (289)

Items 201–285 of 285

  1. Visualization by freeze fracture, in vitro and in vivo, of the products of fat digestion.
    Mark W. Rigler, Richard E. Honkanen, J. Scott Patton · 1988 · Journal of Lipid Research
  2. Lipophilic Prodrugs of SN38: Synthesis and in Vitro Characterization toward Oral Chemotherapy
    Vaskor Bala, Shasha Rao, Peng Li, Shudong Wang, Clive A. Prestidge · 2015 · Molecular Pharmaceutics
  3. Lipid Absorption Triggers Drug Supersaturation at the Intestinal Unstirred Water Layer and Promotes Drug Absorption from Mixed Micelles
    Yan Yan Yeap, Natalie L. Trevaskis, Christopher J. H. Porter · 2013 · Pharmaceutical Research
  4. Analysis of the enhanced oral bioavailability of fenofibrate lipid formulations in fasted humans using an in vitro–in silico–in vivo approach
    Yang Fei, Edmund S. Kostewicz, Ming‐Thau Sheu, Jennifer Dressman · 2013 · European Journal of Pharmaceutics and Biopharmaceutics
  5. Toward an Improved Understanding of the Precipitation Behavior of Weakly Basic Drugs from Oral Lipid-Based Formulations
    Cordula Stillhart, Désirée Dürr, Martin Kuentz · 2014 · Journal of Pharmaceutical Sciences
  6. Insights into Intermediate Phases of Human Intestinal Fluids Visualized by Atomic Force Microscopy and Cryo-Transmission Electron Microscopy ex Vivo
    Anette Müllertz, Dimitrios G. Fatouros, James R. Smith, Maria Vertzoni, Christos I. Reppas · 2011 · Molecular Pharmaceutics
  7. Development of Clinical Dosage Forms for a Poorly Water-Soluble Drug II: Formulation and Characterization of a Novel Solid Microemulsion Preconcentrate System for Oral Delivery of a Poorly Water-Soluble Drug
    Ping Li, Sara Royce Hynes, Thomas Haefele, Madhu Pudipeddi, Alan E. Royce, Abu T.M. Serajuddin · 2008 · Journal of Pharmaceutical Sciences
  8. Comparative bioavailability of neoral and sandimmune in cardiac transplant recipients over 1 year
    Gerard F. Cooney, Valluvan Jeevanandam, S Choudhury, Gilles Feutren, E. Mueller, Howard J. Eisen · 1998 · Transplantation Proceedings
  9. Characterization of mucin – lipid droplet interactions: Influence on potential fate of fish oil-in-water emulsions under simulated gastrointestinal conditions
    Yaoguang Chang, David Julian McClements · 2016 · Food Hydrocolloids
  10. Prediction of dissolution-absorption relationships from a continuous dissolution/Caco-2 system
    Mark J. Ginski, Rajneesh Taneja, James E. Polli · 1999 · AAPS PharmSci
  11. Development of Solid Self-Emulsifying Drug Delivery System (SEDDS) I: Use of Poloxamer 188 as Both Solidifying and Emulsifying Agent for Lipids
    Ankita V. Shah, Abu T.M. Serajuddin · 2012 · Pharmaceutical Research
  12. Cyclosporin absorption from microemulsion formulation in liver transplant recipient
    Andrew K. Trull, Keith Tan, Julie A. Uttridge, T. Bauer, Graeme Alexander, Neville V. Jamieson · 1993 · The Lancet
  13. Association of Halofantrine with Postprandially Derived Plasma Lipoproteins Decreases Its Clearance Relative To Administration in the Fasted State
    Andrew Humberstone, Christopher J. H. Porter, Glenn Anthony Edwards, William N. Charman · 1998 · Journal of Pharmaceutical Sciences
  14. The conflict between in vitro release studies in human biorelevant media and the in vivo exposure in rats of the lipophilic compound fenofibrate
    Thao Do Thi, Michiel Van Speybroeck, Raf Mols, Pieter Annaert, Johan A. Martens, Jan Van Humbeeck, Jan Vermant, Patrick Augustijns, Guy Van den Mooter · 2011 · International Journal of Pharmaceutics
  15. In-vitro permeability of poorly water soluble drugs in the phospholipid vesicle-based permeation assay: the influence of nonionic surfactants
    Sarah Maud Fischer, Gøril Eide Flaten, Ellen Hagesæther, Gert Fricker, Martin Brandl · 2011 · Journal of Pharmacy and Pharmacology
  16. Insights into Drug Precipitation Kinetics during In Vitro Digestion of a Lipid-Based Drug Delivery System Using In-Line Raman Spectroscopy and Mathematical Modeling
    Cordula Stillhart, Georgios Imanidis, Martin Kuentz · 2013 · Pharmaceutical Research
  17. The effect of drug lipophilicity and lipid vehicles on the lymphatic absorption of various testosterone esters
    T. Noguchi, William N. Charman, Valentino J. Stella · 1985 · International Journal of Pharmaceutics
  18. Evaluation of the Structural Determinants of Polymeric Precipitation Inhibitors Using Solvent Shift Methods and Principle Component Analysis
    Dallas B. Warren, Christel A. S. Bergström, Hassan Benameur, Christopher J. H. Porter, Colin William Pouton · 2013 · Molecular Pharmaceutics
  19. Enhancement of Bioavailability of a Hydrophobic Amine Antimalarial by Formulation with Oleic Acid in a Soft Gelatin Capsule
    Valentine J. Stella, John L. Haslam, Noboru Yata, Hiroaki Okada, Siegfried Lindenbaum, Tsunehiko Higuchi · 1978 · Journal of Pharmaceutical Sciences
  20. The effect of digestion and drug load on halofantrine absorption from self-nanoemulsifying drug delivery system (SNEDDS)
    Michaelsen, Maria Høtoft, Wasan, Kishor M., Sivak, Olena, Müllertz, Anette, Rades, Thomas · 2016 · The AAPS Journal
  21. Mechanisms of intestinal fat absorption
    Y. F. Shiau · 1981 · American Journal of Physiology-Gastrointestinal and Liver Physiology
  22. A New Method for Dissolution Studies of Lipid-Filled Capsules Employing Nifedipine as a Model Drug
    Viness Pillay, Reza Fassihi · 1999 · Pharmaceutical Research
  23. Hybrid Nanomaterials that Mimic the Food Effect: Controlling Enzymatic Digestion for Enhanced Oral Drug Absorption
    Angel Tan, Amanda L. Martin, Tri‐Hung Nguyen, Ben J. Boyd, Clive A. Prestidge · 2012 · Angewandte Chemie International Edition
  24. Bioavailability of phenytoin in lipid containing dosage forms in rats
    Sasanka Chakrabarti, F. M. Belpaire · 1978 · Journal of Pharmacy and Pharmacology
  25. Drug release from lipid-based dosage forms. I
    N. Anthony Armstrong, Kenneth James · 1980 · International Journal of Pharmaceutics
  26. Hot-melt extruded ethylcellulose cylinders containing a HPMC–Gelucire® core for sustained drug delivery
    Els Mehuys, Chris Vervaet, Jean Paul Remon · 2004 · Journal of Controlled Release
  27. In Situ Lipolysis and Synchrotron Small-Angle X-ray Scattering for the Direct Determination of the Precipitation and Solid-State Form of a Poorly Water-Soluble Drug During Digestion of a Lipid-Based Formulation
    Jamal Khan, Adrian M. Hawley, Thomas Rades, Ben J. Boyd · 2015 · Journal of Pharmaceutical Sciences
  28. The self-emulsifying action of mixed surfactants in oil.
    Groves Mj, D A de Galindez · 1976 · PubMed
  29. Rapid (1 hour) high performance gel filtration chromatography resolves coexisting simple micelles, mixed micelles, and vesicles in bile.
    DE Cohen, M C Carey · 1990 · Journal of Lipid Research
  30. Impact of Cremophor-EL and Polysorbate-80 on Digoxin Permeability across Rat Jejunum: Delineation of Thermodynamic and Transporter Related Events Using the Reciprocal Permeability Approach
    Kasiram Katneni, Susan A. Charman, Christopher J. H. Porter · 2006 · Journal of Pharmaceutical Sciences
  31. Effects of lipids on bioavailability of sulfisoxazole acetyl, dicumarol, and griseofulvin in rats
    Duane C. Bloedow, William L. Hayton · 1976 · Journal of Pharmaceutical Sciences
  32. Toward the Establishment of Standardized In Vitro Tests for Lipid-Based Formulations, Part 4: Proposing a New Lipid Formulation Performance Classification System
    Hywel D. Williams, Philip Jonas Sassene, Karen Kleberg, Marilyn Calderone, Annabel Igonin, Eduardo Jule, Jan Vertommen, Ross Blundell, Hassan Benameur, Anette Müllertz et al. · 2014 · Journal of Pharmaceutical Sciences
  33. Bioavailability and pharmacokinetics of cyclosporine formulations: Neoral® vs Sandimmune®
    Miles G. Choc · 1997 · International Journal of Dermatology
  34. Development of a high-throughput in vitro intestinal lipolysis model for rapid screening of lipid-based drug delivery systems
    Mette Dalskov Mosgaard, Philip Jonas Sassene, Huiling Mu, Thomas Rades, Anette Müllertz · 2015 · European Journal of Pharmaceutics and Biopharmaceutics
  35. Measurement of the ‘spontaneity’ of self-emulsifiable oils
    Michael J. Groves, R M A Mustafa · 1974 · Journal of Pharmacy and Pharmacology
  36. Characteristics of lipid substances activating the ileal brake in the rat.
    Nicola Jane Brown, N. W. Read, Alan Richardson, R.D.E. Rumsey, Conny B. Bogentoft · 1990 · Gut
  37. Ionic Liquid Versus Prodrug Strategy to Address Formulation Challenges
    Anja Balk, Toni Widmer, Johannes M. Wiest, H. D. Bruhn, J.-C. Rybak, Philipp R. Matthes, Klaus Müller‐Buschbaum, Anastasios Sakalis, Tessa C. Lühmann, Jörg Berghausen et al. · 2014 · Pharmaceutical Research
  38. Drug release from lipid-based dosage forms. II
    N.A. Armstrong, Kenneth James · 1980 · International Journal of Pharmaceutics
  39. Analytical technologies for real-time drug dissolution and precipitation testing on a small scale
    Martin Kuentz · 2014 · Journal of Pharmacy and Pharmacology
  40. In vivo evaluation of tablets and capsules containing spray-dried o/w-emulsions for oral delivery of poorly soluble drugs
    Tue Hansen, Per Holm, Morten Rohde, Kirsten Schultz · 2005 · International Journal of Pharmaceutics
  41. Lipophilic prodrugs of apomorphine I: Preparation, characterisation, and in vitro enzymatic hydrolysis in biorelevant media
    Nrupa Borkar, Boyang Li, René Holm, Anders E. Håkansson, Anette Müllertz, Mingshi Yang, Huiling Mu · 2014 · European Journal of Pharmaceutics and Biopharmaceutics
  42. GASTROINTESTINAL ABSORPTION OF GRISEOFULVIN: I. EFFECT OF PARTICLE SIZE, ADDITION OF SURFACTANTS, AND CORN OIL ON THE LEVEL OF GRISEOFULVIN IN THE SERUM OF RATS
    M. Kraml, Jean Dubuc, Desmond Beall, Nicole L'Heureux · 1962 · Canadian Journal of Biochemistry and Physiology
  43. The Mechanism of Lymphatic Access of Two Cholesteryl Ester Transfer Protein Inhibitors (CP524,515 and CP532,623) and Evaluation of Their Impact on Lymph Lipoprotein Profiles
    Natalie L. Trevaskis, Ravi M. Shanker, William N. Charman, Christopher J. H. Porter · 2010 · Pharmaceutical Research
  44. Pluronic and Tetronic Copolymers with Polyglycolyzed Oils as Self-Emulsifying Drug Delivery Systems
    Marta Fernandez-Tarrio, Fernando Yáñez, Kristof Immesoete, Carmen Alvarez‐Lorenzo, Ángel Concheiro · 2008 · AAPS PharmSciTech
  45. The Potential for Drug Supersaturation during Intestinal Processing of Lipid-Based Formulations May Be Enhanced for Basic Drugs
    Yan Yan Yeap, Natalie L. Trevaskis, Christopher J. H. Porter · 2013 · Molecular Pharmaceutics
  46. Profiling the Role of Deacylation-Reacylation in the Lymphatic Transport of a Triglyceride-Mimetic Prodrug
    Sifei Han, Luojuan Hu, Tim Quach, Jamie S. Simpson, Natalie L. Trevaskis, Christopher J. H. Porter · 2014 · Pharmaceutical Research
  47. Glyceride Lipid Formulations: Molecular Dynamics Modeling of Phase Behavior During Dispersion and Molecular Interactions Between Drugs and Excipients
    Dallas B. Warren, Dylan T. King, Hassan Benameur, Colin William Pouton, David K. Chalmers · 2013 · Pharmaceutical Research
  48. Biorelevant media resistant co-culture model mimicking permeability of human intestine
    Delphine Antoine, Yann Pellequer, Camille Tempesta, Stefan Lorscheidt, Bernadette Kettel, Lana Tamaddon, Vincent Jannin, Frédéric Demarne, Alf Lamprecht, Arnaud Béduneau · 2015 · International Journal of Pharmaceutics
  49. AN EXAMINATION OF THE INTERPLAY BETWEEN ENTEROCYTE-BASED METABOLISM AND LYMPHATIC DRUG TRANSPORT IN THE RAT
    Natalie L. Trevaskis, Christopher J. H. Porter, William N. Charman · 2006 · Drug Metabolism and Disposition
  50. Proposal of stability categories for nano-dispersions obtained from pharmaceutical self-emulsifying formulations
    Andreas Niederquell, Martin Kuentz · 2013 · International Journal of Pharmaceutics
  51. Drug migration into soft gelatin capsule shells and its effect on in-vitro availability
    N A Armstrong, Kenneth James, W K L Pugh · 1984 · Journal of Pharmacy and Pharmacology
  52. Elucidating the Molecular Interactions Occurring during Drug Precipitation of Weak Bases from Lipid-Based Formulations: A Case Study with Cinnarizine and a Long Chain Self-Nanoemulsifying Drug Delivery System
    Philip Jonas Sassene, Mette Dalskov Mosgaard, Korbinian Löbmann, Huiling Mu, Flemming Hofmann Larsen, Thomas Rades, Anette Müllertz · 2015 · Molecular Pharmaceutics
  53. Biopharmaceutical Modeling of Drug Supersaturation During Lipid-Based Formulation Digestion Considering an Absorption Sink
    Cordula Stillhart, Georgios Imanidis, Brendan T. Griffin, Martin Kuentz · 2014 · Pharmaceutical Research
  54. The effect of oral lipids and circulating lipoproteins on the metabolism of drugs
    Jigar P. Patel, Dion R. Brocks · 2009 · Expert Opinion on Drug Metabolism & Toxicology
  55. Lipidic dispersion to reduce food dependent oral bioavailability of fenofibrate: In vitro, in vivo and in silico assessments
    Joseph P. O’Shea, Waleed Faisal, Therese Ruane-O’Hora, Ken J. Devine, Edmund S. Kostewicz, Caitríona M. O’Driscoll, Brendan T. Griffin · 2015 · European Journal of Pharmaceutics and Biopharmaceutics
  56. The disintegration behaviour of capsules in fed subjects: A comparison of hypromellose (carrageenan) capsules and standard gelatin capsules
    Brian E. Jones, Abdul W. Basit, Catherine Tuleu · 2011 · International Journal of Pharmaceutics
  57. Comparison of high-resolution ultrasonic resonator technology and Raman spectroscopy as novel process analytical tools for drug quantification in self-emulsifying drug delivery systems
    Cordula Stillhart, Martin Kuentz · 2011 · Journal of Pharmaceutical and Biomedical Analysis
  58. Effect of food intake and co-administration of placebo self-nanoemulsifying drug delivery systems on the absorption of cinnarizine in healthy human volunteers
    Martin Lau Christiansen, René Holm, Bertil Abrahamsson, Jette Bredahl Jacobsen, Jakob Kristensen, Jens Rikardt Andersen, Anette Müllertz · 2016 · European Journal of Pharmaceutical Sciences
  59. An in Vitro Digestion Test That Reflects Rat Intestinal Conditions To Probe the Importance of Formulation Digestion vs First Pass Metabolism in Danazol Bioavailability from Lipid Based Formulations
    Mette U. Anby, Tri‐Hung Nguyen, Yan Yan Yeap, Orlagh M. Feeney, Hywel D. Williams, Hassan Benameur, Colin William Pouton, Christopher J. H. Porter · 2014 · Molecular Pharmaceutics
  60. In vitro and in vivo evaluation of a matrix-in-cylinder system for sustained drug delivery
    Els Mehuys, Chris Vervaet, Ingrid Gielen, Henri van Bree, Jean Paul Remon · 2004 · Journal of Controlled Release
  61. Tableting Lipid-Based Formulations for Oral Drug Delivery: A Case Study with Silica Nanoparticle–Lipid–Mannitol Hybrid Microparticles
    Kristen E. Bremmell, Angel Tan, Amanda L. Martin, Clive A. Prestidge · 2012 · Journal of Pharmaceutical Sciences
  62. Biopharmaceutical studies of lipid-containing oral dosage forms: Relationship between drug absorption rate and digestibility of vehicles
    Yoshiya Yamahira, Noguchi Takeshi, Hiroshi Takenaka, Maeda Tadao · 1979 · International Journal of Pharmaceutics
  63. Trends in the Assessment of Drug Supersaturation and Precipitation In Vitro Using Lipid-Based Delivery Systems
    Cordula Stillhart, Martin Kuentz · 2016 · Journal of Pharmaceutical Sciences
  64. Acidic mucin layer facilitates micelle dissociation and fatty acid diffusion
    Y. F. Shiau, R. J. Kelemen, M. A. Reed · 1990 · American Journal of Physiology-Gastrointestinal and Liver Physiology
  65. In vitro and in vivo preclinical evaluation of a minisphere emulsion-based formulation (SmPill®) of salmon calcitonin
    Tanira Alessandra Silveira Aguirre, Mónica Rosa, Ivan S. Coulter, David J. Brayden · 2015 · European Journal of Pharmaceutical Sciences
  66. Chemical Drug Stability in Lipids, Modified Lipids, and Polyethylene Oxide-Containing Formulations
    Valentino J. Stella · 2013 · Pharmaceutical Research
  67. In Vivo Formation of Cubic Phase in Situ after Oral Administration of Cubic Phase Precursor Formulation Provides Long Duration Gastric Retention and Absorption for Poorly Water-Soluble Drugs
    Anna C. Pham, Linda Hong, Oliver D. Montagnat, Cameron J. Nowell, Tri‐Hung Nguyen, Ben J. Boyd · 2015 · Molecular Pharmaceutics
  68. Human bioavailability of propranolol from a matrix-in-cylinder system with a HPMC-Gelucire® core
    Els Mehuys, Jean Paul Remon, Annelies E. C. Korst, Luc MAB. Van Bortel, Raf Mols, Patrick Augustijns, Christopher J. H. Porter, Chris Vervaet · 2005 · Journal of Controlled Release
  69. The use of supports in the lyophilization of oil-in-water emulsions
    M Lladser, Claudia Alejandra Medrano, A Arancibia · 1968 · Journal of Pharmacy and Pharmacology
  70. In vitro–in vivo evaluation of lipid based formulations of the CETP inhibitors CP-529,414 (torcetrapib) and CP-532,623
    Claire L. McEvoy, Natalie L. Trevaskis, Glenn Anthony Edwards, Michael E. Perlman, Catherine M. Ambler, Mary Catherine Mack, Barbara Brockhurst, Christopher J. H. Porter · 2014 · European Journal of Pharmaceutics and Biopharmaceutics
  71. In vitro and in vivo evaluations of the performance of an indirubin derivative, formulated in four different self-emulsifying drug delivery systems
    Nasim Heshmati, Xinlai Cheng, Else Dapat, Philip Jonas Sassene, Gerhard Eisenbrand, Gert Fricker, Anette Müllertz · 2014 · Journal of Pharmacy and Pharmacology
  72. A simplified method to screen for in-vivo performance of oral lipid formulations
    Murat Kilic, Jennifer Dressman · 2013 · Journal of Pharmacy and Pharmacology
  73. Study of drug supersaturation for rational early formulation screening of surfactant/co-solvent drug delivery systems
    Cordula Stillhart, Martin Cavegn, Martin Kuentz · 2012 · Journal of Pharmacy and Pharmacology
  74. In Vitro Lipolysis and Intestinal Transport of β-Arteether-Loaded Lipid-Based Drug Delivery Systems
    Patrick B. Memvanga, Pierre Eloy, Éric M. Gaigneaux, Véronique Préat A · 2013 · Pharmaceutical Research
  75. Pancreatic Lipase-Catalyzed Hydrolysis of Esters of Hydroxymethyl Phenytoin Dissolved in Various Metabolizable Vehicles, Dispersed in Micellar Systems, and in Aqueous Suspensions
    Francisco J. Álvarez, Valentine J. Stella · 1989 · Pharmaceutical Research
  76. Physicochemical Characterization of Simulated Intestinal Fed-State Fluids Containing Lyso-Phosphatidylcholine and Cholesterol
    Dimitris G. Fatouros, Isabelle Walrand, Björn Bergenståhl, Anette Müllertz · 2009 · Dissolution Technologies
  77. Biopharmaceutical studies of lipid-containing oral dosage forms: Relationship between drug absorption and gastric emptying of lipid formulations.
    Yoshiya Yamahira, TAKESHI NOGUCHI, Hiroshi Takenaka, TADAO MAEDA · 1978 · Journal of Pharmacobio-Dynamics
  78. A prodrug strategy for the oral delivery of a poorly soluble HCV NS5B thumb pocket 1 polymerase inhibitor using self-emulsifying drug delivery systems (SEDDS)
    Pierre L. Beaulieu, Josie De Marte, Michel Garneau, Laibin Luo, Timothy A. Stammers, Chitra Telang, Dominik Wernic, George Kukolj, Jianmin Duan · 2014 · Bioorganic & Medicinal Chemistry Letters
  79. Preliminary development and evaluation of a parenteral emulsion formulation of penclomedine (NSC-338720; 3,5-dichloro-2,4-dimethoxy-6-trichloromethylpyridine): a novel, practically water insoluble cytotoxic agent.
    R.J. Prankerd, Sylvan G. Frank, Valentine J. Stella · 1989 · PubMed
  80. Novel semisolid SNEDDS based on PEG-30-di-(polyhydroxystearate): Progesterone incorporation and in vitro digestion
    Tamer H. Hassan, Karsten Mäder · 2015 · International Journal of Pharmaceutics
  81. [Research on the spray drying of emulsified medical preparations. 1].
    A RICHTER, K Steiger-Trippi · 1961 · PubMed
  82. Plasma concentrations after oral administration of different pharmaceutical preparations of clomethiazole.
    M Fischler, Frisch Ep, B. Örtengren · 1973 · PubMed
  83. Oral Sulfonamides in Lipid Emulsion
    C. W. Daeschner · 1957 · A M A Journal of Diseases of Children
  84. Steroidal ethers: urinary excretion of pregnanediols in man after ingestion of quingestrone in fasting or non-fasting conditions.
    G Bruni, F Galletti · 1970 · PubMed
  85. Absorption and chemotherapeutic activity of acetyl sulfisoxazole suspended in an oil in water emulsion.
    Svenson Se, W. F. DeLorenzo, Recha Engelberg, MILDRED E. SPOONER, L O RANDALL · 1956 · PubMed