Broad-Spectrum Therapeutic Suppression of Metastatic Melanoma through Nuclear Hormone Receptor Activation
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- Prognostic role of liver X receptor‐alpha in resected stage II and III non‐small‐cell lung cancerGiulio Melloni, Piergiorgio Muriana, Alessandro Bandiera, Raffaella Fontana, Daniela Maggioni, Vincenzo E. A. Russo, Claudio Doglioni, Piero Zannini · 2016 · The Clinical Respiratory Journal
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- RXR signaling targeted cancer therapyWenrui Zhao, Suyao Li, Ruoxue Chen, Junjie Ni, Xuan Huang, Song Li, Xiaoling Lü, Xin Cao · 2023 · The Innovation Life
- New Insights in Prostate Cancer Development and Tumor Therapy: Modulation of Nuclear Receptors and the Specific Role of Liver X ReceptorsLaura Bousset, Amandine Rambur, Allan Fouache, Julio Buñay, Laurent Morel, Jean‐Marc A. Lobaccaro, Silvère Baron, Amalia Trousson, Cyrille de Joussineau · 2018 · International Journal of Molecular Sciences
- The critical function of metabolic reprogramming in cancer metastasisSun‐Zhe Xie, Jun‐Jie Pan, Jianfeng Xu, Wenwei Zhu, Lun–Xiu Qin · 2022 · Aging and Cancer
- The environmental obesogen bisphenol A increases macrophage self-renewalGrace Ampem, Alexandra Junginger, Haidong Yu, Lajos Balogh, Julianna Thuróczy, Marion E. Schneider, Tamás Rőszer · 2019 · Cell and Tissue Research
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- Activation of Liver X Receptor α Sensitizes Mice to T‐Cell Mediated HepatitisLi Gao, Bin Li, Jingyuan Wang, Danhua Shen, Min Yang, Runzi Sun, Hung‐Chun Tung, Meishu Xu, Songrong Ren, Min Zhang et al. · 2020 · Hepatology Communications
- LXR Inhibits Proliferation of Human Breast Cancer Cells through the PI3K-Akt PathwayTreska S. Hassan, Aida Paniccia, Vincenzo E. A. Russo, Knut Rune Steffensen · 2015 · Nuclear Receptor Research
- Brain penetrant liver X receptor (LXR) modulators based on a 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole coreColin M. Tice, Paul Bart Noto, Kristi Yi Fan, Wei Liang Zhao, Stephen D. Lotesta, Chengguo Dong, Andrew P. Marcus, Ya‐Jun Zheng, Guozhou Chen, Zhongren Wu et al. · 2016 · Bioorganic & Medicinal Chemistry Letters
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- Role of the liver X receptors in skin physiology: Putative pharmacological targets in human diseasesZangbéwendé Guy Ouedraogo, Allan Fouache, Amalia Trousson, Silvère Baron, Jean‐Marc A. Lobaccaro · 2017 · Chemistry and Physics of Lipids
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- Reduction of fibrosis and immune suppressive cells in ErbB2-dependent tumorigenesis by an LXR agonistSheng Gao, Hongyan Yuan, Lü Jin, Suman Ranjit, Julia Panov, Xun Lu, Moshe Levi, Robert I. Glazer · 2021 · PLoS ONE
- 1α-Hydroxy derivatives of 7-dehydrocholesterol are selective liver X receptor modulatorsKaori Endo‐Umeda, Atsushi Aoyama, Masato Shimizu, Minoru Ishikawa, Yuichi Hashimoto, Sachiko Yamada, Makoto Makishima · 2017 · The Journal of Steroid Biochemistry and Molecular Biology
- RETRACTED ARTICLE: Liver X receptors constrain tumor development and metastasis dissemination in PTEN-deficient prostate cancerAnthony Alioui, Julie Dufour, Valerio Leoni, Anke Loregger, Martina Moeton, Luigi Iuliano, Chiara Zerbinati, Amandine Septier, Pierre Val, Allan Fouache et al. · 2017 · Nature Communications · Retracted
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- Lipoprotein Deprivation Reveals a Cholesterol-Dependent Therapeutic Vulnerability in Diffuse Glioma MetabolismJames Wood, Salah Abdelrazig, Sergey Evseev, Catherine A. Ortori, Marcos Castellanos‐Uribe, Sean Tobias May, David A. Barrett, Mohammed Diksin, Sajib Chakraborty, Dong‐Hyun Kim et al. · 2022 · Cancers
- A Novel Liver X Receptor Inverse Agonist Impairs Cholesterol and Phospholipid Metabolism and Induces Apoptosis and Necroptosis in Pancreatic Ductal Adenocarcinoma CellsScott Widmann, Shivangi Srivastava, Chin‐Yo Lin · 2023 · Receptors
- ATF4/TXNIP/REDD1/mTOR signaling mediates the antitumor activities of liver X receptor in pancreatic cancersZhikang Chen, Xiaobo Lai, Hui Ding, Aijun Zhang, Yufei Sun, Jianhua Ling, Paul J. Chiao, Zihua Chen, Xuefeng Xia · 2022 · Cancer Innovation
- Liver X receptors induce antiproliferative effects in basal‐like breast cancerMads Haugland Haugen, Hedda von der Lippe Gythfeldt, Eivind Valen Egeland, Lisa Svartdal Normann, Abhilash D. Pandya, Lise‐Lotte Vedin, Siri Juell, Ellen M. Tenstad, Geir Frode Øy, Alexandr Kristian et al. · 2023 · Molecular Oncology
- A Subset of Nuclear Receptors are Uniquely Expressed in Uveal Melanoma CellsKenneth E. Huffman, Ryan M. Carstens, Elisabeth D. Martínez · 2015 · Frontiers in Endocrinology
- In vivo assessment of the vascular disrupting effect of M410 by DCE-MRI biomarker in a rabbit model of liver tumorRUI-MENG YANG, Yong Zou, Danping Huang, Shengsheng Lai, Xiangdong Xu, Xinhua Wei, HAN-ZHENG CHANG, Tongkun Huang, LI WANG, Wenjie Tang et al. · 2014 · Oncology Reports
- Pivotal role of intestinal cholesterol and nuclear receptor LXR in metabolic liver steatohepatitis and hepatocarcinomaElena Piccinin, Maria Arconzo, Emanuela Pasculli, Angela Fulvia Tricase, Silvia Cultrera, Justine Bertrand‐Michel, Nicolas Loiseau, Gaetano Villani, Hervé Guillou, Antonio Moschetta · 2024 · Cell & Bioscience
- Lipids and prostate cancer adenocarcinomaAnthony Alioui, O. Celhay, Silvère Baron, Jean‐Marc A. Lobaccaro · 2014 · Clinical Lipidology
- A new weapon against metastatic melanomaKatie Kingwell · 2014 · Nature Reviews Drug Discovery
- Targeting Liver X Receptors in Cancer Drug DiscoveryAsitha Premaratne, Abhinav Bagchi, Shinjini Basu, Jan-Ακε Gustafsson, Chin‐Yo Lin · 2024 · Receptors
- Transcriptional and non-transcriptional roles of LXRs in cancer cells2015 · Receptors & Clinical Investigation
- A transcriptional mechanism involving R-loop, m6A modification and RNA abasic sites regulates an enhancer RNA of APOEJason A. Watts, Christopher Grunseich, Yesenia Rodriguez, Yaojuan Liu, Dongjun Li, Joshua T. Burdick, Alan Bruzel, Robert J. Crouch, Robert W. Mahley, Samuel H. Wilson et al. · 2022 · bioRxiv (Cold Spring Harbor Laboratory)
- Regulation of neurogenesis and neuronal migration by Rrm2 and Timp3 following seizuresAdebayo Olukayode Adeyeye, Parul Varma, Nico Enerlan, Marissa Olga Coppin, Jenny Hsieh · 2025 · Neurobiology of Disease
- A Stable Luciferase Reporter System to Characterize LXR Regulation by Oxysterols and Novel LigandsSamantha A. Hutchinson, James L. Thorne · 2019 · Methods in molecular biology
- Receptor agonist/antagonist-incorporated anticancer nanodrugs: Design, materials, and strategiesShi-Jie Hao, Shun‐Yu Wu, Yun-Kai Chang, Fu‐Gen Wu · 2024 · Materials Today
- Preclinical Models of Brain MetastasisLucía Zhu, Manuel Valiente · 2020 · Springer eBooks
- Lipid metabolism and signaling in cancerElena Piccinin, James Mukasa Ntambi, Antonio Moschetta · 2020 · Elsevier eBooks
- Immunosuppressive triangle depletion through the combination punches strategy for enhanced immunotherapyQianhua Feng, Huifang Xiao, Cuixia Zheng, Xueli Zhang, Zeying Wang, Lei Wang · 2021 · Applied Materials Today
- Retraction Note: Liver X receptors constrain tumor development and metastasis dissemination in PTEN-deficient prostate cancerAnthony Alioui, Julie Dufour, Valerio Leoni, Anke Loregger, Martina Moeton, Luigi Iuliano, Chiara Zerbinati, Amandine Septier, Pierre Val, Allan Fouache et al. · 2018 · Nature Communications · Retracted
- Nucleolar protein 7 facilitates melanoma progression and metastasis via HIF-1ɑ/PI3K/AKT/ERK axisYumei Li, Fan Chen, Weiyu Shen, Bifei Li, Ning Zheng, Yusheng Lu, Vladimir L. Katanaev, Lee Jia · 2020 · Research Square
- Liver X receptors—a new target for cancer treatmentLiu Xiaowang, Kaiqiang Lu, Ting Xiong, Zhou Zhigang · 2016
- 強心配糖体ウアバインのアグリコン「ウアバゲニン」の新規生理活性Satoru Tamura, Maiko Okada, Minoru Ueda · 2018 · KAGAKU TO SEIBUTSU
- Activation of Lxrβ Causes Metabolic Reprogramming and Sensitizes Solid Tumors to Bcl-xL Inhibition Mediated ApoptosisChiaki Tsuge Ishida, Yiru Zhang, Elena Bianchetti, Chang Shu, Maria J. Sanchez‐Quintero, Catarina Maria Quinzii, Mike‐Andrew Westhoff, Georg Karpel‐Massler, Peter Canoll, Markus David Siegelin · 2018 · SSRN Electronic Journal
- [The direct isotopic cystography in the study of the vesico-ureteral reflux (author's transl)].J C Fombellida Cortázar, J Simón González, M.C. Cano Terol, J Alonso Monfort, I. Zamora Marti · 1978 · PubMed
- Faculty Opinions recommendation of Lxr/apoe activation restricts innate immune suppression in cancer.Philippe Saas, Sylvain Perruche · 2018 · Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
- Data from Neutral Sphingomyelinase 2 Heightens Anti-Melanoma Immune Responses and Anti–PD-1 Therapy EfficacyAnne Montfort, Florie A. Bertrand, Julia Rochotte, Julia Gilhodes, Thomas Filleron, Jean Milhès, Carine Dufau, Caroline Imbert, Joëlle Riond, Marie Tosolini et al. · 2023
- Data from Neutral Sphingomyelinase 2 Heightens Anti-Melanoma Immune Responses and Anti–PD-1 Therapy EfficacyAnne Montfort, Florie A. Bertrand, Julia Rochotte, Julia Gilhodes, Thomas Filleron, Jean Milhès, Carine Dufau, Caroline Imbert, Joëlle Riond, Marie Tosolini et al. · 2023
- Integrated Whole Exome and Transcriptome Sequencing in Cholesterol Metabolism in Melanoma: Systematic ReviewMohamed Mahmoud Nour Eldein, Wesam Ahmed Nasif, Wesam Ahmed Nasif, Amr Ahmed Amin, Gad Allah Modawe, Abdullatif Taha Babakr · 2024 · Sudan Journal of Medical Sciences
- Unlocking the potential of Liver X Receptors: A new era in metabolic regulationImroze Singh, Suman Kalia · 2025 · International Journal of Pharmacology and Clinical Research
- Comprehensive analysis reveals MCM4 as a biomarker for guiding therapies and immunomodulatory role in skin cutaneous melanomaWei Ou, Jiang Zhou, Zhenhua Huang, XinLiang Yang, Xiaohong Liu, Wenjian Zuo, ZhiYong Luo, Min Su · 2025 · Journal of Cancer
- Additional file 1 of Pivotal role of intestinal cholesterol and nuclear receptor LXR in metabolic liver steatohepatitis and hepatocarcinomaElena Piccinin, Maria Arconzo, Emanuela Pasculli, Angela Fulvia Tricase, Silvia Cultrera, Justine Bertrand‐Michel, Nicolas Loiseau, Gaetano Villani, Hervé Guillou, Antonio Moschetta · 2024 · Figshare
- Additional file 2 of Pivotal role of intestinal cholesterol and nuclear receptor LXR in metabolic liver steatohepatitis and hepatocarcinomaElena Piccinin, Maria Arconzo, Emanuela Pasculli, Angela Fulvia Tricase, Silvia Cultrera, Justine Bertrand‐Michel, Nicolas Loiseau, Gaetano Villani, Guillou, Hervé, Antonio Moschetta · 2024 · Figshare
- Epigenetic regulation of gene expression during melanocyte and melanoma developmentPatrick Laurette · 2016 · theses.fr (ABES)
- Nouveaux modèles pour le criblage de modulateurs / perturbateurs des voies de signalisation régulées par les Liver X receptorsAllan Fouache · 2018 · theses.fr (ABES)
- Rôle de la sphingosine kinase-1 dans la réponse immunitaire anti-tumorale et dans le traitement du mélanome par immunothérapieCaroline Imbert · 2018 · theses.fr (ABES)
- Cancer de la prostate et mécanismes de résistance à la castration : étude du rôle des récepteurs nucléaires LXRLaura Bousset · 2019 · theses.fr (ABES)
- MARCH2 prevents doxorubicin-induced cardiomyopathy by stabilizing NR1H2 and promoting clearance of apoptotic cardiomyocytesliu shuolin, Yiran E. Li, Tingfang Zhu, Laihai Zhang, Cong Yang, Yaguang Bi, Chenglong Bao, Ronggui Hu, Junbo Ge, Yingmei Zhang · 2026 · Nature Communications
- Integrating proteomics and metabolomics to reveal MAT2A for metabolic reprogramming in non-small cell lung cancer cellsYimin Chen, Yuxi Liu, Zhenyun Zhu, Anqi Ding, Yuying Suo, Cheng Wang, Xiongjun Wang, Hu Zhou, Qiyu Fang, Qian Liu · 2026 · iScience
- Three decades of liver X receptor agonist chemistry: Structural motifs, structure-activity relationship, and therapeutic prospectsNorberta Delporte, Aurélie Lagarde, Pierre Chalard, Silvère Baron, Amalia Trousson, Jean‐Marc A. Lobaccaro, Isabelle Thomas · 2026 · The Journal of Steroid Biochemistry and Molecular Biology
- BindingDB Entry 50011862: Discovery of new LXRβ agonists as glioblastoma inhibitors.BindingDB · 2022 · UC San Diego
- BindingDB Entry 50008390: Development of novel liver X receptor modulators based on a 1,2,4-triazole scaffold.BindingDB · 2021 · UC San Diego
- BindingDB Entry 50047831: Brain penetrant liver X receptor (LXR) modulators based on a 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole core.BindingDB · 2018 · UC San Diego
- BindingDB Entry 50003012: Recent Advances in the Medicinal Chemistry of Liver X Receptors.BindingDB · 2020 · UC San Diego
- BindingDB Entry 50019169: Discovery of Spiro[pyrrolidine-3,3'-oxindole] LXRβ Agonists for the Treatment of Osteoporosis.BindingDB · 2024 · UC San Diego