Oral epidermal growth factor receptor tyrosine kinase inhibitors for the treatment of non-small cell lung cancer: Comparative pharmacokinetics and drug–drug interactions
Peters, Solange, Zimmermann, Stefan, Adjei, Alex A.·2014·Cancer Treatment Reviews
Cited by (163)
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- BindingDB Entry 50022681: FDA-approved small molecule kinase inhibitors for cancer treatment (2001-2015): Medical indication, structural optimization, and binding mode Part I.BindingDB · 2026 · UC San Diego
- BindingDB Entry 50003219: Recent updates on third generation EGFR inhibitors and emergence of fourth generation EGFR inhibitors to combat C797S resistance.BindingDB · 2020 · UC San Diego
- BindingDB Entry 50009645: Discovery of a Furanopyrimidine-Based Epidermal Growth Factor Receptor Inhibitor (DBPR112) as a Clinical Candidate for the Treatment of Non-Small Cell Lung Cancer.BindingDB · 2021 · UC San Diego
- BindingDB Entry 50013124: Discovery of Dosimertinib, a Highly Potent, Selective, and Orally Efficacious Deuterated EGFR Targeting Clinical Candidate for the Treatment of Non-Small-Cell Lung Cancer.BindingDB · 2022 · UC San Diego
- BindingDB Entry 50017048: Small Molecule Kinase Inhibitor Drugs (1995-2021): Medical Indication, Pharmacology, and Synthesis.BindingDB · 2023 · UC San Diego
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- BindingDB Entry 50023144: Structure-Based Design of New LSD1/EGFRL858R/T790M Dual Inhibitors for Treating EGFR Mutant NSCLC Cancers.BindingDB · 2026 · UC San Diego
- BindingDB Entry 50001303: Design, Synthesis, and Biological Evaluation of Pyrimido[4,5- d]pyrimidine-2,4(1 H,3 H)-diones as Potent and Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors against L858R/T790M Resistance Mutation.BindingDB · 2020 · UC San Diego
- BindingDB Entry 50013716: Design, synthesis and biological evaluation of sulfamoylphenyl-quinazoline derivatives as potential EGFR/CAIX dual inhibitors.BindingDB · 2022 · UC San Diego
- BindingDB Entry 50012225: Design, synthesis and biological evaluation of 2-amino-4-(1,2,4-triazol)pyridine derivatives as potent EGFR inhibitors to overcome TKI-resistance.BindingDB · 2022 · UC San Diego