The Vinylogous Aldol and Related Addition Reactions: Ten Years of Progress

The Vinylogous Aldol Reaction: A Valuable, Yet Understated Carbon−Carbon Bond-Forming Maneuver

Casiraghi, G., Zanardi, F., Appendino, G., & Rassu, G. (2000) · Chemical Reviews · doi:10.1021/cr990247i · Cited by 566

C2-Symmetric Copper(II) Complexes as Chiral Lewis Acids. Scope and Mechanism of Catalytic Enantioselective Aldol Additions of Enolsilanes to (Benzyloxy)acetaldehyde

Evans, D. A., Kozlowski, M. C., Murry, J. A., Burgey, C. S., Campos, K. R., Connell, B. T., & Staples, R. J. (1999) · Journal of the American Chemical Society · doi:10.1021/ja9829822 · Cited by 388

A novel and efficient macrolactonization of ω-hydroxycarboxylic acids using 2-methyl-6-nitrobenzoic anhydride (MNBA)

Shiina, I., Kubota, M., & Ibuka, R. (2002) · Tetrahedron Letters · doi:10.1016/s0040-4039(02)01819-1 · Cited by 275

Chiral Organic Ion Pair Catalysts Assembled Through a Hydrogen-Bonding Network

Uraguchi, D., Ueki, Y., & Ooi, T. (2009) · Science · doi:10.1126/science.1176758 · Cited by 247

Chiral Brønsted Acid Catalyzed Enantioselective Aza‐Diels–Alder Reaction of Brassard's Diene with Imines

Itoh, J., Fuchibe, K., & Akiyama, T. (2006) · Angewandte Chemie International Edition · doi:10.1002/anie.200601345 · Cited by 232

Sol–Gel Polycondensation of Tetraethoxysilane in a Cholesterol-Based Organogel System Results in Chiral Spiral Silica

Jung, J. H., Ono, Y., & Shinkai, S. (2000) · Angewandte Chemie International Edition · doi:10.1002/(sici)1521-3773(20000515)39:10<1799::aid-anie1799>3.0.co;2-z · Cited by 204

Palmerolide A, a Cytotoxic Macrolide from the Antarctic Tunicate Synoicum adareanum

Diyabalanage, T., Amsler, C. D., McClintock, J. B., & Baker, B. J. (2006) · Journal of the American Chemical Society · doi:10.1021/ja0588508 · Cited by 176

Synthesis and Structure Revision of Nakiterpiosin

Gao, S., Wang, Q., & Chen, C. (2008) · Journal of the American Chemical Society · doi:10.1021/ja808110d · Cited by 152

Callipeltoside A: A Cytotoxic Aminodeoxy Sugar-Containing Macrolide of a New Type from the Marine Lithistida Sponge Callipelta sp.

Zampella, A., D’Auria, M. V., Minale, L., Debitus, C., & Roussakis, C. (1996) · Journal of the American Chemical Society · doi:10.1021/ja9621004 · Cited by 148

Total Synthesis and Structural Revision of the Marine Macrolide Neopeltolide

Custar, D., Zabawa, T. P., & Scheidt, K. A. (2007) · Journal of the American Chemical Society · doi:10.1021/ja710080q · Cited by 139

Total Synthesis and Structure Revision of the Marine Metabolite Palmerolide A

Jiang, X., Liu, B., Lebreton, S., & Brabander, J. K. D. (2007) · Journal of the American Chemical Society · doi:10.1021/ja0715142 · Cited by 114

Total Synthesis of the Originally Proposed and Revised Structures of Palmerolide A

Nicolaou, K. C., Guduru, R., Sun, Y., Banerji, B., & Chen, D. Y. ‐. (2007) · Angewandte Chemie International Edition · doi:10.1002/anie.200702243 · Cited by 101

Total Synthesis and Structure−Activity Investigation of the Marine Natural Product Neopeltolide

Custar, D., Zabawa, T. P., Hines, J. F., Crews, C. M., & Scheidt, K. A. (2009) · Journal of the American Chemical Society · doi:10.1021/ja904604x · Cited by 97

The Synthesis of gama-Alkylidenebutenolides

Brückner, R. (2001) · Current Organic Chemistry · doi:10.2174/1385272013375300 · Cited by 93

Chemical and Biological Studies of Nakiterpiosin and Nakiterpiosinone

Gao, S., Wang, Q., Huang, L. J.-S., Lum, L., & Chen, C. (2009) · Journal of the American Chemical Society · doi:10.1021/ja908626k · Cited by 84

Aurilide, a cytotoxic depsipeptide from the sea hare Dolabella auricularia: isolation, structure determination, synthesis, and biological activity

Suenaga, K., Mutou, T., Shibata, T., et al. (2004) · Tetrahedron · doi:10.1016/j.tet.2004.06.125 · Cited by 84

Kulokekahilide-2, a Cytotoxic Depsipeptide from a Cephalaspidean Mollusk Philinopsis speciosa

Nakao, Y., Yoshida, W. Y., Takada, Y., Kimura, J., Liu, Y., Mooberry, S. L., & Scheuer, P. J. (2004) · Journal of Natural Products · doi:10.1021/np049949f · Cited by 82

Catalytic Asymmetric Vinylogous Mukaiyama-Aldol (CAVM) Reactions: The Enolate Activation

Bluet, G., & Campagne, J. (2001) · The Journal of Organic Chemistry · doi:10.1021/jo015567s · Cited by 79

Organocatalytic Direct Vinylogous Michael Addition of α,β‐Unsaturated γ‐Butyrolactam to α,β‐Unsaturated Aldehydes and an Illustration to Scaffold Diversity Synthesis

Feng, X., Cui, H., Xu, S. C., Wu, L., & Chen, Y. (2010) · Chemistry - A European Journal · doi:10.1002/chem.201001350 · Cited by 76

The Structure of Palau'amide, a Potent Cytotoxin from a Species of the Marine Cyanobacterium Lyngbya

Williams, P. G., Yoshida, W. Y., Quon, M. K., Moore, R. E., & Paul, V. J. (2003) · Journal of Natural Products · doi:10.1021/np034001r · Cited by 70

Lewis Acid−Lewis Base Catalyzed Enantioselective Hetero-Diels−Alder Reaction for Direct Access to δ-Lactones

Tiseni, P. S., & Peters, R. (2008) · Organic Letters · doi:10.1021/ol800742d · Cited by 69

Proline Promoted Synthesis of Ring-Fused Homodimers: Self-Condensation of α,β-Unsaturated Aldehydes

Bench, B. J., Liu, C., Evett, C. R., & Watanabe, C. M. H. (2006) · The Journal of Organic Chemistry · doi:10.1021/jo061763t · Cited by 69

Diastereo‐ and Enantioselective Organocatalytic Direct Conjugate Addition of γ‐Butenolide to Chalcones

Zhang, Y., Yu, C., Ji, Y., & Wang, W. (2010) · Chemistry - An Asian Journal · doi:10.1002/asia.201000014 · Cited by 67

Base‐Catalyzed Condensation of 2‐Hydroxybenzaldehydes with α,β‐Unsaturated Aldehydes – Scope and Limitations

Lesch, B., Toräng, J., Vanderheiden, S., & Bräse, S. (2005) · Advanced Synthesis & Catalysis · doi:10.1002/adsc.200404239 · Cited by 66

Convergent and Stereoselective Synthesis of Iminosugar-Containing Galfand UDP-GalfMimicks: Evaluation as Inhibitors of UDP-Gal Mutase

Liautard, V., Desvergnes, V., Itoh, K., Liu, H., & Martin, O. R. (2008) · The Journal of Organic Chemistry · doi:10.1021/jo8001134 · Cited by 66

Total Synthesis of Macquarimicins Using an Intramolecular Diels−Alder Approach Inspired by a Biosynthetic Pathway

Munakata, R., Katakai, H., Ueki, T., et al. (2004) · Journal of the American Chemical Society · doi:10.1021/ja048320w · Cited by 61

The β-elimination route to stereodefined γ-alkylidenebutenolides

Brückner, R. (2001) · Chemical Communications · doi:10.1039/b007590f · Cited by 59

A NEW SYNTHESIS OF VITAMIN A

Mukaiyama, T., & Ishida, A. (1975) · Chemistry Letters · doi:10.1246/cl.1975.1201 · Cited by 57

The Stille Reaction in the Synthesis of Carotenoid Butenolides: Synthesis of 6‘-epi-Peridinin

Vaz, B., Álvarez, R., Brückner, R., & de Lera, Á. R. (2005) · Organic Letters · doi:10.1021/ol0478281 · Cited by 56

Total Synthesis and Cytotoxicity Studies of a Cyclic Depsipeptide with Proposed Structure of Palau'amide

Zou, B., Long, K., & Ma, D. (2005) · Organic Letters · doi:10.1021/ol051685g · Cited by 54

Biomimetic Total Synthesis and Antimicrobial Evaluation of Anachelin H

Gademann, K., Bethuel, Y., Locher, H. H., & Hubschwerlen, C. (2007) · The Journal of Organic Chemistry · doi:10.1021/jo701402b · Cited by 54

The four-carbon elongation of three-carbon chiral synthons using 2-(trimethylsiloxy)furan: highly stereocontrolled entry to enantiomerically pure seven-carbon α,β-unsaturated 2,3-dideoxy-aldonolactones

Casiraghi, G., Colombo, L., Rassu, G., Spanu, P., Fava, G. G., & Belicchi, M. F. (1990) · Tetrahedron · doi:10.1016/s0040-4020(01)87777-2 · Cited by 52

Naphthyl Tetronic Acids as Multi‐Target Inhibitors of Bacterial Peptidoglycan Biosynthesis

Mansour, T. S., Caufield, C. E., Rasmussen, B. A., Chopra, R., Krishnamurthy, G., Morris, K., Svenson, K., Bard, J., Smeltzer, C., Naughton, S., et al. (2007) · ChemMedChem · doi:10.1002/cmdc.200700094 · Cited by 45

A convenient catalytic procedure for the highly enantioselective aldol condensation of O-silyldienolates

Rosa, M. D., Acocella, M. R., Villano, R., Soriente, A., & Scettri, A. (2003) · Tetrahedron Asymmetry · doi:10.1016/s0957-4166(03)00494-4 · Cited by 44

Pronounced asymmetric amplification in the aldol condensation of Chan's diene promoted by a Ti(IV)/BINOL complex

Villano, R., Acocella, M. R., Rosa, M. D., Soriente, A., & Scettri, A. (2004) · Tetrahedron Asymmetry · doi:10.1016/j.tetasy.2004.06.009 · Cited by 43

A Flexible Approach to Azasugars: Asymmetric Total Syntheses of (+)‐Castanospermine, (+)‐7‐Deoxy‐6‐epi‐castanospermine, and (+)‐1‐epi‐Castanospermine

Liu, G., Wu, T., Ruan, Y., & Huang, P. (2010) · Chemistry - A European Journal · doi:10.1002/chem.200903490 · Cited by 36

Total synthesis and stereochemical reassignment of (+)-dolastatin 19, a cytotoxic marine macrolide isolated from Dolabella auricularia

Paterson, I., Findlay, A. D., & Florence, G. J. (2007) · Tetrahedron · doi:10.1016/j.tet.2007.01.048 · Cited by 33

Nonlinear effects and auto-induction in the asymmetric aldol condensation of synthetic equivalents of acetoacetic esters

Villano, R., Rosa, M. D., Salerno, C., Soriente, A., & Scettri, A. (2002) · Tetrahedron Asymmetry · doi:10.1016/s0957-4166(02)00539-6 · Cited by 32

Short and Efficient Synthesis of Cryptophycin Unit A

Eißler, S., Nahrwold, M., Neumann, B., Stammler, H., & Sewald, N. (2007) · Organic Letters · doi:10.1021/ol063032l · Cited by 31

Asymmetric auto-inductive aldol reaction by self-assembly of chiral ligands

Rosa, M. D., Acocella, M. R., Soriente, A., & Scettri, A. (2001) · Tetrahedron Asymmetry · doi:10.1016/s0957-4166(01)00261-0 · Cited by 27

Ti(IV)/BINOL-catalyzed asymmetric aldol reaction of a masked acetoacetic ester: pronounced influence of catalyst concentration on nonlinear effects

Rosa, M. D., Acocella, M. R., Villano, R., Soriente, A., & Scettri, A. (2003) · Tetrahedron Letters · doi:10.1016/s0040-4039(03)01470-9 · Cited by 27

Synthesis of enantiomerically pure 2,3-dideoxy-hept-2-enono-1,4-lactone derivatives diastereoselective addition of 2-(trimethylsiloxy)furan to -glyceraldehyde and -serinal-based three-carbon synthons

Casiraghi, G., Colombo, L., Rassu, G., & Spanu, P. (1989) · Tetrahedron Letters · doi:10.1016/s0040-4039(01)93777-3 · Cited by 27

Asymmetric total synthesis of 1-deoxy-7,8-di-epi-castanospermine

Zambrano, V., Rassu, G., Roggio, A., Pinna, L., Zanardi, F., Curti, C., Casiraghi, G., & Battistini, L. (2010) · Organic & Biomolecular Chemistry · doi:10.1039/b924721a · Cited by 25

Enantioselective aldol condensation of O-silyldienolates derived from alkyl-substituted 2,2-dimethyl-[1,3]-dioxin-4-ones

Rosa, M. D., Acocella, M. R., Rega, M. F., & Scettri, A. (2004) · Tetrahedron Asymmetry · doi:10.1016/j.tetasy.2004.07.020 · Cited by 25

A concise approach to (+)-1-epi-castanospermine

Wu, T., & Huang, P. (2007) · Tetrahedron Letters · doi:10.1016/j.tetlet.2007.11.033 · Cited by 22

5-[1‘-(2‘-N-Arylsulfonyl-1‘,2‘,3‘,4‘-tetrahydroisoquinolyl)]-4,5-dihydro-2(3H)-furanones: Positive Allosteric Modulators of the GABAA Receptor with a New Mode of Action

Razet, R., Thomet, U., Furtmüller, R., Chiaroni, A., Sigel, E., Sieghart, W., & Dodd, R. H. (2000) · Journal of Medicinal Chemistry · doi:10.1021/jm001049i · Cited by 22

Use of bicuculline, a GABA antagonist, as a template for the development of a new class of ligands showing positive allosteric modulation of the GABAA receptor

Razet, R., Thomet, U., Furtmüller, R., Jurský, F., Sigel, E., Sieghart, W., & Dodd, R. H. (2000) · Bioorganic & Medicinal Chemistry Letters · doi:10.1016/s0960-894x(00)00514-x · Cited by 19

Synthetic Approaches to Polyhydroxy Indolizidines and Related Azabicyclic Scaffolds

Hanessian, S., Therrien, É., Warrier, J., & Charron, G. (2006) · Heterocycles · doi:10.3987/com-06-s(w)44 · Cited by 13

Computer‐Assisted Synthetic Planning: The End of the Beginning

Szymkuć, S., Gajewska, E. P., Klucznik, T., Molga, K., Dittwald, P., Startek, M., Bajczyk, M., & Grzybowski, B. A. (2016) · Angewandte Chemie International Edition · doi:10.1002/anie.201506101 · Cited by 611