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Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011)

Wang, Jiang, Sánchez-Roselló, María, Aceña, José Luis, del Pozo, Carlos, Sorochinsky, Alexander E., Fustero, Santos, Soloshonok, Vadim A., Liu, Hong·2014·Chemical Reviews
DOI 10.1021/cr4002879
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Abstract

ADVERTISEMENT RETURN TO ISSUEPREVReviewNEXTFluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011)Jiang Wang†, María Sánchez-Roselló‡§, José Luis Aceña∥, Carlos del Pozo‡, Alexander E. Sorochinsky∥⊥#, Santos Fustero*‡§, Vadim A. Soloshonok*∥⊥, and Hong Liu*†View Author Information† Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zu Chong Zhi Road, Shanghai 201203, China‡ Department of Organic Chemistry, Faculty of Pharmacy, University of Valencia, Av. Vicente Andrés Estellés, 46100 Burjassot, Valencia, Spain§ Laboratorio de Moléculas Orgánicas, Centro de Investigación Príncipe Felipe, C/ Eduardo Primo Yúfera 3, 46012 Valencia, Spain∥ Department of Organic Chemistry I, Faculty of Chemistry, University of the Basque Country UPV/EHU, Paseo Manuel Lardizábal 3, 20018 San Sebastian, Spain⊥ IKERBASQUE, Basque Foundation for Science, Alameda Urquijo, 36-5 Plaza Bizkaia, 48011 Bilbao, Spain# Institute of Bioorganic Chemistry and Petrochemistry, National Academy of Sciences of Ukraine, Murmanska Street 1, 02660 Kyiv-94, Ukraine*E-mail: [email protected]*E-mail: [email protected]*E-mail: [email protected]Cite this: Chem. Rev. 2014, 114, 4, 2432–2506Publication Date (Web):December 3, 2013Publication History Received27 May 2013Published online3 December 2013Published inissue 26 February 2014https://pubs.acs.org/doi/10.1021/cr4002879https://doi.org/10.1021/cr4002879review-articleACS PublicationsCopyright © 2013 American Chemical SocietyRequest reuse permissionsArticle Views48704Altmetric-Citations3850LEARN ABOUT THESE METRICSArticle Views are the COUNTER-compliant sum of full text article downloads since November 2008 (both PDF and HTML) across all institutions and individuals. These metrics are regularly updated to reflect usage leading up to the last few days.Citations are the number of other articles citing this article, calculated by Crossref and updated daily. Find more information about Crossref citation counts.The Altmetric Attention Score is a quantitative measure of the attention that a research article has received online. Clicking on the donut icon will load a page at altmetric.com with additional details about the score and the social media presence for the given article. Find more information on the Altmetric Attention Score and how the score is calculated. Share Add toView InAdd Full Text with ReferenceAdd Description ExportRISCitationCitation and abstractCitation and referencesMore Options Share onFacebookTwitterWechatLinked InRedditEmail Other access optionsGet e-Alertsclose SUBJECTS:Anions,Fluorine,Organic compounds,Pharmaceuticals,Reaction products Get e-Alerts

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Items 201–254 of 254

Research works printed but not linked: 301

  1. Christe K. O., 1986, Inorg. Chem., 25, 3721, 10.1021/ic00241a001 · doi:10.1021/ic00241a001
  2. Moissan H., 1896, C. R. Hebd. Acad. Sci., 128, 1543
  3. Ruff O., 1930, Z. Anorg. Allg. Chem., 190, 270, 10.1002/zaac.19301900127 · doi:10.1002/zaac.19301900127
  4. Baasner B., 2000, Houben-Weyl Methods of Organic Chemistry, 10
  5. Marais J. S. C., 1943, Onderstepoort J. Vet. Sci. Anim. Ind., 18, 203
  6. Marais J. S. C., 1944, Onderstepoort J. Vet. Sci. Anim. Ind., 20, 67
  7. Gribble G. W., 2004, J. Chem. Educ., 81, 1441, 10.1021/ed081p1441 · doi:10.1021/ed081p1441
  8. Fuchikami T., 1982, Tetrahedron Lett., 23, 4099, 10.1016/S0040-4039(00)88357-4 · doi:10.1016/s0040-4039(00)88357-4
  9. Ojima I., 1987, J. Am. Chem. Soc., 109, 7714, 10.1021/ja00259a020 · doi:10.1021/ja00259a020
  10. Ojima I., 1988, J. Am. Chem. Soc., 110, 150, 10.1021/ja00209a024 · doi:10.1021/ja00209a024
  11. Ojima I., 1989, J. Org. Chem., 54, 4511, 10.1021/jo00280a014 · doi:10.1021/jo00280a014
  12. Soloshonok V. A., 1994, Tetrahedron Lett., 35, 5063, 10.1016/S0040-4039(00)73320-X · doi:10.1016/s0040-4039(00)73320-x
  13. Katagiri T., 2001, Chem. Commun., 2054, 10.1039/b105602f · doi:10.1039/b105602f
  14. Fuchikami T., 1982, J. Am. Chem. Soc., 104, 3527, 10.1021/ja00376a057 · doi:10.1021/ja00376a057
  15. Fuchikami T., 1983, J. Org. Chem., 48, 3803, 10.1021/jo00169a040 · doi:10.1021/jo00169a040
  16. Ojima I., 1988, J. Am. Chem. Soc., 110, 5617, 10.1021/ja00225a004 · doi:10.1021/ja00225a004
  17. Soloshonok V. A., 1994, Tetrahedron Lett., 35, 2713, 10.1016/S0040-4039(00)77013-4 · doi:10.1016/s0040-4039(00)77013-4
  18. Soloshonok V. A., 1994, Tetrahedron: Asymmetry, 5, 1091, 10.1016/0957-4166(94)80059-6 · doi:10.1016/0957-4166(94)80059-6
  19. Kobzev S. V., 1989, Zh. Obshch. Khim., 59, 909
  20. Van Niel M. B., 1999, J. Med. Chem., 42, 2087, 10.1021/jm981133m · doi:10.1021/jm981133m
  21. Sparr C., 2009, Angew. Chem., Int. Ed., 48, 3065, 10.1002/anie.200900405 · doi:10.1002/anie.200900405
  22. Soloshonok V. A., 1996, Tetrahedron: Asymmetry, 7, 1547, 10.1016/0957-4166(96)00177-2 · doi:10.1016/0957-4166(96)00177-2
  23. Wakeling A. E., 1991, Cancer Res., 51, 3867
  24. Brazier E. J., 2010, Org. Process Res. Dev., 14, 544, 10.1021/op900315j · doi:10.1021/op900315j
  25. Ballard P., 2006, Bioorg. Med. Chem. Lett., 16, 4908, 10.1016/j.bmcl.2006.06.054 · doi:10.1016/j.bmcl.2006.06.054
  26. 1996, Chem. Abstr., 126, 47235
  27. 2004, Chem. Abstr., 140, 287403
  28. Chandregowda V., 2007, Org. Process Res. Dev., 11, 813, 10.1021/op700054p · doi:10.1021/op700054p
  29. Breitler S., 2011, Org. Lett., 13, 3262, 10.1021/ol201210t · doi:10.1021/ol201210t
  30. Rawling T., 2012, Tetrahedron, 68, 6065, 10.1016/j.tet.2012.05.002 · doi:10.1016/j.tet.2012.05.002
  31. Wagstaff A. J., 2003, Drugs, 63, 217, 10.2165/00003495-200363020-00009 · doi:10.2165/00003495-200363020-00009
  32. McGavin J. K., 2001, Drugs, 61, 2309, 10.2165/00003495-200161150-00015 · doi:10.2165/00003495-200161150-00015
  33. Koukourakis G. V., 2008, Molecules, 13, 1897, 10.3390/molecules13081897 · DOI
  34. Ishitsuka H., 1999, J. Pharm. Soc. Jpn., 119, 881, 10.1248/yakushi1947.119.12_881 · doi:10.1248/yakushi1947.119.12_881
  35. Shimma N., 2000, Bioorg. Med. Chem., 8, 1697, 10.1016/S0968-0896(00)00087-0 · doi:10.1016/s0968-0896(00)00087-0
  36. 1981, Chem. Abstr., 95, 62602
  37. Niedballa U., 1974, J. Org. Chem., 39, 3654, 10.1021/jo00939a008 · doi:10.1021/jo00939a008
  38. Saneyoshi M., 1978, Chem. Pharm. Bull., 26, 2990, 10.1248/cpb.26.2990 · doi:10.1248/cpb.26.2990
  39. Mendel D. B., 2003, Clin. Cancer Res., 9, 327
  40. Manley J. M., 2003, J. Org. Chem., 68, 6447, 10.1021/jo034304q · doi:10.1021/jo034304q
  41. Wang J.-Q., 2005, Bioorg. Med. Chem. Lett., 15, 4380, 10.1016/j.bmcl.2005.06.038 · doi:10.1016/j.bmcl.2005.06.038
  42. Davies J., 2011, Lancet Oncol., 12, 826, 10.1016/S1470-2045(11)70228-5 · doi:10.1016/s1470-2045(11)70228-5
  43. 2004, Chem. Abstr., 140, 77161
  44. Huang W.-S., 2007, Synthesis, 2121, 10.1055/s-2007-983754 · doi:10.1055/s-2007-983754
  45. Ueda S., 2012, J. Am. Chem. Soc., 134, 700, 10.1021/ja2102373 · doi:10.1021/ja2102373
  46. Basuli F., 2011, J. Labelled Compd. Radiopharm., 54, 633, 10.1002/jlcr.1898 · doi:10.1002/jlcr.1898
  47. Wood E. R., 2004, Cancer Res., 64, 6652, 10.1158/0008-5472.CAN-04-1168 · DOI · Paper page
  48. 2002, Chem. Abstr., 137, 119644
  49. Zhong W. Z., 2010, Curr. Drug Metab., 11, 296, 10.2174/138920010791514207 · doi:10.2174/138920010791514207
  50. Pennell N. A., 2012, Am. J. Manag. Care, 18, SP84
  51. 2006, Chem. Abstr., 144, 274297
  52. Ramachandran P. V., 2004, Tetrahedron Lett., 45, 2603, 10.1016/j.tetlet.2004.01.146 · doi:10.1016/j.tetlet.2004.01.146
  53. Xin B., 2012, Bioorg. Med. Chem. Lett., 22, 4783, 10.1016/j.bmcl.2012.05.053 · doi:10.1016/j.bmcl.2012.05.053
  54. Stellwagen J. C., 2011, Bioorg. Med. Chem. Lett., 21, 4436, 10.1016/j.bmcl.2011.06.021 · doi:10.1016/j.bmcl.2011.06.021
  55. Buck J. R., 2012, Tetrahedron Lett., 53, 4161, 10.1016/j.tetlet.2012.05.137 · doi:10.1016/j.tetlet.2012.05.137
  56. Baumann P., 2002, Eur. Neuropsychopharmacol., 12, 433, 10.1016/S0924-977X(02)00051-2 · DOI
  57. Zhang P., 2010, J. Med. Chem., 53, 6112, 10.1021/jm1005034 · doi:10.1021/jm1005034
  58. 1990, Chem. Abstr., 113, 78150
  59. 2009, Chem. Abstr., 150, 144285
  60. 2005, Chem. Abstr., 143, 26491
  61. 2006, Chem. Abstr., 144, 292567
  62. Elati C. R., 2007, Org. Process Res. Dev., 11, 289, 10.1021/op060175e · doi:10.1021/op060175e
  63. 2003, Chem. Abstr., 139, 73997
  64. Solares L. F., 2004, Tetrahedron: Asymmetry, 15, 341, 10.1016/j.tetasy.2003.10.022 · doi:10.1016/j.tetasy.2003.10.022
  65. 2006, Chem. Abstr., 146, 80528
  66. 2007, Chem. Abstr., 147, 211613
  67. Partridge B. M., 2011, Tetrahedron, 67, 10082, 10.1016/j.tet.2011.09.142 · doi:10.1016/j.tet.2011.09.142
  68. Muñoz M., 2012, Expert Opin. Ther. Pat., 22, 735, 10.1517/13543776.2012.697153 · doi:10.1517/13543776.2012.697153
  69. Lin P., 2007, Bioorg. Med. Chem. Lett., 17, 5191, 10.1016/j.bmcl.2007.06.085 · doi:10.1016/j.bmcl.2007.06.085
  70. Jiang J., 2009, J. Med. Chem., 52, 3039, 10.1021/jm8016514 · doi:10.1021/jm8016514
  71. Kolla N., 2007, Org. Process Res. Dev., 11, 455, 10.1021/op700030d · doi:10.1021/op700030d
  72. Vankawala P. J., 2007, Synth. Commun., 37, 3439, 10.1080/00397910701487473 · doi:10.1080/00397910701487473
  73. Pye P. J., 2002, Chem.—Eur. J., 8, 1372, 10.1002/1521-3765(20020315)8:6<1372::AID-CHEM1372>3.0.CO;2-6 · doi:10.1002/1521-3765(20020315)8:6<1372::aid-chem1372>3.0.co;2-6
  74. Zhao M. M., 2002, J. Org. Chem., 67, 6743, 10.1021/jo0203793 · doi:10.1021/jo0203793
  75. Cowden C. J., 2000, Tetrahedron Lett., 41, 8661, 10.1016/S0040-4039(00)01548-3 · doi:10.1016/s0040-4039(00)01548-3
  76. Payack J. F., 2004, Org. Process Res. Dev., 8, 256, 10.1021/op034180j · doi:10.1021/op034180j
  77. 2012, Chem. Abstr., 157, 663055
  78. 2009, Chem. Abstr., 151, 343563
  79. Elati C. R., 2007, Tetrahedron Lett., 48, 8001, 10.1016/j.tetlet.2007.09.051 · doi:10.1016/j.tetlet.2007.09.051
  80. Gangula S., 2010, Synth. Commun., 40, 2254, 10.1080/00397910903221084 · doi:10.1080/00397910903221084
  81. Brands K. M. J., 2006, Org. Process Res. Dev., 10, 109, 10.1021/op0501895 · doi:10.1021/op0501895
  82. Nelson T. D., 2004, Tetrahedron Lett., 45, 8917, 10.1016/j.tetlet.2004.09.185 · doi:10.1016/j.tetlet.2004.09.185
  83. Strupczewski J. T., 1995, J. Med. Chem., 38, 1119, 10.1021/jm00007a009 · doi:10.1021/jm00007a009
  84. Rado J., 2010, Expert Opin. Pharmacother., 11, 2087, 10.1517/14656566.2010.502889 · doi:10.1517/14656566.2010.502889
  85. 1993, Chem. Abstr., 118, 240939
  86. 2008, Chem. Abstr., 148, 308371
  87. 2011, Chem. Abstr., 155, 123430
  88. 2011, Chem. Abstr., 154, 158482
  89. 2011, Chem. Abstr., 155, 123425
  90. 2012, Chem. Abstr., 157, 548664
  91. Janardhana R. V., 2011, Pharm. Lett., 3, 240
  92. 2010, Chem. Abstr., 152, 144708
  93. Strupczewski J. T., 1985, J. Med. Chem., 28, 761, 10.1021/jm00383a012 · doi:10.1021/jm00383a012
  94. 1991, Chem. Abstr., 114, 185553
  95. 1995, Chem. Abstr., 123, 169657
  96. 1995, Chem. Abstr., 123, 314016
  97. 1998, Chem. Abstr., 129, 122674
  98. 2012, Chem. Abstr., 157, 708577
  99. 2010, Chem. Abstr., 152, 405725
  100. Patel D. S., 2011, Res. J. Pharm. Biol. Chem. Sci, 2, 855
  101. Hegde S., 2008, Annu. Rep. Med. Chem., 43, 455
  102. Wang J., 2006, Prog. Nat. Sci., 16, 925, 10.1080/10020070612330017 · DOI
  103. 1987, Chem. Abstr., 106, 156480
  104. 1999, Chem. Abstr., 130, 57245
  105. 2010, Chem. Abstr., 153, 382966
  106. 1998, Chem. Abstr., 128, 140707
  107. Arava V. R., 2011, Pharm. Chem., 3, 381
  108. 2012, Chem. Abstr., 156, 337316
  109. 2012, Chem. Abstr., 156, 390181
  110. Dorange I., 2011, Annu. Rep. Med. Chem., 46, 53
  111. 1993, Chem. Abstr., 119, 225705
  112. 2003, Chem. Abstr., 138, 137040
  113. 2012, Chem. Abstr., 157, 242074
  114. 1998, Chem. Abstr., 129, 104236
  115. Swahn C.-G., 1996, J. Labelled Compd. Radiopharm., 38, 675, 10.1002/(SICI)1099-1344(199607)38:7<675::AID-JLCR880>3.0.CO;2-L · doi:10.1002/(sici)1099-1344(199607)38:7<675::aid-jlcr880>3.0.co;2-l
  116. 2011, Chem. Abstr., 155, 94042
  117. Wu G., 1999, J. Org. Chem., 64, 3714, 10.1021/jo990428k · doi:10.1021/jo990428k
  118. Fu X., 2003, Tetrahedron Lett., 44, 801, 10.1016/S0040-4039(02)02700-4 · doi:10.1016/s0040-4039(02)02700-4
  119. Bertrand B., 2007, Tetrahedron Lett., 48, 2123, 10.1016/j.tetlet.2007.01.118 · doi:10.1016/j.tetlet.2007.01.118
  120. Kysliková E., 2010, J. Mol. Catal. B: Enzym., 67, 266, 10.1016/j.molcatb.2010.09.006 · doi:10.1016/j.molcatb.2010.09.006
  121. Sova M., 2010, Synthesis, 3433
  122. Michalak M., 2011, J. Org. Chem., 76, 6931, 10.1021/jo2010846 · doi:10.1021/jo2010846
  123. Wang X., 2012, Angew. Chem., Int. Ed., 51, 9276, 10.1002/anie.201204925 · doi:10.1002/anie.201204925
  124. aPfefferkorn, J. A.InThe art of drug synthesis;Johnson, D. S.; Li, J. J., Eds.John Wiley & Sons:Hoboken, NJ, 2007; pp169–182.
  125. Quirk J., 2003, Nat. Rev. Drug. Discovery, 2, 769, 10.1038/nrd1205 · doi:10.1038/nrd1205
  126. Konoike T., 1994, J. Org. Chem., 59, 7849, 10.1021/jo00104a049 · doi:10.1021/jo00104a049
  127. Korostylev A., 2008, Eur. J. Org. Chem., 840, 10.1002/ejoc.200701059 · doi:10.1002/ejoc.200701059
  128. Andrushko N., 2008, Eur. J. Org. Chem., 847, 10.1002/ejoc.200700813 · doi:10.1002/ejoc.200700813
  129. Časar Z., 2008, Synlett, 2036, 10.1055/s-2008-1077957 · doi:10.1055/s-2008-1077957
  130. Časar Z., 2009, Synlett, 1144, 10.1055/s-0028-1088152 · doi:10.1055/s-0028-1088152
  131. Hilas O., 2009, Pharm. Ther., 34, 188
  132. Siebert C. D., 2008, Chirality, 20, 103, 10.1002/chir.20509 · doi:10.1002/chir.20509
  133. Bai Y., 2006, J. Chem. Res., 807, 10.3184/030823406780199802 · doi:10.3184/030823406780199802
  134. Johannes C. W., 1998, J. Am. Chem. Soc., 120, 8340, 10.1021/ja981378o · doi:10.1021/ja981378o
  135. Visser M. S., 1996, J. Am. Chem. Soc., 118, 3779, 10.1021/ja960263m · doi:10.1021/ja960263m
  136. Harrity J. P. A., 1997, J. Am. Chem. Soc., 119, 1488, 10.1021/ja9636597 · doi:10.1021/ja9636597
  137. Encinas M. V., 1980, J. Am. Chem. Soc., 102, 1357, 10.1021/ja00524a021 · doi:10.1021/ja00524a021
  138. Trost B. M., 1988, Tetrahedron Lett., 29, 2931, 10.1016/0040-4039(88)85050-0 · doi:10.1016/0040-4039(88)85050-0
  139. Hoveyda A. H., 1993, Chem. Rev., 93, 1307, 10.1021/cr00020a002 · doi:10.1021/cr00020a002
  140. Chandrasekhar S., 2000, Tetrahedron, 56, 6339, 10.1016/S0040-4020(00)00572-X · doi:10.1016/s0040-4020(00)00572-x
  141. Wang N.-X., 2007, Synthesis, 1154, 10.1055/s-2007-965993 · doi:10.1055/s-2007-965993
  142. Carreño M. C., 2008, Eur. J. Org. Chem., 2035, 10.1002/ejoc.200800201 · doi:10.1002/ejoc.200800201
  143. Nakagawa S., 1995, Jpn. J. Pharm., 67, 1, 10.1254/jjp.67.1 · doi:10.1254/jjp.67.1
  144. Müller M., 2005, Angew. Chem., Int. Ed., 44, 362, 10.1002/anie.200460852 · doi:10.1002/anie.200460852
  145. Karanewsky D. S., 1991, J. Org. Chem., 56, 3744, 10.1021/jo00011a064 · doi:10.1021/jo00011a064
  146. Theisen P. D., 1988, J. Org. Chem., 53, 2374, 10.1021/jo00245a051 · doi:10.1021/jo00245a051
  147. Heathcock C. H., 1987, J. Med. Chem., 30, 1858, 10.1021/jm00393a030 · doi:10.1021/jm00393a030
  148. Rosen T., 1985, J. Am. Chem. Soc., 107, 3731, 10.1021/ja00298a062 · doi:10.1021/ja00298a062
  149. Rosen T., 1984, J. Org. Chem., 49, 3657, 10.1021/jo00193a044 · doi:10.1021/jo00193a044
  150. Fernandes R. A., 2002, Eur. J. Org. Chem., 2921, 10.1002/1099-0690(200209)2002:17<2921::AID-EJOC2921>3.0.CO;2-N · doi:10.1002/1099-0690(200209)2002:17<2921::aid-ejoc2921>3.0.co;2-n
  151. Ghosh A. K., 2002, J. Org. Chem., 67, 8783, 10.1021/jo020402k · doi:10.1021/jo020402k
  152. Rosen T., 1984, J. Org. Chem., 49, 3994, 10.1021/jo00195a023 · doi:10.1021/jo00195a023
  153. Kumar P., 2010, Tetrahedron Lett., 51, 5838, 10.1016/j.tetlet.2010.08.093 · doi:10.1016/j.tetlet.2010.08.093
  154. Reddy M. V. R., 2001, J. Organomet. Chem., 624, 239, 10.1016/S0022-328X(01)00665-9 · doi:10.1016/s0022-328x(01)00665-9
  155. Takahashi K., 1993, Tetrahedron Lett., 34, 8263, 10.1016/S0040-4039(00)61406-5 · doi:10.1016/s0040-4039(00)61406-5
  156. Lopp M., 1991, Tetrahedron: Asymmetry, 2, 943, 10.1016/S0957-4166(00)86131-5 · doi:10.1016/s0957-4166(00)86131-5
  157. Minami T., 1992, Tetrahedron Lett., 33, 7525, 10.1016/S0040-4039(00)60814-6 · doi:10.1016/s0040-4039(00)60814-6
  158. Reddy B., 1991, J. Org. Chem., 56, 5752, 10.1021/jo00020a008 · doi:10.1021/jo00020a008
  159. Takano S., 1993, Tetrahedron: Asymmetry, 4, 201, 10.1016/S0957-4166(00)82337-X · doi:10.1016/s0957-4166(00)82337-x
  160. Miyachi N., 1993, Tetrahedron Lett., 34, 8267, 10.1016/S0040-4039(00)61407-7 · doi:10.1016/s0040-4039(00)61407-7
  161. Suzuki M., 2001, Bioorg. Med. Chem., 9, 2727, 10.1016/S0968-0896(01)00198-5 · DOI
  162. Acemoglu M., 2007, Helv. Chim. Acta, 90, 1069, 10.1002/hlca.200790106 · doi:10.1002/hlca.200790106
  163. Fabris J., 2012, Synthesis, 1700
  164. Serebruany V., 2009, Thromb. Haemostasis, 101, 14, 10.1160/TH08-07-0452 · doi:10.1160/th08-07-0452
  165. Huber K., 2009, Nat. Rev. Drug Discovery, 8, 449, 10.1038/nrd2899 · doi:10.1038/nrd2899
  166. Hasegawa M., 2005, Thromb. Haemostasis, 94, 593, 10.1160/TH05-03-0208 · doi:10.1160/th05-03-0208
  167. Dobesh P. P., 2009, Pharmacotherapy, 29, 1393, 10.1592/phco.29.12.1393 · doi:10.1592/phco.29.12.1393
  168. 2009, Chem. Abstr., 151, 266755
  169. Aalla S., 2012, Org. Process Res. Dev., 16, 240, 10.1021/op200325u · doi:10.1021/op200325u
  170. Pan X., 2012, Tetrahedron Lett., 53, 5364, 10.1016/j.tetlet.2012.07.071 · doi:10.1016/j.tetlet.2012.07.071
  171. Zhang H., 2012, Bioorg. Med. Chem. Lett., 22, 3598, 10.1016/j.bmcl.2012.04.050 · doi:10.1016/j.bmcl.2012.04.050
  172. Groll A. H., 1998, Adv. Pharmacol. (San Diego, CA, U.S.), 44, 343
  173. Tasaka A., 1993, Chem. Pharm. Bull., 41, 1035, 10.1248/cpb.41.1035 · doi:10.1248/cpb.41.1035
  174. Richardson K., 1988, Ann. N.Y. Acad. Sci., 544, 6
  175. Tasaka A., 1995, Chem. Pharm. Bull., 43, 441, 10.1248/cpb.43.441 · doi:10.1248/cpb.43.441
  176. Butters M., 2001, Org. Process Res. Dev., 5, 28, 10.1021/op0000879 · doi:10.1021/op0000879
  177. 1997, Chem. Abstr., 127, 262316
  178. 1995, Chem. Abstr., 123, 339705
  179. Butters M., 1992, J. Heterocycl. Chem., 1369, 10.1002/jhet.5570290554 · doi:10.1002/jhet.5570290554
  180. Frampton J. E., 2005, Drugs, 65, 1427, 10.2165/00003495-200565100-00008 · doi:10.2165/00003495-200565100-00008
  181. Molina J. M., 2005, Drugs Today, 41, 241, 10.1358/dot.2005.41.4.900219 · doi:10.1358/dot.2005.41.4.900219
  182. Cahn P., 2004, Expert Opin. Invest. Drugs, 13, 55, 10.1517/13543784.13.1.55 · doi:10.1517/13543784.13.1.55
  183. Bang L. M., 2003, Drugs, 63, 2413, 10.2165/00003495-200363220-00003 · doi:10.2165/00003495-200363220-00003
  184. Gentile I., 2006, Curr. Med. Chem., 13, 2839, 10.2174/092986706778521995 · doi:10.2174/092986706778521995
  185. Nelson M., 2004, Int. J. Clin. Pract., 58, 504, 10.1111/j.1368-5031.2004.00100.x · doi:10.1111/j.1368-5031.2004.00100.x
  186. 1992, Chem. Abstr., 118, 22551
  187. 2000, Chem. Abstr., 132, 166456
  188. Hoong L. K., 1992, J. Org. Chem., 57, 5563, 10.1021/jo00047a004 · doi:10.1021/jo00047a004
  189. Osborne A. P., 2006, Org. Process Res. Dev., 10, 670, 10.1021/op050258f · doi:10.1021/op050258f
  190. Gaede B. J., 2005, Org. Process Res. Dev., 9, 23, 10.1021/op040210m · doi:10.1021/op040210m
  191. Agarwal H. K., 2012, J. Med. Chem., 55, 2672, 10.1021/jm201551m · doi:10.1021/jm201551m
  192. Agarwal H. K., 2013, Mol. Pharmaceutics, 10, 467, 10.1021/mp300361a · doi:10.1021/mp300361a
  193. Rusconi S., 2009, Expert Rev. Clin. Pharmacol., 2, 147, 10.1586/17512433.2.2.147 · doi:10.1586/17512433.2.2.147
  194. Orman J. S., 2008, Drugs, 68, 1435, 10.2165/00003495-200868100-00006 · doi:10.2165/00003495-200868100-00006
  195. Temesgen Z., 2005, Drugs Today, 41, 71, 10.1358/dot.2005.41.11.937960 · doi:10.1358/dot.2005.41.11.937960
  196. Wroblewski A., 1998, Drugs Future, 23, 146, 10.1358/dof.1998.023.02.445832 · doi:10.1358/dof.1998.023.02.445832
  197. Thaisrivongs S., 1996, J. Med. Chem., 39, 4349, 10.1021/jm960541s · doi:10.1021/jm960541s
  198. Turner S. R., 1998, J. Med. Chem., 41, 3467, 10.1021/jm9802158 · doi:10.1021/jm9802158
  199. Judge T. M., 1997, J. Am. Chem. Soc., 119, 3627, 10.1021/ja963434w · doi:10.1021/ja963434w
  200. Soloshonok V. A., 2002, Helv. Chim. Acta, 85, 3616, 10.1002/1522-2675(200211)85:11<3616::AID-HLCA3616>3.0.CO;2-O · doi:10.1002/1522-2675(200211)85:11<3616::aid-hlca3616>3.0.co;2-o

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Metadata

Authors
Wang, J., Sánchez-Roselló, M., Aceña, J. L., del Pozo, C., Sorochinsky, A. E., Fustero, S., Soloshonok, V. A., & Liu, H.
Venue
Chemical Reviews
Publisher
American Chemical Society (ACS)
Published
2013-12-03
Volume
114
Issue
4
Pages
2432-2506
ISSN
  • 0009-2665 (ISSN-L)
  • 1520-6890
DOI
10.1021/cr4002879
OpenAlex
W2333129245
Cited by
4,847
References
254
FWCI
75.99
Type
journal article
Language
en
Open access
closed

About these checks

Registry, retraction, Cites and statistics results are computed, not judged, with one exception: a printed reference that no index lists is read once by a model before it counts as a citation error. Claims are extracted by a model and kept only when their quote appears verbatim in the text; each cited source is then checked, with a model’s help, for whether it says what the claim relies on. Those verdicts can be wrong — read the claim’s quote and the cited source before relying on one.

Statistics and arithmetic are recomputed, not judged.

Confidence bands are shown only for fields calibrated on our annotated test set. None is calibrated yet, so no band is shown.

What counts as a claim ›How we measure confidence ›How we check this ›

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Data sources

Bibliographic data: Semantic Scholar, OpenAlex, Crossref.

Contains information from the Semantic Scholar Academic Graph Datasets, made available under the ODC Attribution License (ODC-BY 1.0).

Semantic Scholar’s data is described in: Kinney, R., et al. (2023). The Semantic Scholar Open Data Platform. arXiv:2301.10140.