TF-PROTACs Enable Targeted Degradation of Transcription Factors

Liu, Jing, Chen, He, Kaniskan, H. Ümit, Xie, Ling, Chen, Xian, Jin, Jian, Wei, Wenyi·2021·Journal of the American Chemical Society

Cited by (251)

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  20. O bi namo ma ronga isi go Galelaka / ditulis Etha Yosafat ; diindonesiakan Robinon Ipol
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  43. BindingDB Entry 50020161: Advances of bioorthogonal coupling reactions in drug development.
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  44. BindingDB Entry 50016839: VHL-based PROTACs as potential therapeutic agents: Recent progress and perspectives.
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  45. BindingDB Entry 50017503: Solid-Phase Synthesis of Cereblon-Recruiting Selective Histone Deacetylase 6 Degraders (HDAC6 PROTACs) with Antileukemic Activity.
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  46. BindingDB Entry 50016515: Nucleic-Acid-Based Targeted Degradation in Drug Discovery.
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  47. BindingDB Entry 50016429: Emerging targeted protein degradation tools for innovative drug discovery: From classical PROTACs to the novel and beyond.
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  48. BindingDB Entry 50021731: Discovery and Characterization of a Novel Cereblon-Recruiting PRC1 Bridged PROTAC Degrader.
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  49. BindingDB Entry 50023360: PROTAC technology: From drug development to probe technology for target deconvolution.
    BindingDB · 2026 · UC San Diego
  50. BindingDB Entry 50020717: A beginner's guide to current synthetic linker strategies towards VHL-recruiting PROTACs.
    BindingDB · 2024 · UC San Diego
  51. BindingDB Entry 50021132: Journey of Von Hippel-Lindau (VHL) E3 ligase in PROTACs design: From VHL ligands to VHL-based degraders.
    BindingDB · 2025 · UC San Diego