Discovery of Novel Antitumor Sulfonamides Targeting G1 Phase of the Cell Cycle

Owa, Takashi, Yoshino, Hiroshi, Okauchi, Tatsuo, Yoshimatsu, Kentaro, Ozawa, Yoichi, Sugi, Naoko Hata, Nagasu, Takeshi, Koyanagi, Nozomu +1 more·1999·Journal of Medicinal Chemistry

Cited by (342)

Items 201–300 of 342

  1. DNA/bovine serum albumin binding and cytotoxicity of transition metal ternary complexes based on sulfamethazine and bromazepam drugs
    Ahmed M. Mansour, Nour Tawfik Abdel-Ghani, Mona S. Ragab · 2020 · Applied Organometallic Chemistry
  2. Role of secondary ligand on Cd complex of sulfamethizole: synthesis, spectroscopic characterization, Hirshfeld surface analysis and DNA interaction
    Mohammed Dawood Alalawy, Bhavesh N. Socha, Bhavin R. Chavda, Taruna J. Padariya, Bharatkumar D. Patel, Urmila H. Patel, Urmila H. Patel, Bhupesh S. Bhatt · 2021 · Journal of Molecular Structure
  3. Benzopyridooxathiazepine derivatives as novel potent antimitotic agents
    Sebastien Gallet, Nathalie Flouquet, Pascal Carato, Bruno Pfeiffer, Pierre Renard, Stéphane Léonce, Alain Pierré, Pascal Berthelot, Nicolas Lebègue · 2008 · Bioorganic & Medicinal Chemistry
  4. Synthesis, crystal structures, characterization and antitumor activities of two copper(II) complexes of a sulfonamide ligand
    Adriana Corina Hangan, Roxana Liana Lucaciu, Alexandru Turza, Luminita Simona Oprean, Emőke Páll, Sînziana Cetean, Bogdan Sevastre · 2017 · Transition Metal Chemistry
  5. 2-[N1-2-Pyrimidyl-aminobenzenesulfonamido] ethyl 4-bis(2-chloroethyl) aminophenyl butyrate
    Zhaohua Richard Huang, Genjin Yang, Zhaoliang Lin, Junlian Huang · 2001 · Bioorganic & Medicinal Chemistry Letters
  6. In vitro pharmacokinetic study of the novel anticancer agent E7070: red blood cell and plasma protein binding in human blood
    H.J.G.D. van den Bongard, Dick Pluim, Robert C.A.M. van Waardenburg, Miroslav Ravic, Jos H. Beijnen, Jan H.M. Schellens · 2003 · Anti-Cancer Drugs
  7. Targeting RNA-binding proteins with small molecules: perspectives and challenges
    Olivier Mpungi Konde, W. B. Balela, T. B. Tshitenge · 2025 · Frontiers in Chemistry
  8. Discovery of novel sulphonamide hybrids that inhibit LSD1 against bladder cancer cells
    Jia Liu, Xingwang Zhu, Yu Liu, Minghuan Mao · 2022 · Journal of Enzyme Inhibition and Medicinal Chemistry
  9. Death inducing and cytoprotective autophagy in T‐47D cells by two common antibacterial drugs: sulphathiazole and sulphacetamide
    Raziye Mohammadpour, Shahrokh Safarian, Nader Sheibani, Saeed Norouzi, Atefeh P. Razazan · 2013 · Cell Biology International
  10. Synthesis and antibacterial activity of new chiral N-sulfamoyloxazolidin-2-ones
    Fouzia Bouchareb, Malika Berredjem, Samira Ait Kaki, AMEL BOUARICHA, Abdeslem Bouzina, Billel Belhani, Nour‐Eddine Aouf · 2015 · Journal of Chemical Sciences
  11. Synthesis, crystal structure and characterization of new biologically active Cu(II) complexes with ligand derived from N-substituted sulfonamide
    Adriana Corina Hangan, Alexandru Turza, Roxana Liana Lucaciu, Bogdan Sevastre, Emőke Páll, Sînziana Cetean, Luminita Simona Oprean · 2016 · Journal of Chemical Sciences
  12. Synthesis, crystal structure, properties, and nuclease activity of a new Cu(II) complex [Cu(L)2(Py)2(H2O)] (HL = N-(5-(4-methylphenyl)-[1,3,4]-thiadiazole-2-yl)toluenesulfonamide)
    Adriana Corina Hangan, Alexandru Turza, R. L. Stan, Răzvan Ștefan, Luminita Simona Oprean · 2015 · Russian Journal of Coordination Chemistry
  13. From serendipity to strategy: molecular glue degraders in cancer therapeutics
    Darling, Sarah, Bajrami, Ilirjana, West, Stephen C. · 2025 · Critical Reviews in Biochemistry and Molecular Biology
  14. Recent advances in anticancer mechanisms of molecular glue degraders: focus on RBM39-dgrading synthetic sulfonamide such as indisulam, E7820, tasisulam, and chloroquinoxaline sulfonamide
    Ji‐Hoon Jang, Joo-Young Kim, Tae Jin Lee · 2024 · Genes & Genomics
  15. Aberrant pre-mRNA processing in cancer
    Jeetayu Biswas, Leora S. Boussi, Eytan M. Stein, Omar Ibrahim Abdel-Wahab · 2024 · The Journal of Experimental Medicine
  16. Indisulam Reduces Viability and Regulates Apoptotic Gene Expression in Pediatric High-Grade Glioma Cells
    Caio César Damasceno Monção, Carlos Alberto Scrideli, Augusto Faria Andrade, Mariano Sebastian Viapiano, Carlos Gilberto Carlotti, Daniel Antunes Moreno, Mirella Baroni, Luíz Gonzaga Tone, Silvia Aparecida Teixeira · 2022 · Biomedicines
  17. Spectroscopic, structural, electrochemical and antimicrobiological studies of Cu(II)-sulfathiazole complex with diethylenetriamine ligand
    Filiz Öztürk, İclal Bulut, Yeliz Genç Bekiroğlu, Ahmet Bulut · 2016 · Polyhedron
  18. The effect of Euphorbia szovitsii Fisch. & C.A.Mey extract on the viability and the proliferation of MDA-MB-231 cell line
    Majid Asadi-Samani, Mahmoud Rafieian‐Kopaei, Zahra Lorigooini, Hedayatollah Shirzad · 2018 · Bioscience Reports
  19. Aryl Sulfonamides Induce Degradation of Aryl Hydrocarbon Receptor Nuclear Translocator through CRL4DCAF15 E3 Ligase
    Sung Ah Kim, Seung-Hyun Jo, Jin Hwa Cho, Min Yeong Yu, Ho‐Chul Shin, Jung‐Ae Kim, Byoung Chul Park, Byoung Chul Park, Jeong‐Hoon Kim, Jeong‐Hoon Kim · 2020 · Molecules and Cells
  20. Development and validation of limited sampling strategies for prediction of the systemic exposure to the novel anticancer agent E7070 (N‐(3‐chloro‐7‐indolyl)‐1,4‐benzenedisulphonamide)
    Charlotte van Kesteren, Ron A. A. Mathôt, Éric Raymond, Jean‐Pierre Armand, P. Fumoleau, Cornelis J.A. Punt, Miroslav Ravic, Jantien Wanders, Jos H. Beijnen, Jan H.M. Schellens · 2002 · British Journal of Clinical Pharmacology
  21. Synthesis and biological evaluation of N-(7-indolyl)-3-pyridinesulfonamide derivatives as potent antitumor agents
    Takashi Owa, Hiroshi Yoshino, Tatsuo Okauchi, Tadashi Okabe, Yoichi Ozawa, Naoko Hata Sugi, Kentaro Yoshimatsu, Takeshi Nagasu, Nozomu Koyanagi, Kyosuke Kitoh · 2002 · Bioorganic & Medicinal Chemistry Letters
  22. A Facile and Efficient Synthesis of Arylsulfonamido‐Substituted 1,5‐Benzodiazepines and N‐[2‐(3‐Benzoylthioureido)aryl]‐3‐oxobutanamide Derivatives
    Abdolali Alizadeh, Nasrin Zohreh · 2010 · Helvetica Chimica Acta
  23. Inhibition of lactate dehydrogenase A by diclofenac sodium induces apoptosis in H e L a cells through activation of AMPK
    Avirup Malla, Suvroma Gupta, Runa Sur · 2024 · FEBS Journal
  24. Targeting strategies for modulating pre-mRNA splicing with small molecules: Recent advances
    Scott J. Barraza, Anuradha Bhattacharyya, Christopher R. Trotta, Matthew G. Woll · 2022 · Drug Discovery Today
  25. Synthesis, Structure, Hirshfeld Surface Analysis, Non-Covalent Interaction, and In Silico Studies of 4-Hydroxy-1-[(4-Nitrophenyl)Sulfonyl]Pyrrolidine-2-Carboxyllic Acid
    David Izuchukwu Ugwu, Florence Uchenna Eze, Chigozie Julius Ezeorah, Lydia Rhyman, Ponnadurai Ramasami, Tania Groutso, Cosmas Chinweike Eze, Chiamaka Peace Uzoewulu, Blessing Chinweotito Ogboo, Obinna C. Okpareke · 2023 · Journal of Chemical Crystallography
  26. Anticancer Agent E7070 Inhibits Amino Acid and Uracil Transport in Fission Yeast
    Kappei Tsukahara, Tatsuo Watanabe, Naoko Hata-Sugi, Kentaro Yoshimatsu, Hiroto Okayama, Takeshi Nagasu · 2001 · Molecular Pharmacology
  27. Substituent Groups
    Patrick Bazzini, Camille Georges Wermuth · 2008 · Elsevier eBooks
  28. Methylation of RBM39 by PRMT6 enhances resistance to Indisulam in non-small cell lung cancer by promoting alternative splicing of proto-oncogenes
    Tongjia Zhang, Shujie Wang, Yue Zhou, Zitao Jiao, Kejia Lu, Xinyi Liu, Hui Li, Wei Jiang, Xiaowei Zhang · 2025 · PLoS Biology
  29. Lead discovery and chemical biology approaches targeting the ubiquitin proteasome system
    Favour A. Akinjiyan, Seth Carbonneau, Nathan T. Ross · 2017 · Bioorganic & Medicinal Chemistry Letters
  30. Indisulam exerts anticancer effects via modulation of transcription, translation and alternative splicing on human cervical cancer cells.
    Zhihui Dou, Xuetian Zhang, Wei Su, Taotao Zhang, Fei Ye, Dapeng Zhao, Xiaohua Chen, Qiang Li, Hong Zhang, Cuixia Di · 2023 · PubMed Central
  31. Synthesis and bioactivity evaluation of some novel sulfonamide derivatives
    Ch. Subramanyam, Sk. Nayab Rasool, D. B. Janakiramudu, S. Rasheed, A. Uday Sankar, Chamarthi Naga Raju · 2017 · Phosphorus, sulfur, and silicon and the related elements
  32. Cytotoxicity of multicellular cancer spheroids, antibacterial, and antifungal of selected sulfonamide derivatives coupled with a salicylamide and/or anisamide scaffold
    Alaaeldin M F Galal, Walid Fayad, Walaa S.A. Mettwally, Sanaa K. Gomaa, Esam R. Ahmed, Heba A. El-Refai, Atef G. Hanna · 2019 · Medicinal Chemistry Research
  33. Uncommon crystallization pattern of a ZnII–sulfathiazole complex: Synthesis, X-ray structural features and TGA calculations of [{Zn(STZ)2(HSTZ)(H2O)}{Zn(STZ)2(H2O)2}3] · 12H2O (STZ = sulfathiazolato anion; sulfathiazole = N1-2-thiazolyl-sulfanilamide)
    Gelson Manzoni de Oliveira, Aline Baraldi, Lenice de Lourenço Marques, Ernesto Schulz Lang, Marcos A. Villetti · 2007 · Inorganica Chimica Acta
  34. Novel N-(aryl/heteroaryl)-2-chlorobenzenesulfonamide derivatives: Synthesis and anticancer activity evaluation
    Anita Bułakowska, Jaroslaw J. Slawinski, Kamila Siedlecka-Kroplewska, Grzegorz Stasiłojć, Marcin Serocki, Mateusz Heldt · 2020 · Bioorganic Chemistry
  35. Human metabolism of [14C]indisulam following i.v. infusion in cancer patients
    Jan Hendrik Beumer, Michel J. X. Hillebrand, Dick Pluim, Hilde Rosing, Karen Foley, S. Murray Yule, Jan H.M. Schellens, Jos H. Beijnen · 2005 · Investigational New Drugs
  36. Design, synthesis, chemical and biological evaluation of 2,5,5-trisubstituted-1,2-thiazepan-6-one 1,1-dioxides
    Demyd S. Milokhov, Mykhailo S. Pomalin, Mykola O. Balabushko, Vladyslav R. Holubnychyi, Vasyl Yu. Hys, Pavlo Virych, Petro Virych, N Yu Lukianova, Vasyl A. Chumachenko, Svitlana Shishkina et al. · 2023 · Results in Chemistry
  37. Synthesis of an RBM39 Degrader That Downregulates CEP192 and Induces Disorganized Spindle Structures
    Xilin Lyu, Xiancheng Wang, Dongze Lin, Yuhan Lu, Chenxu Wang, Ziqin Yan, Zhiyi Wang, Ying Cheng, Jing Cheng, Xuelian Ren et al. · 2025 · Journal of Medicinal Chemistry
  38. Synthesis and Evaluation of N-(3-Trifluoroacetyl-indol-7-yl) Acetamides for Potential In Vitro Antiplasmodial Properties
    Malose J. Mphahlele, Mmakwena Modlicious Mmonwa, Yee Siew Choong · 2017 · Molecules
  39. Design, Synthesis, and in vitro and in vivo Evaluations of (Z)‐3,4,5‐Trimethoxystyrylbenzenesulfonamides/sulfonates as Highly Potent Tubulin Polymerization Inhibitors
    Rasala Mahesh, Vadithe Lakshma Nayak, Korrapati Suresh Babu, Syed Riyaz, Thokhir Basha Shaik, Gajjela Bharath Kumar, Prema Latha Mallipeddi, Challa Ratna Reddy, Kunta Chandra Shekar, Jedy Jose et al. · 2017 · ChemMedChem
  40. Natural stilbenes and analogues as antineoplastic agents
    Fulvia Orsini, Guido Sello · 2008 · Studies in natural products chemistry
  41. Exploring DCAF15 for reprogrammable targeted protein degradation
    Seemon Coomar, Dennis G. Gillingham · 2019 · bioRxiv (Cold Spring Harbor Laboratory)
  42. Molecular Glue Degraders: From Serendipity to Hunting and Design
    Luis Nieto‐Barrado, Ana Domostegui, Cristina Mayor‐Ruiz · 2022 · Wiley eBooks
  43. Solid‐Phase Parallel Synthesis of Photocleavable Bifunctional Molecules Enables Efficient Phenotypic Protein Degrader Discovery
    Baoli Ding, Jiawen Hu, Rongtian Zhang, Binyan Shou, Mengdie Chen, Jiang Li, Meng Yuan, Bo Yang, Qiaojun He, Ji Cao et al. · 2025 · Angewandte Chemie International Edition
  44. Synthesis of 3‐Chloroindoles via Palladium‐Catalyzed Chlorocyclization of Unmasked 2‐Alkynylanilines
    Yongpeng Zheng, Jianxiao Li, Wanqing Wu, Chaorong Qi, Huanfeng Jiang · 2024 · Advanced Synthesis & Catalysis
  45. Methods to characterize and discover molecular degraders in cells
    Zhi Lin, Christina M. Woo · 2022 · Chemical Society Reviews
  46. Chemometric QSAR modeling and in silico design of carbonic anhydrase inhibition of a coral secretory isoform by sulfonamide
    Shalini Thakur Singh, Claudiu Trandafir Supuran · 2012 · Bioorganic & Medicinal Chemistry
  47. New Analogues of the Anticancer E7070: Synthesis and Pharmacology
    Guillaume Laconde, Nicole Pommery, Patrick Depreux, Pascal Berthelot, Jean‐Pierre Hénichart · 2003 · Journal of Enzyme Inhibition and Medicinal Chemistry
  48. SPECIFIC SUBSTITUENT GROUPS
    Camille Georges Wermuth · 2003 · Elsevier eBooks
  49. Spectroscopic, structural characterization and magnetic studies of Cu(II)-sulfathiazole complex with 1,10-Phenanthroline and N-(2-hydroxyethyl)-Ethylenediamine ligands
    Filiz Öztürk, Tuğba Aycan, Ahmet Hilmi Çon · 2019 · Journal of Molecular Structure
  50. Fantastic Molecular Glues and Where to Find them
    Dennis G. Gillingham · 2021 · CHIMIA International Journal for Chemistry
  51. Inducible Protein Degradation to Understand Genome Architecture
    Alexi M Tallan, Benjamin Z. Stanton · 2021 · Biochemistry
  52. Quinazoline-sulfonamides as potential antitumor agents: synthesis and biological testing
    Ahmed Mahmoud Alafeefy, Saleh Ibrahim Alqasoumi, Abdelkader Elbadawy Ashour, Mashael Marzouq AlShebly · 2012 · Journal of Enzyme Inhibition and Medicinal Chemistry
  53. Pharmacokinetic Drug–Drug Interaction of the Novel Anticancer Agent E7070 and Acenocoumarol
    H.J.G.D. van den Bongard, Rolf W. Sparidans, David J.P. Critchley, Jos H. Beijnen, Jan H.M. Schellens · 2004 · Investigational New Drugs
  54. Anti-tumor Activity and Cell Cycle Arrest of a New Diterpene Ester from Daphne mucronata Using K562 Cells
    Heibatollah Sadeghi, Razieh Yazdanparast · 2003
  55. The RBM39 degrader indisulam inhibits acute megakaryoblastic leukemia by altering the alternative splicing of ZMYND8
    Ying Hua Yang, Zhiheng Li, Yang Yang, Peifang Xiao, Zhixu He, Zimu Zhang, Yizhen Li, Lei Shi, Xiaodong Wang, Yanfang Tao et al. · 2025 · Cell & Bioscience
  56. Unlocking DCAFs To Catalyze Degrader Development: An Arena for Innovative Approaches
    Qi Miao, Vilas D. Kadam, Ayan Mukherjee, Zhi Tan, Mingxing Teng · 2023 · Journal of Medicinal Chemistry
  57. Designing symmetrically folded scaffolds of pyridazinone and triazinone derivatives linked via N , N -diethyl-4-nitro-benzenesulfonamide to explore luminescent materials
    Vipin B. Kumar, Krishanu Bandyopadhyay, Manisha Nidhar, Vishal Prasad Sharma, Priyanka Yadav, Suman Gill, Priyanka Sonker, Abhineet Verma, Satyen Saha, Ashish Kumar Tewari · 2025 · Journal of Materials Chemistry C
  58. Synthesis, antibacterial and anticancer activity of azo-based and aminomethylene derivatives of cyclic β-keto sulfones
    Demyd S. Milokhov, Mykola O. Balabushko, Anna Y. Kolomiets, Sofiia D. Rabotnikova, Pavlo Virych, Anton O. Poliudov, Svitlana Valentinovna Shishkina, Yulian M. Volovenko, Alexey V. Dobrydnev · 2025 · Bioorganic & Medicinal Chemistry Letters
  59. Synthesis and biological evaluation of N -alkyl sulfonamides derived from polycyclic hydrocarbon scaffolds using a nitrogen-centered radical approach
    Megan D. Hopkins, Ryan C. Witt, Ann Marie Flusche, John E. Philo, Garett L. Ozmer, Gordon H. Purser, Robert J. Sheaff, Angus A. Lamar · 2022 · Organic & Biomolecular Chemistry
  60. Synthesis and Characterization of Some Metal Complexes with their Sulfamethoxazoleand 4,4'-dimethyl-2,2'-bipyridyl and study Cytotoxic Effect on Hep-2 Cell Line
    Baghdad Science Journal · 2015 · Baghdad Science Journal
  61. A Biomimetic Drug Delivery System Targeting Tumor Hypoxia in Triple-Negative Breast Cancers
    Katyayani Tatiparti, Mohd Ahmar Rauf, Samaresh Sau, Arun K. Iyer · 2020 · Applied Sciences
  62. Overlaid Transcriptional and Proteome Analyses Identify Mitotic Kinesins as Important Targets of Arylsulfonamide-Mediated RBM39 Degradation
    Seemon Coomar, Pedro Mota, Alexander V. Penson, Juerg Schwaller, Omar Ibrahim Abdel-Wahab, Dennis G. Gillingham · 2023 · Molecular Cancer Research
  63. Anticancer Potential of N ‐Sulfonyl Noscapinoids: Synthesis and Evaluation
    Praveen Kumar Reddy Nagireddy, Vamsi Krishna Kommalapati, Vagolu Siva Krishna, Dharmarajan Sriram, Anjana Devi Tangutur, Srinivas Kantevari · 2020 · ChemistrySelect
  64. Structure activity investigation, CT complex analysis and spectroscopic investigation on antibiotic drug; Sulfamethoxazole using quantum chemical calculations
    A. Sathya, S. Ramalingam, P.B. Nagabalasubramanian, J. Karpagam · 2021 · Chemical Physics Impact
  65. The role of machine learning method in the synthesis and biological ınvestigation of heterocyclic compounds
    Arif Mermer · 2021 · Molecular Diversity
  66. Importance of Imidazolidinone Motif in 4-Phenyl-N-arylsulfonylimidazolidinone for their Anticancer Activity
    Vinay Kumar Sharma, K.‐H. LEE, Cheonik Joo, Niti Sharma, Sang‐Hun Jung · 2011 · Bulletin of the Korean Chemical Society
  67. Effect of the isosteric replacement of the phenyl motif with furyl (or thienyl) of 4-phenyl-N-arylsulfonylimidazolones as broad and potent anticancer agents
    Vinay Kumar Sharma, Dang The Hung, K.‐H. LEE, Thanigaimalai Pillaiyar, Jong Seong Kang, Hwan‐Mook Kim, Sang‐Hun Jung · 2011 · MedChemComm
  68. ANTINEOPLASTIC EFFECTS OF DAPHNE MUCRONATA: INHIBITION OF DNA AND RNA SYNTHESIS
    Razieh Yazdanparast, H. Sadeghi · 2003
  69. Solid‐Phase Parallel Synthesis of Photocleavable Bifunctional Molecules Enables Efficient Phenotypic Protein Degrader Discovery
    Baoli Ding, Jiawen Hu, Rongtian Zhang, Binyan Shou, Mengdie Chen, Li Jiang, Meng Yuan, Bo Yang, Qiaojun He, Ji Cao et al. · 2025 · Angewandte Chemie
  70. Sulfonamide-Functionalized Polymeric Nanoparticles for Enhanced In Vivo Colorectal Cancer Therapy
    Rubén D. Sinisterra, Pedro Pires Goulart Guimarães, Celso Tarso Rodrigues Viana, Luciana de Andrade Pereira, Sávio Morato de Lacerda Gontijo, Paula Peixoto Campos, Sílvia Passos Andrade, Robson A.S. Santos · 2021 · Current Drug Delivery
  71. T‐17, a novel cyclin‐dependent kinases/histone deacetylases dual inhibitor, induces cancer cells death through cell cycle arrest and apoptosis
    Lin Zhang, Rui Long, Xiaoli Li, Junhao Jiang, Huali Chen, Binghua Tian, Binyu Long, Yu Yu, Zongjie Gan · 2022 · Drug Development Research
  72. Expedient synthesis of 8-membered azasultams: A combined synthetic, DFT, and in vitro study
    Heorhii V. Posternak, Olena D. Semoshkina, Vasyl Yu. Hys, Demyd S. Milokhov, Pavlo Virych, Svitlana Valentinovna Shishkina, Yulian M. Volovenko, Alexey V. Dobrydnev · 2024 · Tetrahedron Chem
  73. Use of pH-interfering agents as chemosensitizers: Clinical studies survey
    Joonas A. Haapasalo, Kristiina Nordfors, Seppo Parkkila · 2020 · Elsevier eBooks
  74. On the Search of Metallated Sulfonamides: Synthesis and X‐ray Characterization of the New Sulfathiazolato Nickel(II)‐Chelate Complex [Ni(STZ)2(Py)2]·2Py (STZ = Sulfathiazolato Anion; Sulfathiazole = N1‐2‐thiazolyl‐sulfanilamide; Py = Pyridine)
    Gelson Manzoni de Oliveira, Lara Regina Soccol Gris, Lenice de Lourenço Marques, Ernesto Schulz Lang · 2007 · Zeitschrift für anorganische und allgemeine Chemie
  75. Synthesis and Carbonic Anhydrase Inhibition Profiles of N‐(3‐sulfamoylphenyl)propanamide/benzamide Derivatives: Experimental and Computational Insights With Absorption, Distribution, Metabolism, and Excretion Profiling
    Ferhat GÜNEŞ, Uğur Güller, Pınar Güller, Barış Anıl, Mehmet Koca · 2025 · Chemistry & Biodiversity
  76. Synthesis of substituted benzoindolinothiazepines using 5‐ and 6‐nitroindolines
    Guillaume Laconde, Patrick Depreux, Pascal Berthelot, Jean‐Pierre Hénichart · 2005 · Heteroatom Chemistry
  77. Çinko(II)–Sulfatiyazol-Dietilentriamin Kompleksinin Hesaplamalı Kimya Yöntemi ile Spektroskopik Özelliklerinin İncelenmesi: Moleküler Modelleme Çalışması
    Filiz Öztürk, Tuğba Aycan · 2021 · Afyon Kocatepe University Journal of Sciences and Engineering
  78. Biochemical Principles of Targeted Protein Degradation
    Roman V. Agafonov, Richard W. Deibler, W. Austin Elam, Joe Sahil Patel, Stewart L. Fisher · 2022 · Wiley eBooks
  79. Decoding the Therapeutic Potential of Sulfonamide Esters: A Journey of Discovery
    Muhammad Danish, Tehreem Liaquat, Syed Rizwan Shafqat, Shahid Zaman, Emad E. Mahmoud · 2025 · Journal of Molecular and Engineering Materials
  80. Network-driven identification of indisulam neo-substrates for targeted protein degradation
    Andrew F. Jarnuczak, Orli Yogev, Angelo Andres, Stephanie Kay Ashenden, Ye Cheng, Fiona Pachl, Andrew Zhang, Maria Emanuela Cuomo, Meizhong Jin · 2025 · Molecular Omics
  81. A DRUG HUNTER’S APPROACH TO MOLECULAR GLUES
    Daniel S. La, Christopher G. Nasveschuk, Adam M. Gilbert · 2025 · Medicinal chemistry reviews
  82. The sulfonamide anticancer agent indisulam enhances the chemosensitivity of gastric cancer cells by targeting FKBP8
    Yue Li, Chengpiao Lu, Jiaqi Lu, Honglv Jiang, Dan Li, Yuhong Wang, Guoqiang Xu, Xiaohui Wang, Jingjing Ma · 2026 · FEBS Journal
  83. Recent Advances in Targeting RNA Splicing Factors with Small Molecules
    Xinrui Yuan, Chao‐Yie Yang · 2026 · Journal of Medicinal Chemistry
  84. G1 phase arrest and apoptosis induction in human thyroid cancer cell line Thr.C1.PI33 by 3-hydrogenkwadaphnin isolated from Dendrostellera lessertii.
    Azin Nowrouzi, Razieh Yazdanparast · 2007 · PubMed
  85. 2-Amino-5-Bromo-3-Iodoacetophenone and 2-Amino-5-Bromo-3-Iodobenzamide as Synthons for Novel Polycarbo-Substituted Indoles and Their Annulated Derivatives
    Mmakwena Modlicious Mmonwa, Malose J. Mphahlele · 2017 · Springer eBooks
  86. Nano/Micro-Assisted Regenerative Medicine
    Soo-Hong Lee · 2018 · MDPI eBooks
  87. Exploring the Role of Nanotherapeutics for Diagnosis and Treatment of Solid Tumor
    Ravinder Verma, Rokeya Akter, Manish Kumar, Shailendra Bhatt, Abhishek Sunil Tiwari, Varsha Tiwari, Priti Tagde, Parijat Pandey, Vineet Mittal, Deepika Purohit et al. · 2023 · Current Nanoscience
  88. Design and Synthesis of 7-(N-Aryl Pyrrolidinyl) Indoles as Potential DCAF15 Binders
    Ravi Devarajappa, Scarlett Kiyeleko, Sofiane Hocine, Victor Cosson, Remi Calandrino, Timea Baló, Jayson Alves Bordelo, Sébastien Triboulet, Laure Caruana, Laurence Klipfel et al. · 2025 · Reactions
  89. The Tumor Microenvironment: New Insights into Regulation of Tumor pH by Carbonic Anhydrases
    Pawel Swietach, Adrian Llewellyn Harris, Richard D. Vaughan‐Jones · 2010 · Springer eBooks
  90. Discovery of Molecular Glues to Induce Selective Protein Degradation, Leading to Development of New Modalities with Targeted Protein Knockdown Function
    Taisuke Uehara, Takashi Owa · 2020 · Journal of Synthetic Organic Chemistry Japan
  91. Miscellaneous Antineoplastic Agents
    Daniel Lednicer · 2015
  92. Exploiting Chemical Probes for Identifying Drug Target Proteins
    Toshitaka Sato, Yoshiya Oda, Takashi Owa, Takeshi Nagasu · 2003 · Journal of the Mass Spectrometry Society of Japan
  93. Arylsulfonamide mediated RBM39 degradation causes aberrant splicing of mitotic kinesins
    Seemon Coomar, Alexander V. Penson, Juerg Schwaller, Omar Ibrahim Abdel-Wahab, Dennis G. Gillingham · 2021 · bioRxiv (Cold Spring Harbor Laboratory)
  94. CDK Inhibitors
    Laurent Meijer, Eve Damiens · 2002 · Elsevier eBooks
  95. Inhibition of Lactate Dehydrogenase A (LDH-A) by Diclofenac Sodium Induces Apoptosis in HeLa Cells by Activation of AMPK
    Avirup Malla, Suvroma Gupta, Runa Sur · 2023 · bioRxiv (Cold Spring Harbor Laboratory)
  96. Investigational Anticancer Agents Targeting the Microtubule
    Lyudmila A. Vereshchagina, Orit Scharf, Alexander Dimitrios Colevas · 2009 · Humana Press eBooks
  97. Induction of Cell Cycle Arrest in Tumor Tissue And Bone Marrow Of Grafted Mice Treated with Androgen and Antiandrogen. Running title: Effect of androgen and antiandrogen on leukemia cell line
    Souad Aboudkhil, Laurent Henry, Mohammed Nabil Benchekroun, Hassan Filali, Jean Paul Bureau · 2015
  98. Clinical Pharmacokinetics of Anticancer Drugs:focus on E7070, methotrexate and paclitaxel
    H.J.G.D. van den Bongard · 2002
  99. Malignant tumor disease as a sub-chronic, progressive intoxication on the basis of the perpetuation of the release of amino acids, initiated by a retrograde-differentiated muscle degradation protease
    Z. Douvlis · 2002 · Medical Hypotheses
  100. Tumor acidosis in malignant progression and therapy
    Paola Pellegrini · 2016 · Figshare