Discovery of Novel Antitumor Sulfonamides Targeting G1 Phase of the Cell Cycle
Owa, Takashi, Yoshino, Hiroshi, Okauchi, Tatsuo, Yoshimatsu, Kentaro, Ozawa, Yoichi, Sugi, Naoko Hata, Nagasu, Takeshi, Koyanagi, Nozomu +1 more·1999·Journal of Medicinal Chemistry
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- Spectroscopic, structural, electrochemical and antimicrobiological studies of Cu(II)-sulfathiazole complex with diethylenetriamine ligandFiliz Öztürk, İclal Bulut, Yeliz Genç Bekiroğlu, Ahmet Bulut · 2016 · Polyhedron
- The effect of Euphorbia szovitsii Fisch. & C.A.Mey extract on the viability and the proliferation of MDA-MB-231 cell lineMajid Asadi-Samani, Mahmoud Rafieian‐Kopaei, Zahra Lorigooini, Hedayatollah Shirzad · 2018 · Bioscience Reports
- Aryl Sulfonamides Induce Degradation of Aryl Hydrocarbon Receptor Nuclear Translocator through CRL4DCAF15 E3 LigaseSung Ah Kim, Seung-Hyun Jo, Jin Hwa Cho, Min Yeong Yu, Ho‐Chul Shin, Jung‐Ae Kim, Byoung Chul Park, Byoung Chul Park, Jeong‐Hoon Kim, Jeong‐Hoon Kim · 2020 · Molecules and Cells
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- A Facile and Efficient Synthesis of Arylsulfonamido‐Substituted 1,5‐Benzodiazepines and N‐[2‐(3‐Benzoylthioureido)aryl]‐3‐oxobutanamide DerivativesAbdolali Alizadeh, Nasrin Zohreh · 2010 · Helvetica Chimica Acta
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- Anticancer Agent E7070 Inhibits Amino Acid and Uracil Transport in Fission YeastKappei Tsukahara, Tatsuo Watanabe, Naoko Hata-Sugi, Kentaro Yoshimatsu, Hiroto Okayama, Takeshi Nagasu · 2001 · Molecular Pharmacology
- Substituent GroupsPatrick Bazzini, Camille Georges Wermuth · 2008 · Elsevier eBooks
- Methylation of RBM39 by PRMT6 enhances resistance to Indisulam in non-small cell lung cancer by promoting alternative splicing of proto-oncogenesTongjia Zhang, Shujie Wang, Yue Zhou, Zitao Jiao, Kejia Lu, Xinyi Liu, Hui Li, Wei Jiang, Xiaowei Zhang · 2025 · PLoS Biology
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- Indisulam exerts anticancer effects via modulation of transcription, translation and alternative splicing on human cervical cancer cells.Zhihui Dou, Xuetian Zhang, Wei Su, Taotao Zhang, Fei Ye, Dapeng Zhao, Xiaohua Chen, Qiang Li, Hong Zhang, Cuixia Di · 2023 · PubMed Central
- Synthesis and bioactivity evaluation of some novel sulfonamide derivativesCh. Subramanyam, Sk. Nayab Rasool, D. B. Janakiramudu, S. Rasheed, A. Uday Sankar, Chamarthi Naga Raju · 2017 · Phosphorus, sulfur, and silicon and the related elements
- Cytotoxicity of multicellular cancer spheroids, antibacterial, and antifungal of selected sulfonamide derivatives coupled with a salicylamide and/or anisamide scaffoldAlaaeldin M F Galal, Walid Fayad, Walaa S.A. Mettwally, Sanaa K. Gomaa, Esam R. Ahmed, Heba A. El-Refai, Atef G. Hanna · 2019 · Medicinal Chemistry Research
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- Novel N-(aryl/heteroaryl)-2-chlorobenzenesulfonamide derivatives: Synthesis and anticancer activity evaluationAnita Bułakowska, Jaroslaw J. Slawinski, Kamila Siedlecka-Kroplewska, Grzegorz Stasiłojć, Marcin Serocki, Mateusz Heldt · 2020 · Bioorganic Chemistry
- Human metabolism of [14C]indisulam following i.v. infusion in cancer patientsJan Hendrik Beumer, Michel J. X. Hillebrand, Dick Pluim, Hilde Rosing, Karen Foley, S. Murray Yule, Jan H.M. Schellens, Jos H. Beijnen · 2005 · Investigational New Drugs
- Design, synthesis, chemical and biological evaluation of 2,5,5-trisubstituted-1,2-thiazepan-6-one 1,1-dioxidesDemyd S. Milokhov, Mykhailo S. Pomalin, Mykola O. Balabushko, Vladyslav R. Holubnychyi, Vasyl Yu. Hys, Pavlo Virych, Petro Virych, N Yu Lukianova, Vasyl A. Chumachenko, Svitlana Shishkina et al. · 2023 · Results in Chemistry
- Synthesis of an RBM39 Degrader That Downregulates CEP192 and Induces Disorganized Spindle StructuresXilin Lyu, Xiancheng Wang, Dongze Lin, Yuhan Lu, Chenxu Wang, Ziqin Yan, Zhiyi Wang, Ying Cheng, Jing Cheng, Xuelian Ren et al. · 2025 · Journal of Medicinal Chemistry
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- Design, Synthesis, and in vitro and in vivo Evaluations of (Z)‐3,4,5‐Trimethoxystyrylbenzenesulfonamides/sulfonates as Highly Potent Tubulin Polymerization InhibitorsRasala Mahesh, Vadithe Lakshma Nayak, Korrapati Suresh Babu, Syed Riyaz, Thokhir Basha Shaik, Gajjela Bharath Kumar, Prema Latha Mallipeddi, Challa Ratna Reddy, Kunta Chandra Shekar, Jedy Jose et al. · 2017 · ChemMedChem
- Natural stilbenes and analogues as antineoplastic agentsFulvia Orsini, Guido Sello · 2008 · Studies in natural products chemistry
- Exploring DCAF15 for reprogrammable targeted protein degradationSeemon Coomar, Dennis G. Gillingham · 2019 · bioRxiv (Cold Spring Harbor Laboratory)
- Molecular Glue Degraders: From Serendipity to Hunting and DesignLuis Nieto‐Barrado, Ana Domostegui, Cristina Mayor‐Ruiz · 2022 · Wiley eBooks
- Solid‐Phase Parallel Synthesis of Photocleavable Bifunctional Molecules Enables Efficient Phenotypic Protein Degrader DiscoveryBaoli Ding, Jiawen Hu, Rongtian Zhang, Binyan Shou, Mengdie Chen, Jiang Li, Meng Yuan, Bo Yang, Qiaojun He, Ji Cao et al. · 2025 · Angewandte Chemie International Edition
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- Methods to characterize and discover molecular degraders in cellsZhi Lin, Christina M. Woo · 2022 · Chemical Society Reviews
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- The RBM39 degrader indisulam inhibits acute megakaryoblastic leukemia by altering the alternative splicing of ZMYND8Ying Hua Yang, Zhiheng Li, Yang Yang, Peifang Xiao, Zhixu He, Zimu Zhang, Yizhen Li, Lei Shi, Xiaodong Wang, Yanfang Tao et al. · 2025 · Cell & Bioscience
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