Chemistries of bifunctional PROTAC degraders
Cao, Chaoguo, He, Ming, Wang, Liguo, He, Yuna, Rao, Yu·2022·Chemical Society Reviews
Cited by (315)
Items 301–315 of 315
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- BindingDB Entry 50023634: Next-generation cancer therapeutics: PROTACs and the role of heterocyclic warheads in targeting resistance.BindingDB · 2026 · UC San Diego
- BindingDB Entry 50020095: Development of a GC-376 Based Peptidomimetic PROTAC as a Degrader of 3-Chymotrypsin-like Protease of SARS-CoV-2.BindingDB · 2024 · UC San Diego
- BindingDB Entry 50020617: Application of Novel Degraders Employing Autophagy for Expediting Medicinal Research.BindingDB · 2024 · UC San Diego
- Targeted protein degradation in cancer: strategies for undruggable targets and progress towards clinical translationJinxin Tang, Zehao Cheng, Tian Xie, Yan Zhuang, Hongkun Hu, Chenbei Li, Hua Wang, Chengyao Feng, Chao Tu · 2026 · Biomarker Research
- Discovery of the First Orally Bioavailable GLI1 PROTAC for the Treatment of Colorectal CancerYabing Xin, Zi-Yu Yang, Yong-Fu Luo, Yan-Li Du, Rui-Ning Li, Qian Wu, Yangyang Chen, Xiang-Yang Li, Yixue Qiao, Mengchen Lu et al. · 2026 · European Journal of Medicinal Chemistry