THE MECHANISM OF ENZYME-INHIBITOR-SUBSTRATE REACTIONS

Goldstein, Avram·1944·Journal of General Physiology

Cited by (182)

Items 101–182 of 182

  1. FURTHER STUDIES OF INHIBITION OF BACTERIAL GLUTAMIC DECARBOXYLASE
    Eugene Roberts · 1953 · Journal of Biological Chemistry
  2. Small-Molecule Mediated Neuroprotection in an In Situ Model of Tauopathy
    Nicolette S. Honson, Jordan R. Jensen, Aida Abraha, Garth F. Hall, Jeff Kuret · 2009 · Neurotoxicity Research
  3. The esterase activity of bovine carbonic anhydrase B above pH 9. Reversible and cooalent inhibition by acetozolamide.
    JW Wells, S. I. Kandel, Marianne Kandel · 1975 · Journal of Biological Chemistry
  4. Extending the quasi-steady state approximation by changing variables
    José A. M. Borghans · 1996 · Bulletin of Mathematical Biology
  5. Investigation of the effect of calcium ions on the splitting of adenosinetriphosphate by myosin
    L.B. Nanninga · 1959 · Biochimica et Biophysica Acta
  6. Competitive partial inhibitors of serum albumin‐catalyzed sulfur cyanolysis
    Rebecca Jarabak, JOHN W. WESTLEY · 1990 · Journal of Biochemical and Molecular Toxicology
  7. General Theory of Specific Binding: Insights from a Genetic-Mechano-Chemical Protein Model
    John M McBride, Jean‐Pierre Eckmann, Tsvi Tlusty · 2022 · Molecular Biology and Evolution
  8. A comparison of the decarbamoylation rates of physostigmine-inhibited plasma and red cell cholinesterases of man with other species
    Janet R. Wetherell, Mary C. French · 1991 · Biochemical Pharmacology
  9. THE ACTION OF CARBAMIC ESTERS AND TETRAETHYLPYROPHOSPHATE ON NORMAL AND CURARIZED FROG RECTUS MUSCLE
    Franz Hobbiger · 1950 · British Journal of Pharmacology and Chemotherapy
  10. Recent Advances in Enzyme Inhibition: A Pharmacological Review
    Kuldeep Singh, Bharat Bhushan, Nidhi Mittal, Abhishek Kushwaha, Chandan Kumar Raikwar, Arun Kumar Sharma, Dilip Kumar Chanchal, Shivendra Kumar, Mohit Agrawal · 2023 · Current Enzyme Inhibition
  11. Inhibition of squalene synthase in vitro by 3-(biphenyl-4-yl)-quinuclidine
    Walter H.J. Ward, Geoffrey A. Holdgate, S Freeman · 1996 · Biochemical Pharmacology
  12. Kinetics of Active-Site-Directed Irreversible Inhibition
    A. Russell Main · 1973 · Essays in toxicology
  13. In silico and crystallographic studies identify key structural features of biliverdin IXβ reductase inhibitors having nanomolar potency
    Natasha M. Nesbitt, Xiliang Zheng, Zongdong Li, José A. Manso, Wan-Yi Yen, Lisa E. Malone, Jorge Ripoll‐Rozada, Pedro José Barbosa Pereira, Timothy J. Mantle, Jin Wang et al. · 2018 · Journal of Biological Chemistry
  14. Differentiation of three types of competitive cholinesterase inhibitors
    David K. Myers · 1951 · Archives of Biochemistry and Biophysics
  15. The effect of substituents on the hydrolysis of phenyl acetate by wheat germ lipase
    Oscar Gawron, Chester J. Grelecki, Marjorie Duggan · 1953 · Archives of Biochemistry and Biophysics
  16. Chemical Control of Nervous Activity
    David A. Nachmansohn · 1950 · Elsevier eBooks
  17. THE INHIBITION OF CHOLINESTERASES BY 3‐(DIETHOXYPHOSPHINYLOXY)‐N‐METHYLQUINOLINIUM METHYLSULPHATE AND ITS TERTIARY BASE
    Franz Hobbiger · 1954 · British Journal of Pharmacology and Chemotherapy
  18. Incorporation of thymidine and iodeoxyuridine in mammalian cells in vitro
    D. K. Myers, L. E. Feinendegan · 1975 · Journal of Cellular Physiology
  19. Fragment-Based Screening for Enzyme Inhibitors Using Calorimetry
    Michael I. Recht, Vicki L. Nienaber, Francisco E. Torres · 2015 · Methods in enzymology on CD-ROM/Methods in enzymology
  20. The molecular kinetics of the urea-urease system. V. Relationship between activity and concentration of urease solutions
    Mary Colman Wall, Keith J. Laidler · 1953 · Archives of Biochemistry and Biophysics
  21. Phenylethanolamine N-methyltransferase inhibition: re-evaluation of kinetic data
    Qian Wu, Kevin R. Criscione, Gary L. Grunewald · 2004 · Bioorganic & Medicinal Chemistry Letters
  22. The Inhibition of Human Salivary α-Amylase by Type II α-Amylase Inhibitor fromTriticum Aestivum IsCompetitive, Slow and Tight-Binding
    David Judson Goff, F. Jon Kull · 1995 · Journal of enzyme inhibition
  23. Zur Hypothese eines cholinergen Wirkungsmechanismus des Morphins
    W. Schaumann · 1959 · Naunyn-Schmiedeberg s Archives of Pharmacology
  24. Effects of Coordinating Metal Ions on the Mediated Inhibition of Trypsin by Bis(benzimidazoles) and Related Compounds
    Jared J. Paul, Sandra R. Kircus, Thomas N. Sorrell, Patricia A. Ropp, H. Holden Thorp · 2006 · Inorganic Chemistry
  25. A new piecewise spectral homotopy analysisof the Michaelis-Menten enzymatic reactions model
    Stanford Shateyi, S. S. Motsa, Yasir Khan · 2013 · Numerical Algorithms
  26. Influence of enzyme activators and inhibitors, present in an enzyme preparation, on the relations between reaction rate and enzyme concentration
    Masuyuki Katsumata · 1969 · Journal of Theoretical Biology
  27. Properties and behavior of purified human plasma cholinesterase. II. Inactivation by mercuric chloride
    Avram Goldstein, Mary E. Doherty · 1951 · Archives of Biochemistry and Biophysics
  28. A serine protease inhibitor from hemolymph of green mussel, Perna viridis
    Mohd Sajid Khan, U. Goswami, Supada Rambhau Rojatkar · 2008 · Bioorganic & Medicinal Chemistry Letters
  29. The Kinetic Basis of a General Method for the Investigation of Active Site Content of Enzymes and Catalytic Antibodies: First-Order Behaviour under Single-turnover and Cycling Conditions
    Christopher M. Topham, Sheraz Gul, Marina Resmini · 2000 · Journal of Theoretical Biology
  30. A new method for the derivation of rate equations in enzyme kinetics using the maximum rate of product formation
    Ivan G. Darvey, Simon James Prokhovnik, Jim Williams · 1965 · Biochimica et Biophysica Acta (BBA) - Enzymology and Biological Oxidation
  31. Binding of competitive (product) inhibitors to papain in the active and inactive state
    B.G. Wolthers, Kor H. Kalk · 1970 · Biochimica et Biophysica Acta (BBA) - Enzymology
  32. Zur Kinetik der Cholinesterasen-Hemmung durch Prostigmin
    W. Hardegg · 1952 · Naunyn-Schmiedeberg s Archives of Pharmacology
  33. Florasulam Is a Potent Inhibitor of Mycobacterium tuberculosis Acetohydroxyacid Synthase and Possesses In Vivo Antituberculosis Activity
    Shun Jie Wun, Lendl Tan, Thierry G. A. Lonhienne, Yu Shang Low, Peter F. Josh, Andy Kuo, Maree Therese Smith, Yanhua Gao, Gregory K. Pierens, Luke W. Guddat et al. · 2025 · ACS Infectious Diseases
  34. Assessing the Inhibitory Potential of Kinase Inhibitors In Vitro: Major Pitfalls and Suggestions for Improving Comparability of Data Using CK1 Inhibitors as an Example
    Aileen Roth, Adrian Gihring, Florian Göser, Christian Peifer, Uwe Knippschild, Joachim Bischof · 2021 · Molecules
  35. Active centers of microsomal cytochrome P-450 determined with metyrapone by mutual depletion system kinetics
    Ivar Roots, Alfred G. Hildebrandt · 1973 · Naunyn-Schmiedeberg s Archives of Pharmacology
  36. The ATPase activity of avian erythromyeloblastic leukosis virus I. Introductory kinetics
    Irving Green, D. G. Sharp · 1955 · Biochimica et Biophysica Acta
  37. The Mechanism of Action of Hydrolytic Enzymes
    H. Lindley · 1954 · Advances in enzymology and related areas of molecular biology/Advances in enzymology and related subjects
  38. A REWARDING RESEARCH PATHWAY
    Avram Goldstein M. D · 1997 · The Annual Review of Pharmacology and Toxicology
  39. Succinoxidase inhibition studies. II. Mechanism of the binding of a naphthoquinone and of antimycin A by serum albumin
    Arnold E. Reif · 1953 · Archives of Biochemistry and Biophysics
  40. Kinetics of Cofactor-activated Enzyme-catalyzed Reactions
    James O. Alben · 1967 · Journal of Biological Chemistry
  41. Hydrolytic Transformation of Environmental Pollutants
    D. J. Ecobichon · 1977 · Comprehensive physiology
  42. Influence of vitamin-E on liveresterase and cholinesterase
    C. van der Meer, H. T. M. Nieuwerkerk · 1951 · Biochimica et Biophysica Acta
  43. �ber- und unteradditive Wirkung von Herzglykosiden
    W. Schaumann · 1963 · Naunyn-Schmiedeberg s Archives of Pharmacology
  44. DETERMINATION AND PROPERTIES OF SULFHYDRYL GROUPS IN YEAST ALCOHOL DEHYDROGENASE**The original investigations reported were supported by grants from the Office of Naval Research, the National Institutes of Health of the Department of Health, Education and Welfare, and the Howard Hughes Medical Institute.
    Frederic L. Hoch, Bert L. Vallée · 1959 · Elsevier eBooks
  45. Pyridine nucleotide dependent metallodehydrogenases
    Bert L. Vallée, Frederic L. Hoch · 1961 · Reviews of physiology, biochemistry and pharmacology
  46. Drug Design
    Roger L. Lundblad · 2015 · Elsevier eBooks
  47. Thiamin and Cocarboxylase as Inhibitors of Cholinesterases.
    Egil Gjone., Karl Håkon Skramstad · 1955 · Acta Pharmacologica et Toxicologica
  48. Pyridine Nucleotide Dependent Metallodehydrogenases
    Bert L. Vallée, Frederic L. Hoch · 1961 · Springer eBooks
  49. Grundlagen der Kinetik enzymatisch katalysierter Reaktionen
    Ludwig Lumper · 1964 · Enzyme
  50. Novel triazole-based coumarin compounds as acetylcholinesterase inhibitors: Evidence and mechanism of 3-acetyl coumarin tethered (2-bromophenyl)-1,2,3 triazole as a potential mixed type inhibitor
    Naseer Ahmad Dar, Owais Hassan Wani, Yuanyuan Wang, Faez Iqbal Khan, Bilal A. Ganie, Syed Wajaht A. Shah, Tanveer Ali Dar, Tabasum Ismail · 2025 · European Journal of Medicinal Chemistry Reports
  51. Characteristics of Rabbit Muscle Adenylate Kinase Inhibition by Sulfur and Recovery by Dithiothreitol
    Percy J. Russell, Anjana Williams, David Avtla · 1995 · Journal of enzyme inhibition
  52. Direct Identification and Characterization of β-Adrenergic Receptors and Functional Relationship of Adenylyl Cyclase
    Edward Meigs Brown, Allen M. Spiegel, J. D. Gardner · 1978 · Elsevier eBooks
  53. A relationship between the rate of attaining equilibrium and the velocity constant of the reverse reaction in certain enzyme-inhibitor systems
    Avram Goldstein · 1952 · Cellular and Molecular Life Sciences
  54. Extension of the Rate Equations for Enzyme Inhibition
    Mordechai L. Kremer · 1967 · Israel Journal of Chemistry
  55. The effect of an N-methylcarbamate on esterases from snail, mouse and man studied by starch-gel electrophoresis
    Ha ̊kan Tegelstro ̈m, Ha ̊kan Wahren · 1972 · Comparative Biochemistry and Physiology Part B Comparative Biochemistry
  56. Alternative Modes of Prophage Insertion and Excision
    Michael B. Yarmolinsky · 1972 · Elsevier eBooks
  57. Pyridine nucleotide dependent metallodehydrogenases
    Bert L. Vallée, Frederic L. Hoch · 2007 · Springer eBooks
  58. Crippled lung: variations on a theme by Macleod.
    J Quintero, Edward W. Swenson, M Arborelius · 1980 · PubMed
  59. The ATPase activity of avian erythromyeloblastic leukosis virus
    Irving Green · 1955 · Biochimica et Biophysica Acta
  60. Effects of group-selective reagents on monoamine oxidase and cholinesterase in guinea pig ileum
    P. Dal Pra, Letizia De Paolis, Luigi Rossini · 1971 · Pharmacological Research Communications
  61. The plasma proteins and their fractionation
    John Tileston Edsall · 2007 · Springer eBooks
  62. The plasma proteins and their fractionation
    John T. Edsall-Boston · 1950 · Springer eBooks
  63. Genetic variation in the carbonic anhydrase isozymes of macaque monkeys. IV. Degradation by heat and proteolysis of normal and variant carbonic anhydrase isozymes of Macaca nemestrina
    William R.A. Osborne, Richard E. Tashian · 1984 · Archives of Biochemistry and Biophysics
  64. Target: A Useful Model
    Néstor Vicente Torres, Eberhard O. Voit · 2002 · Cambridge University Press eBooks
  65. Enzyme kinetics: Inhibition equations derived from the inelastic collision hypothesis
    John Z. Hearon, Robert Katzman · 1954 · Bulletin of Mathematical Biology
  66. Impiego delle radiazioni ultraviolette per lo studio dei gruppi attivi degli enzimi
    Alessandro Vescia, Enzo Boeri, Serena Traniello · 1960 · Il Nuovo Cimento
  67. An Application of Reverse Quasi Steady State Approximation over SERCA
    Prashant Dwivedi Prashant Dwivedi · 2012 · IOSR Journal of Mathematics
  68. Detailed Unification Equations for Kinetic Parameters: A Case Study on Human Salivary Alpha Amylase
    Ikechukwu Iloh Udema · 2017 · Journal of Analytical & Pharmaceutical Research
  69. Deciphering the Mechanism of Action of Armeniaspirol: A Polyketide Gram-Positive Antibiotic
    Puneet Labana · 2021 · uO Research (University of Ottawa)
  70. The Cybernetic Origins of Life
    Kathleen Alicia Powers · 2020 · eScholarship (California Digital Library)
  71. Cholinesterasen
    W. Hardegg · 1966 · Enzyme
  72. Cholinesterasen
    W. Hardegg · 1966 · Enzyme
  73. Drug Design
    Roger L. Lundblad · 2022 · Elsevier eBooks
  74. Carbamates
    1967 · Elsevier eBooks
  75. TIGHT‐BINDING INHIBITORS
    Robert A. Copeland · 2023
  76. Cholinesterase inhibition
    B.N. Szafran, G.A. Casillas, B.L. Alman · 2023 · Elsevier eBooks
  77. In Vitro Biology: Measuring Pharmacological Activity that Will Translate to Clinical Efficacy
    Iain G. Dougall, Rachel L. Grimley, Per-Erik Strömstedt · 2023 · Royal Society of Chemistry eBooks
  78. Alternatives To Sulphur Dioxide for Inhibiting Tyrosinase and Protecting Grape Must from Browning
    Fernando Zamora, Aitor García-Roldán, Antoni Canalda-Sabaté · 2025 · SSRN Electronic Journal
  79. Study of Possible Alternatives to Sulphur Dioxide for Inhibiting Tyrosinase and Protecting Grape Must from Browning
    Aitor García-Roldán, Antoni Canalda-Sabaté, Jordi Gombau · 2026 · Beverages
  80. Conception et synthèse d’iminosucres multivalents bioactifs à motif glycoimidazole : développement d’une méthode de déshydroxylation sélective
    Maëva M. Pichon · 2018
  81. Development and Stabilization of a Paper-Based Biosensor for the On-Site Detection of Pesticide Residues on Fruits and Vegetables
    Pravin Pokhrel, Krisha Pokharel, Basant Giri · 2026 · Journal of Analytical Chemistry
  82. Polyphosphate Attenuates Oxidative Stress to Support Temperature Adaptability in Hot Spring Cyanobacteria
    Xiaohua Song, Yong’an Wei, Minxiang Xu et al. · 2026 · Plants