Effect of a 28-d treatment with L-796568, a novel β3-adrenergic receptor agonist, on energy expenditure and body composition in obese men
Larsen, Thomas M, Toubro, Søren, van Baak, Marleen A, Gottesdiener, Keith M, Larson, Patrick, Saris, Wim HM, Astrup, Arne·2002·The American Journal of Clinical Nutrition
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- Activating Connexin43 gap junctions primes adipose tissue for therapeutic interventionYi Zhu, Na Li, Mingyang Huang, Xi Chen, Yu An, Jianping Li, Shangang Zhao, Jan‐Bernd Funcke, Jianhong Cao, Zhenyan He et al. · 2022 · Acta Pharmaceutica Sinica B
- Design of a novel pyrrolidine scaffold utilized in the discovery of potent and selective human β3 adrenergic receptor agonistsGregori J. Morriello, Harvey R. Wendt, Alka Bansal, Jerry Di Salvo, Scott D. Feighner, Jiafang He, Amanda L. Hurley, Donna L. Hreniuk, Gino Salituro, Marat Vijay Reddy et al. · 2010 · Bioorganic & Medicinal Chemistry Letters
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- Sympathetic Nervous System Signaling in Heart Failure and Cardiac AgingGaetano Santulli · 2015 · Springer eBooks
- DNA‐mediated UCP1 overexpression in adipose tissue: A promising anti‐obesity gene therapyZewei Zhao, Longyun Hu, Bigui Song, Qian Wu, Jiejing Lin, Qingqing Liu, Siqi Liu, Jin Li, Molin Wang, Jin Li et al. · 2025 · Clinical and Translational Medicine
- The β-adrenergic antagonist propranolol partly abolishes thermogenic response to bioactive food ingredientsAnita Belza, Maj-Britt Gille, Sarah Schultz John, Jens Kondrup · 2009 · Metabolism
- Molecular pharmacology of GPCRsChristopher J. Langmead, Roger J. Summers · 2018 · British Journal of Pharmacology
- Single-nuclei RNA Profiling Reveals Disruption of Adipokine and Inflammatory Signaling in Adipose Tissue of Burn PatientsCarly M. Knuth, Zachary Ricciuti, Dalia Barayan, Sarah Rehou, Abdikarim Abdullahi, Lauar de Brito Monteiro, Marc G. Jeschke · 2023 · Annals of Surgery
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- Potent benzimidazolone based human β3-adrenergic receptor agonistsDon R. Finley, Michael G. Bell, Anthony G. Borel, William E. Bloomquist, Marlene L. Cohen, Mark L. Heiman, Aidas Kriauciunas, Donald P. Matthews, Tania Miles, David A. Neel et al. · 2006 · Bioorganic & Medicinal Chemistry Letters
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- Reduced response to an estrous induction program in postpartum beef cows treated with zilpaterol and gaining body weightAdrian Guzmán, Everardo González-Padilla, Pedro Garces-Yepez, Jorge Víctor Rosete Fernández, René Carlos Calderón Robles, Clara Murcia, Carlos G. Gutiérrez · 2012 · Animal Reproduction Science
- Combination of a Beta Adrenoceptor Modulator and a Norepinephrine-Serotonin Uptake Inhibitor for the Treatment of ObesityCynthia D. Jesudason, James E. Baker, Robert D. Bryant, Jack W. Fisher, Libbey S. O’Farrell, Gregory A. Gaich, Minxia Michelle He, Steven D. Kahl, Aidas Kriauciunas, Mark L. Heiman et al. · 2011 · ACS Medicinal Chemistry Letters
- The Adrenergic System in Cardiovascular Metabolism and AgingGaetano Santulli · 2015 · Springer eBooks
- Approved and Off-Label Uses of Obesity Medications, and Potential New Pharmacologic Treatment OptionsMaría Luisa Isidro, Fernando Cordido · 2010 · Pharmaceuticals
- Angiotensin II type 2 receptor as a novel activator of brown adipose tissue in obesityFabiola Álvarez-Gallego, Raquel González‐Blázquez, Marta Gil‐Ortega, Beatriz Somoza, María Calderón‐Domínguez, Javier Moratinos, Virginia García‐García, Paloma Fernández, Daniel González‐Moreno, Marta Viana et al. · 2023 · BioFactors
- Effect of the β3 adrenoceptor agonist CL 316243 on hypothalamic 5-HT synthesis and suppression of REM sleep in the ratRachel K. Conley, J. Li, M. Ivarsson, Peter H. Hutson · 2006 · Journal of Psychopharmacology
- Longitudinal trends and subgroup analysis in publication patterns for preclinical data of newly approved drugsUrsula Köster, Ingo J. A. Nolte, Martin Christian Michel · 2015 · Naunyn-Schmiedeberg s Archives of Pharmacology
- Plasticity of the Adipose OrganSaverio Cinti · 2010 · Wiley eBooks
- Weight-Loss DrugsGeorge A. Bray, Frank L. Greenway · 2007 · Humana Press eBooks
- Inducible UCP1 silencing: A lentiviral RNA-interference approach to quantify the contribution of beige fat to energy homeostasisNicole Wen Mun Khor, Michael M. Swarbrick, Jenny Elizabeth Gunton · 2019 · PLoS ONE
- Targeting Thermogenesis in the Development of Antiobesity DrugsRuth McPherson, Frédérique Tesson, Robert Dent, Mary‐Ellen Harper · 2004 · CRC Press eBooks
- Thermogenic Targets for Obesity Management in the Era of Incretin-Based TherapiesSahar Soliman, Rebecca Andrews‐Dickert, Petra Ročić, Mihail I. Mitov · 2025 · Pharmaceuticals
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- Brown Adipose Tissue: A New Target for Antiobesity TherapyAnna Meiliana, Andi Wijaya · 2010 · The Indonesian Biomedical Journal
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- Influencing energy expenditure and substrate utilisationJohn C. Clapham, Jonathan R.S. Arch · 2008 · Birkhäuser Basel eBooks
- Drugs with Thermogenic PropertiesArne Vernon Astrup, Søren Toubro · 2008 · CRC Press eBooks
- Evaluating the teratogenicity of the selective ß3-adrenoceptor agonist, CL 316.243 hydrate by employing FETAX (frog embryo teratogenesis assay)Ayper Boğa, Yaşar Sertdemır, Ayşe Doğan · 2016 · Drug and Chemical Toxicology
- A Status of Drugs on the Horizon for Obesity and the Metabolic Syndrome—a Comprehensive Review 2005Frank L. Greenway, George A. Bray · 2007 · Springer eBooks
- Zukunftsperspektiven der medikamentösen Therapie bei AdipositasBirgit Pichler, Bernhard H. Ludvik · 2003 · Journal für Kardiologie (Krause & Pachernegg GmbH)
- Browning of Adipose OrganSaverio Cinti · 2014 · Springer eBooks
- Strategies to activate brown adipose tissue in humansMaarten J. Vosselman · 2015
- EXPLORING BETA 3 ADRENOCEPTORS FOR POTENTIAL CLINICAL APPLICATIONS. Review ArticleArunima Sen, Vikram Narayan Nichani · 2010
- Pericardial fat is a nutritionally regulated depot of brown adipose tissueShalini Ojha · 2015 · Nottingham ePrints (University of Nottingham)
- Genetics of Cardiovascular Risk in ObesityPiers R. Blackett, Dharambir K. Sanghera · 2015 · Springer eBooks
- Brown fat as a therapy for obesity and diabetesRoy Jesse Shephard · 2011 · Yearbook of Sports Medicine
- Distinct Genetic Backgrounds in Quantitative Traits Preceding Type 2 Diabetes: One Reason for Missing HeritabilityPiers R. Blackett, Dharambir K. Sanghera · 2013 · Journal of Advances in Medicine and Medical Research
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- Pathophysiology of Obesity and Cancer: Drugs and Signaling TargetsAhood Khalid, Hira Khalid, Neelam Faiza, Anees Ahmed Khalil, Kiran Shahbaz, Ayesha Aslam, Quratul Ain Shahid, Surajudeen Abiola Abdulrahman, Chukwuebuka Egbuna, Kingsley Chukwuemeka Patrick-Iwuanyanwu · 2021 · Springer eBooks
- I Can Get Fat Where? The Other Types of FatNathan Denton · 2021 · Oxford University Press eBooks
- Review of Al-Qaeda's Armies: Middle East Affiliate Groups and the Next Generation of TerrorAvi Jorisch · 2005 · Middle East Quarterly
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- Phytocompounds That Target White Adipose Tissue for Weight Loss: A Review Spanning From Ucp1 Induction in Rodents to Human Clinical TrialsAnn A. Coulter, Frank L. Greenway, Guru Ramanathan, Jacqueline R. Hubbard, Candida Joan Rebello · 2026 · Obesity Reviews
- BindingDB Entry 50039497: Combination of a Beta adrenoceptor modulator and a norepinephrine-serotonin uptake inhibitor for the treatment of obesity.BindingDB · 2013 · UC San Diego
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- BindingDB Entry 50044030: Biarylaniline phenethanolamines as potent and selective beta3 adrenergic receptor agonists.BindingDB · 2014 · UC San Diego
- BindingDB Entry 50035396: Potent and selective, sulfamide-based human beta 3-adrenergic receptor agonists.BindingDB · 2012 · UC San Diego
- BindingDB Entry 50018277: Potent benzimidazolone based human beta(3)-adrenergic receptor agonists.BindingDB · 2009 · UC San Diego
- BindingDB Entry 50021381: Potent oxindole based human beta3 adrenergic receptor agonists.BindingDB · 2009 · UC San Diego