In vivo characterization of the highly selective monoacylglycerol lipase inhibitor KML 29: antinociceptive activity without cannabimimetic side effects
Ignatowska‐Jankowska, B M, Ghosh, S, Crowe, M S, Kinsey, S G, Niphakis, M J, Abdullah, R A, Tao, Q, O' Neal, S T +4 more·2014·British Journal of Pharmacology
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- Targeting the Endocannabinoid Metabolic Enzymes to Reduce Inflammatory PainSudeshna Ghosh · 2014 · VCU Scholars Compass (Virginia Commonwealth University)
- Analgesic and Anti-Inflammatory Effects of Monoacylglycerol Lipase Inhibition in Mice Subjected to Collagen-Induced ArthritisSara R. Nass · 2015
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- Discriminative Stimulus Properties of Endogenous Cannabinoid Degradative Enzyme InhibitorsOwens, Robert · 2016 · VCU Scholars Compass (Virginia Commonwealth University)
- Development and Preclinical Evaulation of Novel Enzyme-targeting Radiotracers for Positron Emission TomographyJustin W. Hicks · 2015 · TSpace (University of Toronto)
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- Inhibiting the Cannabinoid Catabolic Enzyme MAGL to Potentiate the Anti-Arthritic Properties of the Synthetic Glucocorticoid DexamethasoneSara R. Nass · 2017
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- Role of the type-1 cannabinoid receptor in the control of water intakeZhe Zhao · 2019 · theses.fr (ABES)
- Fatty acid amide hydrolase (FAAH) and the endocannabinoid system in obesity: Mechanistic insights and pharmacological opportunities beyond incretin‐based therapiesIlaria Serra, Elisa Bisconti, Daniele Vergara, Anna Maria Giudetti, Francesco Vari · 2026 · British Journal of Pharmacology
- Advances in Small Molecule Research Targeting Monoacylglycerol Lipase in Drug DiscoveryShuming Chen, Jie Yang, Hu W, Gao Jh, Le Chen, Jifa Zhang, Ben Zhang, Wuyu Mao · 2026 · Medicinal Research Reviews
- BindingDB Entry 50017870: Reversible Monoacylglycerol Lipase Inhibitors: Discovery of a New Class of Benzylpiperidine Derivatives.BindingDB · 2023 · UC San Diego
- BindingDB Entry 50006784: Identification of ABX-1431, a Selective Inhibitor of Monoacylglycerol Lipase and Clinical Candidate for Treatment of Neurological Disorders.BindingDB · 2021 · UC San Diego
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- BindingDB Entry 50023447: Design, synthesis and biological evaluation of naphthyl amide derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors.BindingDB · 2026 · UC San Diego
- BindingDB Entry 50000616: Discovery of 1,5-Diphenylpyrazole-3-Carboxamide Derivatives as Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors.BindingDB · 2019 · UC San Diego
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