Regulatory role of G protein-coupled estrogen receptor for vascular function and obesity
Haas, Elvira, Bhattacharya, Indranil, Brailoiu, Eugen, Damjanović, Marlen, Brailoiu, G. Cristina, Gao, Xin, Mueller-Guerre, Laurence, Marjon, Nicole A. +12 more·2009·Circulation Research
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- The Activation Function-1 of Estrogen Receptor Alpha Prevents Arterial Neointima Development Through a Direct Effect on Smooth Muscle CellsNatalia F. Smirnova, Coralie Fontaine, Mélissa Buscato, Adrien Lupieri, Alexia Vinel, Marie‐Cécile Valera, Maéva Guillaume, Nicole Malet, Jean‐Michel Foidart, Isabelle Raymond‐Letron et al. · 2015 · Circulation Research
- The GPER1 Agonist G-1 Attenuates Endothelial Cell Proliferation by Inhibiting DNA Synthesis and Accumulating Cells in the S and G2 Phases of the Cell CycleAnders Holm, Bo Baldetorp, Björn Olde, L.M. Fredrik Leeb-Lundberg, Bengt‐Olof Nilsson · 2011 · Journal of Vascular Research
- G-1-Activated Membrane Estrogen Receptors Mediate Increased Contractility of the Human MyometriumKaushik Maiti, Jonathan Paúl, M. Read, E.-C. Chan, Simon C. Riley, Pravin Nahar, Roger Smith · 2011 · Endocrinology
- G protein-coupled estrogen receptor 1 mediates relaxation of coronary arteries via cAMP/PKA-dependent activation of MLCPXuan Yu, Fen Li, Enno Klußmann, John N. Stallone, Guichun Han · 2014 · American Journal of Physiology-Endocrinology and Metabolism
- Estrogen receptor subcellular localization and cardiometabolismPierre Gourdy, Maéva Guillaume, Coralie Fontaine, Marine Adlanmérini, Alexandra Montagner, Henrik Laurell, Françoise Lenfant, Jean‐François Arnal · 2018 · Molecular Metabolism
- Signalling mechanisms in the cardiovascular protective effects of estrogen: With a focus on rapid/membrane signalling.Ana-Roberta Niță, Greg A. Knock, Richard J. Heads · 2021 · Current Research in Physiology
- Pregnancy Augments G Protein Estrogen Receptor (GPER) Induced Vasodilation in Rat Uterine Arteries via the Nitric Oxide - cGMP Signaling PathwayTeresa Tropea, Ernestina Marianna De Francesco, Damiano Cosimo Rigiracciolo, Marcello Maggiolini, Mark Wareing, George Osol, Maurizio Mandalà · 2015 · PLoS ONE
- Activation of GPR30 inhibits cardiac fibroblast proliferationHao Wang, Zhuo Zhao, Marina Lin, Leanne Groban · 2015 · Molecular and Cellular Biochemistry
- Emerging evidence of the importance of rapid, non-nuclear estrogen receptor signaling in the cardiovascular systemKazutaka Ueda, Richard H. Karas · 2012 · Steroids
- Regulatory Actions of Estrogen Receptor Signaling in the Cardiovascular SystemUeda, Kazutaka, Adachi, Yusuke, Liu, Pangyen, Fukuma, Nobuaki, Takimoto, Eiki · 2020 · Frontiers in Endocrinology
- History of Estrogen: Its Purification, Structure, Synthesis, Biologic Actions, and Clinical ImplicationsRichard J. Santen, Evan R. Simpson · 2018 · Endocrinology
- Increased estrogen receptor alpha in experimental aortic aneurysms in females compared with malesAdriana Laser, Abhijit Ghosh, Karen J. Roelofs, Omar Sadiq, Brendan McEvoy, Paul D. DiMusto, Jonathan L. Eliason, Gilbert R. Upchurch · 2013 · Journal of Surgical Research
- Chronic Activation of the G Protein-Coupled Receptor 30 with Agonist G-1 Attenuates Heart FailureShoulei Kang, Ying Liu, Di Sun, Chunle Zhou, Aiying Liu, Chuanying Xu, Yanling Hao, Dongye Li, Changdong Yan, Hong Sun · 2012 · PLoS ONE
- Human uterine and placental arteries exhibit tissue-specific acute responses to 17 -estradiol and estrogen-receptor-specific agonistsJemma J. Corcoran, Christopher Nicholson, Michèle Sweeney, Jayne C. Charnock, Stephen Courtenay Robson, Melissa Westwood, Michael John Taggart · 2013 · Molecular Human Reproduction
- Crosstalk between nuclear and G protein-coupled estrogen receptorsShannon N. Romano, Daniel A. Gorelick · 2017 · General and Comparative Endocrinology
- A role for G-protein coupled estrogen receptor (GPER) in estrogen-induced carcinogenesis: Dysregulated glandular homeostasis, survival and metastasisEdward J. Filardo · 2017 · The Journal of Steroid Biochemistry and Molecular Biology
- GPER Mediates Cardiotropic Effects in Spontaneously Hypertensive Rat HeartsErnestina Marianna De Francesco, Tommaso Angelone, Teresa Pasqua, Marco Pupo, Maria Carmela Cerra, Marcello Maggiolini · 2013 · PLoS ONE
- Attenuation of Microbiotal Dysbiosis and Hypertension in a CRISPR/Cas9 Gene Ablation Rat Model of GPER1Harshal Waghulde, Xi Cheng, Sarah Galla, Blair Mell, Jingwei Cai, Shondra M. Pruett‐Miller, Guillermo Vázquez, Andrew D. Patterson, Matam Vijay Kumar, Bina Joe · 2018 · Hypertension
- Estradiol: A Steroid with Multiple FacetsAnita V. Kumar, Antara A. Banerjee, Dipty Singh, Gargi Thakur, Nandini Kasarpalkar, Shubhangi Gavali, Sushama Gadkar, Taruna Madan, Smita D. Mahale, Nafisa Balasinor et al. · 2018 · Hormone and Metabolic Research
- Estrogen Receptors: Therapeutic Perspectives for the Treatment of Cardiac Dysfunction after Myocardial InfarctionJaqueline Soares da Silva, Tadeu Lima Montagnoli, Bruna Rocha, Matheus L. C. A. Tacco, Sophia C. P. Marinho, Gisele Zapata‐Sudo · 2021 · International Journal of Molecular Sciences
- ER , ER , and gpER: novel aspects of oestrogen receptor signalling in atherosclerosisMatthias R. Meyer, Matthias Barton · 2009 · Cardiovascular Research
- G protein-coupled estrogen receptor regulates embryonic heart rate in zebrafishShannon N. Romano, Hailey E. Edwards, Jaclyn Paige Souder, Kevin J. Ryan, Xiangqin Cui, Daniel A. Gorelick · 2017 · PLoS Genetics
- From physiology to pathology: Emerging roles of GPER in cardiovascular diseaseZixuan Wang, Junren Liu, Ying Chen, Yi Tang, Ting Chen, Chang Sheng Zhou, Shuo Wang, Ranbo Chang, Zhongshuai Chen, Wenqing Yang et al. · 2025 · Pharmacology & Therapeutics
- Reduced vasorelaxation to estradiol and G-1 in aged female and adult male rats is associated with GPR30 downregulationSarah Hoffmann Lindsey, Ariel S. da Silva, Mauro S. B. Silva, Mark C. Chappell · 2013 · American Journal of Physiology-Endocrinology and Metabolism
- Not lost in translation: Emerging clinical importance of the G protein-coupled estrogen receptor GPERMatthias Barton · 2016 · Steroids
- G Protein-Coupled Estrogen Receptor in Energy Homeostasis and Obesity PathogenesisHaifei Shi, Shiva Priya Dharshan Senthil Kumar, Xian Liu · 2013 · Progress in molecular biology and translational science
- GPR30 regulates diet-induced adiposity in female mice and adipogenesis in vitroAihua Wang, Jing Luo, William Moore, Hana Alkhalidy, Ling Wu, Jinhua Zhang, Zhen Cheng Wei, Yao Wang, Deborah J. Clegg, Bin Xu et al. · 2016 · Scientific Reports
- The Interface of Nuclear and Membrane Steroid SignalingL. Treviño, Daniel A. Gorelick · 2021 · Endocrinology
- Sex Differences and Regulatory Actions of Estrogen in Cardiovascular SystemKazutaka Ueda, Nobuaki Fukuma, Yusuke Adachi, Genri Numata, Hiroyuki Tokiwa, Masayuki Toyoda, Akira Otani, Masaki Hashimoto, Pang‐Yen Liu, Eiki Takimoto · 2021 · Frontiers in Physiology
- Impaired left-ventricular cardiac function in male GPR30-deficient miceMartina Delbeck · 2010 · Molecular Medicine Reports
- Improvement of Vascular Function by Acute and Chronic Treatment with the GPR30 Agonist G1 in Experimental Diabetes MellitusZi-Lin Li, Jincheng Liu, Shui‐bing Liu, Xiaoqiang Li, Dinghua Yi, Ming Zhao · 2012 · PLoS ONE
- Hetero-oligomeric Complex between the G Protein-coupled Estrogen Receptor 1 and the Plasma Membrane Ca2+-ATPase 4bQuang‐Kim Tran, Mark VerMeer, Michelle Burgard, Ali B. Hassan, Jennifer R. Giles · 2015 · Journal of Biological Chemistry
- Membrane Estrogen Receptors: Their Role in Blood Pressure Regulation and Cardiovascular DiseaseRoopashree Prabhushankar, Caroline Krueger, Camila Margarita Manrique · 2013 · Current Hypertension Reports
- Estrogenic vascular effects are diminished by chronological agingChristopher Nicholson, Michèle Sweeney, Stephen Courtenay Robson, Michael John Taggart · 2017 · Scientific Reports
- Alisol B 23-acetate adjusts bile acid metabolisim via hepatic FXR-BSEP signaling activation to alleviate atherosclerosisYu Fu, Han Feng, Xue Ding, Qing-Hai Meng, Shu-Rui Zhang, Jun Li, Ying Chao, Tingting Ji, Yunhui Bi, Weiwei Zhang et al. · 2022 · Phytomedicine
- Adaptive increases in expression and vasodilator activity of estrogen receptor subtypes in a blood vessel-specific pattern during pregnancyKarina M. Mata, Wěi Li, Ossama M. Reslan, Waleed Tariq Siddiqui, Lauren A. Opsasnick, Raouf Ali Khalil · 2015 · American Journal of Physiology-Heart and Circulatory Physiology
- Activation of GPER Induces Differentiation and Inhibition of Coronary Artery Smooth Muscle Cell ProliferationFen Li, Xuan Yu, Claudia K. Szynkarski, Cong Meng, Beiyan Zhou, Rola Barhoumi, Richard E. White, Cristine L. Heaps, John N. Stallone, Guichun Han · 2013 · PLoS ONE
- Schizophrenia Gene Expression Profile Reverted to Normal Levels by AntipsychoticsBenedicto Crespo‐Facorro, Carlos Alberto Vanegas Prieto, Jesús Sainz · 2015 · The International Journal of Neuropsychopharmacology
- Evolving research in nongenomic actions of aldosteroneJonathan S. Williams · 2013 · Current Opinion in Endocrinology Diabetes and Obesity
- Non-genomic Effects of Estrogen on Cell Homeostasis and Remodeling With Special Focus on Cardiac Ischemia/Reperfusion InjuryRossella Puglisi, Gianfranco Mattia, Alessandra Carè, Giuseppe Marano, Walter Malorni, Paola Matarrese · 2019 · Frontiers in Endocrinology
- The Role of G Protein-Coupled Estrogen Receptor (GPER) in Vascular Pathology and PhysiologyFujie Xu, Jipeng Ma, Xiaowu Wang, Xiaoya Wang, Weiyi Fang, Jingwei Sun, Zilin Li, Jincheng Liu · 2023 · Biomolecules
- Estrogens: Two nuclear receptors, multiple possibilitiesBiason-Lauber, Anna, Lang-Muritano, Mariarosaria · 2022 · Molecular and Cellular Endocrinology
- Sex- and age-dependent effects of Gpr30 genetic deletion on the metabolic and cardiovascular profiles of diet-induced obese miceLuca Meoli, Jörg Isensee, Valeria Zazzu, Christoph S. Nabzdyk, Dian Soewarto, Henning Witt, Anna Foryst‐Ludwig, Ulrich Kintscher, Patricia Ruíz · 2014 · Gene
- Vascular Inflammation and Atherosclerosis: The Role of Estrogen ReceptorsEva N. Kassi, Eliana Spilioti, Narjes Nasiri Ansari, Christos Adamopoulos, Paraskevi Moutsatsou, Angeliki Papapanagiotou, Gerasimos Siasos, Dimitris Tousoulis, Athanasios G. Papavassiliou · 2015 · Current Medicinal Chemistry
- Subtype-specific Estrogen Receptor-mediated Vasodilator Activity in the Cephalic, Thoracic, and Abdominal Vasculature of Female RatOssama M. Reslan, Zongzhi Yin, Graciliano Ramos Alencar do Nascimento, Raouf Ali Khalil · 2013 · Journal of Cardiovascular Pharmacology
- Vasodilatory effects of the selective GPER agonist G-1 is maximal in arteries of postmenopausal womenSamsul Arefin, Tommaso Simoncini, Rebekah S. Wieland, Folke Hammarqvist, Stefania Spina, Lorenzo Goglia, Karolina R. Kublickiene · 2014 · Maturitas
- A common hypofunctional genetic variant of GPER is associated with increased blood pressure in womenRoss D. Feldman, Robert Gros, Qingming Ding, Yasin Hussain, Matthew R. Ban, Adam D. McIntyre, Robert Alexander Hegele · 2014 · British Journal of Clinical Pharmacology
- Evidence for G‐Protein–Coupled Estrogen Receptor as a Pronatriuretic FactorEman Y. Gohar, Elizabeth M. Daugherty, Jeffrey O. Aceves, Randee Sedaka, Ijeoma E. Obi, J. Miller Allan, Reham H. Soliman, Chunhua Jin, Carmen De Miguel, Sarah Hoffmann Lindsey et al. · 2020 · Journal of the American Heart Association
- GPER: A novel target for non-genomic estrogen action in the cardiovascular systemGuichun Han, Fen Li, Xuan Yu, Richard E. White · 2013 · Pharmacological Research
- Activation of novel estrogen receptor GPER results in inhibition of cardiocyte apoptosis and cardioprotectionW M Li, Wei Xiang, Ping Ye · 2015 · Molecular Medicine Reports
- Mechanisms of G Protein-Coupled Estrogen Receptor-Mediated Spinal NociceptionElena Deliu, Gabriela Cristina Brailoiu, Jeffrey B. Arterburn, Tudor Ionel Oprea, Khalid Benamar, Nae J. Dun, Eugen Brailoiu · 2012 · Journal of Pain
- Estrogen Signaling in the Adrenal CortexBrasilina Caroccia, Teresa Maria Seccia, Matthias Barton, Gian Paolo Rossi · 2016 · Hypertension
- G Protein-Coupled Estrogen Receptor Protects From Angiotensin II-Induced Increases in Pulse Pressure and Oxidative StressBenard Ojwang Ogola, Margaret Ann Zimmerman, Venkata N. L. R. Sure, Kaylee M. Gentry, Jennifer L. Duong, Gabrielle L. Clark, Kristin S. Miller, Prasad V. G. Katakam, Sarah Hoffmann Lindsey · 2019 · Frontiers in Endocrinology
- Steroid Receptor Coactivator-1 Mediates Estrogenic Actions to Prevent Body Weight Gain in Female MiceLiangru Zhu, Yongjie Yang, Pingwen Xu, Fang Zou, Xiaofeng Yan, Lan Liao, Jianming Xu, Bert W. O’Malley, Yong Xu · 2012 · Endocrinology
- Activation of G protein-coupled estrogen receptor 1 induces coronary artery relaxation via Epac/Rap1-mediated inhibition of RhoA/Rho kinase pathway in parallel with PKAXuan Yu, Qiao Zhang, Yan Zhao, Benjamin J. Schwarz, John N. Stallone, Cristine L. Heaps, Guichun Han · 2017 · PLoS ONE
- Continuous Exposure of Breast Cancer Cells to Tamoxifen Upregulates GPER-1 and Increases Cell ProliferationLuis Molina, Felipe A. Bustamante, Alexander Ortloff, Iraidi Ramos, Pamela Ehrenfeld, Carlos D. Figueroa · 2020 · Frontiers in Endocrinology
- Mechanism of Cardioprotection: What Can We Learn from Females?Elizabeth Murphy, Cláudia Jacques Lagranha, Anne M. Deschamps, Mark Jeffrey Kohr, Tiffany Tuyen Minh Nguyen, Renee P. Wong, Junhui Sun, Charles Steenbergen · 2011 · Pediatric Cardiology
- G protein‐coupled estrogen receptor‐mediated effects on cytosolic calcium and nanomechanics in brain microvascular endothelial cellsJoseph B. Altmann, Guang Yan, Jeffrey F. Meeks, Mary E. Abood, Eugen Brailoiu, Gabriela Cristina Brailoiu · 2015 · Journal of Neurochemistry
- GPER agonist dilates mesenteric arteries via PI3K-Akt-eNOS and potassium channels in both sexesPollyana Peixoto, Rosária Dias Aires, Virginia Soares Lemos, Nazaré Souza Bissoli, Roger Lyrio dos Santos · 2017 · Life Sciences
- Cardioprotective and anti-inflammatory effects of G-protein coupled receptor 30 (GPR30) on postmenopausal type 2 diabetic ratsHossein Azizian, Mohammad Khaksari, Gholamreza Asadikaram, Mansour Esmailidehaj, Zeinab Farhadi · 2018 · Biomedicine & Pharmacotherapy
- Highly efficient synthesis and characterization of the GPR30-selective agonist G-1 and related tetrahydroquinoline analogsRitwik Burai, Chinnasamy Ramesh, Marvin Shorty, Ramona F. Curpan, Cristian Bologa, Larry A. Sklar, Tudor Ionel Oprea, Eric R. Prossnitz, Jeffrey B. Arterburn · 2010 · Organic & Biomolecular Chemistry
- Hormonal effects on blood vesselsMasahiro Akishita, Jing Yu · 2012 · Hypertension Research
- Role of GPER-Mediated Signaling in Testicular Functions and TumorigenesisAdele Chimento, Arianna De Luca, Marta Claudia Nocito, Paola Avena, Davide La Padula, Lucia Zavaglia, Vincenzo Pezzi · 2020 · Cells
- Reciprocality Between Estrogen Biology and Calcium Signaling in the Cardiovascular SystemQuang‐Kim Tran · 2020 · Frontiers in Endocrinology
- Roles of estrogens, estrogen-like compounds, and endocrine disruptors in adipocytesFernando Lizcano · 2022 · Frontiers in Endocrinology
- Non-genomic vasorelaxant effects of 17β-estradiol and progesterone in rat aorta are mediated by L-type Ca2+ current inhibitionElisa Cairrão, Ezequiel Álvarez, João Miguel Carvas, António José Santos-Silva, Ignácio Verde · 2012 · Acta Pharmacologica Sinica
- Vascular effects of aldosterone: Sorting out the receptors and the ligandsRoss D. Feldman, Robert Gros · 2013 · Clinical and Experimental Pharmacology and Physiology
- Estrogen Receptor Subtypes Mediate Distinct Microvascular Dilation and Reduction in [Ca2+]i in Mesenteric Microvessels of Female RatMarc Q. Mazzuca, Karina M. Mata, Wěi Li, Sridhar S. Rangan, Raouf Ali Khalil · 2014 · Journal of Pharmacology and Experimental Therapeutics
- Unraveling the mechanisms underlying the rapid vascular effects of steroids: sorting out the receptors and the pathwaysRoss D. Feldman, Robert Gros · 2011 · British Journal of Pharmacology
- STX, a Novel Nonsteroidal Estrogenic Compound, Induces Rapid Action in Primate GnRH Neuronal Calcium Dynamics and Peptide ReleaseBrian P. Kenealy, Kim L. Keen, Oline K. Rønnekleiv, E. Terasawa · 2011 · Endocrinology
- Liuwei Dihuang soft capsules attenuates endothelial cell apoptosis to prevent atherosclerosis through GPR30-mediated regulation in ovariectomized ApoE-deficient miceJing Yi, Danfeng Cai, Qi Chen, Qingping Xiong, Tianhui Hu, Yuan Yao, Chao Lin, Xin Sun, Ying Lu, Xueyun Kong et al. · 2017 · Journal of Ethnopharmacology
- G protein-coupled estrogen receptor inhibits vascular prostanoid production and activityMatthias R. Meyer, Natalie C. Fredette, Matthias Barton, Eric R. Prossnitz · 2015 · Journal of Endocrinology
- Estrogen signaling as a bridge between the nucleus and mitochondria in cardiovascular diseasesEmanuel Guajardo-Correa, Juan Francisco Silva-Agüero, Ximena Calle, Mario Chiong, Mauricio Henríquez, Gerardo García‐Rivas, Mauricio Latorre, Valentina Parra · 2022 · Frontiers in Cell and Developmental Biology
- Activation of GPER ameliorates experimental pulmonary hypertension in male ratsAllan K. N. Alencar, Guilherme Carneiro Montes, Tadeu Lima Montagnoli, Ananssa M Silva, Sabrina Teixeira Martinez, Aline Guerra Manssour Fraga, Hao Wang, Leanne Groban, Roberto T. Sudo, Gisele Zapata‐Sudo · 2016 · European Journal of Pharmaceutical Sciences
- Sex Differences, Estrogen Metabolism and Signaling in the Development of Pulmonary Arterial HypertensionYanan Sun, Shreya Sangam, Qiang Guo, Jian Wang, Haiyang Tang, Stephen M. Black, Ankit A. Desai · 2021 · Frontiers in Cardiovascular Medicine
- Evidence That the G Protein–Coupled Membrane Receptor GPR30 Contributes to the Cardiovascular Actions of EstrogenSarah Hoffmann Lindsey, Mark C. Chappell · 2011 · Gender Medicine
- G Protein-Coupled Estrogen Receptor-1 Is Involved in the Protective Effect of Protocatechuic Aldehyde against Endothelial DysfunctionByung Soo Kong, Yoon Hee Cho, Eun Jig Lee · 2014 · PLoS ONE
- G-protein-mediated signaling in vascular smooth muscle cells — implications for vascular diseaseTill F. Althoff, Stefan Offermanns · 2015 · Journal of Molecular Medicine
- Sex and sex steroids as determinants of cardiovascular riskAndrea Cignarella, Chiara Bolego, Matthias Barton · 2024 · Steroids
- Obesity and Cancer: 27-Hydroxycholesterol, the Missing LinkArvand Asghari, Michihisa Umetani · 2020 · International Journal of Molecular Sciences
- Clinical efficacy and safety of angiogenesis inhibitors: sex differences and current challengesAndrea Cignarella, Gian Paolo Fadini, Chiara Bolego, Lucia Trevisi, Carlotta Boscaro, Viola Sanga, Teresa Maria Seccia, Antonio Rosato, Gian Paolo Rossi, Matthias Barton · 2021 · Cardiovascular Research
- Targeting the G protein-coupled estrogen receptor (GPER) in obesity and diabetesSharma, Geetanjali, Prossnitz, Eric R. · 2021 · Endocrine and Metabolic Science
- Release of calcium from endolysosomes increases calcium influx through N-type calcium channels: Evidence for acidic store-operated calcium entry in neuronsLiang Hui, Nicholas H. Geiger, Duncan Bloor-Young, Grant C. Churchill, Jonathan D. Geiger, Xuesong Chen · 2015 · Cell Calcium
- GPER/GPR30 and Regulation of Vascular Tone and Blood PressureMatthias R. Meyer, Eric R. Prossnitz, Matthias Barton · 2011 · Immunology Endocrine & Metabolic Agents - Medicinal Chemistry
- 17β-estradiol promotes acute refeeding in hungry mice via membrane-initiated ERα signalingKaifan Yu, Yanlin He, Ilirjana Hyseni, Zhou Pei, Yongjie Yang, Pingwen Xu, Xing Cai, Hesong Liu, Na Qu, Hailan Liu et al. · 2020 · Molecular Metabolism
- Delineating the receptor mechanisms underlying the rapid vascular contractile effects of aldosterone and estradiolRobert Gros, Qingming Ding, Mark Davis, Rasha Shaikh, Bonan Liu, Jozef Chorazyczewski, J. Geoffrey Pickering, Ross D. Feldman · 2011 · Canadian Journal of Physiology and Pharmacology
- Metabolic impact of endogenously produced estrogens by adipose tissue in females and males across the lifespanLee, Angel A., Den Hartigh, Laura J. · 2025 · Frontiers in Endocrinology
- Progress in the molecular understanding of central regulation of body weight by estrogensKenji Saito, Xuehong Cao, Yanlin He, Yong Xu · 2015 · Obesity
- Calcium signaling in endothelial and vascular smooth muscle cells: sex differences and the influence of estrogens and androgensDaniel Asunción‐Alvarez, Javier C. Palacios, Roberto O. Ybañez‐Julca, Cristhian N. Rodríguez-Silva, Chukwuemeka R. Nwokocha, Fredi Cifuentes, David J. Greensmith · 2024 · American Journal of Physiology-Heart and Circulatory Physiology
- Aldosterone-induced hypertension is sex-dependent, mediated by T cells and sensitive to GPER activationQuynh Nhu Dinh, Antony Vinh, Hyun Ah Kim, Narbada Saini, Brad R. S. Broughton, Sophocles Chrissobolis, Henry Diep, Courtney P Judkins, Grant Raymond Drummond, Christopher Graeme Sobey · 2020 · Cardiovascular Research
- Role of ERβ and GPR30 in the endocrine pancreas: A matter of estrogen dose.Ana B. Ropero, Y. Pang, P. Alonso-Magdalena, P. Thomas, A. Nadal · 2012 · Steroids
- The activation of G protein-coupled estrogen receptor induces relaxation via cAMP as well as potentiates contraction via EGFR transactivation in porcine coronary arteriesXuan Yu, John N. Stallone, Cristine L. Heaps, Guichun Han · 2018 · PLoS ONE
- G protein–coupled estrogen receptor: a promising therapeutic target for aldosterone-induced hypertensionXuehan Li, Wenlong Kuang, Zhihua Qiu, Zihua Zhou · 2023 · Frontiers in Endocrinology
- GPER modulates tone and coronary vascular reactivity in male and female ratsAngelina Rafaela Debortoli Spinassé, Wender do Nascimento Rouver, Nathalie Tristão Banhos Delgado, Vinícius Mengal, Erick Roberto Gonçalves Claudio, Laena Pernomian, Lusiane Maria Bendhack, Margareth Ribeiro Moysés, Roger Lyrio dos Santos · 2017 · Journal of Molecular Endocrinology
- Expression of the oestrogen receptor GPER by testicular peritubular cells is linked to sexual maturation and male fertilityFranziska Sandner, H. Welter, Julia Schwarzer, Frank Michael Köhn, Henryk F. Urbanski, Artur Mayerhofer · 2014 · Andrology
- Calcium supplementation increases circulating cholesterol by reducing its catabolism via GPER and TRPC1-dependent pathway in estrogen deficient womenSongtao Li, Ying Li, Hua Ning, Lixin Na, Yucun Niu, Maoqing Wang, Rennan Feng, Liyan Liu, Fuchuan Guo, Shaoying Hou et al. · 2013 · International Journal of Cardiology
- Bradycardic effects mediated by activation of G protein‐coupled estrogen receptor in rat nucleus ambiguusGabriela Cristina Brailoiu, Jeffrey B. Arterburn, Tudor Ionel Oprea, Vineet Chandra Chitravanshi, Eugen Brailoiu · 2012 · Experimental Physiology
- Discovery of Selective Probes and Antagonists for G Protein-Coupled Receptors FPR/FPRL1 and GPR30Jeffrey B. Arterburn, Tudor Ionel Oprea, Eric R. Prossnitz, Bruce S. Edwards, Larry A. Sklar · 2009 · Current Topics in Medicinal Chemistry
- Impact of Estrogens on the Regulation of White, Beige, and Brown Adipose Tissue DepotsGabriel B. Bernasochi, James R. Bell, Evan R. Simpson, Lea M.D. Delbridge, Wah Chin Boon · 2019 · Comprehensive physiology
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