Stepwise androgen receptor dimerization

van Royen, Martin E., van Cappellen, Wiggert A., de Vos, Carola, Houtsmuller, Adriaan B., Trapman, Jan·2012·Journal of Cell Science

Cited by (144)

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  3. Microfluidics-Based Technologies for the Assessment of Castration-Resistant Prostate Cancer
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  4. Discovery of JNJ-63576253, a Next-Generation Androgen Receptor Antagonist Active Against Wild-Type and Clinically Relevant Ligand Binding Domain Mutations in Metastatic Castration-Resistant Prostate Cancer
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  8. Phase Separation Mediated Sub-Nuclear Compartmentalization of Androgen Receptors
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  10. A high-throughput platform for single-molecule tracking identifies drug interaction and cellular mechanisms
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  11. Structural perspectives on the androgen receptor, the elusive shape-shifter
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  13. The androgen receptor for the radiation oncologist
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  14. A high-throughput platform for single-molecule tracking identifies drug interaction and cellular mechanisms
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  15. Dihydrotestosterone-androgen receptor signaling suppresses EBV-positive gastric cancer through DNA demethylation-mediated viral reactivation
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  16. The evolution of eukaryotic linear motifs governing the function of androgen receptor from fish to Homo sapiens
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  18. Androgen receptor ubiquitination links KCTD13 to genitourinary tract defects
    Ahmed Chahdi, Carolina J. Jorgez, Jill Anne Rosenfeld, Neetu Neetu, Abhishek Seth · 2025 · The FASEB Journal
  19. Androgen Receptor in Health and Disease
    Marco Marcelli · 2017 · Springer eBooks
  20. Dichotomy in the Epigenetic Mark Lysine Acetylation is Critical for the Proliferation of Prostate Cancer Cells
    Ravi Ramesh Pathak, Marc Philizaire, Shiraz Mujtaba · 2015 · Cancers
  21. Androgen Receptor Signaling Interactions Control Epithelial–Mesenchymal Transition (EMT) in Prostate Cancer Progression
    Sarah K. Martin, Michael V. Fiandalo, Natasha Kyprianou · 2013 · Springer eBooks
  22. Deciphering the allosteric control of androgen receptor DNA binding by its disordered N-terminal domain
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  23. Blocking the dimerization of polyglutamine-expanded androgen receptor protects cells from DHT-induced toxicity by increasing AR turnover
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  24. Mutant androgen receptor induces neurite loss and senescence independently of ARE binding in a neuronal model of SBMA
    Jordyn S Karliner, Yuhong Liu, Diane E. Merry · 2024 · Proceedings of the National Academy of Sciences
  25. Bedeutung der Androgenrezeptor-Spleißvariante AR-V7 für Prognose und Therapie des fortgeschrittenen Prostatakarzinoms
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  26. NanoLuc Binary Technology as a methodological approach: an important new tool for studying the localization of androgen receptor and androgen receptor splice variant V7 homo and heterodimers
    Juan Carlos Guzmán, Katrin Weigelt, Angela Neumann, Philipp Tripal, Benjamin Schmid, Zoltán Winter, Ralf Palmisano, Zoran Čulig, Marcus Victor Cronauer, Paul Muschler et al. · 2024 · BMC Cancer
  27. Development of novel small molecule inhibitor of androgen receptor to treat castration-resistant prostate cancer
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  28. The Effects of Legacy and Emerging Persistent Organic Pollutants in Endocrine Signalling Pathways in Mammalian Cancer Cell Lines
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  29. Inhibition of castration resistant prostate cancer by sintokamide A : an antagonist of the amino-terminus of the androgen receptor
    Iran Tavakoli · 2013 · cIRcle (University of British Columbia)
  30. Androgeenireseptorin tumatranslokaatio, FOXA1-vuorovaikutus ja liikkuvuus ihmisen soluissa
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  31. Androgen Receptor Signaling in Castration Resistant Prostate Cancer
    Yu Zhao, Donald J. Tindall, Haojie Huang · 2016 · Springer eBooks
  32. Retroactivity effects dependency on the transcription factors binding mechanisms
    Libertad Pantoja-Hernández, Elena R Alvarez-Buylla, Carlos Fernando Aguilar-Ibañez, Adriana Garay‐Arroyo, A. Soria, Juan Carlos Martínez‐García · 2016 · Journal of Theoretical Biology
  33. Targeting epithelial to mesenchymal transition (EMT) to modulate prostate cancer cell chemoresistance
    Akanksha Upadhyaya · 2020 · Queensland University of Technology
  34. Development of novel androgen receptor inhibitors to overcome castrate-resistant prostate cancer
    Hilal Saraç, Artem R Cherkasov, Nathan A. Lack · 2021 · Elsevier eBooks
  35. Roles of sex phenotype and sex chromosome dosage in sex-biased DNA methylation
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  36. Androgen Receptors in the Pathology of Disease
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  37. Faculty Opinions recommendation of ARv7 Represses Tumor-Suppressor Genes in Castration-Resistant Prostate Cancer.
    Patricia V. Elizalde · 2019 · Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
  38. Supplementary Data 3 from Discovery of JNJ-63576253, a Next-Generation Androgen Receptor Antagonist Active Against Wild-Type and Clinically Relevant Ligand Binding Domain Mutations in Metastatic Castration-Resistant Prostate Cancer
    Jonathan R. Branch, Tammy L. Bush, Vineet Pande, Peter J. Connolly, Zhuming Zhang, Ian Hickson, Janine Ondrus, Steffen Jaensch, James Robert Bischoff, Georges Habineza et al. · 2023
  39. Regulação do promotor SMyHC3 pelos receptores nucleares GR e COUP-TFII
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  40. Drug Repurposing Patent Applications: April–June 2024
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  41. Androgenrezeptor in Gesundheit und Krankheit
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  42. Tracking Transcription Factors on the Genome by their DNase-seq Footprints
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  43. Role of Underutilized Plant-Derived Metal Oxide-Based Nanoparticles Against Prostate Cancer
    Nidhi Bhardwaj, Indu Bhardwaj, Kanika Dulta, Eugenie Nepovimová, Kamil Kuča, Monika Choudhary, Parteek Mandyal, Ambika Choudhary, Lukas Peter · 2026 · Springer eBooks
  44. BindingDB Entry 50013848: Discovery of JNJ-63576253: A Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC).
    BindingDB · 2022 · UC San Diego