Renslo, Adam R.

USP7 small-molecule inhibitors interfere with ubiquitin binding.

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Genetic and Neural Mechanisms that Inhibit Drosophila from Mating with Other Species

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Divergent modes of enzyme inhibition in a homologous structure-activity series.

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Ferrous iron–activatable drug conjugate achieves potent MAPK blockade in KRAS -driven tumors

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Dietary cholesterol activates a Ral-dependent pathway driving LDLR turnover

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