The DOI matches its Crossref record; 7 of the 7 references it cites were found in a registry or an index.
Direct Synthesis of Fluorinated Heteroarylether Bioisosteres
Open accessAbstract
(Bioiso)steering in a new direction: A modular synthesis of reagents (e.g. sodium difluoroethylsulfinate) that can be used for the direct incorporation of difluoroalkyl groups onto heterocycles is reported. The scope and generality of the incorporation of difluoroalkyl groups is exemplified with the difluoroethyl group and a proof of principle is shown for a general synthesis of fluorinated heteroarylether bioisosteres.
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Cites
Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design
Meanwell, N. A. (2011) · Journal of Medicinal Chemistry · doi:10.1021/jm1013693 · Cited by 2,854
Practical and innate carbon–hydrogen functionalization of heterocycles
Fujiwara, Y., Dixon, J. A., O’Hara, F., Funder, E. D., Dixon, D. D., Rodriguez, R. A., Baxter, R. D., Herlé, B., Sach, N., Collins, M. R., et al. (2012) · Nature · doi:10.1038/nature11680 · Cited by 924
Self-citationInnate C-H trifluoromethylation of heterocycles
Ji, Y., Brueckl, T., Baxter, R. D., Fujiwara, Y., Seiple, I. B., Su, S., Blackmond, D. G., & Baran, P. S. (2011) · Proceedings of the National Academy of Sciences · doi:10.1073/pnas.1109059108 · Cited by 757
Self-citationAiming for the Ideal Synthesis
Gaich, T., & Baran, P. S. (2010) · The Journal of Organic Chemistry · doi:10.1021/jo1006812 · Cited by 647
Self-citationA New Reagent for Direct Difluoromethylation
Fujiwara, Y., Dixon, J. A., Rodriguez, R. A., Baxter, R. D., Dixon, D. D., Collins, M. R., Blackmond, D. G., & Baran, P. S. (2012) · Journal of the American Chemical Society · doi:10.1021/ja211422g · Cited by 630
Self-citationLanglois, B. R., Laurent, E., & Roidot, N. (1991) · Tetrahedron Letters · doi:10.1016/0040-4039(91)80524-a · Cited by 439
Coteron, J. M., Marco, M., Esquivias, J., Deng, X., White, K. L., White, J., Koltun, M., El Mazouni, F., Kokkonda, S., Katneni, K., et al. (2011) · Journal of Medicinal Chemistry · doi:10.1021/jm200592f · Cited by 287
Cited by
Successful fluorine-containing herbicide agrochemicals
Fujiwara, T., & O’Hagan, D. (2014) · Journal of Fluorine Chemistry · doi:10.1016/j.jfluchem.2014.06.014 · Cited by 894
Xia, J.-B., Zhu, C., & Chen, C. (2013) · Journal of the American Chemical Society · doi:10.1021/ja410815u · Cited by 560
Tay, N. E. S., Lehnherr, D., & Rovis, T. (2022) · Chemical Reviews · doi:10.1021/acs.chemrev.1c00384 · Cited by 518
Matsui, J. K., Primer, D. N., & Molander, G. A. (2017) · Chemical Science · doi:10.1039/c7sc00283a · Cited by 284
Chemo- and site-selective derivatizations of natural products enabling biological studies
Robles, O., & Romo, D. (2014) · Nat. Prod. Rep. · doi:10.1039/c3np70087a · Cited by 154
Metadata
- Authors
- Zhou, Q., Ruffoni, A., Gianatassio, R., Fujiwara, Y., Sella, E., Shabat, D., & Baran, P. S.
- Venue
- Angewandte Chemie International Edition
- Publisher
- Wiley
- Published
- 2013-03-04
- Volume
- 52
- Issue
- 14
- Pages
- 3949-3952
- ISSN
- 1433-7851 (ISSN-L)
- 1521-3773
- OpenAlex
- W2108835763
- Cited by
- 256
- References
- 7
- FWCI
- 14.66
- Type
- journal article
- Language
- en
- Open access
- green
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- Zhou, Q., Ruffoni, A., Gianatassio, R., Fujiwara, Y., Sella, E., Shabat, D., & Baran, P. S. (2013). Direct Synthesis of Fluorinated Heteroarylether Bioisosteres. Angewandte Chemie International Edition. https://doi.org/10.1002/anie.201300763
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Contains information from the Semantic Scholar Academic Graph Datasets, made available under the ODC Attribution License (ODC-BY 1.0).
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