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Recent Progress in Chemical Modification of Proteins

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Exocyclic Olefinic Maleimides: Synthesis and Application for Stable and Thiol‐Selective Bioconjugation

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Site-Specific Dual Functionalization of Cysteine Residue in Peptides and Proteins with 2-Azidoacrylates

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Thia-Michael addition: the route to promising opportunities for fast and cysteine-specific modification

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Chemical modifications of proteins and their applications in metalloenzyme studies

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Irreversible Cysteine‐Selective Protein Labeling Employing Modular Electrophilic Tetrafluoroethylation Reagents

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Highly Reactive and Tracelessly Cleavable Cysteine‐Specific Modification of Proteins via 4‐Substituted Cyclopentenone

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Site‐Selective Modification of Peptides and Proteins via Interception of Free‐Radical‐Mediated Dechalcogenation

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Silicon-Containing Thiol-Specific Bioconjugating Reagent

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Allene Functionalized Azobenzene Linker Enables Rapid and Light-Responsive Peptide Macrocyclization

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Development and Applications of Water-Compatible Reactions: A Journey to Be Continued

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Peptide and Protein Cysteine Modification Enabled by Hydrosulfuration of Ynamide

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Alkynone β-trifluoroborates: A new class of amine-specific biocompatible click reagents

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Thiol‐Specific Silicon‐Containing Conjugating Reagent: β‐Silyl Alkynyl Carbonyl Compounds

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Computational Study of the Addition of Methanethiol to 40+ Michael Acceptors as a Model for the Bioconjugation of Cysteines

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A Plug-and-Play Platform for the Formation of Trifunctional Cysteine Bioconjugates that also Offers Control over Thiol Cleavability

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Site-Selective Modification of Peptides via Late-Stage Pd-Catalyzed Tandem Reaction of Phenylalanine with Benzoquinone

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Catalyst-free C–N bond formation under biocompatible reaction conditions

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Modified synthetic peptides: from therapeutics to chemosensors

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Photo‐and Electrochemical Modification of Amino Acids, Peptides and Proteins through Cysteine: Recent Advances and Future Perspectives

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Dichloroacetophenone Derivatives: A Class of Bioconjugation Reagents for Disulfide Bridging

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Rapid C–S Coupling in Water via Ion-Pair-Catalyzed Dehydration

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Exocyclic Olefinic Maleimides: Synthesis and Application for Stable and Thiol‐Selective Bioconjugation

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Modulation of protein activity and assembled structure by polymer conjugation: PEGylation vs glycosylation

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Interactive Bioconjugation at N‐Terminal Cysteines by Using O‐Salicylaldehyde Esters towards Dual Site‐Selective Functionalization

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Recent Advances in Chemical Protein Modification via Cysteine

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Allenamides as a Powerful Tool to Incorporate Diversity: Thia‐Michael Lipidation of Semisynthetic Peptides and Access to β‐Keto Amides

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