The N‐Acylethanolamine‐Hydrolyzing Acid Amidase (NAAA)

Tsuboi, Kazuhito, Takezaki, Naoko, Ueda, Natsuo·2007·Chemistry & Biodiversity
DOI 10.1002/cbdv.200790159

Cited by (185)

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  28. Synthesis and Preliminary Evaluation of N-(16-18F-Fluorohexadecanoyl)ethanolamine (18F-FHEA) as a PET Probe of N-Acylethanolamine Metabolism in Mouse Brain
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  72. BindingDB Entry 50030672: beta-Lactams derived from a carbapenem chiron are selective inhibitors of human fatty acid amide hydrolase versus human monoacylglycerol lipase.
    BindingDB · 2010 · UC San Diego
  73. BindingDB Entry 50039848: Lipophilic amines as potent inhibitors of N-acylethanolamine-hydrolyzing acid amidase.
    BindingDB · 2013 · UC San Diego
  74. BindingDB Entry 50014558: Discovery and SAR Evolution of Pyrazole Azabicyclo[3.2.1]octane Sulfonamides as a Novel Class of Non-Covalent
    BindingDB · 2022 · UC San Diego
  75. BindingDB Entry 50041828: Synthesis and structure-activity relationships of N-(2-oxo-3-oxetanyl)amides as N-acylethanolamine-hydrolyzing acid amidase inhibitors.
    BindingDB · 2013 · UC San Diego
  76. BindingDB Entry 50010439: Design and synthesis of cyanamides as potent and selective N-acylethanolamine acid amidase inhibitors.
    BindingDB · 2021 · UC San Diego
  77. BindingDB Entry 50040134: ß-Lactones Inhibit N-acylethanolamine Acid Amidase by S-Acylation of the Catalytic N-Terminal Cysteine.
    BindingDB · 2013 · UC San Diego
  78. BindingDB Entry 50014428: Design and Structure-Activity Relationships of Isothiocyanates as Potent and Selective
    BindingDB · 2022 · UC San Diego
  79. BindingDB Entry 50045459: Novel tail and head group prostamide probes.
    BindingDB · 2016 · UC San Diego
  80. BindingDB Entry 50047146: Potenta-amino-ß-lactam carbamic acid ester as NAAA inhibitors. Synthesis and structure-activity relationship (SAR) studies.
    BindingDB · 2017 · UC San Diego
  81. BindingDB Entry 50043348: Synthesis and structure-activity relationship (SAR) of 2-methyl-4-oxo-3-oxetanylcarbamic acid esters, a class of potent N-acylethanolamine acid amidase (NAAA) inhibitors.
    BindingDB · 2014 · UC San Diego
  82. BindingDB Entry 50001937: Therapeutic Potential of Fatty Acid Amide Hydrolase, Monoacylglycerol Lipase, and N-Acylethanolamine Acid Amidase Inhibitors.
    BindingDB · 2020 · UC San Diego
  83. BindingDB Entry 50044840: Synthesis, biological evaluation, and 3D QSAR study of 2-methyl-4-oxo-3-oxetanylcarbamic acid esters as N-acylethanolamine acid amidase (NAAA) inhibitors.
    BindingDB · 2016 · UC San Diego
  84. BindingDB Entry 50040090: N-(2-oxo-3-oxetanyl)carbamic acid esters as N-acylethanolamine acid amidase inhibitors: synthesis and structure-activity and structure-property relationships.
    BindingDB · 2013 · UC San Diego
  85. BindingDB Entry 50049118: Progress in the development ofß-lactams as N-Acylethanolamine Acid Amidase (NAAA) inhibitors: Synthesis and SAR study of new, potent N-O-substituted derivatives.
    BindingDB · 2019 · UC San Diego