Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY‐876

Siebeneicher, Holger, Cleve, Arwed, Rehwinkel, Hartmut, Neuhaus, Roland, Heisler, Iring, Müller, Thomas, Bauser, Marcus, Buchmann, Bernd·2016·ChemMedChem

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  89. BindingDB Entry 50018672: Discovery and Characterization of the Potent and Highly Selective 1,7-Naphthyridine-Based Inhibitors BAY-091 and BAY-297 of the Kinase PIP4K2A.
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  90. BindingDB Entry 50022625: Ovarian Cancer Relies on Glucose Transporter 1 to Fuel Glycolysis and Growth: Anti-Tumor Activity of BAY-876.
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  91. BindingDB Entry 50015393: Identification of the Highly Active, Species Cross-Reactive Complex I Inhibitor BAY-179.
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  92. BindingDB Entry 50019765: Target Separation and Potential Anticancer Activity of Withanolide-Based Glucose Transporter Protein 1 Inhibitors from
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  93. BindingDB Entry 50007948: The Druggability of Solute Carriers.
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  95. BindingDB Entry 50010394: Discovery and Optimization of Glucose Uptake Inhibitors.
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  96. BindingDB Entry 50008525: Discovery of BAY-985, a Highly Selective TBK1/IKKε Inhibitor.
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  97. BindingDB Entry 50023044: Recent Progress in the Development of Glucose Transporter (GLUT) Inhibitors.
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