PKM2 Phosphorylates Histone H3 and Promotes Gene Transcription and Tumorigenesis

Yang, Weiwei, Xia, Yan, Hawke, David, Li, Xinjian, Liang, Ji, Xing, Dongming, Aldape, Kenneth, Hunter, Tony +2 more·2012·Cell

Cited by (849)

Items 501–600 of 849

  1. Diabetes and PKM2 affect prognosis in patients with intrahepatic cholangiocarcinoma
    Kui Fu, Xiaoli Yang, Hao Wu, Jianping Gong, Xiuyun Li · 2020 · Oncology Letters
  2. Discovery of Functional Alternatively Spliced PKM Transcripts in Human Cancers
    Xiangyü Li, Cheng Zhang, Woonghee Kim, Muhammad Arif, Chunxia Gao, Andreas Hober, David Kotol, Linnéa Strandberg, Björn Forsström, Åsa Sivertsson et al. · 2021 · Cancers
  3. Interplay Between Glucose Metabolism and Chromatin Modifications in Cancer
    Rui Ma, Yinsheng Wu, Shanshan Li, Xilan Yu · 2021 · Frontiers in Cell and Developmental Biology
  4. Pyruvate Kinase M2: A Potential Regulator of Cardiac Injury Through Glycolytic and Non-glycolytic Pathways
    Chenxin Zeng, Jiangfeng Wu, Jun-ming Li · 2024 · Journal of Cardiovascular Pharmacology
  5. Nuclear-localized pyruvate kinases control phosphorylation of histone H3 on threonine 11
    Pengcheng Hu, Yanmei Xu, Yanhua Su, Yuxin Wang, Yan Xiong, Yong Ding · 2024 · Nature Plants
  6. Polychlorinated biphenyls promote cell survival through pyruvate kinase M2-dependent glycolysis in HeLa cells
    Yuting Zhang, Li Juan Song, Zhuoyu Li · 2019 · Toxicology Mechanisms and Methods
  7. Proteins moonlighting in tumor metabolism and epigenetics
    Lei Lv, Qun‐Ying Lei · 2021 · Frontiers of Medicine
  8. Non-metabolic enzyme function of PKM2 in hepatocellular carcinoma: A review
    Shuangxia Zhang, Zhang‐Xiu Liao, Shubo Li, Ying Luo · 2023 · Medicine
  9. PP4R1 promotes glycolysis and gallbladder cancer progression through facilitating ERK1/2 mediated PKM2 nuclear translocation
    Zhiqiang He, Yuhan Zhong, Tian‐Run Lv, Jun-Ke Wang, Yanwen Jin, Fu‐Yu Li, Hai‐Jie Hu · 2024 · Cancer Letters
  10. PKM2 regulates Gli1 expression in hepatocellular carcinoma
    Qiuran Xu, Xin Liu, Xin Min Zheng, Yingmin Yao, Qingguang Liu · 2014 · Oncology Letters
  11. Regulators of carcinogenesis: Emerging roles beyond their primary functions
    Lintao Jia, Rui Zhang, Lan Shen, Angang Yang · 2014 · Cancer Letters
  12. Compartmentation of Metabolites in Regulating Epigenomes of Cancer
    Zhiqiang Zhao, Li Wang, Lijun Di · 2016 · Molecular Medicine
  13. Protein kinase CK2 modulation of pyruvate kinase M isoforms augments the Warburg effect in cancer cells
    Kyung Mi Yang, Kunhong Kim · 2018 · Journal of Cellular Biochemistry
  14. Phenotypic selection with an intrabody library reveals an anti-apoptotic function of PKM2 requiring Mitofusin-1
    Tong Liu, Tomomi Kuwana, Hongkai Zhang, Matthew G. Vander Heiden, Richard Alan Lerner, Donald D. Newmeyer · 2019 · PLoS Biology
  15. Heat shock protein 90 relieves heat stress damage of myocardial cells by regulating Akt and PKM2 signaling in�vivo
    Xiaohui Zhang, Jiaxin Wu, Junzhou Sha, Bo Yang, Jia‑Rui Sun, Endong Bao · 2020 · International Journal of Molecular Medicine
  16. CircMYOF triggers progression and facilitates glycolysis via the VEGFA/PI3K/AKT axis by absorbing miR-4739 in pancreatic ductal adenocarcinoma
    Dandan Zheng, Xianxian Huang, Juanfei Peng, Yanyan Zhuang, Yuanhua Li, Junchi Qu, Shineng Zhang, Fengting Huang · 2021 · Cell Death Discovery
  17. Alteration in glycolytic/cholesterogenic gene expression is associated with bladder cancer prognosis and immune cell infiltration
    Yuying Zhang, Baoyi Zhu, Yi Cai, Sihua Zhu, Hongjun Zhao, Xiaoling Ying, Chonghe Jiang, Jianwen Zeng · 2022 · BMC Cancer
  18. Mechanisms of gene regulation by histone degradation in adaptation of yeast: an overview of recent advances
    Safir Ullah Khan, Munir Ullah Khan, Fadia Kalsoom, Muhammad Imran Khan, Shuang Gao, Ahsanullah Unar, Muhammad Zubair, Muhammad Bilal · 2022 · Archives of Microbiology
  19. A moonlighting function of choline kinase alpha 2 in the initiation of lipid droplet lipolysis in cancer cells
    Qingxia Ma, Zhaoyuan Meng, Ying Meng, Rui Liu, Zhimin Lu · 2021 · 癌症:英文版
  20. Aurora A–mediated pyruvate kinase M2 phosphorylation promotes biosynthesis with glycolytic metabolites and tumor cell cycle progression
    Ya Ping Jiang, Ting Wang, Dandan Sheng, Chaoqiang Han, Xu Tian, Peng Zhang, Weiyi You, Weiwei Fan, Zhiyong Zhang, Tengchuan Jin et al. · 2022 · Journal of Biological Chemistry
  21. Depletion of pyruvate kinase (PK) activity causes glycolytic intermediate imbalances and reveals a PK-TXNIP regulatory axis
    Anna Nieborak, Saulius Lukauskas, Jordi Capellades, Patricia Cristine Heyn, Gabriela S. Silva Santos, Karsten Motzler, Anja Zeigerer, Romina Bester, Ulrike Protzer, Florian Schelter et al. · 2023 · Molecular Metabolism
  22. Epigenetic-based combination therapy and liposomal codelivery overcomes osimertinib-resistant NSCLC via repolarizing tumor-associated macrophages
    Tingting Lin, Wei Xiong, Guihua Chen, Yang He, Long Li, Xinfu Gao, Jialin Zhou, Wen-wen Lv, Yongzhuo Huang · 2023 · Acta Pharmacologica Sinica
  23. Redox proteomics screening cellular factors associated with oxidative stress in hepatocarcinogenesis
    Li Zhou, Wen Ji, Zhao Huang, Edouard Collins Nice, Canhua Huang, Haiyuan Zhang, Qifu Li · 2016 · PROTEOMICS - CLINICAL APPLICATIONS
  24. Anaplerosis in cancer: Another step beyond the warburg effect
    Estefanía Ochoa-Ruiz, Rodrigo Díaz-Ruiz · 2012 · American Journal of Molecular Biology
  25. PKM2 enhances cancer invasion via ETS-1-dependent induction of matrix metalloproteinase in oral squamous cell carcinoma cells
    Young-Jin Park, Jue Young Kim, Doo Young Lee, Xianglan Zhang, Shadavlonjid Bazarsad, Won‐Yoon Chung, Jin Kim · 2019 · PLoS ONE
  26. Sirtuin 6 and metabolic genes interplay in Warburg effect in cancers
    Nosayba Zakariya Al‐Azzam · 2020 · Journal of Clinical Biochemistry and Nutrition
  27. Induction of Apoptosis in Human Leukemic Cell Lines by Diallyl Disulfide via Modulation of EGFR/ERK/PKM2 Signaling Pathways
    Nian Luo, Lv-Cui Zhao, Qing-Qiang Shi, Zi-Qiang Feng, Dilong Chen, Jing Li · 2015 · Asian Pacific Journal of Cancer Prevention
  28. Metabolic enzymes function as epigenetic modulators: A Trojan Horse for chromatin regulation and gene expression
    Xiaoyu Liao, Yifan Guo, Yumin He, Yanxuan Xiao, Jingyi Li, Rui Liu · 2021 · Pharmacological Research
  29. MiR-218-5p/EGFR Signaling in Arsenic-Induced Carcinogenesis
    Ranakul Islam, Lei Zhao, Xiujuan Zhang, L.-Z. Liu · 2023 · Cancers
  30. Targeting PKM2 improves the gemcitabine sensitivity of intrahepatic cholangiocarcinoma cells via inhibiting β-catenin signaling pathway
    Wenna Yu, Fuling Zeng, Yang Xiao, Liuyan Chen, Hengdong Qu, Jian Hong, Chen Qu, Guohua Cheng · 2023 · Chemico-Biological Interactions
  31. Chromatin balances cell redox and energy homeostasis
    Tamaki Suganuma, Jerry L. Workman · 2023 · Epigenetics & Chromatin
  32. Computer‐aided identification of a novel pyruvate kinase M2 activator compound
    Yuanyuan Li, Minyue Bao, Chunlan Yang, Jiao Chen, Shu Wen Zhou, Rong Sun, Chuanfang Wu, Xin Li, Jinku Bao · 2018 · Cell Proliferation
  33. Yeast Nuak1 phosphorylates histone H3 threonine 11 in low glucose stress by the cooperation of AMPK and CK2 signaling
    Seunghee Oh, Jaehyoun Lee, Selene K. Swanson, Laurence A. Florens, Michael P. Washburn, Jerry L. Workman · 2020 · eLife
  34. Ferroxitosis: A cell death from modulation of oxidative phosphorylation and PKM2-dependent glycolysis in melanoma
    Alexander J. Lakhter, James Hamilton, Pierre C. Dagher, Suresh Mukkamala, Takashi Hato, Xiaocheng Charlie Dong, Lindsey D. Mayo, Robert A. Harris, Anantha Shekhar, Mircea Ivan et al. · 2014 · Oncotarget
  35. Non-Metabolic Role of PKM2 in Regulation of the HIV-1 LTR
    Satarupa Sen, Satish L. Deshmane, Rafal Kaminski, Shohreh Amini, Prasun K. Datta · 2016 · Journal of Cellular Physiology
  36. STEAP4 Inhibits HIF-1α/PKM2 Signaling and Reduces High Glucose-Induced Apoptosis of Retinal Vascular Endothelial Cells
    Lei Liu, Hui Xu, Hongyu Zhao, Chunying Jiang · 2020 · Diabetes Metabolic Syndrome and Obesity
  37. TACC3 enhances glycolysis in bladder cancer cells through inducing acetylation of c-Myc
    Zhi-Rui Lin, Falian Liang, Gengde Hong, Xizhen Jiang, Qingling Zhang, Mengyao Wang · 2025 · Cell Death and Disease
  38. A Review on the Role of Pyruvate Kinase M2 in Cancer: From Metabolic Switch to Transcriptional Regulation
    Zulfareen, Aaliya Taiyab, Gulam Mustafa Hasan, Md. Imtaiyaz Hassan · 2025 · International Journal of Biological Macromolecules
  39. Nuclear PKM2 expression, an independent risk factor for ER after curative resection of hepatocellular carcinoma
    Fangtian Fan, Hongyan Wu, Zhaoguo Liu, Xianbang Hou, Wenxin Chen, Aiyun Wang, Yin Lu · 2016 · Biomedicine & Pharmacotherapy
  40. Potential therapies targeting nuclear metabolic regulation in cancer
    Yanjie Chen, Jie Xu, Xiaoyi Liu, Linlin Guo, Ping Yi, Chunming Cheng · 2023 · MedComm
  41. Neurotoxic effects of triclosan in adolescent mice: Pyruvate kinase M2 dimer regulated Signal transducer and activator of transcription 3 phosphorylation mediated microglia activation and neuroinflammation
    Ziyun Wei, XIAO YAN NI, He Cui, Chang Shu, Yuxuan Peng, Yunwei Li, Jieyu Liu · 2024 · The Science of The Total Environment
  42. Copy number amplification of FLAD1 promotes the progression of triple-negative breast cancer through lipid metabolism
    Xiao-Qing Song, Tian‐Jian Yu, Yang Ou-Yang, Jia-Han Ding, Yi‐Zhou Jiang, Zhi‐Ming Shao, Yi Xiao · 2025 · Nature Communications
  43. The glycolytic enzyme PKM2 regulates inflammatory osteoclastogenesis by modulating STAT3 phosphorylation
    Mingjuan Li, Feng Li, Chongjie Zhu, Chi Zhang, Yushi Le, Zubing Li, Qilong Wan · 2025 · Journal of Biological Chemistry
  44. Nuclear functional role of metabolic enzymes and related metabolites: Focus on gene expression regulation
    Simona Todisco, Dominga Iacobazzi, Anna Santarsiero, Paolo Convertini, Vittoria Infantino · 2025 · Molecular Metabolism
  45. C‐MET–dependent signal transduction mediates retinoblastoma growth by regulating PKM2 nuclear translocation
    Hanjun Dai, Weijuan Zeng, Hong Luo · 2019 · Cell Biochemistry and Function
  46. Cell-Free Circulating Epimarks in Cancer Monitoring
    Manon Duforestel, Joséphine Briand, Gwenola Bougras-Cartron, Dominique Heymann, Jean‐Sébastien Frenel, François M. Vallette, Pierre‐François Cartron · 2020 · Epigenomics
  47. SLC7A11 negatively associates with mismatch repair gene expression and endows glioblastoma cells sensitive to radiation under low glucose conditions
    Nan Hu, Weihua Hu, Shaolong Zhou, Zhuo Yang, Wulong Liang, Ruyi Yang, Minghe Li, Zhou Jing, Zian Li, Xudong Fu et al. · 2021 · Neoplasma
  48. RIOX1-demethylated cGAS regulates ionizing radiation-elicited DNA repair
    Yanxuan Xiao, Jingyi Li, Xiaoyu Liao, Yumin He, Tao He, Cuiping Yang, Lu Jiang, So Mi Jeon, Jong-Ho Lee, Yongbin Chen et al. · 2022 · Bone Research
  49. Metabolic Reprogramming in Melanoma: An Epigenetic Point of View
    Sandro Giuliani, Celeste Accetta, Simona Di Martino, Claudia De Vitis, Elena Messina, Edoardo O. Pescarmona, Maurizio Fanciulli, Gennaro Ciliberto, Rita Mancini, Italia Falcone · 2025 · Pharmaceuticals
  50. PKM2 Interacts With the Cdk1-CyclinB Complex to Facilitate Cell Cycle Progression in Gliomas
    Shigeo Ohba, Yongjian Tang, Tor-Christian Aase Johannessen, Joydeep Mukherjee · 2022 · Frontiers in Oncology
  51. Glycolytic Pfkp acts as a Lin41 protein kinase to promote endodermal differentiation of embryonic stem cells
    Leixi Cao, Ruijie Wang, Guangzhi Liu, Yuwei Zhang, Rick Francis Thorne, Xu Dong Zhang, Jinming Li, Yang Xia, Lili Guo, Fengmin Shao et al. · 2023 · EMBO Reports
  52. Muscle‐specific pyruvate kinase isoforms, PKM1 and PKM2 , regulate mammalian SWI / SNF proteins and histone 3 phosphorylation during myoblast differentiation
    Monserrat Olea‐Flores, Tapan Sharma, Odette Verdejo‐Torres, Imaru DiBartolomeo, Paul R. Thompson, Teresita Padilla‐Benavides, Anthony N. Imbalzano · 2024 · The FASEB Journal
  53. A new strategy for overcoming drug resistance in liver cancer: Epigenetic regulation
    Xiaorui Su, Yuxuan Li, Yupeng Ren, Mingbo Cao, Gaoyuan Yang, Jing Luo, Ziyi Hu, Haixia Deng, Meihai Deng, Bo Liu et al. · 2024 · Biomedicine & Pharmacotherapy
  54. Extracellular PKM2 modulates cancer immunity by regulating macrophage polarity
    Guangda Peng, Bin Li, Hongwei Han, Yi Yuan, Falguni Mishra, Yang Huang, Zhi‐Ren Liu · 2025 · Cancer Immunology Immunotherapy
  55. Targeting the interplay between metabolism and epigenetics in cancer
    Emilie Montellier, Jonathan Gaucher · 2018 · Current Opinion in Oncology
  56. Suppressed “Warburg Effect” in Nasopharyngeal Carcinoma Via the Inhibition of Pyruvate Kinase Type M2-Mediated Energy Generation Pathway
    Penglong Zhao, Mengyan Zhou, Ruixiang Chen, Renjie Su · 2020 · Technology in Cancer Research & Treatment
  57. Opposed Interplay between IDH1 Mutations and the WNT/β-Catenin Pathway: Added Information for Glioma Classification
    Alexandre Vallée, Yves Lecarpentier, Jean-Noël Vallée · 2021 · Biomedicines
  58. Pyruvate Kinase M2 Supports Muscle Progenitor Cell Proliferation but Is Dispensable for Skeletal Muscle Regeneration after Injury
    Jamie Blum, Brandon J.F. Gheller, Abigail M. Benvie, Martha S. Field, Elena Panizza, Nathaniel M. Vacanti, Daniel C. Berry, Anna Elizabeth Thalacker‐Mercer · 2021 · Journal of Nutrition
  59. MYC regulates metabolism through vesicular transfer of glycolytic kinases
    Alexia Tsakaneli, V. Carregari, Martina Morini, A. Eva, G. Cangemi, O. Chayka, E. Makarov, Sandra Bibbò, E. Capone, G. Sala et al. · 2021 · Open Biology
  60. Pyruvate Dehydrogenase A1 Phosphorylated by Insulin Associates with Pyruvate Kinase M2 and Induces LINC00273 through Histone Acetylation
    Abu Jubayer Hossain, Rokibul Islam, Jae-Gyu Kim, Oyungerel Dogsom, Kim Cuong Cap, Jae‐Bong Park · 2022 · Biomedicines
  61. FA-SAT ncRNA interacts with PKM2 protein: depletion of this complex induces a switch from cell proliferation to apoptosis
    Daniela Ferreira, Ana Escudeiro, Filomena Adega, Sandra Isabel Anjo, Bruno J. Manadas, Raquel Chaves · 2019 · Cellular and Molecular Life Sciences
  62. PCAF regulates H3 phosphorylation and promotes autophagy in osteosarcoma cells
    Daliang Kong, Boda Ying, Jinrui Zhang, Hongliang Ying · 2019 · Biomedicine & Pharmacotherapy
  63. Pyruvate kinase M2-mediated histone lactylation alters three-dimensional genomic architecture in polycystic ovary syndrome
    Chuanjin Yu, Tingting Liu, Yishu Wang, Xinghui Guo, Yujie Chen, Yifan Zhao, Xia Liu, Weiwei Huang, Shuoyang Zhao, Jiaying Mo et al. · 2025 · Signal Transduction and Targeted Therapy
  64. Calcium Channel α2δ1 is Essential for Pancreatic Tumor-Initiating Cells through Sequential Phosphorylation of PKM2
    Jianwen Liu, Ming Tao, Wei Zhao, Qingru Song, Xiaodan Yang, Meng Li, Yanhua Zhang, Dianrong Xiu, Zhiqian Zhang · 2022 · Cellular and Molecular Gastroenterology and Hepatology
  65. Cardioprotective potential of compound 3K, a selective PKM2 inhibitor in isoproterenol-induced acute myocardial infarction: A mechanistic study
    Mohd Rihan, Shyam Sunder Sharma · 2024 · Toxicology and Applied Pharmacology
  66. Hexokinase 2 nonmetabolic function‐mediated phosphorylation of IκBα enhances pancreatic ductal adenocarcinoma progression
    Yingying Tong, Xin Liu, Lihui Wu, yaoxian Xiang, Jing Wang, Yurong Cheng, Chan Zhang, Baojuan Han, Li Wang, Dong Yan · 2024 · Cancer Science
  67. CHAC1 blockade suppresses progression of lung adenocarcinoma by interfering with glucose metabolism via hijacking PKM2 nuclear translocation
    Junfan Pan, Sixuan Wu, Qihong Pan, Yuan Zhang, He Liu, Qiwei Yao, Jin-Yuan Chen, Jiancheng Li, Yiquan Xu · 2024 · Cell Death and Disease
  68. ERK–USP9X-coupled regulation of thymidine kinase 1 promotes both its enzyme activity-dependent and its enzyme activity-independent functions for tumor growth
    Jingjing Tao, Zheng Wang, Rongkai Shi, Liming Lin, Min Li, Ying Meng, Shudi Luo, Xiaoming Jiang, Zhanpeng Guo, Yongfeng Shang et al. · 2025 · Nature Structural & Molecular Biology
  69. Glucose restriction reverses the Warburg effect and modulates PKM2 and mTOR expression in breast cancer cell lines
    Roula Tahtouh, Layal Wardi, Riad Sarkis, Ray Y Hachem, ISSAM I. RAAD, Nabil El Zein, George Hilal · 2019 · Cellular and Molecular Biology
  70. Cerulenin suppresses ErbB2-overexpressing breast cancer by targeting ErbB2/PKM2 pathway
    Sinan Lv, Yun‐wu Zhang, Jiawei Song, Jingruo Chen, Bohan Huang, Yuhan Luo, Yuhua Zhao · 2022 · Medical Oncology
  71. mTOR activation is critical for betulin treatment in renal cell carcinoma cells
    Wenlong Cheng, Shiqi Ji, Haijian Zhang, Zhixing Han, Qingjun Liu, Jianwen Wang, Hao Ping · 2016 · Biochemical and Biophysical Research Communications
  72. Power of screening tests for colorectal cancer enhanced by high levels of M2-PK in addition to FOBT
    Cristina Zaccaro, Ilaria Maria Saracino, Giulia Fiorini, Natale Figura, John Holton, Valentina Castelli, Valeria Pesci, Luigi Gatta, D. Vaira · 2017 · Internal and Emergency Medicine
  73. Classification of clear cell renal cell carcinoma based on PKM alternative splicing
    Xiangyü Li, Beste Turanlı, Kajetan Juszczak, Woonghee Kim, Muhammad Arif, Yusuke Sato, Seishi Ogawa, Hasan Türkez, Jens Nielsen, Jan Borén et al. · 2020 · Heliyon
  74. Nucleus-located PDK1 regulates growth, invasion and migration of breast cancer cells
    Delu Gan, Shujun Yue, Yulin Jiang, Dian Zhang, He Shi, Husun Qian, Ting Zhou, Wenli Fang, Mengli Yao, Guowei Zuo et al. · 2020 · Life Sciences
  75. Therapeutic Approach of KRAS Mutant Tumours by the Combination of Pharmacologic Ascorbate and Chloroquine
    Orsolya Kapuy, Kinga Makk‐Merczel, András Szarka · 2021 · Biomolecules
  76. Shikonin alleviates choroidal neovascularization by inhibiting proangiogenic factor production from infiltrating macrophages
    Ying Wang, Laiqing Xie, Manhui Zhu, Yang Guo, Yuanyuan Tu, Yamei Zhou, Jia Zeng, Linling Zhu, Shu Du, Zhenzhen Wang et al. · 2021 · Experimental Eye Research
  77. Structural characterization and anti-hepatic fibrosis effects of a novel polysaccharide from Astragalus complanatus seeds.
    Zhi-Fan Zhu, Shuyao Wang, Xiao-Feng Liu, Na Liu, Dianchao Dong, Yan-Chun Qi, Na Li, Nan Wang, Jin Tan, Chang Jia et al. · 2025 · Carbohydrate Polymers
  78. Association of serum levels of antibodies against ALDOA and FH4 with transient ischemic attack and cerebral infarction
    Hao Wang, Hao Lu, Xiao-Meng Zhang, Ken-ichiro Goto, Eiichi Kobayashi, Yoichi Yoshida, Akihiko Adachi, Tomoo Matsutani, Yasuo Iwadate, Seiichiro Mine et al. · 2021 · BMC Neurology
  79. Metabolic Rewiring in Adult-Type Diffuse Gliomas
    Jong‐Whi Park · 2023 · International Journal of Molecular Sciences
  80. Glycolytic enzymes in non-glycolytic web: functional analysis of the key players
    Avirup Malla, Suvroma Gupta, Runa Sur · 2024 · Cell Biochemistry and Biophysics
  81. The role of fructose-1,6-bisphosphatase 1 on regulating the cancer progression and drug resistance
    Mengmeng Wang, Xiaoju Huang, Dan Zhang, Yisan Liu, Pian Liu · 2025 · Discover Oncology
  82. Transcriptional Networks Identify BRPF1 as a Potential Drug Target Based on Inflammatory Signature in Primary Lower-Grade Gliomas
    Mingyang Xia, Huiyao Chen, Tong Chen, Ping Xue, Xinran Dong, Yifeng Lin, Duan Ma, Wenhao Zhou, Wei Shi, Hao Li · 2021 · Frontiers in Oncology
  83. Crosstalk of Epigenetic and Metabolic Signaling Underpinning Glioblastoma Pathogenesis
    Mariam Markouli, Dimitrios Strepkos, Kostas A. Papavassiliou, Athanasios G. Papavassiliou, Christina Piperi · 2022 · Cancers
  84. Pyruvate kinase M2 sustains cardiac mitochondrial quality surveillance in septic cardiomyopathy by regulating prohibitin 2 abundance via S91 phosphorylation
    Yingzhen Du, Jialei Li, Zhe Dai, Yuxin Chen, Yao Zhao, Xiaoman Liu, Tian Xia, Pingjun Zhu, Y Q Wang · 2024 · Cellular and Molecular Life Sciences
  85. Pyruvate kinase M2 represses thermogenic gene expression in brown adipocytes
    Marie Sophie Isidor, Sally Winther, Lasse Kruse Markussen, Astrid Linde Basse, Bjørn Quistorff, Jan Nedergaard, Brice Emanuelli, Jacob Bo Hansen · 2019 · FEBS Letters
  86. Base editing‐mediated perturbation of endogenous PKM1/2 splicing facilitates isoform‐specific functional analysis in vitro and in vivo
    Jianxiang Lin, Susu Wu, Qingmei Shen, Jie Liu, Shisheng Huang, Guangdun Peng, Yunbo Qiao · 2021 · Cell Proliferation
  87. Nucleus-translocated glucokinase functions as a protein kinase to phosphorylate TAZ and promote tumour growth
    Gaoxiang Zhao, Shudi Luo, Hong Chuan Zhao, Qingxia Ma, Hongfei Jiang, Lin Wang, Juanjuan Liu, Dong Sheng Guo, Runze Wang, Qianqian Xu et al. · 2025 · Nature Communications
  88. Hypoxic microenvironment-induced exosomes confer temozolomide resistance in glioma through transfer of pyruvate kinase M2
    Guo‐Fu Li, Ziyu Xiong, Ying Li, Cong Yan, Yingying Cheng, Yuwen Wang, Jingwei Li, Zifeng Dai, Dongdong Zhang, Wenzhong Du et al. · 2024 · Discover Oncology
  89. Tumor Metabolism: A New Field for the Treatment of Glioma
    Xiaoqian Chai, Yingjie Zhang, Wen Zhang, Kuanhan Feng, Yingyu Jiang, Anran Zhu, Xiaojin Chen, Liuqing Di, Ruoning Wang · 2024 · Bioconjugate Chemistry
  90. Defining a Correlative Transcriptional Signature Associated with Bulk Histone H3 Acetylation Levels in Adult Glioblastomas
    Irati Hervás-Corpión, Jorge Navarro-Calvo, Paula Martín-Climent, Marianela Iriarte‐Gahete, Noelia Geribaldi‐Doldán, Carmen Castro, Luis Miguel Valor · 2023 · Cells
  91. Glc7/PP1 dephosphorylates histone H3T11 to regulate autophagy and telomere silencing in response to nutrient availability
    Xinyu Zhang, Qi Yu, Yinsheng Wu, Yuan Zhang, Yi He, Rongsha Wang, Xilan Yu, Shanshan Li · 2023 · Cell Discovery
  92. SH2 domain-containing phosphatase 1 regulates pyruvate kinase M2 in hepatocellular carcinoma
    Wei‐Tien Tai, Man‐Hsin Hung, Pei‐Yi Chu, Yao-Li Chen, Li-Ju Chen, Ming-Hsien Tsai, Min-Husan Chen, Chung‐Wai Shiau, Yin-Pin Boo, Kuen‐Feng Chen · 2016 · Oncotarget
  93. A Cell Engineering Strategy to Enhance the Safety of Stem Cell Therapies
    Elisa Oricchio, Eirini P. Papapetrou, Fabien G. Lafaille, Yosif M. Ganat, Sonja Kriks, Ana Ortega-Molina, Willie H. Mark, Julie Teruya‐Feldstein, Jason T. Huse, Victor E. Reuter et al. · 2014 · Cell Reports
  94. Pantothenate Kinase 4 Governs Lens Epithelial Fibrosis by Negatively Regulating Pyruvate Kinase M2-Related Glycolysis
    Xue Li, Linlin Luo, Ruifeng Li, Chun-Lin Chen, Min Sun, Sen Lin · 2023 · Aging and Disease
  95. N6 ‐isopentenyladenosine inhibits aerobic glycolysis in glioblastoma cells by targeting PKM2 expression and activity
    Cristina Pagano, Laura Coppola, Giovanna Navarra, Giorgio Avilia, Beatrice Savarese, Giovanni Torelli, Sara Bruzzaniti, Erica Piemonte, Mario Galgani, Chiara Laezza et al. · 2024 · FEBS Open Bio
  96. Pyruvate Kinase M2‐Responsive Release of Paclitaxel and Indoleamine 2,3‐Dioxygenase Inhibitor for Immuno‐Chemotherapy of Nonsmall Cell Lung Cancer
    Haisi Wu, Xianbao Sun, Kaiming Li, Jinyu Li, Hui Jiang, Dan Yan, Lin Ya, Yan Ding, Yawen Lu, Xiaole Zhu et al. · 2024 · Advanced Science
  97. PKM2-mediated collagen XVII expression is critical for wound repair
    Yangdan Liu, Chiakang Ho, Dongsheng Wen, Jiaming Sun, Yuxin Liu, Q.F. Li, Yifan Zhang, Ya Gao · 2025 · JCI Insight
  98. In Scarcity and Abundance: Metabolic Signals Regulating Cell Growth
    Shady Saad, Matthias Peter, Reinhard Christoph Dechant · 2013 · Physiology
  99. Constitutive androstane receptor activation evokes the expression of glycolytic genes
    Andrei A. Yarushkin, Yuliya A. Kazantseva, Elena A. Prokopyeva, Diana N. Markova, Yuliya A. Pustylnyak, Vladimir O. Pustylnyak · 2016 · Biochemical and Biophysical Research Communications
  100. Chrysophanol inhibits of colorectal cancer cell motility and energy metabolism by targeting the KITENIN/ErbB4 oncogenic complex
    Mücahit Varlı, Eunae Kim, Songjin Oh, Sultan Pulat, Rui Zhou, Chathurika D. B. Gamage, Barış Gökalsın, Nüzhet Cenk Sesal, Kyung Keun Kim, Man‐Jeong Paik et al. · 2024 · Cancer Cell International