How Ligands Illuminate GPCR Molecular Pharmacology

Cited by (568)

Items 501–568 of 568

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  14. Pharmacological actions of commonly used drugs
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  16. Physiology of GPCRs in the nervous system and the contribution of orphan GPCRs
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  17. Insights into the molecular pharmacology of novel aminotetralins and known drug candidates at serotonin 5-HT1-type receptors
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  18. In Vitro Biology: Measuring Pharmacological Activity that Will Translate to Clinical Efficacy
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  19. Endogenous Promotor-Driven Split Nanoluciferase Biosensor for Assessing G Protein Recruitment
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  20. Caracterização dos mecanismos moleculares envolvidos na ligação e sinalização da angiotensina II no receptor AT1
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  24. Post-translational modifications orchestrate the intrinsic signaling bias of orphan receptor GPR52
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  25. Peptidergic G-Protein-Coupled Receptor Signaling Systems in Cancer: Examination of Receptor Structure and Signaling to Foster Innovative Pharmacological Solutions
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  26. Scaled and Weighted Laplacian Matrices as Functional Descriptors for GPCR Ligands
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  41. Méthodes RMN pour la découverte de nouveaux ligands ciblant les récepteurs couplés aux protéines G
    Claire Raingeval · 2019 · theses.fr (ABES)
  42. Analysis of CXCR4 and ACKR3 oligomerisation
    Joyce Heuninck · 2019 · theses.fr (ABES)
  43. Développement et caractérisation d'outils immunologiques dirigés contre des récepteurs membranaires d'intérêt thérapeutique
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  44. Exploiting G protein-coupled receptors : exploring new possibilities for protein-based biosensors
    Simon Harris · 2019 · theses.fr (ABES)
  45. Numerical modeling of olfaction
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  46. Dynamique structurale de complexes RCPG - neuropeptides
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  48. Démonstration de l’existence des récepteurs mGlu7 hétérodimériques par des approches innovantes
    Kawthar Belkacemi · 2024 · theses.fr (ABES)
  49. Improving AlphaFold2 Performance in Virtual Screens Targeting GPCRs by Enhancing Binding-Site Conformational Sampling
    Núria Mitjavila-Domènech, Alejandro Díaz‐Holguín, Huabin Hu, Nour Aldin Kahlous, Israel Cabeza de Vaca, Björn Wallner, Jens Carlsson · 2026 · Journal of Chemical Information and Modeling
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  51. Translating GPCR Movements into Therapeutic Innovations
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  52. GPCR Drug Development from Preclinical Insights to Clinical Applications
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  54. The Dopamine D3 Receptor as an Emerging Therapeutic Target in Parkinson’s Disease: Structural Advances, Signaling Bias and Neuroprotective Perspectives
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  55. Dynamic interactions in GPCR–G protein coupling: Distinguishing specificity and pluripotency
    Aditya Manoj, Durba Sengupta · 2026 · Elsevier eBooks
  56. Regulation of Translation by PKA Signaling Pathway
    Lele Yang, Kun Hou, Huayu Qi · 2026 · International Journal of Molecular Sciences
  57. Ligand-Dependent Affinity but State-Dominated Efficacy in Structure-Based GPCR Pharmacology Prediction
    Jianxiang Huang, Xin Qiao, Chunhao Zhu, Xiaobing Lan, Shaoyong Lu · 2026 · Journal of Medicinal Chemistry
  58. Thermodynamic, Kinetic, and Structural Determinants of Ligand Selectivity in A2A and A2B Adenosine Receptors
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  59. Peptidomimetics in GPCRs: From structural insights to clinical blockbusters
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  60. BindingDB Entry 50017445: The Pursuit of Enzyme Activation: A Snapshot of the Gold Rush.
    BindingDB · 2023 · UC San Diego
  61. BindingDB Entry 50022489: Covalent-Allosteric Inhibitors to Achieve Akt Isoform-Selectivity.
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  62. BindingDB Entry 50008987: D
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  63. BindingDB Entry 50008908: Defining Structure-Functional Selectivity Relationships (SFSR) for a Class of Non-Catechol Dopamine D
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  64. BindingDB Entry 50016203: Discovery of β-Arrestin-Biased 25CN-NBOH-Derived 5-HT
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  65. BindingDB Entry 50006785: Allosteric Modulation of Class A GPCRs: Targets, Agents, and Emerging Concepts.
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  66. BindingDB Entry 50006764: Small Molecule Allosteric Modulators of G-Protein-Coupled Receptors: Drug-Target Interactions.
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  67. BindingDB Entry 50002445: Discovery of β-Arrestin Biased Ligands of 5-HT
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  68. Structural and functional insights into rhodopsin‐like and secretin‐like GPCR –arrestin interactions and regulation
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