The role of ASCT2 in cancer: A review
Liu, Yang, Zhao, Tingli, Li, Zhengzheng, Wang, Lai, Yuan, Shengtao, Sun, Li·2018·European Journal of Pharmacology
Cited by (162)
Items 101–162 of 162
- Asparagine transport through SLC1A5 / ASCT2 and SLC38A5 / SNAT5 is essential for BCP‐ALL cell survival and a potential therapeutic targetGiuseppe Taurino, Erica Dander, Martina Chiu, Giulia Pozzi, Chiara Maccari, Rita Starace, Daniela Silvestri, Erika Griffini, Massimiliano Giovanni Bianchi, Cecilia Carubbi et al. · 2024 · British Journal of Haematology
- Tumor Metabolism: A New Field for the Treatment of GliomaXiaoqian Chai, Yingjie Zhang, Wen Zhang, Kuanhan Feng, Yingyu Jiang, Anran Zhu, Xiaojin Chen, Liuqing Di, Ruoning Wang · 2024 · Bioconjugate Chemistry
- ASCT2 palmitoylation regulated by JNK1-ZDHHC14 axis orchestrates glutamine metabolism and NSCLC progressionXingyu Chen, Zihao Ke, Shihui Wei, Jiajin Chen, Ke Zhu, Jiaqi Xu, Yun Zhao, Mengyuan Cen, Yan Jin, Zhilei Pan et al. · 2026 · Cell Discovery
- Preclinical radiolabeling, in vivo biodistribution and positron emission tomography of a novel pyrrolobenzodiazepine (PBD)-based antibody drug conjugate targeting ASCT2Christian Werner Wichmann, Ingrid J.G. Burvenich, Nancy Yanan Guo, Angela Rigopoulos, Alexander Franklin McDonald, Diana Cao, Graeme Joseph O'Keefe, Sylvia Jie Gong, Hui Kong Gan, Fiona Elizabeth Scott et al. · 2023 · Nuclear Medicine and Biology
- CircCPA4 induces ASCT2 expression to promote tumor property of non‐small cell lung cancer cells in a miR‐145‐5p ‐dependent mannerZhenhua Zhang, Weiliang Liu, Tao Huang, Junyan Li, Hui Hu, Xinyu Xu, Zhigang Fan · 2024 · Thoracic Cancer
- Circular RNA circ-AGFG1 contributes to esophageal squamous cell carcinoma progression and glutamine catabolism by targeting microRNA-497-5p/solute carrier family 1 member 5 axisSiyang Chen, Zhizhen Liu, Qiang Feng, Jin-shan Zhou, Junchao Huang, Jianghao Yu · 2022 · Anti-Cancer Drugs
- SLC1A5 regulates cell proliferation and self-renewal through β-catenin pathway mediated by redox signaling in arsenic-treated uroepithelial cellsSihao Li, Liang Pei, Qing Zhou, Zhushan Fu, Lei Zhang, Pinya Liu, Nan Yan, Shuhua Xi · 2023 · Ecotoxicology and Environmental Safety
- The Synthesis and Biological Applications of the 1,2,3-Dithiazole ScaffoldAndreas S. Kalogirou, Hans J. Oh, Christopher R. M. Asquith · 2023 · Molecules
- LAT1 and ASCT2 Related microRNAs as Potential New Therapeutic Agents against Colorectal Cancer ProgressionFrancisca Dias, Cristina Almeida, Ana Luísa Teixeira, Mariana Morais, Rui Medeiros · 2021 · Biomedicines
- Metabolism and spatial transcription resolved heterogeneity of glutamine metabolism in cervical carcinomaQian Liu, Jiayu Zhu, Guzhalinuer Abulizi, Ayshamgul Hasim · 2024 · BMC Cancer
- Crosstalk of glutamine metabolism between cancer-associated fibroblasts and cancer cellsTingyu Chen, Yiming Xu, Fan Yang, Yanxin Pan, Ning Ji, Jing Li, Xin Ying Zeng, Qianming Chen, Lu Jiang, Yingqiang Shen · 2025 · Cellular Signalling
- Relationships between Slc1a5 and OsteoclastogenesisHideki Tsumura, Miyuki Shindo, Morihiro Ito, Arisa Igarashi, Kazue Takeda, Kenji Matsumoto, Takashi Ohkura, Kenji Miyado, Fumihiro Sugiyama, Akihiro Umezawa et al. · 2021 · Comparative Medicine
- Synthetic oleanane triterpenoid derivative CDDO‐Me disrupts cellular bioenergetics to suppress pancreatic ductal adenocarcinoma via targeting SLC1A5Percy David Papa Akuetteh, Huimin Huang, Shijia Wu, Hongfei Zhou, Guihua Jin, Welong Hong, Hongbao Yang, Linhua Lan, Fugen Shangguan, Qiyu Zhang · 2022 · Journal of Biochemical and Molecular Toxicology
- Design strategies and recent development of bioactive modulators for glutamine transportersXinying Cheng, Yezhi Wang, Guangyue Gong, Pei Shen, Zhiyu Li, Jinlei Bian · 2024 · Drug Discovery Today
- Metabolic reprogramming in the CLL TME; potential for new therapeutic targetsHelga Simon‐Molas, Chiara Montironi, Anna Kabanova, Eric Eldering · 2024 · Seminars in Hematology
- Alanine-serine-cysteine transporter-targeted small-molecule boron carriers for neutron capture therapy of L-4‑boronophenylalanine-refractory tumorsKazuki Miura, Tomoyuki Araki, Taiki Morita, Kai Nishimura, Satoshi Okada, Minoru Suzuki, Hiroyuki Nakamura · 2025 · Journal of Controlled Release
- Phosphoproteomics Analysis Reveals a Pivotal Mechanism Related to Amino Acid Signals in Goat Fetal FibroblastZheng Xu, Su Huimin, Liping Wang, Ruiyuan Yao, Yuze Ma, Linfeng Bai, Yanfeng Wang, Xudong Guo, Zhigang Wang · 2021 · Frontiers in Veterinary Science
- Circular RNA in Non-small Cell Lung Carcinoma: Identification of Targets and New Treatment ModalitiesUlrich H. Weidle, Fabian Birzele · 2023 · Cancer Genomics & Proteomics
- Elucidation and Regulation of Tyrosine Kinase Inhibitor Resistance in Renal Cell Carcinoma Cells from the Perspective of Glutamine MetabolismKento Morozumi, Yoshihide Kawasaki, Tomonori Sato, Masamitsu Maekawa, Shinya Takasaki, Shuichi Shimada, Takanari Sakai, Shinichi Yamashita, Nariyasu Mano, Akihiro Ito · 2024 · Metabolites
- Metabolism of Tryptophan, Glutamine, and Asparagine in Cancer Immunotherapy—Synergism or Mechanism of Resistance?Kajetan Kiełbowski, Estera Bakinowska, Rafał Becht, Andrzej Pawlik · 2025 · Metabolites
- Monoclonal Antibodies Against Myeloid Leukemia Cells: Current Knowledge and Future DirectionsDaniela Damiani, Mario Tiribelli · 2025 · International Journal of Molecular Sciences
- Useful genes for predicting the efficacy of transarterial chemoembolization in hepatocellular carcinomaYuan Guo, Hongtao Hu, Shi‐Jun Xu, Weili Xia, Hai-Liang Li · 2022 · Journal of Cancer Research and Therapeutics
- The Regulation and Function of the Amino Acid Transporters LAT1, ASCT2, xCT in Urological CancersXue Zhao, Shinichi Sakamoto, Shinpei Saito, Sangjon Pae, Yasutaka Yamada, Sanji Kanaoka, Jiaxing Wei, Yusuke Goto, Tomokazu Sazuka, Yusuke Imamura et al. · 2024 · Receptors
- Imaging the uptake and metabolism of glutamine in prostate tumor models using CEST MRIYuki Hodo, Caitlin M. Tressler, Behnaz Ghaemi, Rebecca L. Thomas, Aliyah S. Webster, Kirsten N. Bains Williams, Yuguo Li, Martin G. Pomper, Chi Van Dang, Zaver M. Bhujwalla et al. · 2025 · npj Imaging
- Glu‐derived Zwitterionic Micelles Conquering the Intestinal Mucosal Barrier toward Oral DeliveryKedong Liu, Yun Chen, Dutao Yang, Yanfei Cai, Zhaoqi Yang, Jian Jin · 2023 · ChemNanoMat
- Diseases & Disorders | Therapies Targeting Glutamine Addiction in CancerNabeel Attarwala, Cissy Zhang, Anne Le · 2020 · Elsevier eBooks
- Integrated stress response-upregulated mitochondrial SLC1A5var enhances glucose dependency in human breast cancer cells in vitroSheng‐Fan Wang, Yu-Chieh Ho, Chian‐Ying Chou, Yuh‐Lih Chang, Hsin‐Chen Lee, Ling‐Ming Tseng · 2024 · The International Journal of Biochemistry & Cell Biology
- Biochemical Markers of Tumor Cell Sensitivity to L-AsparaginaseIlya A. Kislyak, Vadim S. Pokrovsky · 2023 · Biochemistry (Moscow) Supplement Series B Biomedical Chemistry
- Deregulated circRNAs in Epithelial Ovarian Cancer With Activity in PreclinicalIn VivoModels: Identification of Targets and New Modalities for Therapeutic InterventionUlrich H. Weidle, Fabian Birzele · 2024 · Cancer Genomics & Proteomics
- Causality Between Immune Cells, Metabolites and Breast Cancer: Mendelian Randomization and Mediation AnalysisChanglong Wei, Changwang Li, Gongyin Zhang, Honghui Li, Jingsong Li, Jinsheng Zeng · 2024 · Biochemical Genetics
- Therapeutic Targeting of Glutamine Metabolism in Colorectal CancerYashwant Kumar Ratre, Henu Kumar Verma, Arundhati Mehta, Vivek Kumar Soni, Subash Chandra Sonkar, Dhananjay Shukla, Alka Ekka, Santosh Kumar Prajapati, Shakuntala Mahilkar, Naveen Kumar Vishvakarma · 2021 · Springer eBooks
- A Combined SIRT5 Activation and SIRT3 Inhibition Prevents Breast Cancer Spheroids Growth by Reducing HIF-1α and MitophagyFederica Barreca, Michele Aventaggiato, Mario Cristina, Luigi Sansone, Manuel Belli, Maria Beatrice Lista, Gaia Francisci, Sérgio Valente, Dante Rotili, Antonello Mai et al. · 2025 · Pharmaceuticals
- Salubrinal-activated integrated stress response protects against doxorubicin-induced cardiotoxicity via activating transcription factor 4-mediated antioxidant defense and glutathione homeostasisSheng‐Fan Wang, Hsuan-Yu Chou, Pei-Hsun Liu, Hsing-Hui Su, Giun‐Yi Hung, Chian‐Ying Chou, Ling‐Ming Tseng, Yuh‐Chiang Shen, Jiin‐Cherng Yen, Shiang‐Suo Huang et al. · 2026 · Free Radical Biology and Medicine
- CircRNAs as central regulators of Immunometabolic crosstalk in hepatocellular carcinomaSeerwan Hamadameen Sulaiman, Rebaz Anwar Omer, Hemn A.H. Barzani, Hunar Yasin Muhammad, Avan Bazid Qader, Evan Hashm Muhammad, Darya Kaife Muhammad, Sara Wezhawan Ahmad, Hoshyar Saadi Ali · 2026 · Clinica Chimica Acta
- Gallic acid markedly stimulates GLUT1-mediated glucose uptake by the AsPC-1 pancreatic cancer cell lineSílvia M. Torres, Francisca Carmo, Luís C. Monteiro, Cláudia Silva, Nelson Andrade, Fátima Martel · 2023 · Canadian Journal of Physiology and Pharmacology
- In vitro evaluation of (S)-2-amino-3-[3-(2-18F-fluoroethoxy)-4-iodophenyl]-2-methylpropanoic acid (18F-FIMP) as a positron emission tomography probe for imaging amino acid transportersSatoshi Nozaki, Yuka Nakatani, Aya Mawatari, W. Ewan Hume, Hisashi Doi, Yasuyoshi Watanabe · 2023 · EJNMMI Research
- Actividad antitumoral de complejos de cobre(II) con fenantrolina y dipéptidos en células de cáncer de mamaKatherine Seneth Muñoz Garzón, Natalia Álvarez, Gianella Facchin, Beatriz D. Soria, Ana Laura Di Virgilio · 2024 · Revista Colombiana de Hematología y Oncología
- The cytotoxic effect of crocin and chrysin on the AsPC-1 pancreatic cancer cell line is related to inhibition of nutrient uptakeSara Pinto, Nelson Andrade, Francisca Carmo, Cláudia Silva, Fátima Martel · 2025 · PharmaNutrition
- Integrating transcriptomic and metabolomic analyses to characterize the potential function of SLC1A5 in thyroid cancerFengling Shan, Lan Wang, Xinyu Lu, Meihong Zhou, Zi Wang, Jingjing Lou, Xingdang Liu · 2025 · BMC Cancer
- Glutaminase inhibition confers antitumor effects in vitro and in vivo on tyrosine kinase inhibitors-resistant renal cell carcinoma cells by affecting vascular endothelial growth factor signalingKento Morozumi, Yoshihide Kawasaki, Izumi Sakamoto, Tomonori Sato, Masamitsu Maekawa, Shinya Takasaki, Shinichi Yamashita, Nariyasu Mano, Akihiro Ito · 2025 · Biomedicine & Pharmacotherapy
- Recent progress of amino acid transporters as a novel antitumor targetJi-Ye Zhao, Jiayi Lv, Yang Chen, Qi Dong, Hao-Rong Dong · 2022 · Open Chemistry
- Discovery and Synthesis of Hydroxy-l-Proline Blockers of the Neutral Amino Acid Transporters SLC1A4 (ASCT1) and SLC1A5 (ASCT2)Brent R. Lyda, Gregory P. Leary, Jill C. Farnsworth, Derek Silvius, Benjamin Seaver, C. Sean Esslinger, Nicholas R. Natale, Michael P. Kavanaugh · 2024 · Molecules
- Transporter-Mediated Drug DeliveryGergely Gyimesi, Matthias A. Hediger · 2022 · Preprints.org
- Glutamine transporters as effective targets in digestive system malignant tumor treatmentFEI CHU, KAI TONG, Xiang Gu, MEI BAO, Yanfen Chen, Bin Wang, YANHUA SHAO, Ling Wei · 2024 · Oncology Research Featuring Preclinical and Clinical Cancer Therapeutics
- Reproducibility and repeatability of 18F-(2S, 4R)-4-fluoroglutamine PET imaging in preclinical oncology modelsGregory Daniel Ayers, Allison S. Cohen, Seong-Woo Bae, Xiaoxia Wen, Alyssa C. Pollard, Shilpa Sharma, Trey Claus, Adria C. Payne, Ling Geng, Ping Zhao et al. · 2025 · PLoS ONE
- Analysis of a pan‑cancer panel reveals the amino acid metabolism‑related gene MTHFD1 as a potential prognostic and immunotherapeutic biomarkerShunsong Gong, Jiaxue Yang, Chao Pan, Peng Fenglan, Chuan Pan · 2025 · Experimental and Therapeutic Medicine
- Lapatinib induces ferroptosis in osteosarcoma via the SLC1A5-GPX4 axisHaichuan Miao, Xijia Fu, Baolong Liu, Xinfang Pan, Yahao Han, Zhongshen Yu · 2026 · Journal of bone oncology
- Peptides or Amino Acids?—‘The Smaller, the Better?’Christian E. W. Steinberg · 2022 · Springer eBooks
- [Value of prediction models for prognosis prediction of colorectal cancer: an analysis based on TCPA database].H Wen, Weikun Shi, Shuguang Ge, J Li, Lugen Zuo, M Liu · 2021 · PubMed Central
- Glutamine metabolism in prostate cancerTomas Koltai, Stephan J. Reshkin, Fátima Baltazar, Larry Fliegel · 2021 · Elsevier eBooks
- Nutrient Transporters: New Molecular Targets for Triple Negative Breast Cancer in Type 2 DiabeticsCláudia Silva, Fátima Martel · 2022 · Interdisciplinary cancer research
- Expression of Alanine-Serine-Cysteine Transporter 2 (ASCT2) and L-type Amino Acid Transporter 1 (LAT1) in Low-Grade and High-Grade Gliomas: An Analysis of Open-Access Immunohistochemical DataWilliam T Han, Nina H. Cheng, Najib Muhammad, John Y. K. Lee · 2025 · Cureus
- The differential effect of glutamine supplementation on the orthotopic and subcutaneous growth of two syngeneic murine models of gliomaJ Maurer, Purna Mukherjee, Nathan L. Ta, Derek C. Lee, Tomás Duraj, Juan Henao, Michael Kiebish, Devon Van Cura, Marialucia Herdocia, Thomas N. Seyfried · 2025 · ONCOLOGIE
- MRI of ASCT2-mediated amino acid uptake in xenograft tumor modelsBehnaz Ghaemi, Balaji Krishnamachary, Natalie Dillman, Kirsten N. Bains Williams, Yuki Hodo, Yuguo Li, Marie‐France Penet, Martin G. Pomper, Caitlin M. Tressler, Zaver M. Bhujwalla et al. · 2025 · Research Square
- Targeting Glutamine Transporters as a Novel Drug Therapy for Synovial SarcomaThanh Duc Tran, Naoki Takada, Hana Yao, Yoshitaka Ban, Naoto Oebisu, Manabu Hoshi, Nguyen Tran Quang Sang, Nguyen Van Khanh, Dang Minh Quang, Lê Thị Thanh Thủy et al. · 2025 · Cancers
- Additional file 1 of In vitro evaluation of (S)-2-amino-3-[3-(2-18F-fluoroethoxy)-4-iodophenyl]-2-methylpropanoic acid (18F-FIMP) as a positron emission tomography probe for imaging amino acid transportersNozaki, Satoshi, Yuka Nakatani, Aya Mawatari, W. Ewan Hume, Hisashi Doi, Watanabe, Yasuyoshi · 2023 · Figshare
- Additional file 1 of Elevated SLC1A5 associated with poor prognosis and therapeutic resistance to transarterial chemoembolization in hepatocellular carcinomaGuixiong Zhang, 萧贻泰, Jizhou Tan, Hang Liu, Fan, Wenzhe, Jiaping Li · 2024 · Figshare
- Additional file 1 of Blockade of the amino acid transporter SLC6A14 suppresses tumor growth in colorectal CancerLu, Ying, Ziting Jiang, Wang, Kaijing, Yu, Shanshan, Chongbo Hao, Zuan Ma, Fu, Xuelian, Qin, Ming Qing, Xu, Zengguang, 范列英 · 2022 · Figshare
- The tumor immune microenvironment in hepatocellular carcinoma: Its biological role in recurrence and metastasisXia Sheng, Jian-Min Qin · 2026 · World Chinese Journal of Digestology
- Regulation of Amino Acid Transporters by Cell Surface ReceptorsChiara Brignola, Myrhiam Cassese, S. Marrone, Teresa Esposito, Vincenza Barresi, Gabriella Esposito, D. F. Condorelli, Rosario Ammendola, Fabio Cattaneo · 2026 · Antioxidants
- NRF2 / xCT ‐Mediated Antioxidant Adaptation Attenuates Apoptosis Induced by ASCT2 Inhibition in Prostate CancerJiaxing Wei, Yasutaka Yamada, Tomohiro Tamura, Masahiro Sugiura, Xue Zhao, Meng Ni, Adilan Aierken, Tomokazu Sazuka, Yusuke Imamura, Shinichi Sakamoto · 2026 · Cancer Science
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