Rationale, pharmacology and clinical efficacy of partial agonists of α4β2 nACh receptors for smoking cessation
Rollema, Hans, Coe, Jotham W., Chambers, Leslie K., Hurst, Raymond S., Stahl, Stephen M., Williams, Kathryn E.·2007·Trends in Pharmacological Sciences
Cited by (410)
Items 401–410 of 410
- Replication of sex differences in tobacco smoking-induced dopamine responses and extension to nicotine replacement therapyGaelle M. Emvalomenos, Qinlin Gu, Su Jin Kim, Yasmin Zakiniaeiz, Clara Grazian, Steven R. Meikle, Kelly Cosgrove, Evan D. Morris · 2026 · Nicotine & Tobacco Research
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- BindingDB Entry 50038738: Novel acetylcholine and carbamoylcholine analogues: development of a functionally selective alpha4beta2 nicotinic acetylcholine receptor agonist.BindingDB · 2012 · UC San Diego
- BindingDB Entry 50040717: Structure-activity studies of 7-heteroaryl-3-azabicyclo[3.3.1]non-6-enes: a novel class of highly potent nicotinic receptor ligands.BindingDB · 2013 · UC San Diego
- BindingDB Entry 50007946: Discovery of Novel, Potent, Brain-Permeable, and Orally Efficacious Positive Allosteric Modulator of α7 Nicotinic Acetylcholine Receptor [4-(5-(4-Chlorophenyl)-4-methyl-2-propionylthiophen-3-yl)benzenesulfonamide]: Structure-Activity Relationship and Preclinical Characterization.BindingDB · 2021 · UC San Diego
- BindingDB Entry 50043556: TBABindingDB · 2014 · UC San Diego
- BindingDB Entry 50039698: Chemistry and behavioral studies identify chiral cyclopropanes as selectivea4ß2-nicotinic acetylcholine receptor partial agonists exhibiting an antidepressant profile.BindingDB · 2013 · UC San Diego
- BindingDB Entry 50033196: Synthesis of 2-(substituted phenyl)-3,5,5-trimethylmorpholine analogues and their effects on monoamine uptake, nicotinic acetylcholine receptor function, and behavioral effects of nicotine.BindingDB · 2011 · UC San Diego
- BindingDB Entry 50033481: Evaluation of structurally diverse neuronal nicotinic receptor ligands for selectivity at the alpha6( *) subtype.BindingDB · 2011 · UC San Diego
- BindingDB Entry 50039465: Nicotinic Acetylcholine Receptor Efficacy and Pharmacological Properties of 3-(Substituted phenyl)-2ß-substituted Tropanes.BindingDB · 2013 · UC San Diego