Polyhydroxylated alkaloids—Natural occurrence and therapeutic applications

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Total Syntheses of (+)‐Valiolamine and (–)‐1‐epi‐Valiolamine from Naturally Abundant (–)‐Shikimic Acid

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Stereoselective synthesis of (−)-8-epi-swainsonine starting with a chiral aziridine

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Total synthesis of 1-deoxy-7,8a-di-epi-castanospermine and formal synthesis of pumiliotoxin-251D

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Gem-difluoromethylated and trifluoromethylated derivatives of DMDP-related iminosugars: synthesis and glycosidase inhibition

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Concise synthesis of C-1-cyano-iminosugars via a new Staudinger/aza Wittig/Strecker multicomponent reaction strategy

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Atom-economical isocyanide-based multicomponent synthesis of 2,5-dioxopyrrolidines, spirobenzothiazinechromans and 1,5-benzothiazepines

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Crepidtumines A and B, Two Novel Indolizidine Alkaloids from Dendrobium crepidatum

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Cyclisations and Strategies for Stereoselective Synthesis of Piperidine Iminosugars

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Synthesis of polyhydroxylated 7-aminopyrrolizidines and 8-aminoindolizidines

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GANAB and N-Glycans Substrates Are Relevant in Human Physiology, Polycystic Pathology and Multiple Sclerosis: A Review

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Azetidine- and N-carboxylic azetidine-iminosugars as amyloglucosidase inhibitors: synthesis, glycosidase inhibitory activity and molecular docking studies

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Diastereoselective [3 + 2] vs [4 + 2] Cycloadditions of Nitroprolinates with α,β-Unsaturated Aldehydes and Electrophilic Alkenes: An Example of Total Periselectivity

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On the effect of intramolecular H-bonding in the configurational assessment of polyhydroxylated compounds with computational methods. The hyacinthacines case

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Regiochemistry‐Directed Syntheses of Polyhydroxylated Alkaloids from Chiral Aziridines

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Synthesis and reductive desulfurization of chiral non-racemic benzothienoindolizines. An efficient approach to a novel bioactive tylophorine alkaloid analogue and 6-phenylindolizidine

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Stereodivergent Synthesis of Iminosugars from Stannylated Derivatives of (S)-Vinylglycinol

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Double Asymmetric Induction in Organocatalyzed Aldol Reactions: Total Synthesis of (+)‐2‐epi‐Hyacinthacine A2 and (–)‐3‐epi‐Hyacinthacine A1

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Enzymatic and Chemo-Enzymatic Approaches Towards Natural and Non-Natural Alkaloids: Indoles, Isoquinolines, and Others

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Construction of protected hydroxylated pyrrolidines using nitrogen-centered radical cyclizations

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(−)‐(1R,2R,7S,8aR)‐1,2,7‐Trihydroxyindolizidine ((−)‐7S‐OH‐Lentiginosine): Synthesis and Proapoptotic Activity

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Synthesis and Glycosidase Inhibition of Broussonetine M and Its Analogues

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3,4-Dihydroxypyrrolidine as Glycosidase Inhibitor

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Asymmetric syntheses of 6-deoxyfagomin, d-deoxyrhamnojirimycin, and d-rhamnono-1,5-lactam

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Stereoselective Nucleophilic Addition of PhSCF2SiMe3 to Chiral Cyclic Nitrones: Asymmetric Synthesis of gem‐Difluoromethylenated Polyhydroxypyrrolizidines and ‐indolizidines

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α-Glucosidase-inhibitory iminosugars from the leaves of Suregada glomerulata

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Unexpected formation of 3-chloro-1-hydroxy-2,6-diarylpiperidin-4-ones: Synthesis, antibacterial and antifungal activities

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A sort synthesis of polyhydroxylated pyrrolizidines via sequential 1,3-dipolar cycloaddition and reductive amination

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Asymmetric synthesis of 3-amino-4-hydroxy-2-(hydroxymethyl)pyrrolidines as potential glycosidase inhibitors

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Asymmetric Syntheses of (−)-3-epi-Fagomine, (2R,3S,4R)-Dihydroxypipecolic Acid, and Several Polyhydroxylated Homopipecolic Acids

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Highly diastereoselective synthesis of 2-azabicyclo[2.2.1]hept-5-ene derivatives: Bronsted acid catalyzed aza-Diels–Alder reaction between cyclopentadiene and imino-acetates with two chiral auxiliaries

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Development of a practical biocatalytic process for ( S )- N -Boc-3-hydroxypiperidine synthesis

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Flexible approach for the asymmetric synthesis of (−)-hyacinthacine A1 and its 7a-epimer

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Syntheses, characterization and evaluation of novel 2,6-diarylpiperidin-4-ones as potential analgesic-antipyretic agents

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Design and syntheses of some iminosugar derivatives as potential immunosuppressants

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First Total Synthesis of (+)‐Adenophorine, a Naturally Occurring Inhibitor of Glycosidases

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Synthesis of the New 7S‐Aminolentiginosine and Derivatives

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A ring-closing metathesis route to 7-membered aza-heteroannulated sugars

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Polyhydroxylated Pyrrolizidines. Part 7. Stereoselective Synthesis of Unnatural Analogs of (+)‐Casuarine from Partially Protected DGDP

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Total synthesis of pyrrolidine alkaloid, Radicamine-B via Stille coupling

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A divergent asymmetric approach to aza-spiropyran derivative and (1S,8aR)-1-hydroxyindolizidine

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Fluorinated and Conformationally Fixed Derivatives of l -HomoDMDP: Synthesis and Glycosidase Inhibition

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Synthesis and glycosidase inhibition potency of all- trans substituted 1- C -perfluoroalkyl iminosugars

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Phytochemical screening, antibacterial and antioxidant activities of Asparagus laricinus leaf and stem extracts

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Isolation of the pyrrolizidine alkaloid 1-epialexine from Castanospermum australe

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Selenium-promoted synthesis of enantiopure octahydroindolizines, hexahydro-1H-pyrrolizines and hexahydro-3H-pyrrolizin-3-ones

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Enantioselective Syntheses of Rigidiusculamides A and B: Revision of the Relative Stereochemistry of Rigidiusculamide A

Chen, G., Huang, H., Ye, J., Wang, A., Huang, H., Zhang, H., & Huang, P. (2012) · Chemistry - An Asian Journal · doi:10.1002/asia.201100809 · Cited by 16

Spectroscopic techniques investigation on the interaction of glucoamylase with 1-deoxynojirimycin: Mechanistic and conformational study

Wu, H., Zeng, W., Chen, G., Guo, Y., Yao, C., Li, J., & Liang, Z. (2018) · Spectrochimica Acta Part A Molecular and Biomolecular Spectroscopy · doi:10.1016/j.saa.2018.08.013 · Cited by 16

Synthesis of (+)-7a-epi-7-deoxycasuarine via cross metathesis

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Insights into the Activities and Usefulness of Deoxynojirimycin and Morus alba: A Comprehensive Review

Tricase, A. F., Cavalluzzi, M. M., Catalano, A. A., Bellis, M. D., Palma, A. D., Basile, G., Sinicropi, M. S., & Lentini, G. (2025) · Molecules · doi:10.3390/molecules30153213 · Cited by 15

Regio and diastereoselective multicomponent 1,3-dipolar cycloadditions between prolinate hydrochlorides, aldehydes and dipolarophiles for the direct synthesis of pyrrolizidines

Mancebo‐Aracil, J., Nájera, C., Castelló, L. M., Sansano, J. M., Larrañaga, O., de Cózar, A., & Cossío, F. P. (2015) · Tetrahedron · doi:10.1016/j.tet.2015.10.064 · Cited by 15

A route to selective functionalization of polyhydroxypyrrolidines

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An approach to 8 stereoisomers of homonojirimycin from d-glucose via kinetic & thermodynamic azido-γ-lactones

Glawar, A. F. G., Jenkinson, S. F., Newberry, S. J., Thompson, A. L., Nakagawa, S., Yoshihara, A., Akimitsu, K., Izumori, K., Butters, T. D., Kato, A., et al. (2013) · Organic & Biomolecular Chemistry · doi:10.1039/c3ob41334a · Cited by 15

Synthesis of the Proposed Structure of Pentahydroxylated Pyrrolizidine Hyacinthacine C5 and Its C6,C7 Epimer

Tamayo, J. A., Franco, F., & Sánchez‐Cantalejo, F. (2011) · European Journal of Organic Chemistry · doi:10.1002/ejoc.201101126 · Cited by 15

Convenient synthesis of epimeric indolizidines by the intramolecular 1,3-dipolar cycloaddition of a sugar derived N-(3-alkenyl)nitrone

Mironiuk‐Puchalska, E., Rowicki, T., Sas, W., & Koszytkowska‐Stawińska, M. (2013) · Tetrahedron · doi:10.1016/j.tet.2013.09.008 · Cited by 15

Strategy for Designing Selective Lysosomal Acid α-Glucosidase Inhibitors: Binding Orientation and Influence on Selectivity

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Novel one-pot synthesis of 1,2,4-triazolidin-3-thiones comprising piperidine moiety

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Synthesis of polyfunctional quinolizidine alkaloids: development towards selective glycosidase inhibitors

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A Cycloaddition–Cyclization Combined Approach to Enantiopure 3‐Glycinyl‐4‐hydroxypyrrolidines and 3‐Substituted 4‐Hydroxyprolines

Aouadi, K., Abdoul‐Zabar, J., Msaddek, M., & Praly, J. (2014) · European Journal of Organic Chemistry · doi:10.1002/ejoc.201402215 · Cited by 15

Synthesis of thioswainsonine as a potential glycosidase inhibitor

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Synthesis, DFT, in-silico molecular docking, molecular dynamic simulation and ADMET studies of (Z)-2,6-bis(4-bromophenyl)-3,3-dimethyl-4-(2-(2,4,6-trichlorophenyl) hydrazono) piperidine derivatives against the SARS-CoV-2 main-protease

Lorin, S., Rajaraman, D., Selvam, S., Ramakrishnan, J., Kumaradhas, P., Nagaraj, K., & Kaliyaperumal, R. (2024) · Zeitschrift für Physikalische Chemie · doi:10.1515/zpch-2023-0397 · Cited by 15

Stereospecific Cyclization Strategies for α,ε-Dihydroxy-β-amino Esters: Asymmetric Syntheses of Imino and Amino Sugars

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