Systematic Analysis of Helical Protein Interfaces Reveals Targets for Synthetic Inhibitors

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Items 101–196 of 196

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16. Macrocyclic α-Helical Peptide Drug Discovery
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17. Bicyclic Schellman Loop Mimics (BSMs): Rigid Synthetic C-Caps for Enforcing Peptide Helicity
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18. Design, Synthesis, and Conformational Analysis of Trispyrimidonamides as α-Helix Mimetics
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30. Conformationally Controlled sp 3 ‐Hydrocarbon‐Based α‐Helix Mimetics
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31. Streamlined Protein‐Protein Interface Loop Mimicry
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33. A Modular Synthesis of Teraryl‐Based α‐Helix Mimetics, Part 3: Iodophenyltriflate Core Fragments Featuring Side Chains of Proteinogenic Amino Acids
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34. Helix Nucleation via Hydrocarbon Cross‐link Mimicking N‐capping Box
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37. Efficient α‐Helix Induction in a Linear Peptide Chain by N‐Capping with a Bridged‐tricyclic Diproline Analogue
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38. Rational Design Strategies for Developing Synthetic Inhibitors of Helical Protein Interfaces
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40. Salt-bridging effects on short amphiphilic helical structure and introducing sequence-based short beta-turn motifs
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42. Screening a Molecular Fragment Library to Modulate the PED/PEA15-Phospholipase D1 Interaction in Cellular Lysate Environments
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43. Structural Basis for α‐Helix Mimicry and Inhibition of Protein–Protein Interactions with Oligourea Foldamers
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48. X-ray Crystallographic Structure of α-Helical Peptide Stabilized by Hydrocarbon Stapling at i,i + 1 Positions
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