Recent Advances in the Friedländer Reaction

Comprehensive Heterocyclic Chemistry II

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New Conjugated Polymers with Donor−Acceptor Architectures: Synthesis and Photophysics of Carbazole−Quinoline and Phenothiazine−Quinoline Copolymers and Oligomers Exhibiting Large Intramolecular Charge Transfer

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Advances in Heterocyclic Chemistry

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Camptothecin: current perspectives

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Handbook of heterocyclic chemistry

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Heterocyclic Nitrogen Compounds. Part IIA. Hexacyclic Compounds: Pyridine, Quinoline, and Isoquinoline.

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Name Reactions in Heterocyclic Chemistry

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New n-Type Organic Semiconductors: Synthesis, Single Crystal Structures, Cyclic Voltammetry, Photophysics, Electron Transport, and Electroluminescence of a Series of Diphenylanthrazolines

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Heterocyclic Chemistry: Volume I: Principles, Three- and Four-Membered Heterocycles

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Blue‐Light‐Emitting Oligoquinolines: Synthesis, Properties, and High‐Efficiency Blue‐Light‐Emitting Diodes

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The Chemistry of Quinolines.

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Novel Donepezil-Based Inhibitors of Acetyl- and Butyrylcholinesterase and Acetylcholinesterase-Induced β-Amyloid Aggregation

Camps, P., Formosa, X., Galdeano, C., Gómez, T., Muñoz-Torrero, D., Scarpellini, M., Viayna, E., Badia, A., Clos, M. V., Camins, A., et al. (2008) · Journal of Medicinal Chemistry · doi:10.1021/jm8001313 · Cited by 205

New Tacrine−Huperzine A Hybrids (Huprines): Highly Potent Tight-Binding Acetylcholinesterase Inhibitors of Interest for the Treatment of Alzheimer's Disease

Camps, P., El Achab, R., Morral, J., Muñoz-Torrero, D., Badia, A., Baños, J. E., Vivas, N. M., Barril, X., Orozco, M., & Luque, F. J. (2000) · Journal of Medicinal Chemistry · doi:10.1021/jm000980y · Cited by 201

High Mobility Single-Crystal Field-Effect Transistors from Bisindoloquinoline Semiconductors

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Sulfonated cellulose and starch: New biodegradable and renewable solid acid catalysts for efficient synthesis of quinolines

Shaabani, A., Rahmati, A., & Badri, Z. (2008) · Catalysis Communications · doi:10.1016/j.catcom.2007.05.021 · Cited by 176

SAR of 9-Amino-1,2,3,4-tetrahydroacridine-Based Acetylcholinesterase Inhibitors: Synthesis, Enzyme Inhibitory Activity, QSAR, and Structure-Based CoMFA of Tacrine Analogues

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Synthesis and processing of heterocyclic polymers as electronic, optoelectronic, and nonlinear optical materials. 2. New series of conjugated rigid-rod polyquinolines and polyanthrazolines

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Polyquinolines

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Camptothecins: A SAR/QSAR Study

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Plant antitumor agents. 23. Synthesis and antileukemic activity of camptothecin analogs

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Highly Regioselective Friedländer Annulations with Unmodified Ketones Employing Novel Amine Catalysts: Syntheses of 2-Substituted Quinolines, 1,8-Naphthyridines, and Related Heterocycles

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Surfactant-type catalysts in organic reactions

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Streptonigrin and lavendamycin partial structures. Probes for the minimum, potent pharmacophore of streptonigrin, lavendamycin, and synthetic quinoline-5,8-diones

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Novel Multipotent Tacrine−Dihydropyridine Hybrids with Improved Acetylcholinesterase Inhibitory and Neuroprotective Activities as Potential Drugs for the Treatment of Alzheimer's Disease

Marco, J. L., Leon, R. M., Ríos, C. D. L., Guglietta, A., Terencio, J. V., López, M. G., García, A. G., & Villarroya, M. (2006) · Journal of Medicinal Chemistry · doi:10.1021/jm061047j · Cited by 118

Plant antitumor agents. 25. Total synthesis and antileukemic activity of ring A substituted camptothecin analogs. Structure-activity correlations

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Design, Synthesis, and Pharmacological Profile of Novel Fused Pyrazolo[4,3- d ]pyridine and Pyrazolo[3,4- b ][1,8]naphthyridine Isosteres: A New Class of Potent and Selective Acetylcholinesterase Inhibitors

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Novel Tacrine Analogues for Potential Use against Alzheimer's Disease: Potent and Selective Acetylcholinesterase Inhibitors and 5-HT Uptake Inhibitors

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Synthesis of condensed quinolines and quinazolines as DNA ligands

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Ru(II) Complexes of Tetradentate Ligands Related to 2,9-Di(pyrid-2‘-yl)-1,10-phenanthroline

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Acetylcholinesterase inhibitors for potential use in Alzheimer's disease: molecular modeling, synthesis and kinetic evaluation of 11H-indeno-[1,2-b]-quinolin-10-ylamine derivatives

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Naphthyridine-Based Helical Foldamers and Macrocycles: Synthesis, Cation Binding, and Supramolecular Assemblies

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Synthesis, in Vitro Pharmacology, and Molecular Modeling of Very Potent Tacrine−Huperzine A Hybrids as Acetylcholinesterase Inhibitors of Potential Interest for the Treatment of Alzheimer's Disease

Camps, P., Achab, R. E., GOERBIG, D. M., Morral, J., Muñoz‐Torrero, D., Badía, A., Baños, J.-E., Vivas, N. M., Barril, X., Orozco, M., et al. (1999) · Journal of Medicinal Chemistry · doi:10.1021/jm980620z · Cited by 97

Practical Asymmetric Synthesis of (S)-4-Ethyl-7,8-dihydro-4-hydroxy-1H-pyrano[3,4-f]indolizine- 3,6,10(4H)-trione, a Key Intermediate for the Synthesis of Irinotecan and Other Camptothecin Analogs

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Synthesis, biological evaluation and molecular modelling of diversely functionalized heterocyclic derivatives as inhibitors of acetylcholinesterase/butyrylcholinesterase and modulators of Ca2+ channels and nicotinic receptors

Marco, J. L., Rı́os, C. D. L., Garcı́a, A. G., Villarroya, M., Carreiras, M. C., Martins, C., Eleutério, A., Morreale, A., Orozco, M., & Luque, F. J. (2004) · Bioorganic & Medicinal Chemistry · doi:10.1016/j.bmc.2004.02.017 · Cited by 91

Synthesis and biological evaluations of quinoline-based HMG-CoA reductase inhibitors

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Friedländer Synthesis of Quinolines Using a Lewis Acid‐Surfactant‐Combined Catalyst in Water

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Crowded Cu(I) Complexes Involving Benzo[h]quinoline: π-Stacking Effects and Long-Lived Excited States

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Synthesis and evaluation of tacrine–Huperzine a hybrids as acetylcholinesterase inhibitors of potential interest for the treatment of alzheimer’s disease

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Novel fluorinated acridone derivatives. Part 1: Synthesis and evaluation as potential anticancer agents

Fadeyi, O., Adamson, S. T., Myles, E. L., & Okoro, C. O. (2008) · Bioorganic & Medicinal Chemistry Letters · doi:10.1016/j.bmcl.2008.05.078 · Cited by 77

New tacrine-dihydropyridine hybrids that inhibit acetylcholinesterase, calcium entry, and exhibit neuroprotection properties

Leon, R. M., Ríos, C. D. L., Marco, J. L., Huertas, Ó., Barril, X., Luque, F. J., López, M. G., García, A. G., & Villarroya, M. (2008) · Bioorganic & Medicinal Chemistry · doi:10.1016/j.bmc.2008.07.005 · Cited by 74

Thin-film processing and optical properties of conjugated rigid-rod polyquinolines for nonlinear optical applications

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Synthesis and Pharmacological Evaluation of Huprine−Tacrine Heterodimers: Subnanomolar Dual Binding Site Acetylcholinesterase Inhibitors

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Novel quinolinequinone antitumor agents: structure-metabolism studies with NAD(P)H:quinone oxidoreductase (NQO1)

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Synthesis and acetylcholinesterase/butyrylcholinesterase inhibition activity of new tacrine-like analogues

Marco, J. L., Rı́os, C. D. L., Carreiras, M. C., Baños, J.-E., Badı́a, A., & Vivas, N. M. (2001) · Bioorganic & Medicinal Chemistry · doi:10.1016/s0968-0896(00)00284-4 · Cited by 63

Synthesis, acetylcholinesterase inhibition and neuroprotective activity of new tacrine analogues

Leon, R. M., Marco, J. L., Garcı́a, A. G., & Villarroya, M. (2004) · Bioorganic & Medicinal Chemistry · doi:10.1016/j.bmc.2004.11.020 · Cited by 54

Novel tacrine derivatives that block neuronal calcium channels

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The synthesis and in vitro acetylcholinesterase and butyrylcholinesterase inhibitory activity of tacrine (Cognex®) derivaties

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Synthesis, in Vitro Pharmacology, and Molecular Modeling of syn-Huprines as Acetylcholinesterase Inhibitors

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A mild, efficient and improved protocol for the friedländer synthesis of quinolines using lewis acidic ionic liquid

Karthikeyan, G., & Perumal, P. T. (2004) · Journal of Heterocyclic Chemistry · doi:10.1002/jhet.5570410632 · Cited by 52

New multipotent tetracyclic tacrines with neuroprotective activity

Marco, J. L., Leon, R. M., Rı́os, C. D. L., Garcı́a, A. G., López, M. G., & Villarroya, M. (2006) · Bioorganic & Medicinal Chemistry · doi:10.1016/j.bmc.2006.09.025 · Cited by 51

Photoresponsive polyquinolines

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Synthesis and biological evaluation of new 4H-pyrano[2,3-b]quinoline derivatives that block acetylcholinesterase and cell calcium signals, and cause neuroprotection against calcium overload and free radicals

Marco, J. L., Leon, R. M., López, M. G., Garcı́a, A. G., & Villarroya, M. (2006) · European Journal of Medicinal Chemistry · doi:10.1016/j.ejmech.2006.06.016 · Cited by 48

Ruthenium(II) Complexes of 2-Aryl-1,10-phenanthrolines: Synthesis, Structure, and Photophysical Properties

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High-Efficiency Electroluminescence from New Blue-Emitting Oligoquinolines Bearing Pyrenyl or Triphenyl Endgroups

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Dipyrido[4,3-b;5,6-b]acridine Derivatives and Their Ruthenium(II) Complexes

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Acetylcholinesterase inhibition by tacrine analogues

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An Efficient Protocol for the Friedländer Quinoline Synthesis Using the Lewis Acidic Ionic Liquid Choline Chloride•2ZnCl2

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Synthesis and evaluation of tacrine-related compounds for the treatment of Alzheimer's disease

AGUADO, F., Badı́a, A., Baños, J.-E., Bosch, F., Bozzo, C., Camps, P., Contreras, J., Dierssen, M., Escolano, C., GOERBIG, D. M., et al. (1994) · European Journal of Medicinal Chemistry · doi:10.1016/0223-5234(94)90039-6 · Cited by 29

Synthesis and Acetylcholinesterase/Butyrylcholinesterase Inhibition Activity of 4-Amino-2, 3-diaryl-5, 6, 7, 8-tetrahydrofuro(and thieno)[2, 3-b]-quinolines, and 4-Amino-5, 6, 7, 8, 9-pentahydro-2, 3-diphenylcyclohepta[e]furo(and thieno)-[2, 3-b]pyridines

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One‐Pot and Convenient Conversion of 5‐Azidopyrazole‐4‐carboxaldehyde to Pyrazolo[3,4‐b]pyridines

Zheng, A., Zhang, W., & Pan, J. (2006) · Synthetic Communications · doi:10.1080/00397910600588868 · Cited by 25

An Efficient Synthesis of the New Benzo[c]pyrido[2,3,4-kl]acridine Skeleton

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Discovery of Quinolinediones Exhibiting a Heat Shock Response and Angiogenesis Inhibition

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Titanium(IV) chloride promoted condensation of ortho-aminonitriles with δ-valerolactone

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Synthesis and preliminary evaluation of novel analogues of quindolines as potential stabilisers of telomeric G-quadruplex DNA

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Identification of a 3-Hydroxylated Tacrine Metabolite in Rat and Man: Metabolic Profiling Implications and Pharmacology

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On the regioselectivity of the Friedländer reaction leading to huprines: stereospecific acid-promoted isomerization of syn-huprines to their anti-regioisomers

Camps, P., Gómez, E., Muñoz‐Torrero, D., & Arnó, M. (2001) · Tetrahedron Asymmetry · doi:10.1016/s0957-4166(01)00499-2 · Cited by 12

Synthesis of 1,7,10-Anthyridine Derivatives

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Cerium(IV) Ammonium Nitrate as a Catalyst in Organic Synthesis

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Tacrines for Alzheimer's disease therapy. III. The PyridoTacrines

de los Ríos, C., & Marco-Contelles, J. (2019) · European Journal of Medicinal Chemistry · doi:10.1016/j.ejmech.2019.02.005 · Cited by 63