Gemcitabine versus Modified Gemcitabine: A Review of Several Promising Chemical Modifications

Moysan, Elodie, Bastiat, Guillaume, Benoit, Jean-Pierre·2013·Molecular Pharmaceutics

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  1. In vivo Assessment of the Hepatotoxicity of Mixed Gemcitabine and 5-Fluorouracil Loaded on Microemulsion in Mice Bearing Ehrlich Ascites Carcinoma
    Mayson H. Alkhatib, May M. Alasmari, Faiza Abdo · 2017 · Advances in Pharmacology and Pharmacy
  2. Tumor Microenvironment and Intracellular Signal-Activated Nanocomposites for Anticancer Drug Delivery
    Yilan Huang, Yiheng Huang, Yuefei Zhu, Xiaowen Zhu, Zhiqing Pang · 2021 · Materials horizons
  3. Efficacy and Mechanism of Action of a Novel Class of Antic-Cancer Drugs
    Teran, Claudia · 2016 · uO Research (University of Ottawa)
  4. Organofluorine-containing anticancer therapeutics
    Magdalena Ślusarczyk · 2015
  5. PERBANDINGAN INHIBISI BRUSEIN D TERHADAP PROTEIN NFKB PADA SEL KANKER PANKREAS SECARA FLEKSIBEL DAN RIGID DOCKING
    Sekolah Tinggi Teknologi Industri dan Farmasi Bogor, Harry Noviardi, Armi Wulanawati, Institut Pertanian Bogor, Muhammad Sholehuddin malik Ibrohim · 2017 · Jurnal Farmamedika (Pharmamedica Journal)
  6. Self-assembling Phosphoramidate Pronucleotides: Enzymatic Regulation and Application Towards Therapeutic Delivery
    Harrison T. West · 2019 · University of Minnesota Digital Conservancy (University of Minnesota)
  7. Research Progress in Drug Resistance and Structural Modification of Gemcitabine
    悦 万 · 2023 · Pharmacy Information
  8. Targeting Intracranial Tumours with a Combination of RNA and Chemotherapy
    Abdulhamid S. Fatani, Andreas G. Schätzlein, Ijeoma Florence Uchegbu · 2024 · Pharmaceutics
  9. Computational photochemistry: advances in 2022–2023
    Miriam Navarrete‐Miguel, Juliana Cuéllar-Zuquin, Javier Carmona‐García, Abdelazim M. A. Abdelgawwad, Iván Soriano-Díaz, Juan Carlos Roldao, Debabrata Halder, Ana Borrego‐Sánchez, Antonio Francés‐Monerris, Angelo Giussani et al. · 2024 · Royal Society of Chemistry eBooks
  10. Carboxymethyl-β-1,3-D-glucan (CMG)-gemcitabine conjugate improves the anticancer efficacy and alleviate the toxicity of gemcitabine (GEM)
    Maxin Ji, Yudong Zhang, Yilong Duan, Yuqing Zhao, Guangyue Su · 2025 · Natural Product Research
  11. Breast Cancer: Epidemiology, Symptoms, Risk Factors, Pathogenesis, Classification, Current Treatments and Various Approaches in Nano-formulations
    Nitish Kumar, Balram Balram, Gurvirender Singh, Dushyant, Smita Narwal, Ashwani K. Dhingra · 2025 · Current Cancer Therapy Reviews
  12. Some stereoisomers and tautomers of gemcitabine – A DFT treatment
    Lemi Türker · 2025 · Earthline Journal of Chemical Sciences
  13. Challenges in traditional TNBC therapies
    Somdatta Y. Chaudhari, Aishwarya Pandit, Mukund Salunke, Shailaja Jadhav, Aarti Kulkarni, Sachin Namdeo Kothawade · 2025 · Elsevier eBooks
  14. Additional file 2 of Biological evaluation of novel gemcitabine analog in patient-derived xenograft models of pancreatic cancer
    Andriana Inkoom, Ndemazie, Nkafu Bechem, Taylor Smith, Esther Frimpong, Raviteja Bulusu, Rosemary A. Poku, Zhu, Xue, Han, Bo, Trevino, Jose, Edward Agyare · 2024 · Figshare
  15. Additional file 1 of Biological evaluation of novel gemcitabine analog in patient-derived xenograft models of pancreatic cancer
    Andriana Inkoom, Ndemazie, Nkafu Bechem, Taylor Smith, Esther Frimpong, Raviteja Bulusu, Rosemary A. Poku, Zhu, Xue, Bo Han, Trevino, Jose, Edward Agyare · 2024 · Figshare
  16. Nouveau concept de resensibilisation à la chimiothérapie en activant la nucléoside kinase dCK par le masitinib, un inhibiteur de protéines tyrosine kinases
    Kahina Hammam · 2014
  17. Photocaging the C6-carboxylate of β-glucuronide prodrugs enables spatiotemporally controlled release of anticancer agents via a dual activation strategy
    Junjie Fu, Dianya Yong, Jie Liu, Yunying Tan, Hongyu Yang, Jing Hu, Jian Yin · 2026 · Organic & Biomolecular Chemistry
  18. Contribution à l'étude des mécanismes moléculaires de chimiorésistance des cellules cancéreuses pancréatiques
    Marion Gayral · 2015 · theses.fr (ABES)
  19. Hydrogel de nanocapsules lipidiques combinées au peptide de ciblage NFL-TBS.40-63 pour la prévention de récurrences de glioblastome
    Claire Gazaille · 2020
  20. Self-Assembly Regulation, Drug Release Behavior, Anti-Multidrug Resistance of Redox-Responsive Gemcitabine–Quinine Nanoassemblies in Glioblastoma Therapy
    Jiayi Zuo, Shuhui Qu, Haoping Long, Ting Yuan, Jinqiu Liang, Feng Jiang · 2026 · Langmuir
  21. Dual Metabolic Blockade in Pancreatic Cancer: Potent Anticancer Activity of Mitochondria-Targeted Glycolysis and OXPHOS Inhibitors
    闫海波, Dongsheng Li, Min Yang, Mingyang Xu, Ying Yang, Zhenzhen Dai, Jiamin Ou, Yingjie He, Biao Xu, Shaolin Zhang · 2026 · Journal of Medicinal Chemistry
  22. Poly-β-Cyclodextrin as a Superior Host for Gemcitabine: Comparative Supramolecular Characterization and Anticancer Evaluation
    Manickam Sathya, Archana Sumohan Pillai, Varnitha Manikantan, Sengodan Amudha, Ujma Ashapak Tamboli, Ramaraj Rajesh Kumar, Aleyamma Alexander, Israel V.M.V. Enoch · 2026 · Journal of Solution Chemistry
  23. Magadiite-based delivery system with sustained release of gemcitabine and its cytotoxicity against HepG2 cells
    Xuling Weng, Fang Guo, Yu Zhong, Wanyun Feng, Xiaoqiang Shang, Yufeng Chen · 2026 · Chemical Papers
  24. A Dual-Action CXCR4-Targeted Peptide−Drug Conjugate Engineered to Enhance Antitumor Efficacy and Mitigate Myelosuppression in Pancreatic Cancer
    Ke Zhu, Xuanxin Liu, Dapeng Li, Tao Wang, Tao Wen, Xiaocui Fang, Yanlian Yang, Jian Liu, Jie Meng, Chen Wang et al. · 2026 · Molecular Pharmaceutics
  25. HMHLVI: Hybrid Multi-view Hypergraph Learning with Variational Inference for snoRNA-Drug Association Prediction
    Tiyao Liu, Shudong Wang, Dapeng Wang, Shaoqiang Wang, Shanchen Pang · 2026 · Interdisciplinary Sciences Computational Life Sciences
  26. A novel nanoparticle-based co-delivery system of Fritillaria persica L . extract and gemcitabine for inhibiting breast cancer progression
    Reyhaneh Arefimehr, Mehrad Zibaei Moghadam, Negar Jamshidi, Nazanin Jamshidi · 2026 · Beilstein Journal of Nanotechnology
  27. BindingDB Entry 50013685: Development of programmable gemcitabine-GnRH pro-drugs bearing linker controllable "click" oxime bond tethers and preclinical evaluation against prostate cancer.
    BindingDB · 2022 · UC San Diego
  28. BindingDB Entry 50044081: N-Acyl-phosphoramidates as potential novel form of gemcitabine prodrugs.
    BindingDB · 2015 · UC San Diego
  29. BindingDB Entry 50012568: Discovery of a novel chimeric ubenimex-gemcitabine with potent oral antitumor activity.
    BindingDB · 2022 · UC San Diego
  30. BindingDB Entry 50015330: Integrin-Mediated Targeted Cancer Therapy Using c(RGDyK)-Based Conjugates of Gemcitabine.
    BindingDB · 2023 · UC San Diego
  31. BindingDB Entry 50016140: Design, synthesis and antitumor activity study of a gemcitabine prodrug conjugated with a HDAC6 inhibitor.
    BindingDB · 2023 · UC San Diego
  32. BindingDB Entry 50011989: Development of potent CPP6-gemcitabine conjugates against human prostate cancer cell line (PC-3).
    BindingDB · 2022 · UC San Diego