Anandamide suppresses pain initiation through a peripheral endocannabinoid mechanism

Clapper, Jason R, Moreno-Sanz, Guillermo, Russo, Roberto, Guijarro, Ana, Vacondio, Federica, Duranti, Andrea, Tontini, Andrea, Sanchini, Silvano +7 more·2010·Nature Neuroscience

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  11. Efeito da radiação ultravioleta B no sistema endocanabinóide cutâneo
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  14. Encodage de l'information sensorielle nociceptive par la moelle épinière et son implication dans les douleurs neuropathiques et leur traitement
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  15. Role for Endocannabinoids in Spinal Manipulative Therapy Analgesia?
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  16. Interacción del antihelmíntico triclabendazol, el analgésico URB937 y sus derivados con transportadores de membrana dependientes de ATP = Interaction of the anthelmintic triclabendazole, the analgesic URB937 and their derivatives with ATP-dependent membrane transporters
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  21. Role of Cannabinoids in Pain Management
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  22. Faculty Opinions recommendation of Microdeletion in a FAAH pseudogene identified in a patient with high anandamide concentrations and pain insensitivity.
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  24. Perspectives on Neuroscience and Behavior
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  27. Faculty Opinions recommendation of Pharmacological characterization of the peripheral FAAH inhibitor URB937 in female rodents: interaction with the Abcg2 transporter in the blood-placenta barrier.
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  44. BindingDB Entry 50040637: Identification and characterization of carprofen as a multitarget fatty acid amide hydrolase/cyclooxygenase inhibitor.
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  45. BindingDB Entry 8240: Inhibitory properties of ibuprofen and its amide analogues towards the hydrolysis and cyclooxygenation of the endocannabinoid anandamide.
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  46. BindingDB Entry 50047424: Piperidinyl thiazole isoxazolines: A new series of highly potent, slowly reversible FAAH inhibitors with analgesic properties.
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  53. BindingDB Entry 50010033: Peripherally Selective Cannabinoid 1 Receptor (CB1R) Agonists for the Treatment of Neuropathic Pain.
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  54. BindingDB Entry 50043192: Synthesis and structure-activity relationship studies of O-biphenyl-3-yl carbamates as peripherally restricted fatty acid amide hydrolase inhibitors.
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  55. BindingDB Entry 50006534: Design, synthesis and biological evaluation of novel analgesic agents targeting both cyclooxygenase and TRPV1.
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  58. BindingDB Entry 50040090: N-(2-oxo-3-oxetanyl)carbamic acid esters as N-acylethanolamine acid amidase inhibitors: synthesis and structure-activity and structure-property relationships.
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  59. BindingDB Entry 50041943: Biphenyl-3-yl alkylcarbamates as fatty acid amide hydrolase (FAAH) inhibitors: steric effects of N-alkyl chain on rat plasma and liver stability.
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  60. Targeting the endocannabinoid system to reduce nociception
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  61. Cannabinoid Type-1 Receptor Reduces Pain and Neurotoxicity Produced by Chemotherapy
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