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Allosteric Regulation of Proteases

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More Light Please: Daphnia Benefit From Light Pollution by Increased Tolerance Toward Cyanobacterial Chymotrypsin Inhibitors

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Recent advances in patented inhibitors targeting serine proteases in inflammatory diseases

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The literature of heterocyclic chemistry, Part XX, 2020

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Native Metabolomics Unveils Suomilide Analogs with Potent Trypsin Inhibitory Activity

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Side‐Chain Macrocyclization in Ahp‐Bicyclodepsipeptides Biosynthesis Involves Cytochrome P450‐Catalyzed Sequential Aromatic Hydroxylation and C─N Coupling

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Additional file 1 of Distribution and diversity of dimetal-carboxylate halogenases in cyanobacteria

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BindingDB Entry 50018761: Ahp-Cyclodepsipeptides as tunable inhibitors of human neutrophil elastase and kallikrein 7: Total synthesis of tutuilamide A, serine protease selectivity profile and comparison with lyngbyastatin 7.

BindingDB (2024) · UC San Diego · doi:10.7270/q2j96bm5

BindingDB Entry 50007683: Ahp-Cyclodepsipeptide Inhibitors of Elastase: Lyngbyastatin 7 Stability, Scalable Synthesis, and Focused Library Analysis.

BindingDB (2021) · UC San Diego · doi:10.7270/q28p63w5

BindingDB Entry 50017594: Design, synthesis and biological evaluation of P2-modified proline analogues targeting the HtrA serine protease in Chlamydia.

BindingDB (2023) · UC San Diego · doi:10.7270/q29s1w48

Synthese von Ahp-Cyclodepsipeptiden als Inhibitoren für Serinproteasen

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Chemistry and biology of natural product derived protease inhibitors

Stolze, S. C. (2012) · Technische Universität Dortmund Eldorado (Technische Universität Dortmund) · doi:10.17877/de290r-14335

Ahp Cyclodepsipeptides: The Impact of the Ahp Residue on the “Canonical Inhibition” of S1 Serine Proteases

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