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Nickel‐Catalyzed 1,2‐Diarylation of Alkenyl Carboxylates: A Gateway to 1,2,3‐Trifunctionalized Building Blocks

Derosa, J., Kang, T., Tran, V., Wisniewski, S. R., Karunananda, M. K., Jankins, T. C., Xu, K. L., & Engle, K. M. (2019) · Angewandte Chemie · doi:10.1002/ange.201913062 · Cited by 25 · see citing works

Economical Access to Diverse Enantiopure Tetrahydropyridines and Piperidines Enabled by Catalytic Borrowing Hydrogen

Ng, T. W., Tao, R., See, W. W. L., Poh, S. B., & Zhao, Y. (2022) · Angewandte Chemie International Edition · doi:10.1002/anie.202212528 · Cited by 24 · see citing works

Evolution of a Strategy for the Enantioselective Synthesis of (−)-Cajanusine

Guo, R., Witherspoon, B. P., & Brown, M. K. (2020) · Journal of the American Chemical Society · doi:10.1021/jacs.0c00359 · Cited by 24 · see citing works

Photoredox/Cu‐Catalyzed Decarboxylative C(sp3)−C(sp3) Coupling to Access C(sp3)‐Rich gem‐Diborylalkanes

Huang, M., Sun, H., Seufert, F., Friedrich, A., Marder, T. B., & Hu, J. (2024) · Angewandte Chemie International Edition · doi:10.1002/anie.202401782 · Cited by 18 · see citing works

A skeletally diverse library of bioactive natural-product-like compounds enabled by late-stage P450-catalyzed oxyfunctionalization

Bortz, A. R., Bennett, J. M., & Fasan, R. (2024) · Chem · doi:10.1016/j.chempr.2024.08.003 · Cited by 16 · see citing works

Ligand‐Enabled β‐Methylene C(sp 3 )−H Arylation of Masked Aliphatic Alcohols

Xia, G., Zhuang, Z., Liu, L., Schreiber, S. L., Melillo, B. N., & Yu, J. (2020) · Angewandte Chemie · doi:10.1002/ange.202000632 · Cited by 16 · see citing works

Non-natural 3-Arylmorpholino-β-amino Acid as a PPII Helix Inducer

Vaghi, F., Bucci, R., Clerici, F., Contini, A., & Gelmi, M. L. (2020) · Organic Letters · doi:10.1021/acs.orglett.0c02331 · Cited by 16 · see citing works

A Decarboxylative Cross-Coupling Platform To Access 2-Heteroaryl Azetidines: Building Blocks with Application in Medicinal Chemistry

Brewster, J. T., Randall, S. D., Kowalski, J. P., Cruz, C. L., Shoemaker, R. N., Tarlton, E., & Hinklin, R. J. (2022) · Organic Letters · doi:10.1021/acs.orglett.2c03852 · Cited by 15 · see citing works

Advances in amide and thioamide assisted C(sp3)H functionalization

Tan, P. W., & Seayad, J. (2019) · Tetrahedron Letters · doi:10.1016/j.tetlet.2019.151338 · Cited by 15 · see citing works

Enantioconvergent radical addition of racemic alkyl halides to access vicinal stereocentres

Wu, X., Xia, T., Bai, J., Shi, Y., Fang, C., Hu, J., Wu, W., Zhang, C., Wang, Q., Huang, G., et al. (2025) · Nature Chemistry · doi:10.1038/s41557-025-01967-w · Cited by 14 · see citing works

Stereoselective Palladium‐Catalyzed C( sp 3 )−H Mono‐Arylation of Piperidines and Tetrahydropyrans with a C(4) Directing Group

Piticari, A., Antermite, D., Higham, J. I., Moore, J. H., Webster, M. P., & Bull, J. A. (2022) · Advanced Synthesis & Catalysis · doi:10.1002/adsc.202200030 · Cited by 14 · see citing works

Vicinal stereocenters via asymmetric allylic alkylation and Cope rearrangement: a straightforward route to functionally and stereochemically rich heterocycles

Nilova, A., Mannchen, M. D., Noel, A. N., Semenova, E., & Grenning, A. J. (2023) · Chemical Science · doi:10.1039/d2sc07021a · Cited by 14 · see citing works

Di-ortho-C H arylation of phenylalanine: A bimetallic interaction between Pd(IV)-Ag(I)

Tao, Q., Li, Y.-N., Tang, W., Liu, P., Yu, F., & He, Y. (2021) · Tetrahedron Letters · doi:10.1016/j.tetlet.2021.153158 · Cited by 14 · see citing works

MIA-Directed 2-Pyridione-Enabled Selective Ortho-C–H Arylation of Phenylalanine: A Mechanistic Study

Niu, P., Liu, P., Meng, Y., Yu, F., & He, Y. (2021) · The Journal of Organic Chemistry · doi:10.1021/acs.joc.0c02872 · Cited by 14 · see citing works

On the Mechanism and Selectivity of Palladium-Catalyzed C(sp3)–H Arylation of Pyrrolidines and Piperidines at Unactivated C4 Positions: Discovery of an Improved Dimethylaminoquinoline Amide Directing Group

Antermite, D., White, A. J. P., Casarrubios, L., & Bull, J. A. (2023) · ACS Catalysis · doi:10.1021/acscatal.3c01980 · Cited by 13 · see citing works

Nickel-Catalyzed Chemo- and Regioselective Benzylarylation of Unactivated Alkenes with o-Bromobenzyl Chlorides

Wang, H., Huang, H., Gong, C., Diao, Y., Chen, J., Wu, S., & Wang, L. (2021) · Organic Letters · doi:10.1021/acs.orglett.1c03991 · Cited by 11 · see citing works

Alkyl Azetidines Via Batch and Flow Photochemistry

Datsenko, O. P., Baziievskyi, A., Sadkova, I. V., Campos, B., Brewster, J. T., Kowalski, J. P., Hinklin, R. J., & Mykhailiuk, P. K. (2025) · Organic Letters · doi:10.1021/acs.orglett.5c00922 · Cited by 10 · see citing works

Diastereoselective Synthesis of 2,3,4-Trisubstituted Tetrahydrofurans via Thermally Reactive 1,5-Diene- tert -butyl Carbonates

Emmetiere, F., & Grenning, A. J. (2020) · Organic Letters · doi:10.1021/acs.orglett.9b04306 · Cited by 10 · see citing works

Carboxylic Acid-Directed Manganese(I)-Catalyzed Regioselective Hydroarylation of Unactivated Alkenes

Han, J., Yu, H., & Zi, W. (2022) · Organic Letters · doi:10.1021/acs.orglett.2c02309 · Cited by 9 · see citing works

Economical Access to Diverse Enantiopure Tetrahydropyridines and Piperidines Enabled by Catalytic Borrowing Hydrogen

Ng, T. W., Tao, R., See, W. W. L., Poh, S. B., & Zhao, Y. (2022) · Angewandte Chemie · doi:10.1002/ange.202212528 · Cited by 6 · see citing works

Palladium-Catalyzed Intermolecular Functionalization of Unactivated Methylene C(sp3)—H Bonds

Mei, M., & Zhang, Y. (2025) · Chinese Journal of Organic Chemistry · doi:10.6023/cjoc202406012 · Cited by 5 · see citing works

Ready and selective access to 2-arylquinazolines from α-amino acids via a new solvent-free domino transformation under synergistic nano Fe-Mo-Se catalyst

Nguyen, K. X., Pham, P. H., Nguyen, A. C. D., Nguyen, C. T., Nguyen, T. T., Tran, P. D., & Phan, N. T. S. (2020) · Journal of Industrial and Engineering Chemistry · doi:10.1016/j.jiec.2020.08.027 · Cited by 5 · see citing works

Enantioselective Three‐Component Coupling of Heteroarenes, Cycloalkenes and Propargylic Acetates

Teng, S., Chi, Y. R., & Zhou, J. S. (2020) · Angewandte Chemie · doi:10.1002/ange.202014781 · Cited by 4 · see citing works

Pursuing high efficiency in photocatalytic oxidative couplings of heteroarenes and aliphatic C–H bonds

Zhang, L., Zhu, D., Hu, J., Feng, M., Sum, T. C., Sun, H., Hirao, H., Chi, Y. R., & Zhou, J. S. (2023) · Organic Chemistry Frontiers · doi:10.1039/d2qo01558g · Cited by 4 · see citing works

C–H Functionalization of Saturated Heterocycles Beyond the C2 Position

Piticari, A., Larionova, N. I., & Bull, J. A. (2023) · doi:10.1002/9781119774167.ch13 · Cited by 4 · see citing works

Photoredox/Cu‐Catalyzed Decarboxylative C(sp3)−C(sp3) Coupling to Access C(sp3)‐Rich gem‐Diborylalkanes

Huang, M., Sun, H., Seufert, F., Friedrich, A., Marder, T. B., & Hu, J. (2024) · Angewandte Chemie · doi:10.1002/ange.202401782 · Cited by 3 · see citing works

Recent advances in the late-stage modification of complex bioactive molecules with oxetanes and azetidines

Wang, Y., Tian, D., & Zhang, H. (2026) · Tetrahedron Chem · doi:10.1016/j.tchem.2026.100153 · Cited by 2 · see citing works

Azetidine-2-carboxylic Acid and Its Derivatives in Organic Synthesis

Pronina, Y. A., Berezhnaya, E. V., Slesarev, D. S., Drachuk, A., Ponyaev, A. I., Boitsov, V. M., & Stepakov, A. V. (2025) · Russian Journal of General Chemistry · doi:10.1134/s1070363224612559 · Cited by 1 · see citing works

Unlocking Enantioselectivity: Synergy of 2-Pyridone and Chiral Amino Acids in Pd-Catalyzed β-C(sp3)–H Transformations

Mandal, N., Mondal, P., Mandal, S., & Datta, A. (2024) · The Journal of Organic Chemistry · doi:10.1021/acs.joc.4c00078 · Cited by 1 · see citing works

Coupling Reaction Between sp3-Carbon Centers

Iwasaki, T. (2023) · Elsevier eBooks · doi:10.1016/b978-0-323-96025-0.00030-2 · Cited by 1 · see citing works

C–H Activation and Decarboxylative Cross-Coupling of Carboxylic Acids

Trauner, D. H., & Hetzler, B. E. (2019) · Synfacts · doi:10.1055/s-0039-1689765

Correction to “Catalytic Enantioselective Synthesis of a cis-β-Boronyl Cyclobutylcarboxyester Scaffold and Its Highly Diastereoselective Nickel/Photoredox Dual-Catalyzed Csp3–Csp2 Cross-Coupling to Access Elusive trans-β-Aryl/Heteroaryl Cyclobutylcarboxyesters”

Nguyen, K., Clement, H. A., Bernier, L., Coe, J. W., Farrell, W. P., Helal, C. J., Reese, M. R., Sach, N. W., Lee, J. C., & Hall, D. G. (2021) · ACS Catalysis · doi:10.1021/acscatal.1c01255

Arylboration of Enecarbamates for the Synthesis of Borylated Saturated N‐Heterocycles

Trammel, G. L., Kannangara, P. B., Vasko, D., Datsenko, O. P., Mykhailiuk, P. K., & Brown, M. K. (2022) · Angewandte Chemie · doi:10.1002/ange.202212117

Fused-ring α-pyrones from intramolecular C–H activation and their lipids-lowering activity associated with LXR-IDOL-LDLR axis regulation

Mao, Y., Li, J., Tang, C., Ma, B., Xu, Z., Ke, C., Lu, F., Zhang, H., Yao, S., Dai, H., et al. (2022) · European Journal of Medicinal Chemistry · doi:10.1016/j.ejmech.2022.114866

o-Halogenation and -Alkoxylation of Phenylglycine Derivatives by Pd-Mediated C-H Functionalization: Scope and Limitations

Laga, E., Nieto, S., Cativiela, C., & Urriolabeitia, E. P. (2025) · Molecules · doi:10.3390/molecules30020236

Regio‐ and Stereocontrolled‐Synthesis of a Heterocycle Fragment Collection Using Palladium Catalyzed C‐H Arylation

Piticari, A., Antermite, D., Linkhorn, H. J., Larionova, N. A., Webster, M. P., & Bull, J. A. (2025) · Chemistry - A European Journal · doi:10.1002/chem.202503126

Divergent reactivity of azetidine-2-carboxylic acid with amines: access to α-amino-γ-butyrolactams and N -aryl azetidine carboxamides

Sriharsha, C., Ravali, A., Sukumar, G., Jadav, S. S., & Adepu, R. (2026) · Chemical Communications · doi:10.1039/d6cc03205b

C–H Activation and Decarboxylative Cross-Coupling of Carboxylic Acids

Trauner, D. H., & Hetzler, B. E. (2019) · Synfacts · doi:10.1055/s-0039-1689765

Stereoselective C(sp2)–H Alkylation of Enamides with Unactivated Aliphatic Carboxylic Acids via Decarboxylative Cross-Coupling Reactions

Guo, J., Guan, T., Tao, J., Zhao, K., & Loh, T. (2019) · Organic Letters · doi:10.1021/acs.orglett.9b03169 · Cited by 56 · see citing works

Catalytic Decarbonylative Functionalization of C–H Bonds with Carboxylic Acids

Xu, L., Zhao, H., Xu, J., & Yang, J. (2025) · Synlett · doi:10.1055/s-0043-1775457

Carboxylic Acids as Directing Groups for C−H Bond Functionalization

Drapeau, M. P., & Gooßen, L. J. (2016) · Chemistry - A European Journal · doi:10.1002/chem.201603263 · Cited by 308 · see citing works

Recent advances in carboxyl-directed dimerizations and cascade annulations via C–H activations

Li, W.-D., Fan, J., LI, C. ‐., & Shi, X. (2025) · Chemical Communications · doi:10.1039/d4cc06722c · Cited by 14 · see citing works