Death associated with brorphine, an emerging novel synthetic opioid

Fentanyl Law Enforcement Submissions and Increases in Synthetic Opioid–Involved Overdose Deaths — 27 States, 2013–2014

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In vitro functional characterization of a panel of non-fentanyl opioid new psychoactive substances

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Matrix Effect and Cross-Reactivity of Select Amphetamine-Type Substances, Designer Analogues, and Putrefactive Amines using the Bio-Quant Direct ELISA Presumptive Assays for Amphetamine and Methamphetamine

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First Report on Brorphine: The Next Opioid on the Deadly New Psychoactive Substance Horizon?

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Fentanyl- and fentanyl analog-related deaths across five counties in Central New York between 2013 and 2017

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The Rise and Fall of Isotonitazene and Brorphine: Two Recent Stars in the Synthetic Opioid Firmament

Vandeputte, M. M., Krotulski, A. J., Papsun, D. M., Logan, B. K., & Stove, C. P. (2022) · Journal of Analytical Toxicology · doi:10.1093/jat/bkab082 · Cited by 71 · see citing works

Reports of Adverse Events Associated with Use of Novel Psychoactive Substances, 2017–2020: A Review

Mohr, A. L. A., Logan, B. K., Fogarty, M. F., Krotulski, A. J., Papsun, D. M., Kacinko, S. L., Huestis, M. A., & Ropero‐Miller, J. D. (2022) · Journal of Analytical Toxicology · doi:10.1093/jat/bkac023 · Cited by 72 · see citing works

Non-Fentanyl New Synthetic Opioids—An Update

Zawilska, J. B., Adamowicz, P., Kurpeta, M., & Wojcieszak, J. (2023) · Forensic Science International · doi:10.1016/j.forsciint.2023.111775 · Cited by 55 · see citing works

Proliferation of Novel Synthetic Opioids in Postmortem Investigations After Core-Structure Scheduling for Fentanyl-Related Substances

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New Psychoactive Substances Intoxications and Fatalities during the COVID-19 Epidemic

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In vitro functional assays as a tool to study new synthetic opioids at the μ-opioid receptor: Potential, pitfalls and progress

Vandeputte, M. M., Vasudevan, L., & Stove, C. P. (2022) · Pharmacology & Therapeutics · doi:10.1016/j.pharmthera.2022.108161 · Cited by 22 · see citing works

Pharmacological and metabolic characterization of the novel synthetic opioid brorphine and its detection in routine casework

Grafinger, K. E., Wilde, M., Otte, L., & Auwärter, V. (2021) · Forensic Science International · doi:10.1016/j.forsciint.2021.110989 · Cited by 21 · see citing works

Characteristics of fatal ‘novel’ synthetic opioid toxicity in Australia

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Elucidating the harm potential of brorphine analogues as new synthetic opioids: Synthesis, in vitro, and in vivo characterization

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Blood concentrations of new synthetic opioids

Adamowicz, P., & Nowak, K. (2021) · International Journal of Legal Medicine · doi:10.1007/s00414-021-02729-2 · Cited by 13 · see citing works

Application of Fabric Phase Sorptive Extraction (FPSE) Engaged to Tandem LC-MS/MS for Quantification of Brorphine in Oral Fluid

Florou, D., Vlachou, T., Sakkas, V. A., & Boumba, V. A. (2022) · Journal of Xenobiotics · doi:10.3390/jox12040025 · Cited by 9 · see citing works

Interpol review of toxicology 2019–2022

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Multi-analytical identification of the synthetic opioids cychlorphine and methiodone (IC-26) in drug seizures: first detection in Europe

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Brorphine and Its Analogues: Pharmacology, Toxicology, and Biomonitoring

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Fentanyl

(2021) · Reactions Weekly · doi:10.1007/s40278-021-02537-3

Metabolism of brorphine, chlorphine, fluorphine and N-propionitrile chlorphine in human hepatocytes and authentic N-propionitrile chlorphine case studies using high-resolution mass spectrometryPreprint

Gameli, P. S., Kronstrand, R., & Gréen, H. (2026) · Research Square · doi:10.21203/rs.3.rs-11241883/v1

In Vivo Pharmaco-Toxicological Characterization of Brorphine and its Possible Emerging Analogues Orphine, Fluorphine, Chlorphine and Iodorphine

Bilel, S., Vandeputte, M. M., Tirri, M., Corli, G., Stove, C. P., & Marti, M. (2024) · Emerging Trends in Drugs, Addictions, and Health · doi:10.1016/j.etdah.2023.100073 · Cited by 1 · see citing works

Death cases involving certain new psychoactive substances: A review of the literature

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Life (and death) in Pink: The dangerous rise of synthetic opioids in the new psychoactive substances panorama

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Novel Synthetic Opioids: The Pathologist’s Point of View

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The Rise and Fall of Isotonitazene and Brorphine: Two Recent Stars in the Synthetic Opioid Firmament

Vandeputte, M. M., Krotulski, A. J., Papsun, D. M., Logan, B. K., & Stove, C. P. (2022) · Journal of Analytical Toxicology · doi:10.1093/jat/bkab082 · Cited by 71 · see citing works