The DOI matches its Crossref record; 192 of the 192 references it cites were found in a registry or an index.
Update on melatonin receptors: IUPHAR Review 20
Open accessAbstract
Melatonin receptors are seven transmembrane‐spanning proteins belonging to the GPCR superfamily. In mammals, two melatonin receptor subtypes exist ‐ MT 1 and MT 2‐ encoded by the MTNR1A and MTNR1B genes respectively. The current review provides an update on melatonin receptors by the corresponding subcommittee of the International Union of Basic and Clinical Pharmacology. We will highlight recent developments of melatonin receptor ligands, including radioligands, and give an update on the latest phenotyping results of melatonin receptor knockout mice. The current status and perspectives of the structure of melatonin receptor will be summarized. The physiological importance of melatonin receptor dimers and biologically important and type 2 diabetes‐associated genetic variants of melatonin receptors will be discussed. The role of melatonin receptors in physiology and disease will be further exemplified by their functions in the immune system and the CNS. Finally, antioxidant and free radical scavenger properties of melatonin and its relation to melatonin receptors will be critically addressed.
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Cites
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Cited by
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Metadata
- Authors
- Jockers, R., Delagrange, P., Dubocovich, M. L., Markus, R. P., Renault, N., Tosini, G., Cecon, E., & Zlotos, D. P.
- Venue
- British Journal of Pharmacology
- Publisher
- Wiley
- Published
- 2016-08-08
- Volume
- 173
- Issue
- 18
- Pages
- 2702-2725
- ISSN
- 0007-1188 (ISSN-L)
- 1476-5381
- OpenAlex
- W2442143867
- Cited by
- 422
- References
- 192
- FWCI
- 18.60
- Type
- journal article
- Language
- en
- Open access
- bronze
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- Jockers, R., Delagrange, P., Dubocovich, M. L., Markus, R. P., Renault, N., Tosini, G., Cecon, E., & Zlotos, D. P. (2016). Update on melatonin receptors: IUPHAR Review 20. British Journal of Pharmacology. https://doi.org/10.1111/bph.13536
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Contains information from the Semantic Scholar Academic Graph Datasets, made available under the ODC Attribution License (ODC-BY 1.0).
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