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BindingDB Entry 50035383: Investigation of novel fumagillin analogues as angiogenesis inhibitors.

BindingDB (2012) · UC San Diego · doi:10.7270/q27p8zxd

BindingDB Entry 50021193: Emerging and Re-emerging Warheads for Targeted Covalent Inhibitors: An Update.

BindingDB (2025) · UC San Diego · doi:10.7270/q2vm4hvh

BindingDB Entry 50001481: Identification of the Histidine Residue in Vitamin D Receptor That Covalently Binds to Electrophilic Ligands.

BindingDB (2020) · UC San Diego · doi:10.7270/q2cf9snz

BindingDB Entry 50043055: Pyridinylpyrimidines selectively inhibit human methionine aminopeptidase-1.

BindingDB (2014) · UC San Diego · doi:10.7270/q290256x

BindingDB Entry 4625: Fumagillin and fumarranol interact with P. falciparum methionine aminopeptidase 2 and inhibit malaria parasite growth in vitro and in vivo.

BindingDB (2011) · UC San Diego · doi:10.7270/q2ws8rq5

BindingDB Entry 50042935: Pyridinylquinazolines selectively inhibit human methionine aminopeptidase-1 in cells.

BindingDB (2014) · UC San Diego · doi:10.7270/q2sj1n1z

BindingDB Entry 50011328: Structure-based optimisation of orally active & reversible MetAP-2 inhibitors maintaining a tight 'molecular budget'.

BindingDB (2022) · UC San Diego · doi:10.7270/q2n58qzh

BindingDB Entry 50018496: Anticancer fungal natural products: Mechanisms of action and biosynthesis.

BindingDB (2024) · UC San Diego · doi:10.7270/q2n58rmf

BindingDB Entry 50014379: 3-Amino-2-hydroxyamides and related compounds as inhibitors of methionine aminopeptidase-2.

BindingDB (2009) · UC San Diego · doi:10.7270/q2z31z3n

BindingDB Entry 50014030: Peptidyl hydroxamic acids as methionine aminopeptidase inhibitors.

BindingDB (2009) · UC San Diego · doi:10.7270/q2dv1j90

BindingDB Entry 50007812: Emerging and Re-Emerging Warheads for Targeted Covalent Inhibitors: Applications in Medicinal Chemistry and Chemical Biology.

BindingDB (2021) · UC San Diego · doi:10.7270/q2959mwn

BindingDB Entry 2187: The 1.15A crystal structure of the Staphylococcus aureus methionyl-aminopeptidase and complexes with triazole based inhibitors.

BindingDB (2007) · UC San Diego · doi:10.7270/q2c53j49

BindingDB Entry 50045953: Metabolites of PPI-2458, a selective, irreversible inhibitor of methionine aminopeptidase-2: structure determination and in vivo activity.

BindingDB (2016) · UC San Diego · doi:10.7270/q2nc62xh

BindingDB Entry 7157: Spiroepoxytriazoles Are Fumagillin-like Irreversible Inhibitors of MetAP2 with Potent Cellular Activity.

BindingDB (2016) · UC San Diego · doi:10.7270/q23j3bqr

Protonation States of Methionine Aminopeptidase Studied by QM/MM Car-Parrinello Molecular Dynamics Simulations

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Spiroepoxytriazoles Are Fumagillin-like Irreversible Inhibitors of MetAP2 with Potent Cellular Activity

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