Receptor-independent actions of PPAR thiazolidinedione agonists: Is mitochondrial function the key?

Feinstein, D.L., Spagnolo, A., Akar, C., Weinberg, G., Murphy, P., Gavrilyuk, V., Russo, C. Dello·2005·Biochemical Pharmacology

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  44. Design and Synthesis of Biotinylated Troglitazone as an Active Affinity Probe
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  48. Efecto hipoglicemiante coadyuvante del extracto etanólico de hojas de Annona muricata L (guanábana), en pacientes con diabetes tipo 2 bajo tratamiento de glibenclamida Coadjuvant hypoglycemiant effect of Annona muricata L (guanabana) leaves ethanolic extract in patients with type 2 diabetes mellitus receiving glibenclamide treatment
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  69. Additional file 2 of The troglitazone derivative EP13 disrupts energy metabolism through respiratory chain complex I inhibition in breast cancer cells and potentiates the antiproliferative effect of glycolysis inhibitors
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  70. Additional file 1 of The troglitazone derivative EP13 disrupts energy metabolism through respiratory chain complex I inhibition in breast cancer cells and potentiates the antiproliferative effect of glycolysis inhibitntriors
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  75. BindingDB Entry 50004305: Structure-based design of a thiazolidinedione which targets the mitochondrial protein mitoNEET.
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  76. BindingDB Entry 50023020: Rational design and synthesis of novel N-benzylindole-based epalrestat analogs as selective aldose reductase inhibitors: An unexpected discovery of a new glucose-lowering agent (AK-4) acting as a mitochondrial uncoupler.
    BindingDB · 2026 · UC San Diego
  77. BindingDB Entry 50033824: A novel binding assay identifies high affinity ligands to the rosiglitazone binding site of mitoNEET.
    BindingDB · 2012 · UC San Diego
  78. BindingDB Entry 50003080: PPARγ-sparing thiazolidinediones as insulin sensitizers. Design, synthesis and selection of compounds for clinical development.
    BindingDB · 2020 · UC San Diego