The DOI matches its Crossref record; 23 of the 23 references it cites were found in a registry or an index.
Progress with covalent small-molecule kinase inhibitors
Open accessAbstract
With reduced risk of toxicity and high selectivity, covalent small-molecule kinase inhibitors (CSKIs) have emerged rapidly. Through the lens of structural system pharmacology, here we review this rapid progress by considering design strategies and the challenges and opportunities offered by current CSKIs.
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Cited by
Advances in covalent drug discovery
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Rapid Covalent-Probe Discovery by Electrophile-Fragment Screening
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Advances in covalent kinase inhibitors
Abdeldayem, A., Raouf, Y. S., Constantinescu, S. N., Moriggl, R., & Gunning, P. T. (2020) · Chemical Society Reviews · doi:10.1039/c9cs00720b · Cited by 317
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Covalent Inhibition in Drug Discovery
Ghosh, A. K., Samanta, I., Mondal, A., & Liu, W. R. (2019) · ChemMedChem · doi:10.1002/cmdc.201900107 · Cited by 265
Metadata
- Authors
- Zhao, Z., & Bourne, P. E.
- Venue
- Drug Discovery Today
- Publisher
- Elsevier BV
- Published
- 2018-03
- Volume
- 23
- Issue
- 3
- Pages
- 727-735
- ISSN
- 1359-6446 (ISSN-L)
- OpenAlex
- W2783904016
- Cited by
- 194
- References
- 23
- FWCI
- 9.50
- Type
- journal article
- Language
- en
- Open access
- hybrid
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Contains information from the Semantic Scholar Academic Graph Datasets, made available under the ODC Attribution License (ODC-BY 1.0).
Semantic Scholar’s data is described in: Kinney, R., et al. (2023). The Semantic Scholar Open Data Platform. arXiv:2301.10140.
