Peptide Coupling Reagents, More than a Letter Soup

Controlled Microwave Heating in Modern Organic Synthesis

Kappe, C. O. (2004) · Angewandte Chemie International Edition · doi:10.1002/anie.200400655 · Cited by 3,628 · see citing works

Amide bond formation: beyond the myth of coupling reagents

Valeur, E., & Bradley, M. (2008) · Chemical Society Reviews · doi:10.1039/b701677h · Cited by 2,209 · see citing works

Amide bond formation and peptide coupling

Montalbetti, C., & Falque, V. M. (2005) · Tetrahedron · doi:10.1016/j.tet.2005.08.031 · Cited by 1,789 · see citing works

Eine neue Methode zur Synthese von Peptiden: Aktivierung der Carboxylgruppe mit Dicyclohexylcarbodiimid unter Zusatz von 1‐Hydroxy‐benzotriazolen

König, W., & Geiger, R. (1970) · Chemische Berichte · doi:10.1002/cber.19701030319 · Cited by 1,580 · see citing works

1-Hydroxy-7-azabenzotriazole. An efficient peptide coupling additive

Carpino, L. A. (1993) · Journal of the American Chemical Society · doi:10.1021/ja00063a082 · Cited by 1,494 · see citing works

A New Method of Forming Peptide Bonds

Sheehan, J. C., & Hess, G. P. (1955) · Journal of the American Chemical Society · doi:10.1021/ja01609a099 · Cited by 1,264 · see citing works

The Use of Esters of N-Hydroxysuccinimide in Peptide Synthesis

Anderson, G. W., Zimmerman, J. E., & Callahan, F. M. (1964) · Journal of the American Chemical Society · doi:10.1021/ja01063a037 · Cited by 1,241 · see citing works

Chemical Synthesis of Natural Product Peptides: Coupling Methods for the Incorporation of Noncoded Amino Acids into Peptides

Humphrey, J. M., & Chamberlin, A. R. (1997) · Chemical Reviews · doi:10.1021/cr950005s · Cited by 1,165 · see citing works

New coupling reagents in peptide chemistry

Knorr, R., Trzeciak, A., Bannwarth, W., & Gillessen, D. (1989) · Tetrahedron Letters · doi:10.1016/s0040-4039(00)99616-3 · Cited by 996 · see citing works

Tertiary Phosphane/Tetrachloromethane, a Versatile Reagent for Chlorination, Dehydration, and PN Linkage

Appel, R. (1975) · Angewandte Chemie International Edition in English · doi:10.1002/anie.197508011 · Cited by 944 · see citing works

Über ein allgemeines Verfahren der Peptid‐Synthese

Bergmann, M. F., & Zervas, L. (1932) · Berichte der deutschen chemischen Gesellschaft (A and B Series) · doi:10.1002/cber.19320650722 · Cited by 785 · see citing works

Recent development of peptide coupling reagents in organic synthesis

Han, S., & Kim, Y. (2004) · Tetrahedron · doi:10.1016/j.tet.2004.01.020 · Cited by 776 · see citing works

Reactifs de couplage peptidique I (1) - l'hexafluorophosphate de benzotriazolyl N-oxytrisdimethylamino phosphonium (B.O.P.)

CASTRO, B., Dormoy, J., Evin, G. M., & Selve, C. (1975) · Tetrahedron Letters · doi:10.1016/s0040-4039(00)72100-9 · Cited by 647 · see citing works

PyBOP®: A new peptide coupling reagent devoid of toxic by-product

Coste, J. H., Le‐Nguyen, D., & CASTRO, B. (1990) · Tetrahedron Letters · doi:10.1016/s0040-4039(00)94371-5 · Cited by 626 · see citing works

Chemistry and Biology of Peptides

Gitu, P. M., Hruby, V., Brown, W. S., & Muscio, F. (1972) · Cited by 614 · see citing works

Peptides: Chemistry and Biology

Sewald, N., & Jakubke, H. (2009) · Wiley eBooks · doi:10.1002/9783527626038 · Cited by 451 · see citing works

Principles of Peptide Synthesis

Bodanszky, M. (1993) · Springer eBooks · doi:10.1007/978-3-642-78056-1 · Cited by 439 · see citing works

Oxyma: An Efficient Additive for Peptide Synthesis to Replace the Benzotriazole‐Based HOBt and HOAt with a Lower Risk of Explosion ^[1]

Subirós‐Funosas, R., Prohens, R., Barbas, R., El‐Faham, A., & Albericio, F. (2009) · Chemistry – A European Journal · doi:10.1002/chem.200900614 · Cited by 421 · see citing works

New convenient reagent for peptide syntheses

Belleau, B., & Mälek, G. (1968) · Journal of the American Chemical Society · doi:10.1021/ja01008a045 · Cited by 415 · see citing works

Reinvestigation of the mixed carbonic anhydride method of peptide synthesis

Anderson, G. W., Zimmerman, J. E., & Callahan, F. M. (1967) · Journal of the American Chemical Society · doi:10.1021/ja00995a032 · Cited by 407 · see citing works

Une nouvelle méthode de synthèse peptidique

Boissonnas, R. A. (1951) · Helvetica Chimica Acta · doi:10.1002/hlca.19510340318 · Cited by 389 · see citing works

Advantageous applications of azabenzotriazole (triazolopyridine)-based coupling reagents to solid-phase peptide synthesis

Carpino, L. A., El‐Faham, A., Minor, C. A., & Alberício, F. (1994) · Journal of the Chemical Society Chemical Communications · doi:10.1039/c39940000201 · Cited by 352 · see citing works

Ueber die Glycin‐carbonsäure

Leuchs, H. (1906) · Berichte der deutschen chemischen Gesellschaft · doi:10.1002/cber.190603901133 · Cited by 331 · see citing works

N,N'-Carbonyldiimidazole, a New Peptide Forming Reagent1

Paul, R., & Anderson, G. W. (1960) · Journal of the American Chemical Society · doi:10.1021/ja01502a038 · Cited by 308 · see citing works

COMU: A Safer and More Effective Replacement for Benzotriazole‐Based Uronium Coupling Reagents

El‐Faham, A., Subirós‐Funosas, R., Prohens, R., & Alberício, F. (2009) · Chemistry - A European Journal · doi:10.1002/chem.200900615 · Cited by 306 · see citing works

Über Peptid‐Synthesen. 3. Mitteilung. Die Verwendung von Anhydriden aus N‐acylierten Aminosäuren und Derivaten anorganischer Säuren

Wieland, T., & Bernhard, H. (1951) · Justus Liebig s Annalen der Chemie · doi:10.1002/jlac.19515720115 · Cited by 290 · see citing works

The Preparation of Peptides Using Mixed Carbonic—Carboxylic Acid Anhydrides

Vaughan, J. R., & Osato, R. L. (1952) · Journal of the American Chemical Society · doi:10.1021/ja01123a028 · Cited by 288 · see citing works

Backbone Amide Linker (BAL) Strategy for Solid-Phase Synthesis of C-Terminal-Modified and Cyclic Peptides1,2,3

Jensen, K. J., Alsina, J., Songster, M. F., Vágner, J., Alberício, F., & Bárány, G. (1998) · Journal of the American Chemical Society · doi:10.1021/ja974116f · Cited by 275 · see citing works

O-Benzotriazolyl-N,N,N′,N′-tetramethyluronium Hexafluorophosphate as Coupling Reagent for the Synthesis of Peptides of Biological Interest

Dourtoglou, V. G., Gross, B., Lambropoulou, V., & Zioudrou, C. (1984) · Synthesis · doi:10.1055/s-1984-30895 · Cited by 275 · see citing works

Use of Onium Salt-Based Coupling Reagents in Peptide Synthesis1

Alberício, F., Bofill, J. M., El‐Faham, A., & Kates, S. A. (1998) · The Journal of Organic Chemistry · doi:10.1021/jo980807y · Cited by 273 · see citing works

Extending the Applicability of Native Chemical Ligation

Canne, L. E., Bark, S. J., & Kent, S. B. H. (1996) · Journal of the American Chemical Society · doi:10.1021/ja960398s · Cited by 268 · see citing works

Synthesis of Peptides by Aminolysis of Nitrophenyl Esters

BODÁNSZKY, M. (1955) · Nature · doi:10.1038/175685a0 · Cited by 268 · see citing works

ACYLALKYLCARBONATES AS ACYLATING AGENTS FOR THE SYNTHESIS OF PEPTIDES

Vaughan, J. R. (1951) · Journal of the American Chemical Society · doi:10.1021/ja01151a554 · Cited by 263 · see citing works

Tetramethylfluoroformamidinium Hexafluorophosphate: A Rapid-Acting Peptide Coupling Reagent for Solution and Solid Phase Peptide Synthesis

Carpino, L. A., & El‐Faham, A. (1995) · Journal of the American Chemical Society · doi:10.1021/ja00124a040 · Cited by 262 · see citing works

New Amine-masking Groups for Peptide Synthesis

McKay, F. C., & Albertson, N. F. (1957) · Journal of the American Chemical Society · doi:10.1021/ja01574a029 · Cited by 256 · see citing works

Principles of Peptide Synthesis

Bodanszky, M. (1984) · Reactivity and structure · doi:10.1007/978-3-642-96763-4 · Cited by 242 · see citing works

Recent developments in the carbodiimide chemistry

lajczyk, M. M. X., & lbasiński, P. K. X. (1981) · Tetrahedron · doi:10.1016/s0040-4020(01)92010-1 · Cited by 241 · see citing works

Methodological implications of simultaneous solid-phase peptide synthesis. 1. Comparison of different coupling procedures

Hudson, D. (1988) · The Journal of Organic Chemistry · doi:10.1021/jo00238a026 · Cited by 239 · see citing works

[(9-Fluorenylmethyl)oxy]carbonyl (FMOC) amino acid fluorides. Convienient new peptide coupling reagents applicable to the FMOC/tert-butyl strategy for solution and solid-phase syntheses.

Carpino, L. A., Sadat-Aalaee, D., Chao, H. G., & DeSelms, R. H. (1990) · Journal of the American Chemical Society · doi:10.1021/ja00182a041 · Cited by 234 · see citing works

3-(Diethoxyphosphoryloxy)-1,2,3- benzotriazin-4(3H)-one (DEPBT): A New Coupling Reagent with Remarkable Resistance to Racemization

Li, H., Jiang, X., Ye, Y., Fan, C., Romoff, T. T., & Goodman, M. (1999) · Organic Letters · doi:10.1021/ol990573k · Cited by 232 · see citing works

Peptide Synthesis via Amino Acid Halides

Carpino, L. A., Beyermann, M., Wenschuh, H., & Bienert, M. (1996) · Accounts of Chemical Research · doi:10.1021/ar950023w · Cited by 227 · see citing works

PyBOP® and PyBroP: Two reagents for the difficult coupling of the α,α-dialkyl amino acid, Aib.

Frérot, E., Coste, J. H., Pantaloni, A., Dufour, M.-N., & Jouin, P. (1991) · Tetrahedron · doi:10.1016/s0040-4020(01)80922-4 · Cited by 227 · see citing works

A New Reagent for Activating Carboxyl Groups; Preparation and Reactions ofN,N-Bis[2-oxo-3-ox-azolidinyl]phosphorodiamidic Chloride

Diago-Meseguer, J., PALOMO‐COLL, A. L., Fernández-Lizarbe, J. R., & Zugaza-Bilbao, A. (1980) · Synthesis · doi:10.1055/s-1980-29116 · Cited by 223 · see citing works

Racemization studies during solid-phase peptide synthesis using azabenzotriazole-based coupling reagents

Carpino, L. A., El‐Faham, A., & Alberício, F. (1994) · Tetrahedron Letters · doi:10.1016/0040-4039(94)85198-0 · Cited by 212 · see citing works

N-Acylbenzotriazoles: Neutral Acylating Reagents for the Preparation of Primary, Secondary, and Tertiary Amides

KATRITZKY, A. R., He, H., & Suzuki, K. (2000) · The Journal of Organic Chemistry · doi:10.1021/jo000792f · Cited by 208 · see citing works

Synthesis of acyl halides under very mild conditions

Devos, A., REMION, J., FRISQUE‐HESBAIN, A. ‐., Colens, A., & Ghosez, L. (1979) · Journal of the Chemical Society Chemical Communications · doi:10.1039/c39790001180 · Cited by 203 · see citing works

Synthesis and characterization of 4-(4,6-dimethoxy-1,3,5-triazin-2-yl)-4-methylmorpholinium chloride

Kunishima, M., Kawachi, C., Iwasaki, F., Terao, K., & Tani, S. (1999) · Tetrahedron Letters · doi:10.1016/s0040-4039(99)00968-5 · Cited by 198 · see citing works

Solvent-free preparation of amides from acids and primary amines under microwave irradiation

Perreux, L., Loupy, A., & Volatron, F. (2002) · Tetrahedron · doi:10.1016/s0040-4020(02)00085-6 · Cited by 196 · see citing works

(Fluoren-9-ylmethoxy)carbonyl (Fmoc) amino acid chlorides. Synthesis, characterization, and application to the rapid synthesis of short peptide segments

Carpino, L. A., Cohen, B. J., STEPHENS, K. E. J., Sadat-Aalaee, S. Y., Tien, J. H., & Langridge, D. C. (1986) · The Journal of Organic Chemistry · doi:10.1021/jo00369a042 · Cited by 195 · see citing works

Efficiency in Peptide Coupling: 1-Hydroxy-7-azabenzotriazole vs 3,4-Dihydro-3-hydroxy-4-oxo-1,2,3-benzotriazine

Carpino, L. A., El‐Faham, A., & Alberício, F. (1995) · The Journal of Organic Chemistry · doi:10.1021/jo00116a054 · Cited by 195 · see citing works

L'hexafluorophosphate de O-benzotriazolyl-N,N-tetramethyluronium: Un reactif de couplage peptidique nouveau et efficace

Dourtoglou, V. G., Ziegler, J.-C., & Gross, B. (1978) · Tetrahedron Letters · doi:10.1016/0040-4039(78)80103-8 · Cited by 192 · see citing works

New Peptide Synthesis

Wissmann, H., & Kleiner, H. (1980) · Angewandte Chemie International Edition in English · doi:10.1002/anie.198001331 · Cited by 186 · see citing works

The 9-fluorenylmethyloxycarbonyl family of base-sensitive amino-protecting groups

Carpino, L. A. (1987) · Accounts of Chemical Research · doi:10.1021/ar00143a003 · Cited by 185 · see citing works

Solid-Phase Synthesis of Difficult Peptide Sequences at Elevated Temperatures: A Critical Comparison of Microwave and Conventional Heating Technologies

Bacsa, B., Horváti, K., Bősze, S. E., Andreae, F., & Kappe, C. O. (2008) · The Journal of Organic Chemistry · doi:10.1021/jo8013897 · Cited by 180 · see citing works

Explosive properties of 1-hydroxybenzotriazoles

Wehrstedt, K., Wandrey, P., & Heitkamp, D. (2005) · Journal of Hazardous Materials · doi:10.1016/j.jhazmat.2005.05.044 · Cited by 175 · see citing works

On the use of PyAOP, a phosphonium salt derived from HOAt, in solid-phase peptide synthesis

Alberício, F., Cases, M., Alsina, J., Triolo, S. A., Carpino, L. A., & Kates, S. A. (1997) · Tetrahedron Letters · doi:10.1016/s0040-4039(97)01011-3 · Cited by 171 · see citing works

Synthetische Versuche mit Hippurazid

Curtius, T. (1902) · Berichte der deutschen chemischen Gesellschaft · doi:10.1002/cber.190203503125 · Cited by 170 · see citing works

Cyclization ofall- l -Pentapeptides by Means of 1-Hydroxy-7-azabenzotriazole-Derived Uronium and Phosphonium Reagents

Ehrlich, A., Heyne, H., Winter, R., Beyermann, M., Haber, H., Carpino, L. A., & Bienert, M. (1996) · The Journal of Organic Chemistry · doi:10.1021/jo951108d · Cited by 158 · see citing works

THE PEPTIDES: Analysis, Synthesis, Biology

(1979) · Elsevier eBooks · doi:10.1016/b978-0-12-304201-9.50001-1 · Cited by 158 · see citing works

Coupling Reagents in Peptide Synthesis

Klausner, Y. S., & Bodansky, M. (1972) · Synthesis · doi:10.1055/s-1972-21899 · Cited by 157 · see citing works

Novel Amine Chemistry Based on DMAP-Catalyzed Acylation

Ragnarsson, U., & Grehn, L. (1998) · Accounts of Chemical Research · doi:10.1021/ar980001k · Cited by 156 · see citing works

Coupling N-Methylated Amino Acids Using PyBroP and PyCloP Halogenophosphonium Salts: Mechanism and Fields of Application

Coste, J. H., Frérot, E., & Jouin, P. (1994) · The Journal of Organic Chemistry · doi:10.1021/jo00088a027 · Cited by 156 · see citing works

<i>N</i>-Triazinylammonium Tetrafluoroborates. A New Generation of Efficient Coupling Reagents Useful for Peptide Synthesis

Kamiński, Z. J., Kolesińska, B., Kolesińska, J., Sabatino, G., Chelli, M., Rovero, P., Błaszczyk, M., Główka, M. L., & Papini, A. M. (2005) · Journal of the American Chemical Society · doi:10.1021/ja054260y · Cited by 155 · see citing works

Preparation and Applications of Pentafluorophenyl Esters of 9-Fluorenylmethyloxycarbonyl Amino Acids for Peptide Synthesis

KISFALUDY, L., & Schön, I. (1983) · Synthesis · doi:10.1055/s-1983-30327 · Cited by 151 · see citing works

Preparation of Peptides Using Mixed Carboxylic Acid Anhydrides

Vaughan, J. R., & Osato, R. L. (1951) · Journal of the American Chemical Society · doi:10.1021/ja01156a011 · Cited by 150 · see citing works

Reaktionsfähige Heterocyclische Diamide Der Kohlensäure

Staab, H. A. (1957) · Justus Liebig s Annalen der Chemie · doi:10.1002/jlac.19576090108 · Cited by 148 · see citing works

NEW TRENDS IN PEPTIDE COUPLING REAGENTS

Alberício, F., Chinchílla, R., Dodsworth, D. J., & Nájera, C. (2001) · Organic Preparations and Procedures International · doi:10.1080/00304940109356592 · Cited by 143 · see citing works

Darstellung von Imidazoliden. Synthese von Amiden, Hydraziden und Hydroxamsäuren nach der Imidazolidmethode

Staab, H. A., Lüking, M., & Dürr, F. H. (1962) · Chemische Berichte · doi:10.1002/cber.19620950526 · Cited by 142 · see citing works

Peptide Coupling Reagents VI1. A Novel, Cheaper Preparation of Benzotriazolyloxytris[dimethylamino]phosphonium Hexafluorophosphate (BOP Reagent)

CASTRO, B., Dormoy, J., DOURTOGLOU, B., Evin, G. M., Selve, C., & Ziegler, J.-C. (1976) · Synthesis · doi:10.1055/s-1976-24189 · Cited by 137 · see citing works

The diisopropylcarbodiimide/ 1-hydroxy-7-azabenzotriazole system: Segment coupling and stepwise peptide assembly

Carpino, L. A., & El‐Faham, A. (1999) · Tetrahedron · doi:10.1016/s0040-4020(99)00344-0 · Cited by 135 · see citing works

Side Reactions in Peptide Synthesis

Bodanszky, M., & Martínez, J. (1981) · Synthesis · doi:10.1055/s-1981-29442 · Cited by 133 · see citing works

A FACILE SYNTHESIS OF CARBOXAMIDES BY USING 1-METHYL-2-HALOPYRIDINIUM IODIDES AS COUPLING REAGENTS

Bald, E., Saigo, K., & Mukaiyama, T. (1975) · Chemistry Letters · doi:10.1246/cl.1975.1163 · Cited by 131 · see citing works

Stepwise Automated Solid Phase Synthesis of Naturally Occurring Peptaibols Using FMOC Amino Acid Fluorides

Wenschuh, H., Beyermann, M., Haber, H., Seydel, J. K., Krause, E., Bienert, M., Carpino, L. A., El‐Faham, A., & Alberício, F. (1995) · The Journal of Organic Chemistry · doi:10.1021/jo00107a020 · Cited by 129 · see citing works

tert-Butyloxycarbonyl and benzyloxycarbonyl amino acid fluorides. New, stable rapid-acting acylating agents for peptide synthesis

Carpino, L. A., Mansour, E. M. E., & Sadat-Aalaee, D. (1991) · The Journal of Organic Chemistry · doi:10.1021/jo00008a005 · Cited by 128 · see citing works

Urethane protected amino acid N-carboxyanhydrides and their use in peptide synthesis

Fuller, W. D., Cohen, M. P., Shabankareh, M., Blair, R. K., Goodman, M., & Naider, F. R. (1990) · Journal of the American Chemical Society · doi:10.1021/ja00176a063 · Cited by 127 · see citing works

A NOVEL ACTIVATED ESTER IN PEPTIDE SYNTHESES

Nefkens, G. H. L., & TESSER, G. I. (1961) · Journal of the American Chemical Society · doi:10.1021/ja01466a068 · Cited by 126 · see citing works

A Study on the Activation of Carboxylic Acids by Means of 2-Chloro-4,6-dimethoxy-1,3,5-triazine and 2-Chloro-4,6-diphenoxy-1,3,5-triazine

Kaminski, Z. J., Paneth, P., & Rudziński, J. (1998) · The Journal of Organic Chemistry · doi:10.1021/jo972020y · Cited by 124 · see citing works

Cyanuric chloride : a useful reagent for converting carboxylic acids into chlorides, esters, amides and peptides

Venkataraman, K., & Wagle, D. R. (1979) · Tetrahedron Letters · doi:10.1016/s0040-4039(00)71006-9 · Cited by 123 · see citing works

Evolving Strategies for Protein Synthesis Converge on Native Chemical Ligation

Macmillan, D. (2006) · Angewandte Chemie International Edition · doi:10.1002/anie.200602945 · Cited by 123 · see citing works

Polymer bound EDC (P-EDC): A convenient reagent for formation of an amide bond

Desai, M. C., & Stramiello, L. M. S. (1993) · Tetrahedron Letters · doi:10.1016/s0040-4039(00)61539-3 · Cited by 122 · see citing works

Reaction of tert-butyldimethylsilyl esters with oxalyl chloride-dimethylformamide: preparation of carboxylic acid chlorides under neutral conditions

Wissner, A., & Grudzinskas, C. V. (1978) · The Journal of Organic Chemistry · doi:10.1021/jo00414a041 · Cited by 120 · see citing works

Peptide synthesis

Atherton, E., Cameron, L. R., & Sheppard, R. C. (1988) · Tetrahedron · doi:10.1016/s0040-4020(01)86121-4 · Cited by 115 · see citing works

Fmoc Amino Acid Fluorides: Convenient Reagents for the Solid-PhaseAssembly of Peptides Incorporating Sterically Hindered Residues

Wenschuh, H., Beyermann, M., Krause, E., Brudel, M., Winter, R., Schuemann, M., Carpino, L. A., & Bienert, M. (1994) · The Journal of Organic Chemistry · doi:10.1021/jo00091a011 · Cited by 115 · see citing works

Preparation of Acyl Halides under Very Mild Conditions

Lee, J. B. (1966) · Journal of the American Chemical Society · doi:10.1021/ja00966a052 · Cited by 109 · see citing works

Structural studies of reagents for peptide bond formation: Crystal and molecular structures of HBTU and HATU

Abdelmoty, I., Alberício, F., Carpino, L. A., Foxman, B. M., & Kates, S. A. (1994) · Letters in Peptide Science · doi:10.1007/bf00126274 · Cited by 105 · see citing works

Simple method for the synthesis of amides

Barstow, L. E., & Hruby, V. J. (1971) · The Journal of Organic Chemistry · doi:10.1021/jo00808a033 · Cited by 102 · see citing works

2-Chloro-4,6-dimethoxy-1,3,5-triazine. A New Coupling Reagent for Peptide Synthesis

Kaminski, Z. J. (1987) · Synthesis · doi:10.1055/s-1987-28122 · Cited by 98 · see citing works

Water-Soluble Phosphinothiols for Traceless Staudinger Ligation and Integration with Expressed Protein Ligation

Tam, A., Soellner, M. B., & Raines, R. T. (2007) · Journal of the American Chemical Society · doi:10.1021/ja073204p · Cited by 98 · see citing works

A CONVENIENT METHOD FOR THE CONSTRUCTION OF β-LACTAM COMPOUNDS FROM β-AMINO ACIDS USING 2-CHLORO-1-METHYLPYRIDINIUM IODIDE AS CONDENSING REAGENT

Huang, H., Iwasawa, N., & Mukaiyama, T. (1984) · Chemistry Letters · doi:10.1246/cl.1984.1465 · Cited by 96 · see citing works

Versatile Acylation ofN-Nucleophiles Using a New Polymer-Supported 1-Hydroxybenzotriazole Derivative

Pop, I. E., Deprez, B. P., & Tartar, A. L. (1997) · The Journal of Organic Chemistry · doi:10.1021/jo961761g · Cited by 96 · see citing works

The use of N-hydroxy-5-norbornene-2,3-dicarboximide acitive esters in peptide synthesis.

Fujino, M., Kobayashi, S., OBAYASHI, M., Fukuda, T., Shinagawa, S., & Nishimura, O. (1974) · Chemical and Pharmaceutical Bulletin · doi:10.1248/cpb.22.1857 · Cited by 96 · see citing works

Polypeptides with Known Repeating Sequence of Amino Acids. Synthesis of Poly-L-glutamyl-L-alanyl-L-glutamic Acid and Polyglycylglycyl-L-phenylalanine through Pentachlorophenyl Active Ester1

Kovacs, J. A., Giannotti, R., & Kapoor, A. (1966) · Journal of the American Chemical Society · doi:10.1021/ja00962a035 · Cited by 96 · see citing works

Polymeric reagents I. Synthesis of an insoluble polymeric carbodiimide

Weinshenker, N. M., & Shen, C. M. (1972) · Tetrahedron Letters · doi:10.1016/s0040-4039(01)94023-7 · Cited by 94 · see citing works

Peptide Coupling in the Presence of Highly Hindered Tertiary Amines

Carpino, L. A., Ionescu, D., & El‐Faham, A. (1996) · The Journal of Organic Chemistry · doi:10.1021/jo950912x · Cited by 93 · see citing works

Solid-Phase Peptide Synthesis in Water Using Microwave-Assisted Heating

Galanis, A., Alberício, F., & Grøtli, M. (2009) · Organic Letters · doi:10.1021/ol901893p · Cited by 91 · see citing works

Über Peptidsynthesen V. Über eine bequeme Darstellungsweise von Acylthiophenolen und ihre Verwendung zu Amid‐ und Peptid‐Synthesen

Wieland, T., Schäfer, W., & Bokelmann, E. (1951) · Justus Liebig s Annalen der Chemie · doi:10.1002/jlac.19515730110 · Cited by 91 · see citing works

1-Ethyl 2-Halopyridinium Salts, Highly Efficient Coupling Reagents for Hindered Peptide Synthesis both in Solution and the Solid-Phase

Li, P., & Xu, J. (2000) · Tetrahedron · doi:10.1016/s0040-4020(00)00657-8 · Cited by 90 · see citing works

New Useful Reagents for Peptide Synthesis. Insoluble Active Esters of Polystyrene-Bound 1-Hydroxybenzotriazole

Kalir, R., Warshawsky, A., Fridkin, M., & Patchornik, A. (1975) · European Journal of Biochemistry · doi:10.1111/j.1432-1033.1975.tb02424.x · Cited by 88 · see citing works

A Novel Organophosphorus Compound as a Coupling Reagent for Peptide Synthesis

Fan, C., Hao, X., & Ye, Y. (1996) · Synthetic Communications · doi:10.1080/00397919608003508 · Cited by 88 · see citing works

Efficient Conversion of Carboxylic Acids intoN-Acylbenzotriazoles

KATRITZKY, A. R., Zhang, Y., & Singh, S. K. (2003) · Synthesis · doi:10.1055/s-2003-42462 · Cited by 85 · see citing works

A mild and efficient procedure for the preparation of acid chlorides from car☐ylic acids

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