Multigram-Scale Synthesis of Short Peptides via a Simplified Repetitive Solution-Phase Procedure

Solid Phase Peptide Synthesis. I. The Synthesis of a Tetrapeptide

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From Production of Peptides in Milligram Amounts for Research to Multi-Tons Quantities for Drugs of the Future

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Analytical uses of ultrasound I. Sample preparation

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[1] Concept and early development of solid-phase peptide synthesis

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Solid‐phase synthesis of C‐terminal modified peptides

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Naturally-Occurring Cyclopeptides: Structures and Bioactivity

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Inhibition of angiogenesis in vitro by Arg-Gly-Asp-containing synthetic peptide.

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The 1,1-Dioxobenzo[b]thiophene-2-ylmethyloxycarbonyl (Bsmoc) Amino-Protecting Group

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Slurry Nebulization in Plasmas for Analysis of Inorganic Materials

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Tris(2-aminoethyl)amine as substitute for 4-(aminomethyl)piperidine in the FMOC/polyamine approach to rapid peptide synthesis

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Carbodiimide-Mediated Amide Formation in a Two-Phase System. A High-Yield and Low-Racemization Procedure for Peptide Synthesis

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Rapid, Continuous Solution-Phase Peptide Synthesis: Application to Peptides of Pharmaceutical Interest

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Sulfur-containing polypeptides. XIV. Removal of the tert-butyloxycarbonyl group with boron trifluoride etherate

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Exploiting natural peptide diversity: novel research tools and drug leads

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Development of HIV fusion inhibitors

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Isolation, structure and synthesis of mahafacyclin B, a cyclic heptapeptide from the latex of Jatropha mahafalensis

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Rapid Peptide Synthesis in Liquid Phase. Preparation of Angiotensin II and Delta-sleep-inducing Peptide by the “Hold-in-Solution” Method

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N,O-Isopropylidenated Threonines as Tools for Peptide Cyclization: Application to the Synthesis of Mahafacyclin B

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A novel method for repetitive peptide synthesis in solution without isolation of intermediates

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β‐Lactam‐Containing Cyclopeptide Analogs

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DioRaSSP: Diosynth Rapid Solution Synthesis of Peptides

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Pentafluorophenol: A Superior Reagent for Condensations in Heterocyclic Chemistry

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Industrial production of an oxytocin antagonist: Synthetic approaches to the development of a multi-kilogram scale solution synthesis

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Sustainability in peptide chemistry: current synthesis and purification technologies and future challenges

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Ynamide Coupling Reagents: Origin and Advances

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Inverse Peptide Synthesis Using Transient Protected Amino Acids

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Site-Specific Modification of Amino Acids and Peptides by Aldehyde–Alkyne–Amine Coupling under Ambient Aqueous Conditions

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A green protocol for peptide bond formation in WEB

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Peptide Bond Formation of Amino Acids by Transient Masking with Silylating Reagents

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Peptide‐Chain Elongation Using Unprotected Amino Acids in a Micro‐Flow Reactor

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Recent Advances in The Fabrication and Bio-Medical Applications of Self-Assembled Dipeptide Nanostructures

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Synthesis and Mechanochemical Activity of Peptide-Based Cu(I) Bis(N-heterocyclic carbene) Complexes

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Peptide Bond Formation Between Unprotected Amino Acids: Convergent Synthesis of Oligopeptides

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From precision synthesis to cross-industry applications: The future of emerging peptide technologies

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Isostearyl Mixed Anhydrides for the Preparation ofN-Methylated Peptides UsingC-Terminally UnprotectedN-Methylamino Acids

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Kilogram-Scale Synthesis of Osteogenic Growth Peptide (10–14) Using a Fragment Coupling Approach

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Process Development toward a Key Fragment of the PCSK9 Inhibitor Enlicitide Decanoate

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α‐N‐Protected dipeptide acids: a simple and efficient synthesis via the easily accessible mixed anhydride method using free amino acids in DMSO and tetrabutylammonium hydroxide

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Effect of Brønsted Acids on the Activation of Mixed Anhydride/Mixed Carbonic Anhydride and C‐Terminal‐Free N‐Methylated Peptide Synthesis in a Micro‐Flow Reactor

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Synthesis of BDNF-mimetic dimeric dipeptide GSB-106, a potential neuroprotector drug

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Chemical ligation from O-acyl isopeptides via 8- and 11-membered cyclic transition states

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Physiological effects of a novel artificially synthesized antimalarial cyclic peptide: Mahafacyclin B

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Peptide Synthesis Using Unprotected Amino AcidsPreprint

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Production of Atosiban’s Key Intermediate Pentapeptide: Synthetic Approaches to the Development of a Peptide Synthesis with Less Racemization and Simplifier Purification Process

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Accelerated Synthesis of Internally Functionalized Dendrimers

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Rapid microwave-assisted solution-phase peptide synthesis

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A novel method for repetitive peptide synthesis in solution without isolation of intermediates

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A new method for rapid solution synthesis of shorter peptides by use of PyBOP®

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Rapid, Continuous Solution-Phase Peptide Synthesis: Application to Peptides of Pharmaceutical Interest

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Microwave irradiated high-speed solution synthesis of peptide acids employing Fmoc-amino acid pentafluorophenyl esters as coupling agents

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