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Expedient Enantioselective Synthesis of Cermizine D

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Rhodium/Chiral Diene Complexes in the Catalytic Asymmetric Arylation of β-Pyrazol-1-yl Acrylates

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Model Based Targeting of IL-6-Induced Inflammatory Responses in Cultured Primary Hepatocytes to Improve Application of the JAK Inhibitor Ruxolitinib

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γ-Amino Alcohols via Organocascade Reactions Involving Dienamine Catalysis

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Highly Enantioselective Direct Michael Addition of 1H‐Benzotriazole to Chalcones Catalyzed by Sc(OTf)3/N,N′‐Dioxide Complex

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Development of an NH4Cl-Catalyzed Ethoxy Ethyl Deprotection in Flow for the Synthesis of Merestinib

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Metal Azolate/Carboxylate Frameworks as Catalysts in Oxidative and C–C Coupling Reactions

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Synthesis and clinical application of small-molecule inhibitors of Janus kinase

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Design, Synthesis and Structure-Activity Relationships of Novel Diaryl Urea Derivatives as Potential EGFR Inhibitors

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Synthesis, SAR study, and biological evaluation of novel quinoline derivatives as phosphodiesterase 10A inhibitors with reduced CYP3A4 inhibition

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Enantioselective N-alkylation of isatins and synthesis of chiral N-alkylated indoles

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Azole‐Directed Cobalt‐Catalyzed Asymmetric Hydrogenation of Alkenes

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Proline Derivatives

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Chapter 12 Advances in the Discovery of Small Molecule JAK3 Inhibitors

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An efficient strategy for the general synthesis of 3-aryl substituted pyrazolo[5,1-c][1,4]benzoxazines and pyrazolo[1,5-a][1,4]benzodiazepin-6(4H)-ones

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Suppression of Autoimmune Arthritis by Small Molecule Inhibitors of the JAK/STAT Pathway

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Synthesis of Chiral Pyrazoles: A 1,3‐Dipolar Cycloaddition/[1,5] Sigmatropic Rearrangement with Stereoretentive Migration of a Stereogenic Group

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Modification of Pyrrolo[2,3‐d]pyrimidines by C–H Borylation Followed by Cross‐Coupling or Other Transformations: Synthesis of 6,8‐Disubstituted 7‐Deazapurine Bases

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Enantioselective Reaction Using Palladium Pincer Complexes with C2-Symmetric Chiral Bis(imidazoline)s

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Synthesis and Anticancer Activity of Novel Dual Inhibitors of Human Protein Kinases CK2 and PIM-1

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Ruxolitinib induces autophagy in chronic myeloid leukemia cells

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Metalation of Pyrazoles and Indazoles

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Selective Janus Kinase 1 Inhibition Resolves Inflammation and Restores Hair Growth Offering a Viable Treatment Option for Alopecia Areata

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The Timing and Magnitude of the Type I Interferon Response Are Correlated with Disease Tolerance in Arbovirus Infection

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Improved Synthesis of 1H-Pyrazole-4-carbaldehyde

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Epigenetic changes in inflammatory arthritis monocytes contribute to disease and can be targeted by JAK inhibition

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Enantioselective Aza-Michael Reactions of Pyrazoles: Synthesis of INCB0184124

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Cinchona-Functionalized Crown-Ether-Pinioned Calix[4]arene for a Scalable Asymmetric Organocatalytic Aza-Michael Addition Reaction

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Asymmetric One‐Pot Synthesis of 1,4‐Dihydroquinolines via an Organocatalytic Aza‐Michael/Michael Cascade Strategy

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A Concise Enantioselective Synthesis of Fluorinated Pyrazolo-Piperidine GSK3901383A Enabled by an Organocatalytic Aza-Michael Addition

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Enantioselective Synthesis of Azaflavanones Using Organocatalytic 6‐endo Aza‐Michael Addition

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