Sites of alcohol and volatile anaesthetic action on GABAA and glycine receptors

Molecular and cellular mechanisms of general anaesthesia

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The actions of propofol on inhibitory amino acid receptors of bovine adrenomedullary chromaffin cells and rodent central neurones

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Binding of Xenon to Sperm Whale Myoglobin

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Mapping of general anaesthetic target sites provides a molecular basis for cutoff effects

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A relationship between alcohol intoxication and the disordering of brain membranes by a series of short-chain alcohols.

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Enhancement of homomeric glycine receptor function by longchain alcohols and anaesthetics

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Identification of channel-lining residues in the M2 membrane-spanning segment of the GABA(A) receptor alpha1 subunit.

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Effects of volatile anesthetics on the kinetics of inhibitory postsynaptic currents in cultured rat hippocampal neurons

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Positive modulation of human gamma-aminobutyric acid type A and glycine receptors by the inhalation anesthetic isoflurane.

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Up-regulation of γ-aminobutyric acid transporter I mediates ethanol sensitivity in mice

Hu, J. H., Ma, Y.-H., Yang, N., Mei, Z., Zhang, M.-H., Fei, J., & Guo, L. H. (2004) · Neuroscience · doi:10.1016/j.neuroscience.2003.11.018 · Cited by 20

Ethanol Inhibition of Glycine-Activated Responses in Neurons of Ventral Tegmental Area of Neonatal Rats

Ye, J. H., Tao, L., Zhu, L., Krnjević, K., & McArdle, J. J. (2001) · Journal of Neurophysiology · doi:10.1152/jn.2001.86.5.2426 · Cited by 20

Effects of Halothane on Phosphatidylcholine, -ethanolamine, -glycerol, and -serine Monolayer Order at a Liquid/Liquid Interface

Watry, M. R., & Richmond, G. L. (2002) · Langmuir · doi:10.1021/la020463d · Cited by 20

Mechanism of anesthetic action: oxygen pathway perturbation hypothesis

Hu, H. P., & Wu, M. X. (2001) · Medical Hypotheses · doi:10.1054/mehy.2001.1419 · Cited by 20

Clinical Pharmacology

Grimm, K. A., & Lamont, L. A. (2007) · doi:10.1002/9780470376478.ch1 · Cited by 20

Modulation of Presynaptic β3-Containing GABAA Receptors Limits the Immobilizing Actions of GABAergic Anesthetics

Grasshoff, C., Jurd, R., Rudolph, U., & Antkowiak, B. (2007) · Molecular Pharmacology · doi:10.1124/mol.107.037648 · Cited by 19

Evidence for α-Helices in the Large Intracellular Domain Mediating Modulation of the α1-Glycine Receptor by Ethanol and Gβγ

Burgos, C. F., Castro, P. A., Mariqueo, T. A., Bunster, M. C., Guzmán, L., & Aguayo, L. G. (2014) · Journal of Pharmacology and Experimental Therapeutics · doi:10.1124/jpet.114.217976 · Cited by 19

A Novel Alcohol-Sensitive Position in the N-Methyl-d-Aspartate Receptor GluN2A Subunit M3 Domain Regulates Agonist Affinity and Ion Channel Gating

Ren, H., Zhao, Y., Wu, M., & Peoples, R. W. (2013) · Molecular Pharmacology · doi:10.1124/mol.113.085993 · Cited by 19

Cell surface expression of homomeric GABAA receptors depends on single residues in subunit transmembrane domains

Hannan, S. B., & Smart, T. G. (2018) · Journal of Biological Chemistry · doi:10.1074/jbc.ra118.002792 · Cited by 20

Divergence of Volatile Anesthetic Effects in Inhibitory Neurotransmitter Receptors

Greenblatt, E. P., & Meng, X. (2001) · Anesthesiology · doi:10.1097/00000542-200106000-00017 · Cited by 19

Four-α-Helix Bundle with Designed Anesthetic Binding Pockets. Part I: Structural and Dynamical Analyses

Ma, D., Brandon, N. R., Cui, T., Bondarenko, V., Canlas, C. P., Johansson, J. S., Tang, P. S., & Xu, Y. (2008) · Biophysical Journal · doi:10.1529/biophysj.107.117838 · Cited by 19

Linking of Glycine Receptor Transmembrane Segments Three and Four Allows Assignment of Intrasubunit-Facing Residues

McCracken, L. M., McCracken, M. L., Gong, D. H., Trudell, J. R., & Harris, R. A. (2010) · ACS Chemical Neuroscience · doi:10.1021/cn100019g · Cited by 19

Occupancy of a Single Anesthetic Binding Pocket Is Sufficient to Enhance Glycine Receptor Function

Roberts, M. T., Phelan, R., Erlichman, B., Pillai, R. N., Ma, L., Lopreato, G. F., & Mihic, S. J. (2005) · Journal of Biological Chemistry · doi:10.1074/jbc.m502000200 · Cited by 19

PET quantification of muscarinic cholinergic receptors with [N‐11C‐methyl]‐benztropine and application to studies of propofol‐induced unconsciousness in healthy human volunteers

Xie, G., Gunn, R. N., Dagher, A., Daloze, T., Plourde, G., Backman, S. B., Dikšić, M., & Fiset, P. (2003) · Synapse · doi:10.1002/syn.10292 · Cited by 19

Meyer and Overton Revisited

Lynch, C. I. (2008) · Anesthesia & Analgesia · doi:10.1213/ane.0b013e3181706c7e · Cited by 19

Aging of Whiskey Increases the Potentiation of GABAAReceptor Response

Kôda, H., Hossain, S. J., Kiso, Y., & Aoshima, H. (2003) · Journal of Agricultural and Food Chemistry · doi:10.1021/jf030111s · Cited by 19

Effects of Ethanol on Adenosine 5′‐Triphosphate–Gated Purinergic and 5‐Hydroxytryptamine3Receptors

Davies, D. L., Asatryan, L., Kuo, S. T., Woodward, J. J., King, B. F., Alkana, R. L., Xiao, C., Ye, J. H., Sun, H., Zhang, L., et al. (2006) · Alcoholism Clinical and Experimental Research · doi:10.1111/j.1530-0277.2006.00023.x · Cited by 19

Interaction of Serotonin1A Receptors from Bovine Hippocampus with Tertiary Amine Local Anesthetics

Kalipatnapu, S., & Chattopadhyay, A. (2004) · Cellular and Molecular Neurobiology · doi:10.1023/b:cemn.0000022771.33702.85 · Cited by 19

The Effects of Isoflurane on Acetylcholine Receptor Channels: 3. Effects of Conservative Polar-to-Nonpolar Mutations within the Channel Pore

Wenningmann, I., Barann, M., Vidal, A. M., & Dilger, J. P. (2001) · Molecular Pharmacology · doi:10.1016/s0026-895x(24)12622-3 · Cited by 19

Molecular Approaches to Improving General Anesthetics

Forman, S. A. (2010) · Anesthesiology Clinics · doi:10.1016/j.anclin.2010.08.004 · Cited by 18

Zinc-Dependent Modulation of α2- and α3-Glycine Receptor Subunits by Ethanol

McCracken, L. M., Trudell, J. R., McCracken, M. L., & Harris, R. A. (2013) · Alcoholism Clinical and Experimental Research · doi:10.1111/acer.12192 · Cited by 19

A possible mechanism for pressure reversal of general anaesthetics from molecular simulations

Chau, P. ‐., Hoang, P. N. M., Picaud, S., & Jedlovszky, P. (2007) · Chemical Physics Letters · doi:10.1016/j.cplett.2007.02.071 · Cited by 18

Characterization of sevoflurane effects on Per2 expression using ex vivo bioluminescence imaging of the suprachiasmatic nucleus in transgenic rats

Matsuo, I., Iijima, N., Takumi, K., Higo, S., Aikawa, S., Anzai, M., Ishii, H., Sakamoto, A., & Ozawa, H. (2015) · Neuroscience Research · doi:10.1016/j.neures.2015.11.010 · Cited by 18

Contributions of dipole moments, quadrupole moments, and molecular polarizabilities to the anesthetic potency of fluorobenzenes

Trudell, J. R. (1998) · Biophysical Chemistry · doi:10.1016/s0301-4622(98)00161-6 · Cited by 18

Argon gas: a potential neuroprotectant and promising medical therapy

Nowrangi, D., Tang, J., & Zhang, J. H. (2014) · Medical Gas Research · doi:10.1186/2045-9912-4-3 · Cited by 19

Determinants of the Anesthetic Sensitivity of Neuronal Nicotinic Acetylcholine Receptors

Downie, D. L., Vicente‐Agulló, F., Campos‐Caro, A., Bushell, T. J., Lieb, W. R., & Franks, N. P. (2002) · Journal of Biological Chemistry · doi:10.1074/jbc.m107847200 · Cited by 18

Subunit-specific potentiation of recombinant glycine receptors by NV-31, a bilobalide-derived compound

Lynch, J. W., & Chen, X. (2008) · Neuroscience Letters · doi:10.1016/j.neulet.2008.02.022 · Cited by 18

Anions and the anaesthetist

Maloney, D. G., Appadurai, I. R., & Vaughan, R. S. (2002) · Anaesthesia · doi:10.1046/j.1365-2044.2002.02274.x · Cited by 18

NT-3 delivered by an adenoviral vector induces injured dorsal root axons to regenerate into the spinal cord of adult rats

Zhang, Y., Dijkhuizen, P. A., Anderson, P. N., Lieberman, A. R., & Verhaagen, J. (1998) · Journal of Neuroscience Research · doi:10.1002/(sici)1097-4547(19981115)54:4 · Cited by 99

Dual Action of Isoflurane on the γ-aminobutyric Acid (GABA)-Mediated Currents Through Recombinant α1β2γ2L-GABAA-Receptor Channels

Neumahr, S., Hapfelmeier, G., Scheller, M., Schneck, H., Franke, C., & Kochs, E. F. (2000) · Anesthesia & Analgesia · doi:10.1097/00000539-200005000-00035 · Cited by 18

Acute Effects of Ethanol on Kainate Receptors with Different Subunit Compositions

Valenzuela, C. F., & Cardoso, R. A. (1999) · Journal of Pharmacology and Experimental Therapeutics · doi:10.1016/s0022-3565(24)38074-7 · Cited by 18

Structure, Diversity, Pharmacology, and Pathology of Glycine Receptor Chloride Channels

Harvey, R. J., & Betz, H. (2000) · Handbook of experimental pharmacology · doi:10.1007/978-3-642-57083-4_18 · Cited by 18

Important amino acids for function of the insect Rdl GABA receptor

Nakao, T., & Banba, S. (2020) · Pest Management Science · doi:10.1002/ps.6121 · Cited by 17

Selective potentiation of alpha 1 glycine receptors by ginkgolic acid

Maleeva, G., Buldakova, S., & Bregestovski, P. D. (2015) · Frontiers in Molecular Neuroscience · doi:10.3389/fnmol.2015.00064 · Cited by 17

Effects of ethanol on glycinergic synaptic currents in mouse spinal cord neurons

Mariqueo, T. A., Agurto, A., Muñoz, B., Martín, L. S., Coronado, C., Fernández-Pérez, E. J., Murath, P., Sánchez, A., Homanics, G. E., & Aguayo, L. G. (2014) · Journal of Neurophysiology · doi:10.1152/jn.00789.2013 · Cited by 17

Thiocolchicoside inhibits the activity of various subtypes of recombinant GABAA receptors expressed in Xenopus laevis oocytes

Mascia, M. P., E), B., Obili, N., Maciocco, E., Cocco, G. A., Sechi, G., & Biggio, G. (2006) · European Journal of Pharmacology · doi:10.1016/j.ejphar.2006.11.076 · Cited by 17

The role of NMDA and GABAA receptors in the inhibiting effect of 3 MPa nitrogen on striatal dopamine level

Lavoûte, C., Weiss, M., & Rostain, J. (2007) · Brain Research · doi:10.1016/j.brainres.2007.07.085 · Cited by 17

The L293 residue in transmembrane domain 2 of the 5-HT3A receptor is a molecular determinant of allosteric modulation by 5-hydroxyindole

Hu, X., & Dm, L. (2008) · Neuropharmacology · doi:10.1016/j.neuropharm.2008.03.009 · Cited by 17

Comparison of kinetic and pharmacological profiles of recombinant α1γ2L and α1β2γ2L GABAA receptors – A clue to the role of intersubunit interactions

Brodzki, M., Rutkowski, R., Jatczak-Śliwa, M., Kisiel, M., Czyzewska, M. M., & Mozrzymas, J. W. (2016) · European Journal of Pharmacology · doi:10.1016/j.ejphar.2016.05.015 · Cited by 17

Effect of general anesthetics on the properties of lipid membranes of various compositions

Hantal, G., Fábián, B., Sega, M., Jójárt, B., & Jedlovszky, P. (2018) · Biochimica et Biophysica Acta (BBA) - Biomembranes · doi:10.1016/j.bbamem.2018.12.008 · Cited by 17

Nicotinic Receptor Pore Mutations Create a Sensitive Inhibitory Site for Ethanol

Forman, S. A., & Zhou, Q. (2000) · Alcoholism Clinical and Experimental Research · doi:10.1111/j.1530-0277.2000.tb02104.x · Cited by 17

Molecular volume determines the activity of the halogenated alkane bromoform at wild-type and mutant GABAA receptors

Kash, T. L., Jenkins, A., & Harrison, N. L. (2003) · Brain Research · doi:10.1016/s0006-8993(02)03748-4 · Cited by 17

G Protein βγ Gating Confers Volatile Anesthetic Inhibition to Kir3 Channels

Styer, A. M., Mirshahi, U. L., Wang, C., Girard, L., Jin, T., Logothetis, D. E., & Mirshahi, T. (2010) · Journal of Biological Chemistry · doi:10.1074/jbc.m110.178541 · Cited by 16

Protein Kinase C Modulation of Ethanol Inhibition of Glycine-Activated Current in Dissociated Neurons of Rat Ventral Tegmental Area

Tao, L., & Ye, J. H. (2002) · Journal of Pharmacology and Experimental Therapeutics · doi:10.1124/jpet.300.3.967 · Cited by 17

Dual cooperative allosteric modulation of binding to ionotropic glycine receptors

Maksay, G., & Bı́ró, T. (2002) · Neuropharmacology · doi:10.1016/s0028-3908(02)00213-7 · Cited by 17

Formation of water polyhedrons in propofol–water clusters

León, Í., Cocinero, E. J., Rijs, A. M., Millán, J., Alonso, E. E., Lesarri, A. G., & Fernández, J. A. (2012) · Physical Chemistry Chemical Physics · doi:10.1039/c2cp42304a · Cited by 16

A possible molecular mechanism for the pressure reversal of general anaesthetics: Aggregation of halothane in POPC bilayers at high pressure

Tu, K.-M., Matubayasi, N., Liang, K. K., Todorov, I. T., Chan, S. L.-F., & Chau, P. ‐. (2012) · Chemical Physics Letters · doi:10.1016/j.cplett.2012.06.044 · Cited by 16

Charge and Geometry of Residues in the Loop 2 β Hairpin Differentially Affect Agonist and Ethanol Sensitivity in Glycine Receptors

Perkins, D. I., Trudell, J. R., Asatryan, L., Davies, D. L., & Alkana, R. L. (2012) · Journal of Pharmacology and Experimental Therapeutics · doi:10.1124/jpet.111.190942 · Cited by 16

Sleep Homeostasis and General Anesthesia

Gardner, B., Strus, E., Meng, Q. C., Coradetti, T., Naidoo, N. N., Kelz, M. B., & Williams, J. A. (2015) · Anesthesiology · doi:10.1097/aln.0000000000000939 · Cited by 16

GABAA Receptor Subtype Mechanisms and the Abuse-Related Effects of Ethanol: Genetic and Pharmacological Evidence

Chandler, C. M., Overton, J. S., Rüedi‐Bettschen, D., & Platt, D. M. (2017) · Handbook of experimental pharmacology · doi:10.1007/164_2017_80 · Cited by 16

Neuroendocrine, epigenetic, and intergenerational effects of general anesthetics

Martynyuk, A. E., Ju, L.-S., Morey, T. E., & Zhang, J. (2020) · World Journal of Psychiatry · doi:10.5498/wjp.v10.i5.81 · Cited by 16

Function of hyperekplexia‐causing α1R271Q/L glycine receptors is restored by shifting the affected residue out of the allosteric signalling pathway

Shan, Q., Han, L., & Lynch, J. W. (2011) · British Journal of Pharmacology · doi:10.1111/j.1476-5381.2011.01701.x · Cited by 17

Trifluoroacetate is an allosteric modulator with selective actions at the glycine receptor

Tipps, M. E., Iyer, S. V., & Mihic, S. J. (2012) · Neuropharmacology · doi:10.1016/j.neuropharm.2012.04.011 · Cited by 16

Volatile anesthetics affect the morphology of rat glioma C6 cells via RhoA, ERK, and Akt activation

Tas, P. W. L., Gambaryan, S. P., & Roewer, N. (2007) · Journal of Cellular Biochemistry · doi:10.1002/jcb.21294 · Cited by 16

Contaminating levels of zinc found in commonly-used labware and buffers affect glycine receptor currents

Cornelison, G. L., & Mihic, S. J. (2013) · Brain Research Bulletin · doi:10.1016/j.brainresbull.2013.10.012 · Cited by 16

Review of Functional Studies of Beverage Components Acting on the Recombinant GABAANeuroreceptor, and Na+/Glucose Cotransporter-Response Using theXenopusOocyte Expression System and Electrophysiological Measurements

Hossain, S. J., Aoshima, H., Kôda, H., & Kiso, Y. (2007) · Food Biotechnology · doi:10.1080/08905430701534081 · Cited by 16

The TM2 6′ Position of GABAA Receptors Mediates Alcohol Inhibition

Johnson, W. D., Howard, R. J., Trudell, J. R., & Harris, R. A. (2011) · Journal of Pharmacology and Experimental Therapeutics · doi:10.1124/jpet.111.188037 · Cited by 16

The novel hyperekplexia allele GLRA1(S267N) affects the ethanol site of the glycine receptor

Becker, K., Breitinger, H., Humeny, A., Meinck, H., Dietz, B., Aksu, F., & Becker, C. (2007) · European Journal of Human Genetics · doi:10.1038/sj.ejhg.5201958 · Cited by 16

Mutations of L293 in transmembrane two of the mouse 5‐hydroxytryptamine3A receptor alter gating and alcohol modulatory actions

Hu, X., Hayrapetyan, V. Y., Gadhiya, J. J., Rhubottom, H. E., Lovinger, D. M., & Machu, T. K. (2006) · British Journal of Pharmacology · doi:10.1038/sj.bjp.0706685 · Cited by 16

Molecular Modeling and Mutagenesis Reveals a Tetradentate Binding Site for Zn2+in GABAAαβ Receptors and Provides a Structural Basis for the Modulating Effect of the γ Subunit

Trudell, J. R., Yue, M. E., Bertaccini, E. J., Jenkins, A., & Harrison, N. L. (2008) · Journal of Chemical Information and Modeling · doi:10.1021/ci700324a · Cited by 16

Effects of Volatile Anesthetic on Channel Structure of Gramicidin A

Tang, P. S., Mandal, P. K., & Zegarra, M. (2002) · Biophysical Journal · doi:10.1016/s0006-3495(02)73912-x · Cited by 16

Effects of a mutation in the TM2–TM3 linker region of the glycine receptor α1 subunit on gating and allosteric modulation

Dupre, M. L., Broyles, J. M., & Mihic, S. J. (2007) · Brain Research · doi:10.1016/j.brainres.2007.03.031 · Cited by 16

The Plasticizer Di(2-ethylhexyl) Phthalate Modulates γ-Aminobutyric Acid Type A and Glycine Receptor Function

Yang, L., Milutinovic, P. S., Brosnan, R. J., Eger, E. I., & Sonner, J. M. (2007) · Anesthesia & Analgesia · doi:10.1213/01.ane.0000267336.37735.d7 · Cited by 16

Effects of isoflurane and ketamine on ATP-sensitive K channels in rat substantia nigra

Ishiwa, D., Kamiya, Y., Itoh, H., Saito, Y., Ohtsuka, T., Yamada, Y., & Andoh, T. (2004) · Neuropharmacology · doi:10.1016/j.neuropharm.2004.01.012 · Cited by 16

Xenon-induced inhibition of synchronized bursts in a rat cortical neuronal network

Uchida, T., Suzuki, S., Hirano, Y., Ito, D., Nagayama, M., & Gohara, K. (2012) · Neuroscience · doi:10.1016/j.neuroscience.2012.03.063 · Cited by 16

A Caenorhabditis elegans Pheromone Antagonizes Volatile Anesthetic Action Through a Go-Coupled Pathway

van Swinderen, B., Metz, L. B., Shebester, L., & Crowder, C. M. (2002) · Genetics · doi:10.1093/genetics/161.1.109 · Cited by 16

Disruption of an intersubunit electrostatic bond is a critical step in glycine receptor activation

Todorović, J., Welsh, B. T., Bertaccini, E. J., Trudell, J. R., & Mihic, S. J. (2010) · Proceedings of the National Academy of Sciences · doi:10.1073/pnas.1001845107 · Cited by 16

Volatile anesthetics directly activate baseline S K+ channels in Aplysia neurons

Winegar, B. D., & Yost, C. S. (1998) · Brain Research · doi:10.1016/s0006-8993(98)00687-8 · Cited by 16

Effects of a low dose of ethanol in an animal model of premenstrual anxiety

Smith, S. S., Ruderman, Y., Gong, Q. H., & Gulinello, M. E. (2004) · Alcohol · doi:10.1016/j.alcohol.2004.04.003 · Cited by 16

Large Intracellular Domain-Dependent Effects of Positive Allosteric Modulators on Glycine Receptors

Lara, C. O., Burgos, C. F., Silva-Grecchi, T., Muñoz-Montesino, C., Aguayo, L. G., Fuentealba, J., Castro, P. A., Guzmán, J. L., Corringer, P., Yévenes, G. E., et al. (2019) · ACS Chemical Neuroscience · doi:10.1021/acschemneuro.9b00050 · Cited by 15

Probing the pharmacological properties of distinct subunit interfaces within heteromeric glycine receptors reveals a functional ββ agonist‐binding site

Dutertre, S., Drwal, M. N., Laube, B., & Betz, H. (2012) · Journal of Neurochemistry · doi:10.1111/j.1471-4159.2012.07755.x · Cited by 15

State-dependent vs. central motor effects of ethanol on breathing

Vecchio, L. M., Grace, K. P., Liu, H., Harding, S. E., Lê, A. D., & Horner, R. L. (2009) · Journal of Applied Physiology · doi:10.1152/japplphysiol.00797.2009 · Cited by 15

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Koob, G. F., & Moal, M. L. (2006) · Elsevier eBooks · doi:10.1016/b978-012419239-3/50042-4 · Cited by 15

Ethanol Enhances Taurine‐Activated Glycine Receptor Function

Welsh, B. T., Kirson, D., Allen, H. M., & Mihic, S. J. (2010) · Alcoholism Clinical and Experimental Research · doi:10.1111/j.1530-0277.2010.01249.x · Cited by 15

Volatile anesthetics and endogenous cannabinoid anandamide have additive and independent inhibitory effects on α7-nicotinic acetylcholine receptor-mediated responses in Xenopus oocytes

Jackson, S. N., Singhal, S. K., Woods, A. S., Morales, M., Shippenberg, T. S., Zhang, L., & Öz, M. (2008) · European Journal of Pharmacology · doi:10.1016/j.ejphar.2007.12.023 · Cited by 15

Anesthetic-Like Modulation of Receptor Function by Surfactants: A Test of the Interfacial Theory of Anesthesia

Yang, L., & Sonner, J. M. (2008) · Anesthesia & Analgesia · doi:10.1213/ane.0b013e31817ee500 · Cited by 15

Pressure reversal of general anaesthetics: A possible mechanism from molecular dynamics simulations

Chau, P. ‐., Jedlovszky, P., Hoang, P. N. M., & Picaud, S. (2008) · Journal of Molecular Liquids · doi:10.1016/j.molliq.2008.09.005 · Cited by 15

Recreational concentrations of alcohol enhance synaptic inhibition of cerebellar unipolar brush cells via pre- and postsynaptic mechanisms

Richardson, B. D., & Rossi, D. J. (2017) · Journal of Neurophysiology · doi:10.1152/jn.00963.2016 · Cited by 15

Ethanol effects on GABA-gated current in a model of increased α4βδ GABAA receptor expression depend on time course and preexposure to low concentrations of the drug

Smith, S. S., & Gong, Q. H. (2007) · Alcohol · doi:10.1016/j.alcohol.2007.04.007 · Cited by 15

Positive allosteric modulatory effects of ajulemic acid at strychnine-sensitive glycine α1- and α1β-receptors

Ahrens, J., Leuwer, M., Demir, R., Krampfl, K., de la Roche, J., Foadi, N., Karst, M., & Haeseler, G. (2008) · Naunyn-Schmiedeberg s Archives of Pharmacology · doi:10.1007/s00210-008-0366-8 · Cited by 15

Embryonic exposure to ethanol disturbs regulation of mitotic spindle orientation via GABAA receptors in neural progenitors in ventricular zone of developing neocortex

Tochitani, S., Sakata‐Haga, H., & Fukui, Y. (2010) · Neuroscience Letters · doi:10.1016/j.neulet.2010.01.071 · Cited by 15

Phylogenetic shadowing of a histamine-gated chloride channel involved in insect vision

Iovchev, M. I., Boutanaev, A. M., Ivanov, I., Wolstenholme, A. J., Nurminsky, D. I., & Semenov, E. (2005) · Insect Biochemistry and Molecular Biology · doi:10.1016/j.ibmb.2005.09.002 · Cited by 15

Separate Domains for Desensitization of GABA ρ 1 and β 2 Subunits Expressed in Xenopus Oocytes

Lu, L., & Huang, Y. (1998) · The Journal of Membrane Biology · doi:10.1007/s002329900398 · Cited by 15

Increased Ro15-4513–Induced Seizures Following Multiple Ethanol Withdrawals

Mhatre, M. (1999) · Pharmacology Biochemistry and Behavior · doi:10.1016/s0091-3057(98)00257-3 · Cited by 14

Ethanol Modulates the Interaction of the Endogenous Neurosteroid Allopregnanolone with the α1β2γ2L GABAA Receptor

Akk, G., Li, P., Manion, B. D., Evers, A. S., & Steinbach, J. H. (2006) · Molecular Pharmacology · doi:10.1124/mol.106.029942 · Cited by 15

Bioinspired Bi2S3 Thin Films on 4-Mercaptobenzoic Acid Functionalized Self-Assembled Monolayers

Liufu, S., Chen, L., Wang, Q., & Yao, Q. (2007) · Crystal Growth & Design · doi:10.1021/cg060319g · Cited by 15

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Differential Sensitivity of Expressed L-Type Calcium Channels and Muscarinic M1 Receptors to Volatile Anesthetics inXenopus Oocytes

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Allosteric modulation in spontaneously active mutant γ-aminobutyric acidA receptors in frogs

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Characterisation of thymol effects on RDL receptors from the bee parasite Varroa destructor

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GIRK Channels

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Amyotrophic lateral sclerosis—A case report and mechanistic review of the association with toluene and other volatile organic compounds

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Unexpected Properties of δ-Containing GABAA Receptors in Response to Ligands Interacting with the α+ β− Site

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Brucine suppresses ethanol intake and preference in alcohol-preferring Fawn-Hooded rats

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The Anesthetic Interaction Between Adenosine Triphosphate and N-methyl-D-Aspartate Receptor Antagonists in the Rat

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A Cysteine Substitution Probes β3H267 Interactions with Propofol and Other Potent Anesthetics in α1β3γ2L γ-Aminobutyric Acid Type A Receptors

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Glycine and GABAA Ultra-Sensitive Ethanol Receptors as Novel Tools for Alcohol and Brain Research

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Binary combinations of propofol and barbiturates on human α1 glycine receptors expressed in Xenopus oocytes

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The Molecular Mechanisms of Anesthetic Action: Updates and Cutting Edge Developments from the Field of Molecular Modeling

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Sevoflurane-induced Reduction of Hypoxic Drive Is Sex-independent

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Allosteric Modulation of GABAA Receptor Function by General Anesthetics and Alcohols

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Antagonism of Inhalant and Volatile Anesthetic Enhancement of Glycine Receptor Function

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Anaesthetics set their sites on ion channels

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Inhibition of rho1 receptor GABAergic currents by alcohols and volatile anesthetics.

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