Characterization of the Biological Roles of the Estrogen Receptors, ERα and ERβ, in Estrogen Target Tissues in Vivo through the Use of an ERα-Selective Ligand

Comparison of the Ligand Binding Specificity and Transcript Tissue Distribution of Estrogen Receptors α and β

Kuiper, G. G. J. M., Carlsson, B., Grandien, K., Enmark, E., Häggblad, J., Nilsson, S., & Gustafsson, J.-A. (1997) · Endocrinology · doi:10.1210/endo.138.3.4979 · Cited by 4,442

Estrogen Receptor Null Mice: What Have We Learned and Where Will They Lead Us?

Couse, J. F., & Korach, K. S. (1999) · Endocrine Reviews · doi:10.1210/edrv.20.3.0370 · Cited by 2,045

Estrogen Actions in the Central Nervous System

McEwen, B. S., & Alves, S. E. (1999) · Endocrine Reviews · doi:10.1210/edrv.20.3.0365 · Cited by 1,504

The Estrogen Receptor β-Isoform (ERβ) of the Human Estrogen Receptor Modulates ERα Transcriptional Activity and Is a Key Regulator of the Cellular Response to Estrogens and Antiestrogens1

Hall, J. M., & McDonnell, D. P. (1999) · Endocrinology · doi:10.1210/endo.140.12.7179 · Cited by 1,078

Effect of single and compound knockouts of estrogen receptors α (ERα) and β (ERβ) on mouse reproductive phenotypes

Dupont, S., Krust, A., Gansmuller, A., Dierich, A., Chambon, P., & Mark, M. (2000) · Development · doi:10.1242/dev.127.19.4277 · Cited by 1,064

Pyrazole Ligands: Structure−Affinity/Activity Relationships and Estrogen Receptor-α-Selective Agonists

Stauffer, S. R., Coletta, C. J., Tedesco, R., Nishiguchi, G., Carlson, K. E., Sun, J., Katzenellenbogen, B. S., & Katzenellenbogen, J. A. (2000) · Journal of Medicinal Chemistry · doi:10.1021/jm000170m · Cited by 760

Role of Estrogen Receptor Beta in Estrogen Action

Pettersson, K., & Gustafsson, J.-Α. (2001) · Annual Review of Physiology · doi:10.1146/annurev.physiol.63.1.165 · Cited by 491

Analysis of transcription and estrogen insensitivity in the female mouse after targeted disruption of the estrogen receptor gene

Couse, J. F., Curtis, S. W., Washburn, T. F., Lindzey, J. K., GOLDING, T. S., Lubahn, D. B., Smithies, O., & Korach, K. S. (1995) · Molecular Endocrinology · doi:10.1210/mend.9.11.8584021 · Cited by 454

The Estrogen Receptor β Subtype: A Novel Mediator of Estrogen Action in Neuroendocrine Systems

Kuiper, G. G. J. M., Shughrue, P. J., Merchenthaler, I. J., & Gustafsson, J.-Α. (1998) · Frontiers in Neuroendocrinology · doi:10.1006/frne.1998.0170 · Cited by 438

Oestrogen receptors – an overview

Enmark, E., & Gustafsson, J.-Α. (1999) · Journal of Internal Medicine · doi:10.1046/j.1365-2796.1999.00545.x · Cited by 377

Strategies to treat sepsis: old and new

LaRosa, S. P., & Opal, S. M. (2011) · Clinical Investigation · doi:10.4155/cli.10.19 · Cited by 2

The role of estrogen receptor subtypes for induction of delayed effects on the estrous cycle and female reproductive organs in rats

Takahashi, M., Ichimura, R., Inoue, K., Morikawa, T., Kuwata, K., Watanabe, G., & Yoshida, M. (2017) · Reproductive Biology · doi:10.1016/j.repbio.2017.01.007 · Cited by 2

Estrogen Action and Breast Cancer

Fox, J., Liu, H., & Jordan, V. (2000) · Humana Press eBooks · doi:10.1007/978-1-59259-664-5_10 · Cited by 2

Effects of Alternate Treatment of Estrogen Receptor Antagonist and Agonist on Morphology of Male Reproductive Organs of Adult Mice

Choi, H., Seong, C. N., Park, M., & Cho, H. W. (2013) · Han-guk hyeonmigyeong hakoeji/Applied microscopy · doi:10.9729/am.2013.43.3.103 · Cited by 2

Regulation of Bone Cell Function by Estrogens

Komm, B. S., Cheskis, B. J., & Bodine, P. V. N. (2010) · Elsevier eBooks · doi:10.1016/b978-0-12-375098-3.50015-9 · Cited by 2

Biological Effects and Markers of Exposure to Xenosteroids and Selective Estrogen Receptor Modulators (SERMs) at the Hypothalamic-Pituitary Unit

Tena‐Sempere, M., & Aguilarl, E. (2005) · Springer eBooks · doi:10.1007/3-540-26940-1_6 · Cited by 2

Estrogen Receptor Pathways and Breast Cancer

Peng, J., & Jordan, V. C. (2008) · Humana Press eBooks · doi:10.1007/978-1-59745-470-4_9 · Cited by 2

Entwicklung eines Screeningsystems zur Identifizierung hochaktiver und selektiver Hemmstoffe der 17beta-Hydroxysteroid-Dehydrogenase Typ 1 (17betaHSD1)

Kruchten, P. (2009) · Publications of the UdS (Saarland University) · doi:10.22028/d291-22614 · Cited by 2

SFRP1 Is Estrogen Inducible in Bone Marrow Stromal Cells and Suppresses the Earliest Events in Lymphopoiesis.

Yokota, T., Oritani, K., Garrett, K. P., Kouro, T., Nishida, M., Takahashi, I., Ichii, M., Matsumura, I., Kincade, P. W., & Kanakura, Y. (2007) · Blood · doi:10.1182/blood.v110.11.611.611 · Cited by 2

Isoflavones and breast cancer

Woodside, J. V., & Campbell, M. J. (2001) · Research Portal (Queen's University Belfast) · Cited by 2

The median preoptic nucleus is a key site for estradiol regulation of sleep–wake behaviors in females rats

Kruk, K., Smith, P. D. C., Cusmano, D. M., Viechweg, S. S., Byrd, C., Huddleson, A. M., Schwartz, & Mong, J. A. (2026) · SLEEP · doi:10.1093/sleep/zsaf387 · Cited by 1

Nutritional phytoestrogens and bone health

Wuttke, W., Jarry, H., & Seidlová‐Wuttke, D. (2009) · Elsevier eBooks · doi:10.1533/9781845695743.1.83 · Cited by 1

Differential Responses of Various Pharmaceuticals to Human Estrogen Receptors α and β in Newly-constructed Yeast Reporter Assays

Chu, W.-L., Shiizaki, K., Kawanishi, M., & Yagi, T. (2009) · Genes and Environment · doi:10.3123/jemsge.31.80 · Cited by 1

The phytoestrogen biochaninA weakens acute cardiac allograft rejection without affecting the reproductive system

Schrepfer, S., Deuse, T., Schäfer, H., Koch‐Nolte, F., Braendle, W. L., & Reichenspurner, H. C. (2005) · Transplant Immunology · doi:10.1016/j.trim.2005.03.017 · Cited by 1

Trauma-hemorrhage and dendritic cell functions: A critical review of splenic dendritic cell dysfunction following trauma-hemorrhage and therapeutic approach

Kawasaki, T., & Sata, T. (2013) · OA Anaesthetics · doi:10.13172/2052-7853-1-2-979 · Cited by 1

Estrogen receptor beta is a negative regulator of mammary cell proliferation

Song, X. (2014) · ScholarWorks -A service of University of Vermont Libraries (University of Vermont) · Cited by 1

Assessment of Endocrine Toxicity

(2009) · CRC Press eBooks · doi:10.1201/9781420080124.ch10 · Cited by 1

Genotoxicity of Endogenous Estrogens

Wright, J. S. (2009) · Wiley eBooks · doi:10.1002/9783527628100.ch35 · Cited by 1

Phytoestrogenic extracts of Cyclopia modulate molecular targets involved in the prevention and treatment of breast cancer

Visser, J. A. K. (2014) · SUNScholar (Stellenbosch University) · Cited by 1

CHAPTER 14 – Regulation of Bone Cell Function by Estrogens

Komm, B., Cheskis, B., & Bodine, P. (2008) · Elsevier eBooks · doi:10.1016/b978-012370544-0.50016-1

Estrogen Action in Normal Prostate Epithelium and in Prostate Cancer

Prins, G. S., & Korach, K. S. (2008) · Humana Press eBooks · doi:10.1007/978-1-60327-079-3_9 · Cited by 1

Effects of estrogen receptor activation on post-exercise muscle satellite cell proliferation

Bunyan, K. (2009) · Scholars Commons (Wilfrid Laurier University)

17BETA-ESTRADIOL regulates immunoglobulin M production through interaction with estrogen receptors

Nakaya, M., Tachibana, H., & Yamada, K. (2006) · Springer eBooks · doi:10.1007/1-4020-4457-7_33

Molecular mechanisms of antidiabetic effects of estrogen

Bryzgalova, G. (2008) · Figshare

The Influence of Propyl Pyrazole Triol on the Post-Exercise Alpha Estrogen Receptor-Mediated Activation of Satellite Cells in Skeletal Muscle of Ovariectomized Rats

Thomas, A. E. (2009) · Scholars Commons (Wilfrid Laurier University)

Vascular biology of estrogen receptors alpha and beta : -An experimental approach to restenosis and transplant arteriosclerosis

Savolainen-Peltonen, H. M. (2004) · Työväentutkimus Vuosikirja

Molecular characterization of estrogen receptors with focus on breast cancer

Putnik, M. (2012) · Figshare

ESTROGEN RECEPTOR REGULATION OF GLUCOSE AND FAT METABOLISM IN THE SKELETAL MUSCLE AND ADIPOSE TISSUE

Gorres, B. K. (2011) · KU ScholarWorks (The University of Kansas)

The effect of pomegranate on postmenopausal syndrome in ovariectomized rats

Ahn, K. H., Yi, K. W., Park, H. T., Shin, J., Hur, J. Y., Kim, Y. T., Kim, S. H., Lee, K. W., Bae, C. S., & Kim, T. (2010) · Korean Journal of Obstetrics & Gynecology · doi:10.5468/kjog.2010.53.4.354

The role of gonadal hormones in mesencephalic dopaminergic systems

Johnson, M. L. (2008) · DukeSpace (Duke University)

Estrogen receptor expression in relation to pain modulation and transmission : experimental studies in rats

Amandusson, Å. (2009) · DiVA (Linkoping University)

Melanoma y esteroides sexuales: ¿tienen relación?

Lozano, J. R., González, A. D. L. F., & Fonseca, E. (2007) · Piel · doi:10.1016/s0213-9251(07)73114-3

THE ROLE OF ANGIOTENSIN-(1-7) IN CARDIOVASCULAR PHYSIOLOGY

Grobe, J. L. (2006)

ESTROGEN ACTION IN RELATION TO METABOLIC DISEASE

Lundholm, L. (2007)

The effects of the selective estrogen receptor modulators MPP and raloxifene in normal and cancerous human and murine uterine tissue

Davis, A. (2007) · doi:10.32469/10355/4999

Studies on molecular mechanisms of persistent vaginal abnormalities induced by neonatal estrogen exposure in mice

中村, 武. (2014) · Institutional Repositories DataBase (IRDB)

Investigation of the mechanisms of estrogen receptor activation by phosphorylation

Halliday, A. C. (2009) · Spiral (Imperial College London) · doi:10.25560/4348

The nuclear hormone receptor ERα plays a critical role in determining estrogen-induced cholesterol gallstones

Wang, H. H., Portincasa, P., & Wang, D. Q.-H. (2009) · Springer eBooks · doi:10.1007/978-1-4020-9644-0_17

Évaluation biologique in vitro d'inhibiteurs de la stéroïde sulfatase ayant un effet SERM

Ouellet, C. (2013) · Corpus Université Laval (Université Laval)

Effects of Short-Term Treatment with Estrogen Receptor Agonist on Morphological Changes in Reproductive Organs of Adult Male Mice

Choi, H., Mo, Y. J., Lee, M., Choe, E. S., Yee, S. T., & Cho, H. W. (2016) · Han-guk hyeonmigyeong hakoeji/Applied microscopy · doi:10.9729/am.2016.46.4.193

Estrogenic Modulation of Fear Generalization

Lynch, J. F. (2016) · OhioLink ETD Center (Ohio Library and Information Network)

Zebrafish as a Model for Studying Estrogen Signaling and Estrogenic Endocrine Disruption

Hao, R. (2013)

Estrogen Receptor Modulators

Rosales, C. I., Gutgesell, L. M., Ratia, K. M., & Thatcher, G. R. J. (2021) · Wiley eBooks · doi:10.1002/0471266949.bmc054.pub2

Low dose of propyl-pyrazole-triol, an agonist of estrogen receptor alpha, administration stimulates the Coolidge effect in fadrozole-treated male rats

Corre, P. H. C., Mainwaring, J. M., Peralta, K. K. Z., Lokman, P. M., Porteous, R. W., & Wibowo, E. (2024) · Hormones and Behavior · doi:10.1016/j.yhbeh.2024.105520

Additional file 5 of Sex and interspecies differences in ESR2-expressing cell distributions in mouse and rat brains

Morishita, M., Higo, S., Iwata, K., & Hirotaka, I. (2024) · Figshare · doi:10.6084/m9.figshare.26655556

Additional file 10 of Sex and interspecies differences in ESR2-expressing cell distributions in mouse and rat brains

Morishita, M., Higo, S., Iwata, K., & Ishii, H. (2024) · Figshare · doi:10.6084/m9.figshare.26655574

Additional file 1 of Sex and interspecies differences in ESR2-expressing cell distributions in mouse and rat brains

Morishita, M., Higo, S., Iwata, K., & Ishii, H. (2024) · Figshare · doi:10.6084/m9.figshare.26655544

Additional file 7 of Sex and interspecies differences in ESR2-expressing cell distributions in mouse and rat brains

Morishita, M., Higo, S., Iwata, K., & Hirotaka, I. (2024) · Figshare · doi:10.6084/m9.figshare.26655565

Additional file 9 of Sex and interspecies differences in ESR2-expressing cell distributions in mouse and rat brains

Morishita, M., Higo, S., Iwata, K., & Ishii, H. (2024) · Figshare · doi:10.6084/m9.figshare.26655571

Additional file 3 of Sex and interspecies differences in ESR2-expressing cell distributions in mouse and rat brains

Morishita, M., Higo, S., Iwata, K., & Hirotaka, I. (2024) · Figshare · doi:10.6084/m9.figshare.26655550

Additional file 4 of Sex and interspecies differences in ESR2-expressing cell distributions in mouse and rat brains

Morishita, M., Higo, S., Iwata, K., & Hirotaka, I. (2024) · Figshare · doi:10.6084/m9.figshare.26655553

Additional file 6 of Sex and interspecies differences in ESR2-expressing cell distributions in mouse and rat brains

Morishita, M., Higo, S., Iwata, K., & Hirotaka, I. (2024) · Figshare · doi:10.6084/m9.figshare.26655559

Additional file 8 of Sex and interspecies differences in ESR2-expressing cell distributions in mouse and rat brains

Morishita, M., Higo, S., Iwata, K., & Ishii, H. (2024) · Figshare · doi:10.6084/m9.figshare.26655568

Additional file 2 of Sex and interspecies differences in ESR2-expressing cell distributions in mouse and rat brains

Morishita, M., Higo, S., Iwata, K., & Hirotaka, I. (2024) · Figshare · doi:10.6084/m9.figshare.26655547

BindingDB Entry 50018042: Tetrahydrofluorenones with conformationally restricted side chains as selective estrogen receptor beta ligands.

BindingDB (2009) · UC San Diego · doi:10.7270/q2v124dh

BindingDB Entry 50017953: Triazolo-tetrahydrofluorenones as selective estrogen receptor beta agonists.

BindingDB (2009) · UC San Diego · doi:10.7270/q2mp52wg

BindingDB Entry 50015171: 7-Substituted 2-phenyl-benzofurans as ER beta selective ligands.

BindingDB (2009) · UC San Diego · doi:10.7270/q2tm79k8

BindingDB Entry 50017728: The discovery of tetrahydrofluorenones as a new class of estrogen receptor beta-subtype selective ligands.

BindingDB (2009) · UC San Diego · doi:10.7270/q2r2110x

BindingDB Entry 50002976: Estrogen Receptor (ER) Subtype Selectivity Identifies 8-Prenylapigenin as an ERβ Agonist from Glycyrrhiza inflata and Highlights the Importance of Chemical and Biological Authentication.

BindingDB (2020) · UC San Diego · doi:10.7270/q2dv1nkt

BindingDB Entry 50011085: Optimisation of estrogen receptor subtype-selectivity of a 4-Aryl-4H-chromene scaffold previously identified by virtual screening.

BindingDB (2021) · UC San Diego · doi:10.7270/q2wd4457

BindingDB Entry 50017889: Estrogen receptor beta-subtype selective tetrahydrofluorenones: use of a fused pyrazole as a phenol bioisostere.

BindingDB (2009) · UC San Diego · doi:10.7270/q24t6j01

BindingDB Entry 50015847: Structure-activity relationships and sub-type selectivity in an oxabicyclic estrogen receptor alpha/beta agonist scaffold.

BindingDB (2009) · UC San Diego · doi:10.7270/q25h7fr7

BindingDB Entry 50016247: Estrogen receptor ligands: design and synthesis of new 2-arylindene-1-ones.

BindingDB (2009) · UC San Diego · doi:10.7270/q25q4vmb

Gene-environment interaction in age-related macular degeneration: Exogenous estrogen, cigarette smoking, and VEGF pathway polymorphisms

Courtenay, M. D. (2014)

Response-Specific and Ligand Dose-Dependent Modulation of Estrogen Receptor (ER) α Activity by ERβ in the Uterus

Frasor, J. M., Barnett, D., Danes, J. M., Hess, R., Parlow, A. F., & Katzenellenbogen, B. S. (2003) · Endocrinology · doi:10.1210/en.2002-0143 · Cited by 232

Dissecting Physiological Roles of Estrogen Receptor α and β with Potent Selective Ligands from Structure-Based Design

Hillisch, A., Peters, O., Kosemund, D., Müller, G. A., Walter, A., Schneider, B., Reddersen, G., Elger, W. A. G., & Fritzemeier, K. (2004) · Molecular Endocrinology · doi:10.1210/me.2004-0050 · Cited by 171

Activities of estrogen receptor alpha- and beta-selective ligands at diverse estrogen responsive gene sites mediating transactivation or transrepression

Harrington, W. R., Sheng, S., Barnett, D., Petz, L. N., Katzenellenbogen, J. A., & Katzenellenbogen, B. S. (2003) · Molecular and Cellular Endocrinology · doi:10.1016/s0303-7207(03)00255-7 · Cited by 301

Die Wirkung von selektiven Östrogenrezeptor [alpha] und [beta]-Agonisten auf Ovar und Uterus am Nagetier

Siebel, P., & Hegele‐Hartung, C. (2005) · RWTH Publications (RWTH Aachen)

Effects of selective estrogen receptor agonists on estrogen receptor expression in the uterus of ovariectomized rats

Blesson, C. S., Masironi, B., & Sahlin, L. (2012) · Open Journal of Molecular and Integrative Physiology · doi:10.4236/ojmip.2012.22006 · Cited by 6