Aureobasidins, new antifungal antibiotics. Taxonomy, fermentation, isolation, and properties.

The genera of fungi sporulating in pure culture

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Studies on aculeacin. I. Isolation and characterization of aculeacin A.

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The black yeasts and allied hyphomycetes.

de Hoog, S., & Hermanides-Nijhof, E. J. (1977) · Studies in Mycology · Cited by 114

L-671,329, a new antifungal agent. I. Fermentation and isolation.

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Structure of aureobasidin A.

IKAI, K., Takesako, K., Shiomi, K., MORIGUCHI, M., UMEDA, Y., Yamamoto, J., Kato, I., & NAGANAWA, H. (1991) · The Journal of Antibiotics · doi:10.7164/antibiotics.44.925 · Cited by 96

A taxonomic study in the “black yeasts”

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Struktur des cyclopeptid-antibiotikums sl 7810 (= echinocandinb)

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Mulundocandin, a new lipopeptide antibiotic. I Taxonomy, fermentation, isolation and characterization.

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Structures of aureobasidins B to R.

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The structure of lipopeptin a

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The influence of moisture on the suppression of Pseudomonas syringae by Aureobasidium pullulans on an artificial leaf surface

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Chapter 14. Progress with antifungal agents and approaches to combat fungal resistance

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Integrative and replicative genetic transformation of Aureobasidium pullulans

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Total Synthesis of Aureobasidin A, an Antifungal Cyclic Depsipeptide

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Emerging Approaches to Inhibit Botrytis cinerea

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Laboratory effect of Boni Protect containing Aureobasidium pullulans (de Bary) Arnoud in the control of some fungal diseases of apple fruit

Wagner, A., Hetman, B., Kopacki, M., Jamiołkowska, A., Krawiec, P., & Lipa, T. (2013) · Acta Agrobotanica · doi:10.5586/aa.2013.009 · Cited by 12

Solution cis-Proline Conformation of IPCs Inhibitor Aureobasidin A Elucidated via NMR-Based Conformational Analysis

Gao, Q., Cleves, A. E., Wang, X., Liu, Y., Bowen, S., Williamson, R. T., Jain, A. N., Sherer, E. C., & Reibarkh, M. (2022) · Journal of Natural Products · doi:10.1021/acs.jnatprod.1c01071 · Cited by 11

Contribution to the synthesis of aureobasidin A. Synthesis of cyclopeptolides containing the sequence leucyl‐N‐methyl‐β‐hydroxyvalyl‐ (2R)‐oxy‐(3R)‐methyl‐pentanoic acid *

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Macrocyclic N-Methylated Cyclic Peptides and Depsipeptides

Maharani, R., Sleebs, B. E., & Hughes, A. B. (2015) · Studies in natural products chemistry · doi:10.1016/b978-0-444-63460-3.00004-3 · Cited by 9

Gγ recruitment system incorporating a novel signal amplification circuit to screen transient protein‐protein interactions

福田, 展., Ishii, J., & Kondo, A. (2011) · FEBS Journal · doi:10.1111/j.1742-4658.2011.08232.x · Cited by 9

A novel species of Aureobasidium (Dothioraceae) recovered from Acer pseudosieboldianum in Korea

Lee, D., Cho, S., Oh, J. Y., Cho, E.-J., & Kwon, S. G. (2021) · Journal of Asia-Pacific Biodiversity · doi:10.1016/j.japb.2021.08.005 · Cited by 9

Total synthesis of the antifungal cyclic depsipeptides Sch 57697 and aureobasidin A

Jao, E., Cooper, A. B., Rane, D. F., Saksena, A. K., Desai, J. A., Wang, J., GIRIJAVALLABHAN, V. M., & Ganguly, A. K. (1996) · Tetrahedron Letters · doi:10.1016/0040-4039(96)01199-9 · Cited by 9

Biological activities of organic extracts of four Aureobasidium pullulans varieties isolated from extreme marine and terrestrial habitats

Botić, T., Kunčič, M. K., Sepčić, K., Batista, U., Zalar, P., Knez, Ž., & Gunde‐Cimerman, N. (2014) · Natural Product Research · doi:10.1080/14786419.2014.888554 · Cited by 9

Non-β-Lactam Antibiotics

Erkel, G. (2010) · Springer eBooks · doi:10.1007/978-3-642-11458-8_6 · Cited by 9

Dibenzylideneacetone Overcomes Botrytis cinerea Infection in Cherry Tomatoes by Inhibiting Chitinase Activity

Niu, X., Wang, Z., Wang, C., & Wang, H. (2023) · Journal of Agricultural and Food Chemistry · doi:10.1021/acs.jafc.3c05695 · Cited by 8

Conformational feature of aureobasidin E, a new type of potent antifungal antibiotic

Ishida, T., In, Y., Fujikawa, A., Urata, H., Inoue, M., IKAI, K., Takesako, K., & Kato, I. (1992) · Journal of the Chemical Society Chemical Communications · doi:10.1039/c39920001231 · Cited by 8

Aureobasidins as New Inhibitors of P-Glycoprotein in Multidrug Resistant Tumor Cells.

Kurome, T., Takesako, K., Kato, I., & Tsuruo, T. (1998) · The Journal of Antibiotics · doi:10.7164/antibiotics.51.353 · Cited by 7

Antimicrobial Activity of Indigenous Strains of Aureobasidium Isolated From Santalum Album Leaves

Kalantar, E., Deopurkar, R. L., & Kapadnis, B. P. (2006) · Iranian journal of pharmaceutical research · doi:10.22037/ijpr.2010.654 · Cited by 7

Aldol-Promoted Reaction of R106-Sarcosine: Synthesis and Conformational Analysis of Novel R106 Analogs

Rodriguez, M. J., Zweifel, M. J., & Loncharich, R. J. (1996) · The Journal of Organic Chemistry · doi:10.1021/jo951485q · Cited by 7

Development of Applied Microbiology to Modern Biotechnology in Japan

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Origin and characterization of cyclodepsipeptides: Comprehensive structural approaches with focus on mass spectrometry analysis of alkali‐cationized molecular species

Liuu, S., Damont, A., Perret, A., Firmesse, O., Bécher, F., Lavison‐Bompard, G., Hueber, A., Woods, A. S., Darii, E., Fenaille, F., et al. (2024) · Mass Spectrometry Reviews · doi:10.1002/mas.21904 · Cited by 4

Mechanisms of antifungal resistance

Delgado, J., Núñez, F., Bermúdez, E., & Asensio, M. A. (2024) · Elsevier eBooks · doi:10.1016/b978-0-12-818619-0.00156-8 · Cited by 5

Diastereoselective synthesis of syn,syn- and syn,anti-2,4-diamino-3-hydroxyglutaric acid derivatives from ethyl α-acyl alaninates

Alvarez‐Ibarra, C., Csákÿ, A. G., MARTINEZ‐SANTOS, E., QUIROGA, M. L., & Tejedor, J. (1999) · Tetrahedron · doi:10.1016/s0040-4020(99)00065-4 · Cited by 5

The Role of Plasma Membrane Pleiotropic Drug Resistance Transporters in the Killer Activity of Debaryomyces hansenii and Wickerhamomyces anomalus Toxins

Czarnecka, M., Połomska, X., Restuccia, C., & Żarowska, B. (2022) · Toxins · doi:10.3390/toxins14030180 · Cited by 5

Site-specific ring opening of depsipeptide aureobasidin A in hydrogen fluoride

Inami, K., Kurome, T., Takesako, K., Kato, I., & Shiba, T. (1996) · Tetrahedron Letters · doi:10.1016/0040-4039(96)00213-4 · Cited by 5

Chapter 16. Recent Advances in Antifungal Agents

Barrett, J. F., & Klaubert, D. H. (1992) · Annual reports in medicinal chemistry · doi:10.1016/s0065-7743(08)60414-5 · Cited by 5

Role of Antifungal Drugs in Combating Invasive Fungal Diseases

Dutt, K. (2019) · Wiley eBooks · doi:10.1002/9781119460053.ch5 · Cited by 4

Characteristics of Aureobasidium pullulans (de Bary et Lowenthal) G. Arnaud isolated from apples and pears with symptoms of sooty blotch in Poland

Mirzwa-Mróz, E., Wińska-Krysiak, M., Dzięcioł, R., & Miekus, A. (2014) · DOAJ (DOAJ: Directory of Open Access Journals) · Cited by 3

Total Synthesis of Pleofugin A, a Potent Inositol Phosphorylceramide Synthase Inhibitor

Kiho, T., Yokoyama, M., & Kogen, H. (2018) · Organic Letters · doi:10.1021/acs.orglett.8b01930 · Cited by 3

Glycans of the Pathogenic Yeast Cryptococcus neoformans and Related Opportunities for Therapeutic Advances

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Aureobasidium sp. from cardamom plant as a potential biocontrol for Fusarium equiseti infecting tomato plants

Rai, G. B., Kayastha, S., Dahal, S., Subba, B., & Malla, S. (2026) · Biological Control · doi:10.1016/j.biocontrol.2026.106077 · Cited by 2

Antimicrobial activity and optimization of Aureobasidin A production by Aureobasidium pullulans PA-2 against Escherichia coli and Staphylococcus aureus

Cheng, L., Yue, D., Wei, Y., Zhu, H., Weng, H., Guo, L., & Guo, Q. (2023) · Plant Protection Science · doi:10.17221/173/2021-pps · Cited by 2

Disruption of Fungi Cell Membranes by Polyenes, Azoles, Allylamines, Amino Acids and Peptides

Aderiye, B. I. (2015) · International Scientific Research Journal · doi:10.18483/irjsci.13 · Cited by 2

Essential Genes inAspergillus fumigatus

Hu, W., Jiang, B., & Roemer, T. (2014) · ASM Press eBooks · doi:10.1128/9781555815523.ch5 · Cited by 1

ANTIBACTERIAL ACTIVITY OF AUREOBASIDIUM PULLULANS

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Overview of Structural Study on Conformations and Intermolecular Interactions of Biomolecules

Ishida, T. (2012) · YAKUGAKU ZASSHI · doi:10.1248/yakushi.132.785 · Cited by 1

PEG-4000 Increased the Mating Efficiency of Yeast-Two Hybrid Screening Process using PmF-box1 as Bait

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Total synthesis of aureobasidin a, an antifungal cyclic depsipeptide

Kurome, T., Inami, K., Inoue, T., IKAI, K., Takesako, K., Kato, I., & Shiba, T. (1994) · Springer eBooks · doi:10.1007/978-94-011-0683-2_114 · Cited by 1

A synthetic intermediate of enantiopureN-protected β-hydroxyvaline, (2R)-2-[N-(tert-butoxycarbonyl)amino]-3-methylbutane-1,3-diol

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Real-Time Monitoring of Relative Peptide–Protein Interaction Strengths in the Yeast Two-Hybrid System

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A synthetic fragment of a cyclic depsipeptide, aureobasidine A:tert-butoxycarbonyl- L -allo-isoleucyl-N-methyl- L -valine (Boc- L -allo-Ile- L -MeVal-OH)

Oku, H., Naito, R., Yamada, K., & Katakai, R. (2004) · Acta Crystallographica Section E Structure Reports Online · doi:10.1107/s1600536804028089

Antimicrobial activity of a thermotolerant Aureobasidium pullulans strain isolated from Faizabad region of Uttar Pradesh in India

Singh, R. K., Gaur, R., Gaur, M. K., Pandey, P. K., & Jamal, F. (2015)

Application of factorial design for the optimized production of antistaphylococcal metabolite by Aureobasidium pullulans

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Cellular and molecular aspects of the interaction betwen maize and the anthracnose pathogen Colletotrichum graminicola

Jiménez, M. F. T. (2013) · UKnowledge (University of Kentucky)

Issues in the Development of Drugs for Treating Deep-Seated Mycosis.

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Stereostructure of aureobasidine E, a new type of potent antifungal antibiotic

Fujikawa, A., In, Y., Urata, H., Inoue, M., Ishida, T., Nemoto, N., Kobayashi, Y., IKAI, K., Takesako, K., & Kato, I. (1993) · Springer eBooks · doi:10.1007/978-94-011-1474-5_73

Synthesis of α-Hydroxyisovaleric acid (Hiv) and α-Acetyloxyisovaleric Acid (Ac-Hiv), Precursors of Aureobasidin B, with Improved Yield

Maharani, R., Rahim, A., Rizqullah, H., Miftah, N. M., Hidayat, A. T., Zainuddin, A., Nurlelasari, N., Harneti, D., & Supratman, U. (2018) · Chimica et Natura Acta · doi:10.24198/cna.v6.n3.20855

Annotated References

(1994) · Expert Opinion on Investigational Drugs · doi:10.1517/13543784.3.2.197

Cyclic Peptides and Betalains

Mofasser, A. Z. M., Howlader, M. I., Alam, M. M., Sayed, N. I., & Mia, R. (2025) · Wiley eBooks · doi:10.1002/9781394287888.ch14

BindingDB Entry 50032683: Inhibition of inositol phosphorylceramide synthase by the cyclic peptide aureobasidin A.

BindingDB (2011) · UC San Diego · doi:10.7270/q27h1jv5

BindingDB Entry 50036824: Aureobasidins: structure-activity relationships for the inhibition of the human MDR1 P-glycoprotein ABC-transporter.

BindingDB (2012) · UC San Diego · doi:10.7270/q2pg1sfc

BindingDB Entry 50037081: Cyclosporins: structure-activity relationships for the inhibition of the human MDR1 P-glycoprotein ABC transporter.

BindingDB (2012) · UC San Diego · doi:10.7270/q29024hj

Isolation, structures, and antifungal activities of new aureobasidins.

Yoshikawa, Y., IKAI, K., UMEDA, Y., OGAWA, A., Takesako, K., Kato, I., & NAGANAWA, H. (1993) · The Journal of Antibiotics · doi:10.7164/antibiotics.46.1347 · Cited by 29

Structures and Antifungal Activities of New Aureobasidins.

AWAZU, N., IKAI, K., Yamamoto, J., NISHIMURA, K., Mizutani, S., Takesako, K., & Kato, I. (1995) · The Journal of Antibiotics · doi:10.7164/antibiotics.48.525 · Cited by 26

Biological properties of aureobasidin A, a cyclic depsipeptide antifungal antibiotic.

Takesako, K., KURODA, H., INOUE, T., HARUNA, F., Yoshikawa, Y., Kato, I., Uchida, K., Hiratani, T., & Yamaguchi, H. (1993) · The Journal of Antibiotics · doi:10.7164/antibiotics.46.1414 · Cited by 189

Structure of aureobasidin A.

IKAI, K., Takesako, K., Shiomi, K., MORIGUCHI, M., UMEDA, Y., Yamamoto, J., Kato, I., & NAGANAWA, H. (1991) · The Journal of Antibiotics · doi:10.7164/antibiotics.44.925 · Cited by 96

Antifungal agents from tropical isolates of Aureobasidium pullulans

Deenarn, P., Lotrakul, P., Prasongsuk, S., & Punnapayak, H. (2006) · doi:10.11556/msj7abst.50.0.181.0