Release and absorption rates of intramuscularly and subcutaneously injected pharmaceuticals (II)

Effect of the cholesterol content of small unilamellar liposomes on their stability in vivo and in vitro

Kirby, C. J., Clarke, J., & Gregoriadis, G. (1980) · Biochemical Journal · doi:10.1042/bj1860591 · Cited by 592 · see citing works

The effect of particle size and charge on the clearance rates of liposomes and liposome encapsulated drugs

Juliano, R. L., & Stamp, D. (1975) · Biochemical and Biophysical Research Communications · doi:10.1016/s0006-291x(75)80433-5 · Cited by 521 · see citing works

Serum-induced leakage of liposome contents

Allen, T. M., & Cleland, L. G. (1980) · Biochimica et Biophysica Acta (BBA) - Biomembranes · doi:10.1016/0005-2736(80)90118-2 · Cited by 472 · see citing works

Liposomal and Lipid Formulations of Amphotericin B

Janknegt, R., de Marie, S., Bakker‐Woudenberg, I. A. J. M., & Crommelin, D. J. A. (1992) · Clinical Pharmacokinetics · doi:10.2165/00003088-199223040-00004 · Cited by 272 · see citing works

Disintegration of phosphatidylcholine liposomes in plasma as a result of interaction with high-density lipoproteins

Scherphof, G. L., Roerdink, F. H., Waite, M. B., & Parks, J. S. (1978) · Biochimica et Biophysica Acta (BBA) - General Subjects · doi:10.1016/0304-4165(78)90025-9 · Cited by 246 · see citing works

Lymphatic Transport of Drugs

Charman, W. N., & Stella, V. J. (2019) · Routledge eBooks · doi:10.1201/9780203748572 · Cited by 195 · see citing works

Properties and Biological Effects of Liposomes and their uses in Pharmacology and Toxicology

Kimelberg, H. K., Mayhew, E. G., & Gregoriadis, G. (1978) · Critical Reviews in Toxicology · doi:10.3109/10408447809029333 · Cited by 165 · see citing works

Effect of liposome size and drug release properties on pharmacokinetics of encapsulated drug in rats.

Allen, T. M., & Everest, J. M. (1983) · Journal of Pharmacology and Experimental Therapeutics · doi:10.1016/s0022-3565(25)21638-x · Cited by 137 · see citing works

Biopharmaceutical Considerations in Subcutaneous and Intramuscular Drug Administration

Ballard, B. E. (1968) · Journal of Pharmaceutical Sciences · doi:10.1002/jps.2600570301 · Cited by 136 · see citing works

The phospholipid component of small unilamellar liposomes controls the rate of clearance of entrapped solutes from the circulation

Gregoriadis, G. C., & Senior, J. (1980) · FEBS Letters · doi:10.1016/0014-5793(80)80994-x · Cited by 133 · see citing works

Interaction of unilamellar liposomes with serum lipoproteins and apolipoproteins

Guo, L., Hamilton, R. L., Goerke, J., et al. (1980) · Journal of Lipid Research · doi:10.1016/s0022-2275(20)34759-3 · Cited by 127 · see citing works

Serum opsonins and phagocytosis of saturated and unsaturated phospholipid liposomes

Moghimi, S. M., & Patel, H. M. (1989) · Biochimica et Biophysica Acta (BBA) - Biomembranes · doi:10.1016/0005-2736(89)90307-6 · Cited by 119 · see citing works

The pharmacokinetics of artemisinin after oral, intramuscular and rectal administration to volunteers

Titulaer, H. A. C., Zuidema, J., Kager, P. A., Wetsteyn, J. C. F. M., Lugt, C. B., & Merkus, F. W. H. M. (1990) · Journal of Pharmacy and Pharmacology · doi:10.1111/j.2042-7158.1990.tb07030.x · Cited by 116 · see citing works

Interaction of Liposomes with Blood Plasma Proteins

BLACK, C. D. V., & Gregoriadis, G. C. (1976) · Biochemical Society Transactions · doi:10.1042/bst0040253a · Cited by 99 · see citing works

Enzyme replacement via liposomes variations in lipid composition determine liposomal integrity in biological fluids

Finkelstein, M. C., & Weissmann, G. (1979) · Biochimica et Biophysica Acta (BBA) - General Subjects · doi:10.1016/0304-4165(79)90354-4 · Cited by 93 · see citing works

Leakage of sucrose from phosphatidylcholine liposomes induced by interaction with serum albumin

Zborowski, J., Roerdink, F. H., & Scherphof, G. L. (1977) · Biochimica et Biophysica Acta (BBA) - General Subjects · doi:10.1016/0304-4165(77)90151-9 · Cited by 81 · see citing works

The effect of serum protein fractions on liposome-cell interactions in cultured cells and the perfused rat liver

Tyrrell, D. A. J., Richardson, V. J., & Ryman, B. E. (1977) · Biochimica et Biophysica Acta (BBA) - General Subjects · doi:10.1016/0304-4165(77)90204-5 · Cited by 76 · see citing works

Incorporation of phosphatidylcholine into spherical and discoidal lipoproteins during incubation of egg phosphatidylcholine vesicles with isolated high density lipoproteins or with plasma.

Tall, A. R., & Green, P. H. (1981) · Journal of Biological Chemistry · doi:10.1016/s0021-9258(19)69912-6 · Cited by 74 · see citing works

Release and absorption rate aspects of intramuscularly injected pharmaceuticals

Zuidema, J., Pieters, F. A. J. M., & Duchateau, G. S. M. J. E. (1988) · International Journal of Pharmaceutics · doi:10.1016/0378-5173(88)90209-8 · Cited by 72 · see citing works

Effect of fetal calf serum and serum protein fractions on the uptake of liposomal phosphatidylcholine by rat hepatocytes in primary monolayer culture

Hoekstra, D., & Scherphof, G. L. (1979) · Biochimica et Biophysica Acta (BBA) - Biomembranes · doi:10.1016/0005-2736(79)90357-2 · Cited by 67 · see citing works

Bioavailability and single‐dose pharmacokinetics of intramuscular phenytoin

Kostenbauder, H. B., Rapp, R. P., McGovren, J. P., et al. (1975) · Clinical Pharmacology & Therapeutics · doi:10.1002/cpt1975184449 · Cited by 65 · see citing works

Liposomes disposition in vivo V. Liposome stability in plasma and implications for drug carrier function

Hunt, C. A. (1982) · Biochimica et Biophysica Acta (BBA) - General Subjects · doi:10.1016/0304-4165(82)90233-1 · Cited by 61 · see citing works

Bioavailability of Oral and Intramuscular Phenobarbital

Viswanathan, C. T., Booker, H. E., & Welling, P. G. (1978) · The Journal of Clinical Pharmacology · doi:10.1002/j.1552-4604.1978.tb02428.x · Cited by 49 · see citing works

Liposomes and biotherapeutics

Storm, G., Wilms, H. P., & Crommelin, D. J. A. (1991) · Biotherapy · doi:10.1007/bf02175097 · Cited by 43 · see citing works

Effect of lipoprotein-free plasma on the interaction of human plasma high density lipoprotein with egg yolk phosphatidylcholine liposomes

Damen, J., Dijkstra, J., Regts, J., et al. (1980) · Biochimica et Biophysica Acta (BBA) - Lipids and Lipid Metabolism · doi:10.1016/0005-2760(80)90188-5 · Cited by 41 · see citing works

Premedication with midazolam in out‐patient general anaesthesia. A comparison with morphine‐scopolamine and placebo

Raeder, J. C., & Breivik, H. (1987) · Acta Anaesthesiologica Scandinavica · doi:10.1111/j.1399-6576.1987.tb02612.x · Cited by 41 · see citing works

The Determination of Absorption Rates from Rat Muscles: an Experimental Approach to Kinetic Descriptions

Sund, R. B., & Schou, J. S. (1964) · Acta Pharmacologica et Toxicologica · doi:10.1111/j.1600-0773.1964.tb01796.x · Cited by 36 · see citing works

Studies of Human Peripheral Blood Flow: The Effect of Injection Volume on the Intramuscular Radiosodium Clearance Rate

WARNER, G. F., Dobson, E. L., Pace, N., et al. (1953) · Circulation · doi:10.1161/01.cir.8.5.732 · Cited by 36 · see citing works

Studies on the absorption of practically water-insoluble drugs following injection. II. Intramuscular absorption from aqueous suspensions in rats.

Hirano, K., Ichihashi, T., & Yamada, H. (1981) · Chemical and Pharmaceutical Bulletin · doi:10.1248/cpb.29.817 · Cited by 36 · see citing works

Intramuscular Absorption of Drugs from Oily Solutions in the Rat

Tanaka, T., Kobayashi, H., Okumura, K., Muranishi, S., & Sezaki, H. (1974) · Chemical and Pharmaceutical Bulletin · doi:10.1248/cpb.22.1275 · Cited by 31 · see citing works

LOCAL EFFECTS AND MECHANISM OF ABSORPTION OF IRON PREPARATIONS ADMINISTERED INTRAMUSCULARLY

BERESFORD, C. R., Golberg, L., & Smith, J. P. (1957) · British Journal of Pharmacology and Chemotherapy · doi:10.1111/j.1476-5381.1957.tb01371.x · Cited by 27 · see citing works

PLASMA-DIAZEPAM LEVELS FOLLOWING INTRAMUSCULAR INJECTION BY NURSES AND DOCTORS

Dundee, J. W., Gamble, J. A. S., & ASSAF, R. A. E. (1974) · The Lancet · doi:10.1016/s0140-6736(74)90130-5 · Cited by 27 · see citing works

The Parenteral Controlled Release of Liposome Encapsulated Chloroquine in Mice

Titulaer, H. A. C., Eling, W. M. C., Crommelin, D. J. A., et al. (1990) · Journal of Pharmacy and Pharmacology · doi:10.1111/j.2042-7158.1990.tb07052.x · Cited by 27 · see citing works

Interaction of plasma apolipoproteins with lipid monolayers

Jackson, R. L., Pattus, F., & DEMEL, R. A. (1979) · Biochimica et Biophysica Acta (BBA) - Biomembranes · doi:10.1016/0005-2736(79)90126-3 · Cited by 25 · see citing works

Absorption of Atropine From Muscle

Schriftman, H., & Kondritzer, A. A. (1957) · American Journal of Physiology-Legacy Content · doi:10.1152/ajplegacy.1957.191.3.591 · Cited by 23 · see citing works

A Rheological Study of Procaine Penicillin G Depot Preparations**Research Division, Abbott Laboratories, North Chicago, Ill.

Ober, S. S., Vincent, H. C., Simon, D. E., & Frederick, K. J. (1958) · Journal of the American Pharmaceutical Association (Scientific ed ) · doi:10.1002/jps.3030470915 · Cited by 22 · see citing works

Influence of solvent on the availability of testosterone propionate from oily, intramuscular injections in the rat

Al-Hindawi, M. K., James, K., & Nicholls, P. J. (1987) · Journal of Pharmacy and Pharmacology · doi:10.1111/j.2042-7158.1987.tb06951.x · Cited by 22 · see citing works

Factors affecting the absorption of ampicillin administered intramuscularly in dwarf goats

Groothuis, D. G., Werdler, M. E. B., Mifrt, A. S. J. P. A. M. V., et al. (1980) · Research in Veterinary Science · doi:10.1016/s0034-5288(18)32699-7 · Cited by 21 · see citing works

The in vivo release of cortisone esters from liposomes and the intramuscular clearance of liposomes

Arrowsmith, M., Hadgraft, J., & Kellaway, I. W. (1984) · International Journal of Pharmaceutics · doi:10.1016/0378-5173(84)90181-9 · Cited by 21 · see citing works

Effect of Albumin and Methylated Albumin on the Glucose Permeability of Lipid Membranes

Kitagawa, T., Inoue, K., & Nojima, S. (1976) · The Journal of Biochemistry · doi:10.1093/oxfordjournals.jbchem.a131169 · Cited by 20 · see citing works

Multivesicular liposomes containing cytarabine for slow-release Sc administration.

Kim, S., & Howell, S. B. (1987) · PubMed · Cited by 20 · see citing works

Clearance concept in salivary drug excretion. Part I: theory.

Zuidema, J., & van Ginneken, C. A. M. (1983) · PubMed · Cited by 20 · see citing works

Studies on the Absorption of Practically Water-Insoluble Drugs Following Injection VI: Subcutaneous Absorption from Aqueous Suspensions in Rats

Hirano, K., & Hideo, Y. (1982) · Journal of Pharmaceutical Sciences · doi:10.1002/jps.2600710506 · Cited by 18 · see citing works

Liposomes and immunoliposomes for controlled release or site specific delivery of anti-parasitic drugs and cytostatics

Crommelin, D. J. A., Eling, W. M. C., Steerenberg, P. A., Nässander, U. K., Storm, G., de Jong, W. H., van Hoesel, Q. G. C. M., & Zuidema, J. (1991) · Journal of Controlled Release · doi:10.1016/0168-3659(91)90038-f · Cited by 17 · see citing works

A Residue Study and Comparison of Penicillin and Dihydrostreptomycin Concentrations After Intramuscular and Subcutaneous Administration in Cattle

Mercer, H. D., Rollins, L. D., Garth, M. A., et al. (1971) · Journal of the American Veterinary Medical Association · doi:10.2460/javma.1971.158.06.776 · Cited by 17 · see citing works

Effect of Dosing Volume on Intramuscular Absorption Rate of Aminoglycosides

Pfefferx, M., & Harken, D. R. V. (1981) · Journal of Pharmaceutical Sciences · doi:10.1002/jps.2600700428 · Cited by 15 · see citing works

Influence of injection volume on the release kinetics of liposomal chloroquine administered subcutaneously or intramuscularly to mice

Kadir, F., Eling, W. M. C., Crommelin, D. J. A., & Zuidema, J. (1991) · Journal of Controlled Release · doi:10.1016/0168-3659(91)90146-5 · Cited by 15 · see citing works

Absorption of Drugs from the Skeletal Muscle of the Rats.(3). Effect of Watersoluble Adjuvants and Vehicles on the Intramuscular Absorption

Kakemi, K., Sezaki, H., Okumura, K., et al. (1972) · Chemical and Pharmaceutical Bulletin · doi:10.1248/cpb.20.443 · Cited by 15 · see citing works

Drug lipophilicity and release pattern of some β-blocking agents after intra-adipose injection in pigs

Kadir, F., Zuidema, J., Pijpers, A., Vulto, A. G., & Verheijden, J. H. M. (1990) · International Journal of Pharmaceutics · doi:10.1016/0378-5173(90)90266-7 · Cited by 15 · see citing works

Pharmacokinetic and Pharmacodynamic Aspects of Artelinic Acid in Rodents

Titulaer, H. A. C., Eling, W. M. C., & Zuidema, J. (1993) · Journal of Pharmacy and Pharmacology · doi:10.1111/j.2042-7158.1993.tb05695.x · Cited by 15 · see citing works

Pharmacokinetics of intravenously, intramuscularly and intra‐adiposely administered carazolol in pigs

Kadir, F., Zuidema, J., Pijpers, A., Meléndez-Arce, R., Vulto, A. G., & Verheijden, J. H. M. (1990) · Journal of Veterinary Pharmacology and Therapeutics · doi:10.1111/j.1365-2885.1990.tb00788.x · Cited by 13 · see citing works

Prolonged elimination of midazolam after i. m. administration

Rærder, J. C., & Nilsen, O. G. (1988) · Acta Anaesthesiologica Scandinavica · doi:10.1111/j.1399-6576.1988.tb02767.x · Cited by 12 · see citing works

Kinetics and prophylactic efficacy of increasing dosages of liposome-encapsulated chloroquine after intramuscular injection into mice

Kadir, F., Eling, W. M. C., Crommelin, D. J. A., et al. (1992) · Journal of Controlled Release · doi:10.1016/0168-3659(92)90138-h · Cited by 12 · see citing works

Clearance concept in salivary drug excretion. Part II: Experiments.

Zuidema, J., & van Ginneken, C. A. M. (1983) · PubMed · Cited by 12 · see citing works

Studies on the Absorption of Practically Water-Insoluble Drugs Following Injection VII: Plasma Concentration after Different Subcutaneous Doses of a Drug in Aqueous Suspension in Rats

Hirano, K., & Yamada, H. (1983) · Journal of Pharmaceutical Sciences · doi:10.1002/jps.2600720607 · Cited by 11 · see citing works

Influence of the injection volume on the release pattern of intramuscularly administered propranolol to rats

Kadir, F., Seijsener, C. B. J., & Zuidema, J. (1992) · International Journal of Pharmaceutics · doi:10.1016/0378-5173(92)90011-p · Cited by 8 · see citing works

Bioavailability of parenteral drugs I. Intravenous and intramuscular doses.

Tse, F. L. S., & Welling, P. G. (1981) · PubMed · Cited by 8 · see citing works

Effect of Propylene Glycol on Subcutaneous Absorption of a Benzimidazole Hydrochloride

Yu, C.-D., & Kent, J. S. (1982) · Journal of Pharmaceutical Sciences · doi:10.1002/jps.2600710434 · Cited by 7 · see citing works

Effect of ethanol on the intramuscular absorption of water-soluble drugs in the rat.

Kobayashi, H., Miyoshi, Y., KITAMURA, K., et al. (1977) · Chemical and Pharmaceutical Bulletin · doi:10.1248/cpb.25.2862 · Cited by 5 · see citing works

Bioavailability in human volunteers of three intramuscular formulations of cefonicid: A long‐acting cephalosporin

Brumfitt, W., Hamilton-Miller, J. M. T., Grady, D., et al. (1988) · Biopharmaceutics & Drug Disposition · doi:10.1002/bod.2510090303 · Cited by 1 · see citing works

Subcutaneous Administration of Biotherapeutics: An Overview of Current Challenges and Opportunities

Bittner, B., Richter, W., & Schmidt, J. (2018) · BioDrugs · doi:10.1007/s40259-018-0295-0 · Cited by 447 · see citing works

Subcutaneous drug delivery and the role of the lymphatics

McLennan, D. N., Porter, C. J. H., & Charman, S. A. (2005) · Drug Discovery Today: Technologies · doi:10.1016/j.ddtec.2005.05.006 · Cited by 259 · see citing works

Formulation and pharmacology of long-acting cabotegravir

Trezza, C., Ford, S. L., Spreen, W., Pan, R., & Piscitelli, S. (2015) · Current Opinion in HIV and AIDS · doi:10.1097/coh.0000000000000168 · Cited by 179 · see citing works

Population Pharmacokinetics of Intramuscular Paliperidone Palmitate in Patients with Schizophrenia: A Novel Once-Monthly, Long-Acting Formulation of an Atypical Antipsychotic

Samtani, M. N., Vermeulen, A., & Stuyckens, K. (2009) · Clinical Pharmacokinetics · doi:10.2165/11316870-000000000-00000 · Cited by 170 · see citing works

Prediction of Lipophilicity of Orthopramides by Comparative Molecular Field Analysis (CoMFA)

유성은, & 신영아 (1995) · Bulletin of the Korean Chemical Society · Cited by 1 · see citing works

A New Straightforward Method for Lipophilicity (logP) Measurement using 19F NMR Spectroscopy

Wang, Z., Jeffries, B. F., Felstead, H. R., et al. (2019) · Journal of Visualized Experiments · doi:10.3791/58567 · Cited by 6 · see citing works

Lipophilicity and antiproliferative activity profiling of 2-benzylidencycloalkanones

Hallgas, B., Dobos, Z., Agócs, A., et al. (2007) · Journal of Chromatography B · doi:10.1016/j.jchromb.2007.05.027 · Cited by 12 · see citing works

A New Straightforward Method for Lipophilicity (logP) Measurement using 19F NMR Spectroscopy

Wang, Z., Jeffries, B. F., Felstead, H. R., et al. (2019) · Journal of Visualized Experiments · doi:10.3791/58567-v

The Comparison Between the Calculated and HPLC-Predicted Lipophilicity Parameters for Selected Groups of Drugs

Stasiak, J., Koba, M., Bober, L., et al. (2013) · Combinatorial Chemistry & High Throughput Screening · doi:10.2174/1386207311316080003 · Cited by 5 · see citing works