σ-1 Receptors (σ1 Binding Sites) Form Raft-Like Microdomains and Target Lipid Droplets on the Endoplasmic Reticulum: Roles in Endoplasmic Reticulum Lipid Compartmentalization and Export

Lipid rafts and signal transduction

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Purification, molecular cloning, and expression of the mammalian sigma1-binding site.

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Adipose differentiation-related protein is an ubiquitously expressed lipid storage droplet-associated protein

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Mechanisms of lipid-body formation

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Steroid Binding at σ Receptors Suggests a Link Between Endocrine, Nervous, and Immune Systems

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Evidence for sigma opioid receptor: binding of [3H]SKF-10047 to etorphine-inaccessible sites in guinea-pig brain.

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Epidermal Growth Factor-induced Vacuolar (H+)-ATPase Assembly

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Access of viral proteins to mitochondria via mitochondria‐associated membranes

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Molecular Dysfunctions of Mitochondria-Associated Membranes (MAMs) in Alzheimer’s Disease

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Sigma‐2 Receptor Agonists as Possible Antitumor Agents in Resistant Tumors: Hints for Collateral Sensitivity

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Behavioural phenotyping of knockout mice for the sigma-1 (σ 1 ) chaperone protein revealed gender-related anxiety, depressive-like and memory alterations

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Attenuation of methamphetamine-induced effects through the antagonism of sigma (σ) receptors: Evidence from in vivo and in vitro studies

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Juxtaposition of the Steroid Binding Domain-like I and II Regions Constitutes a Ligand Binding Site in the σ-1 Receptor

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A Variant of the Sigma Receptor Type-1 Gene Is a Protective Factor for Alzheimer Disease

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Dysregulation of Neuronal Calcium Signaling via Store-Operated Channels in Huntington's Disease

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Emerging Benefits: Pathophysiological Functions and Target Drugs of the Sigma-1 Receptor in Neurodegenerative Diseases

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Cocaine and HIV-1 Interplay: Molecular Mechanisms of Action and Addiction

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Analogues of σ Receptor Ligand 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) with Added Polar Functionality and Reduced Lipophilicity for Potential Use as Positron Emission Tomography Radiotracers

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The molecular chaperone sigma 1 receptor mediates rescue of retinal cone photoreceptor cells via modulation of NRF2

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Sigma-1 Receptor Regulates Early Steps of Viral RNA Replication at the Onset of Hepatitis C Virus Infection

Friesland, M., Mingorance, L., Chung, J., Chisari, F. V., & Gastaminza, P. (2013) · Journal of Virology · doi:10.1128/jvi.03557-12 · Cited by 51

Sigma-1 Receptor (S1R) Interaction with Cholesterol: Mechanisms of S1R Activation and Its Role in Neurodegenerative Diseases

Zhemkov, V., Geva, M., Hayden, M. R., & Борисович, Б. И. (2021) · International Journal of Molecular Sciences · doi:10.3390/ijms22084082 · Cited by 50

Palmitoylated CKAP4 regulates mitochondrial functions through an interaction with VDAC2 at ER–mitochondria contact sites

Harada, T., Sada, R., Osugi, Y., Matsumoto, S., Matsuda, T., Hayashi, M., Nagai, T., Harada, A., & Kikuchi, A. (2020) · Journal of Cell Science · doi:10.1242/jcs.249045 · Cited by 49

Antinociception by Sigma-1 Receptor Antagonists

Romero, L. I., Merlos, M., & Vela, J. M. (2016) · Advances in pharmacology · doi:10.1016/bs.apha.2015.11.003 · Cited by 47

Ligand-dependent localization and intracellular stability of sigma-1 receptors in CHO-K1 ce

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Immunohistochemical localization of the sigma1 receptor in Schwann cells of rat sciatic nerve

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Effects of the Sigma-1 Receptor Agonist 1-(3,4-Dimethoxyphenethyl)-4-(3-Phenylpropyl)-Piperazine Dihydro-Chloride on Inflammation after Stroke

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Regulators of mitochondrial Ca2+ homeostasis in cerebral ischemia

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The Functional Role of Voltage-Gated Sodium Channel Nav1.5 in Metastatic Breast Cancer

Luo, Q., Wu, T., Wu, W., Chen, G., Luo, X., Jiang, L., Tao, H., Rong, M., Kang, S., & Deng, M. (2020) · Frontiers in Pharmacology · doi:10.3389/fphar.2020.01111 · Cited by 46

Structure of the σ1 Receptor and Its Ligand Binding Site

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ADRP is dissociated from lipid droplets by ARF1-dependent mechanism

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Purification and characterization of the guinea pig sigma-1 receptor functionally expressed in Escherichia coli

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Overview of Sigma-1R Subcellular Specific Biological Functions and Role in Neuroprotection

Lachance, V., Bélanger, S.-M., Hay, C., Corvec, V. L., Banouvong, V., Lapalme, M., Tarmoun, K., Beaucaire, G., Lussier, M. P., & Kourrich, S. (2023) · International Journal of Molecular Sciences · doi:10.3390/ijms24031971 · Cited by 46

Cognitive evaluation of disease-modifying efficacy of donepezil in the APP23 mouse model for Alzheimer’s disease

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Organelle Communication at Membrane Contact Sites (MCS): From Curiosity to Center Stage in Cell Biology and Biomedical Research

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Progesterone and Allopregnanolone Rapidly Attenuate Estrogen-Associated Mechanical Allodynia in Rats with Persistent Temporomandibular Joint Inflammation

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Cancer: Untethering Mitochondria from the Endoplasmic Reticulum?

Herrera-Cruz, M. S., & Simmen, T. (2017) · Frontiers in Oncology · doi:10.3389/fonc.2017.00105 · Cited by 45

Targeting Nanocarriers with Anisamide: Fact or Artifact?

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APEX2- tagging of Sigma 1-receptor indicates subcellular protein topology with cytosolic N-terminus and ER luminal C-terminus

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Lovastatin-induced cholesterol depletion affects both apical sorting and endocytosis of aquaporin-2 in renal cells

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The evolutionary appearance of signaling motifs in PGRMC1

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Effects of the selective sigma‐1 receptor antagonist S1 RA on formalin‐induced pain behavior and neurotransmitter release in the spinal cord in rats

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Circulating low density lipoprotein (LDL)

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Chaperone Sigma1R and Antidepressant Effect

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The emerging role of the sigma-1 receptor in autophagy: hand-in-hand targets for the treatment of Alzheimer’s

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The Human Cytomegalovirus Protein UL37 Exon 1 Associates with Internal Lipid Rafts

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A role for sigma receptors in stimulant self-administration and addiction

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Sigma-1 Receptor Signaling: In Search of New Therapeutic Alternatives for Cardiovascular and Renal Diseases

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Loss of Sigma‐1 Receptor Chaperone Promotes Astrocytosis and Enhances the Nrf2 Antioxidant Defense

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Sigma-1 receptors and animal studies centered on pain and analgesia

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The Ligand Binding Region of the Sigma-1 Receptor: Studies Utilizing Photoaffinity Probes, Sphingosine and N-Alkylamines

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Connection Lost, MAM: Errors in ER–Mitochondria Connections in Neurodegenerative Diseases

Johri, A., & Chandra, A. (2021) · Brain Sciences · doi:10.3390/brainsci11111437 · Cited by 34

Protein Kinase A Activation Down-Regulates, Whereas Extracellular Signal-Regulated Kinase Activation Up-Regulates σ-1 Receptors in B-104 Cells: Implication for Neuroplasticity

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High prevalence for obesity in severe COVID-19: Possible links and perspectives towards patient stratification

Dugail, I., Amri, E., & Vitale, N. (2020) · Biochimie · doi:10.1016/j.biochi.2020.07.001 · Cited by 34

Sigma–1 receptor activation alleviates blood–brain barrier disruption post cerebral ischemia stroke by stimulating the GDNF–GFRα1–RET pathway

Liu, D., Yang, L., Liu, P., Ji, X., Qi, X., Wang, Z., Chi, T., & Zou, L. (2021) · Experimental Neurology · doi:10.1016/j.expneurol.2021.113867 · Cited by 33

Involvement of the sigma1(σ1) receptor in the anti‐amnesic, but not antidepressant‐like, effects of the aminotetrahydrofuran derivative ANAVEX1‐41

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Sigma-1 Receptor Regulates Mitochondrial Function in Glucose- and Oxygen-Deprived Retinal Ganglion Cells

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Sigma 1 Receptor and Its Pivotal Role in Neurological Disorders

Shokr, M. M., Badawi, G. A., Elshazly, S. M., Zaki, H. F., & Mohamed, A. F. (2024) · ACS Pharmacology & Translational Science · doi:10.1021/acsptsci.4c00564 · Cited by 33

Trafficking of PrPcto mitochondrial raft-like microdomains during cell apoptosis

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Pharmacophore and docking-based sequential virtual screening for the identification of novel Sigma 1 receptor ligands

Alamri, M. A. (2019) · Bioinformation · doi:10.6026/97320630015586 · Cited by 32

Pridopidine reduces mutant huntingtin‐induced endoplasmic reticulum stress by modulation of the Sigma‐1 receptor

Shenkman, M., Geva, M., Gershoni‐Emek, N., Hayden, M. R., & Lederkremer, G. Z. (2021) · Journal of Neurochemistry · doi:10.1111/jnc.15366 · Cited by 31

Endomembrane remodeling in SARS-CoV-2 infection

Chen, D., Zhao, Y. G., & Zhang, H. (2022) · Cell Insight · doi:10.1016/j.cellin.2022.100031 · Cited by 33

Sigma-1 (σ1) receptor deficiency reduces β-amyloid25–35-induced hippocampal neuronal cell death and cognitive deficits through suppressing phosphorylation of the NMDA receptor NR2B

Yin, J., Sha, S., Chen, T., Wang, C., Hong, J., Jie, P., Zhou, R., Li, L., Sokabe, M., & Chen, L. (2014) · Neuropharmacology · doi:10.1016/j.neuropharm.2014.09.027 · Cited by 30

Aberrant Subcellular Dynamics of Sigma-1 Receptor Mutants Underlying Neuromuscular Diseases

Wong, A. Y. C., Hristova, E., Ahlskog, N., Tassé, L.-A., Ngsee, J. K., Chudalayandi, P., & Bergeron, R. (2016) · Molecular Pharmacology · doi:10.1124/mol.116.104018 · Cited by 30

The Sigma-1 Receptor: When Adaptive Regulation of Cell Electrical Activity Contributes to Stimulant Addiction and Cancer

Soriani, O., & Kourrich, S. (2019) · Frontiers in Neuroscience · doi:10.3389/fnins.2019.01186 · Cited by 29

Findings questioning the involvement of Sigma-1 receptor in the uptake of anisamide-decorated particles

Dasargyri, A., Hervella, P., Christiansen, A. J., Proulx, S. T., Detmar, M. J., & Leroux, J. (2016) · Journal of Controlled Release · doi:10.1016/j.jconrel.2016.01.021 · Cited by 29

The Sigma Enigma: A Narrative Review of Sigma Receptors

Pergolizzi, J. V., Varrassi, G., Coleman, M., Breve, F., Christo, D. K., Christo, P. J., & Moussa, C. (2023) · Cureus · doi:10.7759/cureus.35756 · Cited by 29

Sigma-1 receptors amplify dopamine D1 receptor signaling at presynaptic sites in the prelimbic cortex

Fu, Y., Zhao, Y., Luan, W., Dong, L.-Y., Dong, Y. W., Lai, B., Zhu, Y., & Zheng, P. (2010) · Biochimica et Biophysica Acta (BBA) - Molecular Cell Research · doi:10.1016/j.bbamcr.2010.08.005 · Cited by 28

Scouting new sigma receptor ligands: Synthesis, pharmacological evaluation and molecular modeling of 1,3-dioxolane-based structures and derivatives

Franchini, S., Battisti, U. M., Prandi, A., Tait, A., Borsari, C., Cichero, E., Fossa, P., Cilia, A., Prezzavento, O., Ronsisvalle, S., et al. (2016) · European Journal of Medicinal Chemistry · doi:10.1016/j.ejmech.2016.01.059 · Cited by 27

Sigma-1 receptor activation mediates the sustained antidepressant effect of ketamine in mice via increasing BDNF levels

Ma, H., Li, J., Qiao, X., Zhang, Y., Hou, X.-J., Chen, H., Chen, H., Zhang, Y., & Li, Y. (2023) · Acta Pharmacologica Sinica · doi:10.1038/s41401-023-01201-8 · Cited by 28

Astrocytic mobilization of glutathione peroxidase-1 contributes to the protective potential against cocaine kindling behaviors in mice via activation of JAK2/STAT3 signaling

Nhu, H., Nguyen, L. T. T., Shin, E., Kim, D.-J., Jeong, J. H., Chung, Y. H., Lei, X. G., Sharma, N., Jang, C., Nabeshima, T., et al. (2018) · Free Radical Biology and Medicine · doi:10.1016/j.freeradbiomed.2018.12.027 · Cited by 27

Interaction of Afobazole with σ1-Receptors

Середенин, С. Б., Антипова, Т. А., Воронин, М. В., Kurchashova, S., & Kuimov, A. N. (2009) · Bulletin of Experimental Biology and Medicine · doi:10.1007/s10517-009-0624-x · Cited by 26

The essential roles of protein–protein interaction in sigma-1 receptor functions

Pabba, M. (2013) · Frontiers in Cellular Neuroscience · doi:10.3389/fncel.2013.00050 · Cited by 25

Overexpression of Sigma1 Receptor and Its Positive Associations With Pathologic TNM Classification in Esophageal Squamous Cell Carcinoma

Xu, Q., Li, E., Zhang, Y.-F., Liao, L., Xu, X., Wu, Z., Shen, J., & Xu, L. (2012) · Journal of Histochemistry & Cytochemistry · doi:10.1369/0022155412443542 · Cited by 25

A Role for Sigma Receptors in Stimulant Self-Administration and Addiction

Katz, J. L., Hiranita, T., Hong, W. C., Job, M. O., & McCurdy, C. R. (2016) · Handbook of experimental pharmacology · doi:10.1007/164_2016_94 · Cited by 23

Involvement of Chaperone Sigma1R in the Anxiolytic Effect of Fabomotizole

Воронин, М. В., Vakhitova, Y. V., Tsypysheva, I. P., Tsypyshev, D. O., Rybina, I. V., Kurbanov, R. D., Абрамова, Е. В., & Середенин, С. Б. (2021) · International Journal of Molecular Sciences · doi:10.3390/ijms22115455 · Cited by 22

Modulation of mesenteric collecting lymphatic contractions by σ1-receptor activation and nitric oxide production

Trujillo, A. N., Katnik, C. P., Cuevas, J., Jake, B., Taylor‐Clark, T. E., & Breslin, J. W. (2017) · American Journal of Physiology-Heart and Circulatory Physiology · doi:10.1152/ajpheart.00702.2016 · Cited by 20

The Mitochondrial-associated ER membrane (MAM) compartment and its dysregulation in Amyotrophic Lateral Sclerosis (ALS)

Parakh, S., & Atkin, J. D. (2021) · Seminars in Cell and Developmental Biology · doi:10.1016/j.semcdb.2021.02.002 · Cited by 20

Pharmacological and Pathological Implications of Sigma-1 Receptor in Neurodegenerative Diseases

Drewes, N. B., Fang, X., Gupta, N., & Nie, D. (2025) · Biomedicines · doi:10.3390/biomedicines13061409 · Cited by 22

GLP-1/Sigma/RAGE receptors: An evolving picture of Alzheimer's disease pathology and treatment

Neha, N., Wali, Z., Pinky, P., Hattiwale, S. H., Jamal, A., & Parvez, S. (2023) · Ageing Research Reviews · doi:10.1016/j.arr.2023.102134 · Cited by 19

DGAT2 stability is increased in response to DGAT1 inhibition in gene edited HepG2 cells

McFie, P. J., Chumala, P., Katselis, G. S., & Stone, S. J. (2021) · Biochimica et Biophysica Acta (BBA) - Molecular and Cell Biology of Lipids · doi:10.1016/j.bbalip.2021.158991 · Cited by 18

Isolation and characterization of alternatively spliced variants of the mouse sigma1 receptor gene, Sigmar1

Pan, L., Pasternak, D. A., Xu, J., Xu, M., Lu, Z., Pasternak, G. W., & Pan, Y. (2017) · PLoS ONE · doi:10.1371/journal.pone.0174694 · Cited by 18

The molecular role of Sigmar1 in regulating mitochondrial function through mitochondrial localization in cardiomyocytes

Abdullah, C. S., Aishwarya, R., Alam, S., Remex, N. S., Morshed, M., Nitu, S. S., Miriyala, S., Panchatcharam, M., Hartman, B., King, J., et al. (2021) · Mitochondrion · doi:10.1016/j.mito.2021.12.002 · Cited by 18

A Medicinal‐Chemistry‐Guided Approach to Selective and Druglike Sigma 1 Ligands

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Sigma-1 receptor as a potential pharmacological target for the treatment of neuropathology

Bolshakova, A. V., Kukanova, E. O., Gainullina, A. N., Zhemkov, V., Korban, S. A., & Борисович, Б. И. (2016) · St Petersburg Polytechnical University Journal Physics and Mathematics · doi:10.1016/j.spjpm.2016.03.003 · Cited by 17

Annexins Bridging the Gap: Novel Roles in Membrane Contact Site Formation

Enrich, C., Lu, A., Tebar, F., Rentero, C., & Grewal, T. (2022) · Frontiers in Cell and Developmental Biology · doi:10.3389/fcell.2021.797949 · Cited by 18

Improving mitochondria-associated endoplasmic reticulum membranes integrity as converging therapeutic strategy for rare neurodegenerative diseases and cancer

Cagalinec, M., Mohd, A., Borecká, S., Bultynck, G., Choubey, V., Yanovsky‐Dagan, S., Ezer, S., Gašperíková, D., Harel, T., Jurkovičová, D., et al. (2025) · Biochimica et Biophysica Acta (BBA) - Molecular Cell Research · doi:10.1016/j.bbamcr.2025.119954 · Cited by 15

Design and Synthesis of Orally Active Quinolyl Pyrazinamides as Sigma 2 Receptor Ligands for the Treatment of Pancreatic Cancer

Roy, J., Kyani, A., Hanafi, M., Xu, Y., Takyi‐Williams, J., Sun, D., Osman, E. E. A., & Neamati, N. (2023) · Journal of Medicinal Chemistry · doi:10.1021/acs.jmedchem.2c01769 · Cited by 15

Gaining in pan-affinity towards sigma 1 and sigma 2 receptors. SAR studies on arylalkylamines

Rossi, D., Rui, M., Giacomo, M. D., Schepmann, D., Wünsch, B., Monteleone, S., Liedl, K. R., & Collina, S. (2016) · Bioorganic & Medicinal Chemistry · doi:10.1016/j.bmc.2016.10.005 · Cited by 13

Differential Responses to Sigma-1 or Sigma-2 Receptor Ablation in Adiposity, Fat Oxidation, and Sexual Dimorphism

Li, J., Félix‐Soriano, E., Wright, K. R., Shen, H., Baer, L. A., Stanford, K. I., & Guo, L. (2022) · International Journal of Molecular Sciences · doi:10.3390/ijms231810846 · Cited by 13

Novel sugar-cholestanols as anticancer agents against peritoneal dissemination of tumor cells

Hahismoto, S., Yazawa, S., Asao, T., Faried, A., Nishimura, T., Tsuboi, K., Nakagawa, T., Yamauchi, T., Koyama, N., Umehara, K., et al. (2008) · Glycoconjugate Journal · doi:10.1007/s10719-008-9108-x · Cited by 13

Deconstruction of 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline moiety to separate P-glycoprotein (P-gp) activity from σ2 receptor affinity in mixed P-gp/σ2 receptor agents

Pati, M. L., Abate, C., Contino, M., Ferorelli, S., Luisi, R., Carroccia, L., Niso, M., & Berardi, F. (2014) · European Journal of Medicinal Chemistry · doi:10.1016/j.ejmech.2014.11.001 · Cited by 13

The effects of new sigma (σ) receptor ligands, PB190 and PB212, in the models predictive of antidepressant activity

Skuza, G., Sadaj, W., Kabziński, M., Cassano, G., Gasparre, G., Abate, C., & Berardi, F. (2014) · Pharmacological Reports · doi:10.1016/j.pharep.2013.12.002 · Cited by 13

Benzomorphan and non-benzomorphan agonists differentially alter sigma-1 receptor quaternary structure, as does types of cellular stress

Couly, S., Yasui, Y., Foncham, S., Grammatikakis, I., Lal, A., Shi, L., & Su, T. (2024) · Cellular and Molecular Life Sciences · doi:10.1007/s00018-023-05023-z · Cited by 13

Amylovis-201 is a new dual-target ligand, acting as an anti-amyloidogenic compound and a potent agonist of the σ1 chaperone protein

García-Pupo, L., Crouzier, L., Bencomo-Martínez, A., Meunier, J., Morilleau, A., Delprat, B., Sablón-Carrazana, M., Menéndez, R., Maurice, T., & Rodríguez‐Tanty, C. (2024) · Acta Pharmaceutica Sinica B · doi:10.1016/j.apsb.2024.06.013 · Cited by 12

Sigma-1 receptor concentration in plasma of patients with late-life depression: a preliminary study

Tani, M., Shimizu, H., Takebayashi, M., Tanaka, H., Yamagata, B., Kurosawa, K., Yamada, H., Hachisu, M., Hisaoka‐Nakashima, K., Okada‐Tsuchioka, M., et al. (2013) · Neuropsychiatric Disease and Treatment · doi:10.2147/ndt.s53386 · Cited by 12

Identification, pharmacological evaluation and binding mode analysis of novel chromene and chromane based σ1 receptor ligands

Laurini, E., Harel, D., Marson, D., Schepmann, D., Schmidt, T. J., Pricl, S., & Wünsch, B. (2014) · European Journal of Medicinal Chemistry · doi:10.1016/j.ejmech.2014.06.054 · Cited by 12

The Effects of Terminal Tagging on Homomeric Interactions of the Sigma 1 Receptor

Yano, H., Liu, L., Naing, S., & Shi, L. (2019) · Frontiers in Neuroscience · doi:10.3389/fnins.2019.01356 · Cited by 12

Despite Transcriptional and Functional Coordination, Cyclooxygenase-2 and Microsomal Prostaglandin E Synthase-1 Largely Reside in Distinct Lipid Microdomains in WISH Epithelial Cells

Ackerman, W. E., Robinson, J. M., & Kniss, D. A. (2005) · Journal of Histochemistry & Cytochemistry · doi:10.1369/jhc.5a6710.2005 · Cited by 12

Pharmacological Analysis of GABAA Receptor and Sigma1R Chaperone Interaction: Research Report I―Investigation of the Anxiolytic, Anticonvulsant and Hypnotic Effects of Allosteric GABAA Receptors’ Ligands

Воронин, М. В., Шангин, С. В., Литвинова, С. А., Абрамова, Е. В., Kurbanov, R. D., Rybina, I. V., Vakhitova, Y. V., & Середенин, С. Б. (2023) · International Journal of Molecular Sciences · doi:10.3390/ijms24119580 · Cited by 11

The Emerging Role of Sigma Receptors in Pain Medicine

Pergolizzi, J. V., & Varrassi, G. (2023) · Cureus · doi:10.7759/cureus.42626 · Cited by 11

Allosteric Modulation of Opioid G-Protein Coupled Receptors by Sigma1 Receptors

Pasternak, G. W. (2017) · Handbook of experimental pharmacology · doi:10.1007/164_2017_34 · Cited by 11

Sigma1 Regulates Lipid Droplet–Mediated Redox Homeostasis Required for Prostate Cancer Proliferation

Oyer, H. M., Steck, A. R., Longen, C. G., Venkat, S., Bayrak, K., Munger, E. B., Fu, D., Castagnino, P. A., Sanders, C. M., Tancler, N. A., et al. (2023) · Cancer Research Communications · doi:10.1158/2767-9764.crc-22-0371 · Cited by 11

Convolamine, a tropane alkaloid extracted from Convolvulus plauricalis, is a potent sigma‐1 receptor‐positive modulator with cognitive and neuroprotective properties

Crouzier, L., Meunier, J., Carles, A., Morilleau, A., Vrigneau, C., Schmitt, M., Bourguignon, J., Delprat, B., & Maurice, T. (2023) · Phytotherapy Research · doi:10.1002/ptr.8068 · Cited by 11

Neuroprotective targets through which 6-acetyl-3-(4-(4-(4-fluorophenyl)piperazin-1-yl)butyl)benzo[d]oxazol-2(3H)-one (SN79), a sigma receptor ligand, mitigates the effects of methamphetamine in vitro

Kaushal, N., Robson, M. J., Rosen, A., McCurdy, C. R., & Matsumoto, R. R. (2014) · European Journal of Pharmacology · doi:10.1016/j.ejphar.2013.12.039 · Cited by 10

Deferred Administration of Afobazole Induces Sigma1R-Dependent Restoration of Striatal Dopamine Content in a Mouse Model of Parkinson’s Disease

Андреевич, К. И., Verbovaya, E. R., Воронков, Д. Н., Воронин, М. В., & Середенин, С. Б. (2020) · International Journal of Molecular Sciences · doi:10.3390/ijms21207620 · Cited by 11

What is the role of lipids in prion conversion and disease?

Conceição, C. A., de Lemos, G. A., Barros, C. A., & Vieira, T. C. R. G. (2023) · Frontiers in Molecular Neuroscience · doi:10.3389/fnmol.2022.1032541 · Cited by 10

Intracellular Dynamics of σ-1 Receptors (σ1 Binding Sites) in NG108-15 Cells

Hayashi, T., & Su, T. (2003) · Journal of Pharmacology and Experimental Therapeutics · doi:10.1124/jpet.103.051292 · Cited by 189

The potential role of sigma-1 receptors in lipid transport and lipid raft reconstitution in the brain: Implication for drug abuse

Hayashi, T., & Su, T. (2005) · Life Sciences · doi:10.1016/j.lfs.2005.05.009 · Cited by 92

Detergent-Resistant Microdomains Determine the Localization of σ-1 Receptors to the Endoplasmic Reticulum-Mitochondria Junction

Hayashi, T., & Fujimoto, M. (2010) · Molecular Pharmacology · doi:10.1124/mol.109.062539 · Cited by 224

Sigma-1 Receptor Remodels Endoplasmic Reticulum Membrane

Zhemkov, V., & Борисович, Б. И. (2020) · Biophysical Journal · doi:10.1016/j.bpj.2019.11.1416

Subcellular Localization and Interacellular Dynamics of σ1 Receptors

Hayashi, T., & Su, T. (2007) · Springer eBooks · doi:10.1007/978-0-387-36514-5_8 · Cited by 2