Development of a second-generation antiandrogen for treatment of advanced prostate cancer.

Tran, Chris, Ouk, Samedy, Clegg, Nicola J., Chen, Yu, Watson, Philip A., Arora, Vivek, Wongvipat, John, Smith-Jones, Peter M. +11 more·2009·Science

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  55. An update on androgen deprivation therapy for prostate cancer
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  58. Loss of CHD1 Promotes Heterogeneous Mechanisms of Resistance to AR-Targeted Therapy via Chromatin Dysregulation
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  62. Nuclear receptors: recent drug discovery for cancer therapies.
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  67. Minireview: Alternative Activation Pathways for the Androgen Receptor in Prostate Cancer
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  68. Androgen-induced Long Noncoding RNA (lncRNA) SOCS2-AS1 Promotes Cell Growth and Inhibits Apoptosis in Prostate Cancer Cells
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  69. Natural-Products-Inspired Use of the gem -Dimethyl Group in Medicinal Chemistry
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  70. Biologic and clinical significance of androgen receptor variants in castration resistant prostate cancer
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  71. Second generation androgen receptor antagonists and challenges in prostate cancer treatment
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  72. Enzalutamide: targeting the androgen signalling pathway in metastatic castration‐resistant prostate cancer
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  74. Androgen Receptor on the Move: Boarding the Microtubule Expressway to the Nucleus
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