Quetiapine Nanoemulsion for Intranasal Drug Delivery: Evaluation of Brain-Targeting Efficiency

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Excipients Used for Modified Nasal Drug Delivery: A Mini-Review of the Recent Advances

Protopapa, C., Siamidi, A., Pavlou, P., & Vlachou, M. (2022) · Materials · doi:10.3390/ma15196547 · Cited by 22 · see citing works

NIOSOMES AS AN EMERGING FORMULATION TOOL FOR DRUG DELIVERY-A REVIEW

S., S. T., Mothilal, M., & Jaganathan, M. K. (2019) · International Journal of Applied Pharmaceutics · doi:10.22159/ijap.2019v11i2.30534 · Cited by 21 · see citing works

Mathematical Modeling and Simulation to Investigate the CNS Transport Characteristics of Nanoemulsion-Based Drug Delivery Following Intranasal Administration

Kadakia, E., Bottino, D. C., & Amiji, M. M. (2019) · Pharmaceutical Research · doi:10.1007/s11095-019-2610-y · Cited by 20 · see citing works

Nanocarriers for effective drug delivery

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Antipsychotics-Loaded Nanometric Emulsions for Brain Delivery

Pires, P. C., Paiva‐Santos, A. C., & Veiga, F. (2022) · Pharmaceutics · doi:10.3390/pharmaceutics14102174 · Cited by 18 · see citing works

Development and characterization of CD73-siRNA-loaded nanoemulsion: effect on C6 glioma cells and primary astrocytes

Teixeira, F. C., Bruxel, F., Azambuja, J. H., Berenguer, A. M., Stefani, M. A., Sévigny, J., Spanevello, R. M., Battastini, A. M. O., Teixeira, H. F., & Braganhol, E. (2019) · Pharmaceutical Development and Technology · doi:10.1080/10837450.2019.1705485 · Cited by 16 · see citing works

Development and Comparative In Vitro and In Vivo Study of BNN27 Mucoadhesive Liposomes and Nanoemulsions for Nose-to-Brain Delivery

Kannavou, M., Karali, K., Κάτσιλα, Θ., Siapi, E., Marazioti, A., Klepetsanis, P. G., Calogeropoulou, T., Charalampopoulos, I., & Antimisiaris, S. G. (2023) · Pharmaceutics · doi:10.3390/pharmaceutics15020419 · Cited by 16 · see citing works

Surface Modification of Nanoparticles to Oppose Uptake by the Mononuclear Phagocyte System

Parmar, K. R., & Patel, J. K. (2019) · Springer eBooks · doi:10.1007/978-3-030-06115-9_12 · Cited by 16 · see citing works

Exploring the potential of site-specific co-delivery of Berberine alongside 5-fluorouracil in oral cancer: Formulation development, in-vitro apoptosis, ex-vivo permeability and in-vivo biocompatibility studies

Tamane, P., Mahadik, K. R., & Pokharkar, V. (2022) · Journal of Drug Delivery Science and Technology · doi:10.1016/j.jddst.2022.103105 · Cited by 15 · see citing works

Nose to Brain Drug Delivery: A Recent Update

Chatterjee, B. (2018) · Journal of Formulation Science & Bioavailability · doi:10.4172/2577-0543.1000105 · Cited by 14 · see citing works

Design and Fabrication of Brain-Targeted Drug Delivery

Soni, V., Pandey, V., Asati, S., Jain, P., & Tekade, R. K. (2019) · Elsevier eBooks · doi:10.1016/b978-0-12-817909-3.00014-5 · Cited by 14 · see citing works

Dissolving Microneedles Patch: A Promising Approach for Advancing Transdermal Delivery of Antischizophrenic Drug

Umar, Q.-U.-A., Khan, M. I., Ahmad, Z., Akhtar, M. F., Sohail, M. F., Madni, A., Erum, A., Ayesha, B. T., Ain, Q. U., & Mushtaq, A. (2024) · Journal of Pharmaceutical Sciences · doi:10.1016/j.xphs.2024.08.011 · Cited by 12 · see citing works

Intranasal delivery of transferrin conjugated chitosan nanoparticles to the brain: A comparative analysis of conjugated and un-conjugated nanoparticles in vivo

Annu, Sartaj, A., Qamar, Z., Aldosari, E., Baboota, S., & Ali, J. (2024) · Journal of Drug Delivery Science and Technology · doi:10.1016/j.jddst.2024.106550 · Cited by 12 · see citing works

W/O/W Microemulsions for Nasal Delivery of Hydrophilic Compounds: A Preliminary Study

Cimino, C., Bonaccorso, A., Tomasello, B., Alberghina, G. A., Musumeci, T., Puglia, C., Pignatello, R., Marrazzo, A., & Carbone, C. (2024) · Journal of Pharmaceutical Sciences · doi:10.1016/j.xphs.2024.01.013 · Cited by 11 · see citing works

An Updated Review on Nanoemulsion: Factory for Food and Drug Delivery

Kumar, V., Garg, V., Saini, N., Aggarwal, N., Kumar, H., Kumar, D., Chopra, H., Kamal, M. A., & Dureja, H. (2024) · Current Pharmaceutical Biotechnology · doi:10.2174/0113892010267771240211124950 · Cited by 11 · see citing works

BBD assisted in-situ nanoliposomes of esculin hydrate via intranasal delivery for the amelioration of Parkinson's disease

Ansari, M. S., Ali, A., Rashid, M. A., Alhamhoom, Y., Sultana, N., Waheed, A., Alam, M. S., Aqil, M., & Sultana, Y. (2024) · Journal of Drug Delivery Science and Technology · doi:10.1016/j.jddst.2024.105658 · Cited by 10 · see citing works

Nanotechnology-Based Drug Delivery System

Bhutta, Z. A., Shoaib, M., Kanwal, A., Ashar, A., Mahfooz, A., Huma, H., Ahmed, R., Ali, M., Kulyar, M. F., & Li, K. (2022) · Advances in bioinformatics and biomedical engineering book series · doi:10.4018/978-1-7998-8908-3.ch005 · Cited by 10 · see citing works

Investigating the potential of highly porous zopiclone-loaded 3D electrospun nanofibers for brain targeting via the intranasal route

Taha, E., Nour, S. A. E.-K., Mamdouh, W., & Naguib, M. J. (2024) · International Journal of Pharmaceutics · doi:10.1016/j.ijpharm.2024.124230 · Cited by 9 · see citing works

Revolutionizing nanomedicine: Expanding horizons of nanoemulsions in drug delivery and beyond

Kumar, M., Chauhan, N., Kumar, D., Mahmood, S., Chopra, S., & Bhatia, A. (2024) · Journal of Dispersion Science and Technology · doi:10.1080/01932691.2024.2369835 · Cited by 9 · see citing works

Nose-to-brain delivery of biologics and stem cells

Agrawal, M., Konwar, A. N., Alexander, A., & Borse, V. B. (2021) · Elsevier eBooks · doi:10.1016/b978-0-12-822522-6.00015-1 · Cited by 9 · see citing works

Nanomaterials-mediated lysosomal regulation: a robust protein-clearance approach for the treatment of Alzheimer’s disease

Hao, M., Chu, J., Zhang, T., Yin, T., Gu, Y., Liang, W., Ji, W., Zhuang, J., Liu, Y., Gao, J., et al. (2024) · Neural Regeneration Research · doi:10.4103/nrr.nrr-d-23-01736 · Cited by 8 · see citing works

Polymer–lipid hybrid nanostructures for drug delivery

Gusmão, L. A., & Tedesco, A. C. (2022) · Elsevier eBooks · doi:10.1016/b978-0-323-85754-3.00003-4 · Cited by 8 · see citing works

Applications of innovative technologies to the delivery of antipsychotics

Bergonzi, M. C., Bilia, A. R., & Landucci, E. (2021) · Drug Discovery Today · doi:10.1016/j.drudis.2021.09.019 · Cited by 8 · see citing works

Phytomedicine nanoformulations for Parkinson's disease

Saji, C. V., Mohanakumar, K. P., & Shenoi, R. A. (2024) · Phytomedicine Plus · doi:10.1016/j.phyplu.2024.100704 · Cited by 7 · see citing works

Applications of nanoemulsions as drug delivery vehicle for phytoconstituents

Attama, A. A., Agbo, C. P., Onokala, O. B., Kenechukwu, F. C., Ugwueze, M. E., Mbah, C. C., Umeyor, C. E., Uronnachi, E., & Nnamani, P. O. (2023) · Elsevier eBooks · doi:10.1016/b978-0-323-99527-6.00017-3 · Cited by 7 · see citing works

Applications of Polymeric Nanoparticle in Nose to Brain Drug Delivery

Sunena, S., Kumar, S., Sulekha, S., Tomar, D., Kumar, D., & Kishore, V. (2023) · Research Journal of Pharmacy and Technology · doi:10.52711/0974-360x.2023.00988 · Cited by 6 · see citing works

Microfluidic Preparation and Evaluation of Multivesicular Liposomes Containing Gastrodin for Oral Delivery across the Blood–Brain Barrier

Luo, Y., Che, X., Zheng, G., Liu, Z., Xie, D., & Wang, L. (2024) · Molecular Pharmaceutics · doi:10.1021/acs.molpharmaceut.4c00582 · Cited by 6 · see citing works

Application of Nano-based Drug Loading Systems in the Treatment of Neurological Infections: An Updated Review

Sadigh‐Eteghad, S., Shahi, S., Mahmoudi, J., Farjami, A., Bazmani, A., Naghili, B., Dizaj, S. M., & Salatin, S. (2022) · Current Pharmaceutical Design · doi:10.2174/1381612828666220728092336 · Cited by 8 · see citing works

In vitro characterization of statistically optimized quetiapine-loaded self-nanoemulsified systems with quality by design

Katamreddy, J. D., Yalavarthi, P. R., Rao, D. S., Teja, S. S., & Battu, S. (2018) · International Journal of Pharmaceutical Investigation · doi:10.4103/jphi.jphi_9_18 · Cited by 6 · see citing works

Challenges in Targeting Nasal Passage and Nose-to-Brain Delivery via Nanoemulsions

Bahadur, S., & Pathak, K. (2023) · Springer eBooks · doi:10.1007/978-3-031-23112-4_5 · Cited by 6 · see citing works

Formulation and characterization of dolutegravir sodium-loaded nanostructured lipid carrier in situ gel for targeted brain delivery via intranasal route

Taher, S. S., & Al-Kinani, K. K. (2025) · OpenNano · doi:10.1016/j.onano.2025.100270 · Cited by 5 · see citing works

Preparations, Applications, Patents, and Marketed Formulations of Nanoemulsions - A Comprehensive Review

Chauhan, M., Mazumder, R., Rani, A., Mishra, R., & Pal, R. S. (2024) · Pharmaceutical Nanotechnology · doi:10.2174/0122117385325186240912110731 · Cited by 5 · see citing works

Pharmacokinetics of intranasal drugs, still a missed opportunity?

Sardu, M. L., & Poggesi, I. (2024) · Xenobiotica · doi:10.1080/00498254.2024.2349046 · Cited by 4 · see citing works

Surface-engineered Niosomes of Esculin Hydrate for the management of depression via intranasal route: Optimization, In vitro, Ex vivo and pharmacokinetic assessment

Alhowyan, A., Imran, M., Haque, A., & Kalam, M. A. (2024) · Journal of Drug Delivery Science and Technology · doi:10.1016/j.jddst.2024.106417 · Cited by 4 · see citing works

A nanochitosan-D-galactose formulation increases the accumulation of primaquine in the liver

Gomes, F., Ribeiro, A. C. D. M., Sanches, G. S., Borges, H. S., Takahashi, L. A. U., Daniel‐Ribeiro, C. T., Tedesco, A. C., Nascimento, J. W. L., & Carvalho, L. J. M. (2024) · Antimicrobial Agents and Chemotherapy · doi:10.1128/aac.00915-23 · Cited by 4 · see citing works

Formulation, Optimization and In Vitro Studies of Flutamide-loaded Nanostructured Lipid Carrier Based Oral Drug Delivery for Enhanced Anticancer Activity

Sabale, V., Nikam, M., & Sabale, P. (2024) · Journal of Pharmaceutical Innovation · doi:10.1007/s12247-024-09859-1 · Cited by 4 · see citing works

Optimization and Evaluation of Functionally Engineered Paliperidone Nanoemulsions for Improved Brain Delivery via Nasal Route

Sawant, N. D., Tatke, P. A., & Desai, N. D. (2025) · Molecular Pharmaceutics · doi:10.1021/acs.molpharmaceut.5c00786 · Cited by 4 · see citing works

Application of nanoemulsion in pharmaceuticals industry

Jadhav, K., Singh, R., Ray, E., & Verma, R. K. (2024) · Elsevier eBooks · doi:10.1016/b978-0-323-90047-8.00011-x · Cited by 4 · see citing works

DESIGN, OPTIMIZATION AND EVALUATION OF INTRANASAL NANOTHERAPEUTIC OF ATYPICAL ANTIPSYCHOTIC DRUG

(2023) · European Chemical Bulletin · doi:10.48047/ecb/2023.12.si4.437 · Cited by 3 · see citing works

Systematic Approach in the Development of Chitosan Functionalized Iloperidone Nanoemulsions for Transnasal Delivery, In Vitro and In Vivo Studies

Sawant, N. D., Tatke, P. A., & Desai, N. D. (2024) · AAPS PharmSciTech · doi:10.1208/s12249-024-02964-x · Cited by 3 · see citing works

Effective Brain Targeting Using the Self-Emulsifying Drug Delivery Systems

Gawde, S., Bachhav, Y. G., & Kumar, M. S. (2026) · AAPS PharmSciTech · doi:10.1208/s12249-026-03398-3 · Cited by 2 · see citing works

Approaches for the delivery of anti-parkinsonian therapeutic agents via the intranasal route

Banyyounes, J., & Obeid, M. A. (2026) · Discover Neuroscience · doi:10.1186/s13064-026-00258-5 · Cited by 2 · see citing works

Intranasal Delivery of Piceatannol-Loaded Liposomes for Glioblastoma Management: Formulation Optimization, In Vitro, Ex Vivo, In Ovo and LC-MS/MS- Based In Vivo Pharmacokinetic and Brain Distribution Assessment

Sikder, A., Katarpawar, S. N., Phatale, V., Kumar, R., Vambhurkar, G. B., Wagh, S. S., Pandey, G., Kolipaka, T., Dikundwar, A. G., & Srivastava, S. (2026) · BioNanoScience · doi:10.1007/s12668-026-02757-5 · Cited by 2 · see citing works

Drug Delivery System and Technologies

Guo, W., Ding, P., Okoro, O. V., Sun, Y., Jiang, G., Shavandi, A., & Nie, L. (2025) · Smart nanomaterials technology · doi:10.1007/978-981-97-8086-0_3 · Cited by 2 · see citing works

An Emerging Prospective of Antipsychotics for Treating Neurodegenerative Disorders

Kumar, B., Sahoo, A., Singhal, M., Varshney, G., Halder, T., & Bali, V. (2025) · Current Pharmaceutical Design · doi:10.2174/0113816128344910241211112452 · Cited by 2 · see citing works

Approaches in Barriers, Modifications, Route of Administrations, and Formulations of Therapeutic Agents for Brain Delivery

Kotha, A. K., Ghosh, S., Komanduri, N., Wang, R., Bhowmick, S., & Chougule, M. B. (2019) · Springer eBooks · doi:10.1007/978-981-13-3642-3_11 · Cited by 2 · see citing works

Evaluation of wound healing potential and biochemical estimation of sage oil nanoemulsion on animal model.

Alam, M. S., Ali, M. D., Ahmad, S., Banu, N., Ali, M. S., Alam, N., Ali, M. S., Ansari, M. S., Shamim, M., & Mujtaba, M. A. (2021) · PubMed · Cited by 2 · see citing works

Controlled Drug Delivery via the Nasal Route

Conway, B. R., & Ghori, M. U. (2021) · doi:10.1002/9781119769644.ch16 · Cited by 2 · see citing works

Intranasal carvacrol nanoemulsion: Stroke imaging and neuroprotective study

Mahajan, H. S., & Girnar, G. (2025) · ADMET & DMPK · doi:10.5599/admet.2967 · Cited by 1 · see citing works

Intranasal nanoemulsion for targeted medication delivery to the brain: a novel approach to treat psychotic disorder

Das, S., Sarkar, M., Bagchi, A., & Bahadur, S. (2026) · Drug Delivery and Translational Research · doi:10.1007/s13346-026-02054-4 · Cited by 1 · see citing works

In Vitro and In Vivo Evaluation of Quetiapine Fumarate Nanoemulsion for Brain Targeting Through Intranasal Route

Priya, S., Sequira, S., Shetty, S. S., Jyothi, D., James, J. P., Koland, M., & Merugumolu, V. K. (2024) · Indian Journal of Pharmaceutical Sciences · doi:10.36468/pharmaceutical-sciences.1352

DEVELOPMENT AND CHARACTERIZATION OF QUETIAPINE NANOEMULSION: A COMPREHENSIVE REVIEW OF FORMULATION STRATEGIES, CHARACTERIZATION TECHNIQUES, BRAIN TARGETING, AND THERAPEUTIC APPLICATIONS

B. Premkumar*, D. D. (2026) · Zenodo (CERN European Organization for Nuclear Research) · doi:10.5281/zenodo.21702229

Brain Targeting of Quetiapine Fumarate via Intranasal Delivery of Loaded Lipospheres: Fabrication, In-Vitro Evaluation, Optimization, and In-Vivo Assessment

Zaki, R. M., Aldawsari, M. F., Alossaimi, M. A., Alzaid, S. F., Seshadri, V. D., Almurshedi, A. S., Aldosari, B. N., Yusif, R. M., & Sayed, O. M. (2022) · Pharmaceuticals · doi:10.3390/ph15091083 · Cited by 12 · see citing works

Quetiapine Fumarate Loaded Mucoadhesive Nanoemulsion: Formulation, Optimization & Brain Delivery via Intranasal Administration

Setia, A., & Ahlawat, S. (2017) · Drug Delivery Letters · doi:10.2174/2210303106666160808113114 · Cited by 4 · see citing works

Non-invasive intranasal delivery of quetiapine fumarate loaded microemulsion for brain targeting: Formulation, physicochemical and pharmacokinetic consideration

Shah, B. M., Khunt, D., Misra, M., & Padh, H. (2016) · European Journal of Pharmaceutical Sciences · doi:10.1016/j.ejps.2016.05.008 · Cited by 92 · see citing works